Brief Information of the Cell Line and Protein
Cell Line ID: CL000043 , U2OS
Synonyms
U-2 OS
U-2OS
U-2-OS
U2-OS
U20-S
U20S
2T
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0042
Protein ID: PT01779 , Sphingosine 1-phosphate receptor 4
Gene Name S1PR4
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID O95977
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000043  Protein ID: PT01779
 
Compound ID Compound Name Compound Formula
CP0496074
(2S,3R,5R)-5-[(hydrogen phosphonatooxy)methyl]-2-(hydroxymethyl)-3-(4-octylphenyl)pyrrolidin-1-ium
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C20H34NO5P
 1
1
EC50 = 7.4 nM
   TI
   LI
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   TS
CP0417200
(2R)-2-amino-3-[[4-(2-benzylphenyl)-1H-indole-2-carbonyl]amino]propanoic acid
   Show/Hide
C25H23N3O3
 1
1
EC50 = 10 nM
   TI
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   TS
CP0917730
(R)-2-amino-2-(6-octyl-1H-benzo[d]imidazol-2-yl)ethyl dihydrogenphosphate, 2,2,2-trifluoroacetate salt
   Show/Hide
C19H29F3N3O6P
 1
1
EC50 = 36 nM
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CP0440054
2-chloro-3-[2-(2,4-dichlorophenoxy)ethoxy]-6-(fluoromethyl)pyridine
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C14H11Cl3FNO2
 1
1
EC50 = 45 nM
   TI
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CP0397480
2,6-dibromo-3-[2-(2,4-dichlorophenoxy)ethoxy]pyridine
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C13H9Br2Cl2NO2
 1
1
EC50 = 46 nM
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CP0476125
2-bromo-3-[2-(2,4-dichlorophenoxy)ethoxy]-6-methyl-pyridine
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C14H12BrCl2NO2
 1
1
EC50 = 52 nM
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CP0461436
3-[2-(2,4-dichlorophenoxy)ethoxy]-2-iodo-6-methylpyridine
   Show/Hide
C14H12Cl2INO2
 1
1
EC50 = 54 nM
   TI
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   TS
CP0403196
(5Z)-5-[[1-(2,4-difluorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-(2-methoxyethylimino)-3-methyl-1,3-thiazolidin-4-one
   Show/Hide
C20H21F2N3O2S
 1
1
EC50 = 56 nM
   TI
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   TS
CP0399349
(5Z)-5-[(1-benzyl-2,5-dimethylpyrrol-3-yl)methylidene]-2-(2-methoxyethylimino)-3-methyl-1,3-thiazolidin-4-one
   Show/Hide
C21H25N3O2S
 1
1
EC50 = 68 nM
   TI
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CP0500471
(5Z)-5-[[1-[(2-fluorophenyl)methyl]-2,5-dimethylpyrrol-3-yl]methylidene]-3-methyl-2-methylimino-1,3-thiazolidin-4-one
   Show/Hide
C19H20FN3OS
 1
1
EC50 = 72 nM
   TI
   LI
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   TS
CP0440265
(5Z)-5-[[1-[(2,6-difluorophenyl)methyl]-2,5-dimethylpyrrol-3-yl]methylidene]-3-methyl-2-methylimino-1,3-thiazolidin-4-one
   Show/Hide
C19H19F2N3OS
 1
1
EC50 = 92 nM
   TI
   LI
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   TS
CP0391052
(5Z)-5-[[1-(2,4-difluorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-3-ethyl-2-ethylimino-1,3-thiazolidin-4-one
   Show/Hide
C20H21F2N3OS
 1
1
EC50 = 104 nM
   TI
   LI
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   TS
CP0440267
(5Z)-5-[[1-[(2,4-difluorophenyl)methyl]-2,5-dimethylpyrrol-3-yl]methylidene]-3-methyl-2-methylimino-1,3-thiazolidin-4-one
