Compound ID |
Compound Name |
Compound Formula |
CP0219930
|
3-[(2R)-6-[3-fluoro-4-methoxy-6-(3-methoxycyclobutyl)oxypyridin-2-yl]-3,4-dihydro-2H-chromen-2-yl]propanoic acid
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|
C23H26FNO6
|
1
|
1 |
EC50 = 4.6 nM
|
|
|
CP0048202
|
3-[(2R)-6-[3,4-difluoro-6-(3-methoxycyclobutyl)oxypyridin-2-yl]-3,4-dihydro-2H-chromen-2-yl]propanoic acid
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|
C22H23F2NO5
|
1
|
1 |
EC50 = 6.8 nM
|
|
|
CP0172418
|
2-[3-[2-chloro-5-(trifluoromethoxy)phenyl]-3-azaspiro[5.5]undecan-9-yl]acetic acid
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|
C19H23ClF3NO3
|
1
|
1 |
EC50 = 54 nM
|
|
|
CP0396176
|
2-[3-(3,5-dichlorophenyl)-3-azaspiro[5.5]undecan-9-yl]acetic acid
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|
C18H23Cl2NO2
|
1
|
1 |
EC50 = 120 nM
|
|
|
CP0464379
|
2-[3-[3-cyano-5-(trifluoromethylsulfanyl)phenyl]-3-azaspiro[5.5]undecan-9-yl]acetic acid
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|
C20H23F3N2O2S
|
1
|
1 |
EC50 = 140 nM
|
|
|
CP0464376
|
2-[3-[2-cyano-5-(trifluoromethoxy)phenyl]-3-azaspiro[5.5]undecan-9-yl]acetic acid
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|
C20H23F3N2O3
|
1
|
1 |
EC50 = 290 nM
|
|
|
CP0466653
|
2-[3-[2-fluoro-5-(trifluoromethoxy)phenyl]-3-azaspiro[5.5]undecan-9-yl]acetic acid
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|
C19H23F4NO3
|
1
|
1 |
EC50 = 470 nM
|
|
|
CP0006743
|
4-methoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamide
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|
C16H19NO3S
|
1
|
1 |
EC50 = 630.96 nM
|
|
|
CP0461738
|
2-[3-(3-chloro-2,5-difluorophenyl)-3-azaspiro[5.5]undecan-9-yl]acetic acid
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|
C18H22ClF2NO2
|
1
|
1 |
EC50 = 1100 nM
|
|
|
CP0396175
|
2-[3-[2-fluoro-5-(trifluoromethyl)phenyl]-3-azaspiro[5.5]undecan-9-yl]acetic acid
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|
C19H23F4NO2
|
1
|
1 |
EC50 = 3000 nM
|
|
|
CP0516513
|
2-[3-(5-chloro-2,2-dimethyl-3H-1-benzofuran-7-yl)-3-azaspiro[5.5]undecan-9-yl]acetic acid
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|
C22H30ClNO3
|
1
|
1 |
EC50 = 4000 nM
|
|
|
CP0500271
|
2-[3-[4-(trifluoromethyl)pyridin-2-yl]-3-azaspiro[5.5]undecan-9-yl]acetic acid
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|
C18H23F3N2O2
|
1
|
1 |
EC50 = 4200 nM
|
|
|
CP0503952
|
2-[3-(2-chloro-5-methoxyphenyl)-3-azaspiro[5.5]undecan-9-yl]acetic acid
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|
C19H26ClNO3
|
1
|
1 |
EC50 = 5300 nM
|
|
|
CP0469180
|
2-[3-(2-chlorophenyl)-3-azaspiro[5.5]undecan-9-yl]acetic acid
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|
C18H24ClNO2
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0379890
|
4-methyl-N-(9H-xanthen-9-yl)benzenesulfonamide
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|
C20H17NO3S
|
1
|
1 |
IC50 = 7.943 nM
|
|
|