| Compound ID |
Compound Name |
Compound Formula |
|
CP0034742
|
(R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-amide: 0.1C4H10O
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|
C25H20N4O2
|
1
|
| 1 |
Ki = 0.02344 nM
|
|
|
|
CP0160764
|
(R)-1-(1-(3,3-dimethyl-2-oxobutyl)-2-oxo-5-(pyridin-2-yl)-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-(3-(methylamino)phenyl)urea
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|
C28H30N6O3
|
1
|
| 1 |
Ki = 30.2 nM
|
|
|
|
CP0036767
|
S-L-365,260
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|
C24H22N4O2
|
1
|
| 1 |
Ki = 173.78 nM
|
|
|
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CP0399462
|
3-[[2-[5-(1-adamantyl)-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
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|
C33H38N4O5
|
1
|
| 1 |
Ki = 371.54 nM
|
|
|
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CP0445812
|
2-[3-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]phenyl]sulfanylacetic acid
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|
C30H36N4O5S
|
1
|
| 1 |
Ki = 645.65 nM
|
|
|
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CP0915570
|
2-((R)-5-cyclohexyl-2,3-dihydro-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1H-benzo[e][1,4]diazepin-3-yl)-N-(3-(methylamino)phenyl)-acetamide
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|
C30H38N4O3
|
1
|
| 1 |
Ki = 724.44 nM
|
|
|
|
CP0918905
|
2-((S)-5-cyclohexyl-2,3-dihydro-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1H-benzo[e][1,4]diazepin-3-yl)-N-(3-(methylamino)phenyl)-acetamide
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|
C30H38N4O3
|
1
|
| 1 |
Ki = 1174.9 nM
|
|
|
|
CP0437076
|
3-[[2-[1-[2-(1-adamantyl)-2-oxoethyl]-5-cyclohexyl-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
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|
C35H40N4O5
|
1
|
| 1 |
Ki = 1905.46 nM
|
|
|
|
CP0374443
|
3-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]-N-methylsulfonylbenzamide
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|
C30H37N5O6S
|
1
|
| 1 |
Ki = 2951.21 nM
|
|
|
|
CP0374442
|
2-[3-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]phenoxy]acetic acid
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|
C30H36N4O6
|
1
|
| 1 |
Ki = 4073.8 nM
|
|
|
|
CP0435584
|
3-[[2-[5-cycloheptyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
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|
C30H36N4O5
|
1
|
| 1 |
Ki = 5754.4 nM
|
|
|
|
CP0911234
|
2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-hydroxymethyl-phenyl)-acetamide
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|
C29H36N4O4
|
1
|
| 1 |
Ki = 5888.44 nM
|
|
|
|
CP0374445
|
2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]-N-[3-[methyl(2H-tetrazol-5-yl)amino]phenyl]acetamide
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|
C30H37N9O3
|
1
|
| 1 |
Ki = 6456.54 nM
|
|
|
|
CP0435586
|
3-[[2-[1-(3,3-dimethyl-2-oxobutyl)-2-oxo-5-propan-2-yl-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
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|
C26H30N4O5
|
1
|
| 1 |
Ki = 7079.46 nM
|
|
|
|
CP0512402
|
2-[3-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]anilino]acetic acid;hydrochloride
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|
C30H37N5O5
|
1
|
| 1 |
Ki = 8511.38 nM
|
|
|
|
CP0435604
|
2-[3-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]phenyl]acetic acid
Show/Hide
|
C30H36N4O5
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0077676
|
3-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
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|
C29H34N4O5
|
2
|
| 1 |
Ki = 11220.18 nM
|
|
|
| 2 |
Ki < 10000 nM
|
|
|
|
CP0044497
|
3-[[5-(1-adamantyloxymethyl)-2-cyclohexyl-1H-imidazole-4-carbonyl]amino]benzoic acid
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|
C28H35N3O4
|
1
|
| 1 |
Ki < 10000 nM
|
|
|
|
CP0374437
|
3-[[2-[5-cyclohexyl-1-(2-cyclopentyl-2-oxoethyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
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|
C30H34N4O5
|
1
|
| 1 |
Ki < 10000 nM
|
|
|
|
CP0377903
|
2-[3-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]phenyl]sulfonylacetic acid
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|
C30H36N4O7S
|
1
|
| 1 |
Ki < 10000 nM
|
|
|
|
CP0384935
|
3-[[2-[5-cyclohexyl-1-[2-(2-methylphenyl)-2-oxoethyl]-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
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|
C32H32N4O5
|
1
|
| 1 |
Ki < 10000 nM
|
|
|
|
CP0384937
|
3-[[2-(5-cyclohexyl-1-methyl-2-oxo-1,3,4-benzotriazepin-3-yl)acetyl]amino]benzoic acid
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|
C24H26N4O4
|
1
|
| 1 |
Ki < 10000 nM
|
|
|
|
CP0435585
|
3-[[2-[5-cyclopentyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
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|
C28H32N4O5
|
1
|
| 1 |
Ki < 10000 nM
|
|
|
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CP0437070
|
3-[[2-[5-cyclohexyl-2-oxo-1-(2-oxo-2-pyrrolidin-1-ylethyl)-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
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|
C29H33N5O5
|
1
|
| 1 |
Ki < 10000 nM
|
|
|
|
CP0443146
|
3-[[2-[5-cyclohexyl-2-oxo-1-(2-oxopropyl)-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
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|
C26H28N4O5
|
1
|
| 1 |
Ki < 10000 nM
|
|
|
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CP0486210
|
3-[[2-[5-cyclohexyl-1-(3-methylbutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
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|
C28H34N4O4
|
1
|
| 1 |
Ki < 10000 nM
|
|
|
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CP0911235
|
2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-pyrrolidin-1-yl-phenyl)-acetamide
Show/Hide
|
C32H41N5O3
|
1
|
| 1 |
Ki < 10000 nM
|
|
|
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CP0918907
|
2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-(2-ethoxy-ethylamino)-phenyl)-acetamide
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|
C32H43N5O4
|
1
|
| 1 |
Ki < 10000 nM
|
|
|
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CP0918908
|
2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-methylamino-phenyl)-acetamide
Show/Hide
|
C29H37N5O3
|
1
|
| 1 |
Ki < 10000 nM
|
|
|