   Show/Hide
C19H19F2N3OS
 1
1
EC50 = 147 nM
   TI
   LI
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   TS
CP0262193
3-[2-(2,4-dichlorophenoxy)ethoxy]-6-methyl-2-nitro-pyridine
   Show/Hide
C14H12Cl2N2O4
 1
1
EC50 = 162 nM
   TI
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   TS
CP0456636
(5Z)-5-[[1-(2-fluorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-3-methyl-2-methylimino-1,3-thiazolidin-4-one
   Show/Hide
C18H18FN3OS
 1
1
EC50 = 205 nM
   TI
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CP0463524
2-bromo-3-[2-(2,4-dichlorophenoxy)ethoxy]-6-fluoropyridine
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C13H9BrCl2FNO2
 1
1
EC50 = 208 nM
   TI
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   TS
CP0428024
(5Z)-5-[[1-(2,4-difluorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-3-methyl-2-methylimino-1,3-thiazolidin-4-one
   Show/Hide
C18H17F2N3OS
 1
1
EC50 = 210 nM
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CP0501354
3-[2-(4-bromo-2-chlorophenoxy)ethoxy]-6-methyl-2-nitropyridine
   Show/Hide
C14H12BrClN2O4
 1
1
EC50 = 220 nM
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   TS
CP0523518
3-[2-(2-bromo-4-chlorophenoxy)ethoxy]-6-methyl-2-nitropyridine
   Show/Hide
C14H12BrClN2O4
 1
1
EC50 = 232 nM
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   TS
CP0438093
(5Z)-3-ethyl-2-ethylimino-5-[[1-(2-fluorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-1,3-thiazolidin-4-one
   Show/Hide
C20H22FN3OS
 1
1
EC50 = 250 nM
   TI
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   TS
CP0500477
(5Z)-5-[(1-benzyl-2,5-dimethylpyrrol-3-yl)methylidene]-3-methyl-2-methylimino-1,3-thiazolidin-4-one
   Show/Hide
C19H21N3OS
 1
1
EC50 = 262 nM
   TI
   LI
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CP0523521
[5-[2-(2,4-dichlorophenoxy)ethoxy]-6-iodopyridin-2-yl]methanol
   Show/Hide
C14H12Cl2INO3
 1
1
EC50 = 287 nM
   TI
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   TS
CP0496134
6-chloro-3-[2-(2,4-dichlorophenoxy)ethoxy]-2-nitropyridine
   Show/Hide
C13H9Cl3N2O4
 1
1
EC50 = 304 nM
   TI
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   TS
CP0475354
(5Z)-5-[[1-(2-fluorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-(2-hydroxyethylimino)-3-methyl-1,3-thiazolidin-4-one
   Show/Hide
C19H20FN3O2S
 1
1
EC50 = 306 nM
   TI
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   TS
CP0391050
(5Z)-5-[[1-[(2,6-difluorophenyl)methyl]-2,5-dimethylpyrrol-3-yl]methylidene]-3-ethyl-2-ethylimino-1,3-thiazolidin-4-one
   Show/Hide
C21H23F2N3OS
 1
1
EC50 = 314 nM
   TI
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   TS
CP0391053
(5Z)-5-[(1-benzyl-2,5-dimethylpyrrol-3-yl)methylidene]-2-(2-hydroxyethylimino)-3-methyl-1,3-thiazolidin-4-one
   Show/Hide
C20H23N3O2S
 1
1
EC50 = 396 nM
   TI
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   TS
CP0387901
(5Z)-5-[[1-(4-fluorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-3-methyl-2-methylimino-1,3-thiazolidin-4-one
   Show/Hide
C18H18FN3OS
 1
1
EC50 = 433 nM
   TI
   LI
   LO
   TS
CP0432808
(5Z)-5-[[1-(4-chloro-2-fluorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-3-methyl-2-methylimino-1,3-thiazolidin-4-one
   Show/Hide
C18H17ClFN3OS
 1
1
EC50 = 440 nM
   TI
   LI
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   TS
CP0425059
6-methyl-2-nitro-3-[2-(2,4,6-trichlorophenoxy)ethoxy]pyridine
   Show/Hide
C14H11Cl3N2O4
 1
1
EC50 = 570 nM
   TI
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   TS
CP0465762
3-[2-[4-bromo-2-(trifluoromethyl)phenoxy]ethoxy]-6-methyl-2-nitropyridine
   Show/Hide
C15H12BrF3N2O4
 1
1
EC50 = 601 nM
   TI
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   TS
CP0496076
(5Z)-5-[(2,5-dimethyl-1-phenylpyrrol-3-yl)methylidene]-3-ethyl-2-ethylimino-1,3-thiazolidin-4-one
   Show/Hide
C20H23N3OS
 1
1
EC50 = 602 nM
   TI
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CP0499464
2-chloro-3-[2-(2,4-dichlorophenoxy)ethoxy]-6-ethenylpyridine
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C15H12Cl3NO2
 1
1
EC50 = 658 nM
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CP0391051
(5Z)-5-[[2,5-dimethyl-1-(2-phenylethyl)pyrrol-3-yl]methylidene]-3-methyl-2-methylimino-1,3-thiazolidin-4-one
   Show/Hide
C20H23N3OS
 1
1
EC50 = 660 nM
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CP0873702
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-l,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-3-hydroxyazetidine-1-carboxamide
   Show/Hide
C25H25N5O4
 1
1
EC50 = 739 nM
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CP0452391
3-[3-(2,4-dichlorophenyl)propoxy]-6-methyl-2-nitropyridine
   Show/Hide
C15H14Cl2N2O3
 1
1
EC50 = 920 nM
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CP0399348
(5Z)-5-[[1-(2,4-difluorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-methylimino-1,3-thiazolidin-4-one
   Show/Hide
C17H15F2N3OS
 1
1
EC50 = 1000 nM
   TI
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CP0845580
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-l,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-hydroxyethanesulfonamide
   Show/Hide
C23H24N4O5S
 1
1
EC50 = 1210 nM
   TI
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CP0461435
2-bromo-3-[2-(2,4-dichlorophenoxy)ethoxy]pyridine
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C13H10BrCl2NO2
 1
1
EC50 = 1300 nM
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CP0462703
1-[2-(2,4-dichlorophenoxy)ethoxy]-4-methyl-2-nitrobenzene
   Show/Hide
C15H13Cl2NO4
 1
1
EC50 = 1300 nM
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CP0496135
[6-chloro-5-[2-(2,4-dichlorophenoxy)ethoxy]pyridin-2-yl]methanol
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C14H12Cl3NO3
 1
1
EC50 = 1500 nM
   TI
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CP0496075
(5Z)-5-[[1-(3-fluorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-3-methyl-2-methylimino-1,3-thiazolidin-4-one
   Show/Hide
C18H18FN3OS
 1
1
EC50 = 1600 nM
   TI
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CP0883372
(R)-5-(3-(1-(2-hydroxyethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazo1-5-yl)-2-isopropoxybenzonitrile
   Show/Hide
C23H24N4O3
 1
1
EC50 = 1610 nM
   TI
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CP0506142
(5Z)-5-[[1-(2,4-difluorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-3-(2-methoxyethyl)-2-methylimino-1,3-thiazolidin-4-one
   Show/Hide
C20H21F2N3O2S
 1
1
EC50 = 1700 nM
   TI
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CP0496077
(5Z)-5-[(2,5-dimethyl-1-pyridin-2-ylpyrrol-3-yl)methylidene]-3-methyl-2-methylimino-1,3-thiazolidin-4-one
   Show/Hide
C17H18N4OS
 1
1
EC50 = 1800 nM
   TI
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   TS
CP0452392
6-chloro-5-[2-(2,4-dichlorophenoxy)ethoxy]pyridine-2-carbaldehyde
   Show/Hide
C14H10Cl3NO3
 1
1
EC50 = 1800 nM
   TI
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CP0500476
(2Z,5Z)-5-[[1-(2-fluorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-pyridin-2-ylimino-1,3-thiazolidin-4-one
   Show/Hide
C21H17FN4OS
 1
1
EC50 = 2100 nM
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CP0478400
5-[2-(2,4-dichlorophenoxy)ethoxy]-6-iodopyridine-2-carbaldehyde
   Show/Hide
C14H10Cl2INO3
 1
1
EC50 = 2100 nM
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CP0461437
3-[2-(2,4-dichlorophenoxy)ethoxy]-2,6-dimethylpyridine
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C15H15Cl2NO2
 1
1
EC50 = 2600 nM
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CP0523520
3-[2-(2-chloro-4-fluorophenoxy)ethoxy]-6-methyl-2-nitropyridine
   Show/Hide
C14H12ClFN2O4
 1
1
EC50 = 2600 nM
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CP0399079
(5Z)-5-[[1-(2-fluorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-3-methyl-2-phenylimino-1,3-thiazolidin-4-one
   Show/Hide
C23H20FN3OS
 1
1
EC50 = 2800 nM
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CP0501356
3-[2-(2-fluoro-4-nitrophenoxy)ethoxy]-6-methyl-2-nitropyridine
   Show/Hide
C14H12FN3O6
 1
1
EC50 = 2800 nM
   TI
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CP0496338
3-[2-(2,4-dichlorophenoxy)ethoxy]-2-nitro-pyridine
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C13H10Cl2N2O4
 1
1
EC50 = 2980 nM
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CP0496078
(5Z)-5-[[1-(3-fluoropyridin-2-yl)-2,5-dimethylpyrrol-3-yl]methylidene]-3-methyl-2-methylimino-1,3-thiazolidin-4-one
   Show/Hide
C17H17FN4OS
 1
1
EC50 = 3100 nM
   TI
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CP0523519
3-[2-(4-chloro-2-fluorophenoxy)ethoxy]-6-methyl-2-nitropyridine
   Show/Hide
C14H12ClFN2O4
 1
1
EC50 = 3100 nM
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CP0466840
5-[2,5-dimethyl-3-[(Z)-(3-methyl-2-methylimino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]pyrrol-1-yl]-2-fluorobenzonitrile
   Show/Hide
C19H17FN4OS
 1
1
EC50 = 3200 nM
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CP0871095
(+/-)-2-((4-(5-(3,4,diethoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)amino)ethanol
   Show/Hide
C23H27N3O4
 1
1
EC50 = 3250 nM
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CP0467453
3-[2-(3-chloro-5-nitrophenoxy)ethoxy]-6-methyl-2-nitropyridine
   Show/Hide
C14H12ClN3O6
 1
1
EC50 = 3500 nM
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CP0495907
(5Z)-5-[[1-(2-fluorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-methylimino-1,3-thiazolidin-4-one
   Show/Hide
C17H16FN3OS
 1
1
EC50 = 3600 nM
   TI
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CP0496080
(5Z)-5-[[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]methylidene]-2-methylimino-1,3-thiazolidin-4-one
   Show/Hide
C15H13FN4OS
 1
1
EC50 = 3800 nM
   TI
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CP0473474
3-[2-(2-chloranyl-4-methoxy-phenoxy)ethoxy]-6-methyl-2-nitro-pyridine
   Show/Hide
C15H15ClN2O5
 1
1
EC50 = 3900 nM
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CP0248629
Ozanimod
   Show/Hide
C23H24N4O3
 1
1
EC50 = 4192 nM
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CP0461433
methyl 3-[2-(2,4-dichlorophenoxy)ethoxy]-6-methylpyridine-2-carboxylate
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C16H15Cl2NO4
 1
1
EC50 = 4800 nM
   TI
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   TS
CP0525009
(5Z)-3-ethyl-2-ethylimino-5-[[1-(3-fluoropyridin-2-yl)-2,5-dimethylpyrrol-3-yl]methylidene]-1,3-thiazolidin-4-one
   Show/Hide
C19H21FN4OS
 1
1
EC50 = 5400 nM
   TI
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CP0465761
3-[2-(4-chloro-2-methoxyphenoxy)ethoxy]-6-methyl-2-nitropyridine
   Show/Hide
C15H15ClN2O5
 1
1
EC50 = 5400 nM
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CP0861107
(+/-)-4-(5-(3,4,diethoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ol
   Show/Hide
C21H22N2O4
 1
1
EC50 = 5500 nM
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CP0492507
2-bromo-3-[2-(2,4-dichlorophenoxy)ethoxy]-6-phenylpyridine
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C19H14BrCl2NO2
 1
1
EC50 = 6000 nM
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CP0480520
3-[2-(2,4-dimethylphenoxy)ethoxy]-6-methyl-2-nitro-pyridine
   Show/Hide
C16H18N2O4
 1
1
EC50 = 7200 nM
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CP0463523
3-[2-(2,4-dichlorophenoxy)ethoxy]-2-ethyl-6-methylpyridine
   Show/Hide
C16H17Cl2NO2
 1
1
EC50 = 7300 nM
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CP0871098
(S)-5-(3-(1-amino-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
   Show/Hide
C21H20N4O2
 1
1
EC50 = 7866 nM
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CP0883375
(R)-5-(3-(1-amino-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxy-benzonitrile hydrochloride
   Show/Hide
C21H21ClN4O2
 1
1
EC50 = 9034 nM
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CP0845581
(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-methoxyethanesulfonamide
   Show/Hide
C24H26N4O5S
 1
1
EC50 > 10000 nM
   TI
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   TS
CP0848219
(R)-2-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazo1-3-yl)-2,3-dihydro-1H-inden-1-ylamino)-N,N-dimethylacetamide hydrochloride
   Show/Hide
C25H28ClN5O3
 1
1
EC50 > 10000 nM
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CP0848223
(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-3-hydroxyazetidine-1-carboxamide
   Show/Hide
C25H25N5O4
 1
1
EC50 > 10000 nM
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CP0861106
(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-hydroxyethanesulfonamide
   Show/Hide
C23H24N4O5S
 1
1
EC50 > 10000 nM
   TI
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CP0906147
(S)-2-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazo1-3-yl)-2,3-dihydro-1H-inden-1-ylamino)-N,N-dimethylacetamide
   Show/Hide
C25H27N5O3
 1
1
EC50 > 10000 nM
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   TS
CP0906148
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-meth-oxyethanesulfonamide
   Show/Hide
C24H26N4O5S
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0037883
5-(2,5-dichlorophenyl)-N-(4-(hydroxymethyl)-2,6-dimethylphenyl)furan-2-carboxamide
   Show/Hide
C20H17Cl2NO3
 1
1
IC50 = 21 nM
   TI
   LI
   LO
   TS
CP0037886
N-[4-(aminomethyl)-2,6-dimethylphenyl]-5-(2,5-dichlorophenyl)furan-2-carboxamide
   Show/Hide
C20H18Cl2N2O2
 1
1
IC50 = 25 nM
   TI
   LI
   LO
   TS
CP0037885
N-[4-(hydroxymethyl)-2,6-dimethylphenyl]-5-(3-methylthiophen-2-yl)furan-2-carboxamide
   Show/Hide
C19H19NO3S
 1
1
IC50 = 34 nM
   TI
   LI
   LO
   TS
CP0524460
4-(5-(2,5-dichlorophenyl)furan-2-carboxamido)-3,5-dimethylbenzyl acetate
   Show/Hide
C22H19Cl2NO4
 1
1
IC50 = 34 nM
   TI
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   LO
   TS
CP0164917
5-(2,5-dichlorophenyl)-N-(2-ethyl-6-methylphenyl)furan-2-carboxamide
   Show/Hide
C20H17Cl2NO2
 1
1
IC50 = 41 nM
   TI
   LI
   LO
   TS
CP0037887
5-(2,5-dichlorophenyl)-N-(4-(2-hydroxyethoxy)-2,6-dimethylphenyl)furan-2-carboxamide
   Show/Hide
C21H19Cl2NO4
 1
1
IC50 = 44 nM
   TI
   LI
   LO
   TS
CP0075105
N-(4-hydroxy-2,6-dimethylphenyl)-5-(3-methylthiophen-2-yl)furan-2-carboxamide
   Show/Hide
C18H17NO3S
 1
1
IC50 = 46 nM
   TI
   LI
   LO
   TS
CP0524458
N-[4-(2-amino-2-oxoethoxy)-2,6-dimethylphenyl]-5-(2,5-dichlorophenyl)furan-2-carboxamide
   Show/Hide
C21H18Cl2N2O4
 1
1
IC50 = 52 nM
   TI
   LI
   LO
   TS
CP0075101
5-(2,5-dichlorophenyl)-N-(4-hydroxy-2,6-dimethylphenyl)furan-2-carboxamide
   Show/Hide
C19H15Cl2NO3
 1
1
IC50 = 58 nM
   TI
   LI
   LO
   TS
CP0272018
5-(2,5-dimethylphenyl)-N-(2,6-dimethylphenyl)thiophene-2-carboxamide
   Show/Hide
C21H21NOS
 1
1
IC50 = 59 nM
   TI
   LI
   LO
   TS
CP0488392
5-(2,5-dichlorophenyl)-N-mesitylfuran-2-carboxamide
   Show/Hide
C20H17Cl2NO2
 1
1
IC50 = 63 nM
   TI
   LI
   LO
   TS
CP0378115
5-(2,5-dimethylphenyl)-N-(2,6-dimethylphenyl)furan-2-carboxamide
   Show/Hide
C21H21NO2
 1
1
IC50 = 64 nM
   TI
   LI
   LO
   TS
CP0191730
3-(2,5-dimethylphenyl)-N-(2,6-dimethylphenyl)benzamide
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C23H23NO
 1
1
IC50 = 75 nM
   TI
   LI
   LO
   TS
CP0291357
5-(2,5-dichlorophenyl)-N-(2,6-dimethylphenyl)-2-furamide
   Show/Hide
C19H15Cl2NO2
 1
1
IC50 = 78 nM
   TI
   LI
   LO
   TS
CP0190953
5-(2,5-dichlorophenyl)-N-(4-methoxy-2,6-dimethylphenyl)furan-2-carboxamide
   Show/Hide
C20H17Cl2NO3
 1
1
IC50 = 80 nM
   TI
   LI
   LO
   TS
CP0199380
5-(2,5-dichlorophenyl)-N-(2,6-diethylphenyl)-2-furamide
   Show/Hide
C21H19Cl2NO2
 1
1
IC50 = 89 nM
   TI
   LI
   LO
   TS
CP0075104
N-(2,6-dimethylphenyl)-5-(3-methylthiophen-2-yl)furan-2-carboxamide
   Show/Hide
C18H17NO2S
 1
1
IC50 = 93 nM
   TI
   LI
   LO
   TS
CP0459514
N-[4-(acetamidomethyl)-2,6-dimethylphenyl]-5-(2,5-dichlorophenyl)furan-2-carboxamide
   Show/Hide
C22H20Cl2N2O3
 1
1
IC50 = 94 nM
   TI
   LI
   LO
   TS
CP0373149
5-(2,5-dichlorophenyl)-N-(2,6-diisopropylphenyl)-2-furamide
   Show/Hide
C23H23Cl2NO2
 1
1
IC50 = 105 nM
   TI
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   TS
CP0524461
5-(2,5-dichlorophenyl)-N-(3,5-dimethylbiphenyl-4-yl)furan-2-carboxamide
   Show/Hide
C25H19Cl2NO2
 1
1
IC50 = 115 nM
   TI
   LI
   LO
   TS
CP0505019
N-(2,6-dimethylphenyl)-5-thiophen-2-ylfuran-2-carboxamide
   Show/Hide
C17H15NO2S
 1
1
IC50 = 118 nM
   TI
   LI
   LO
   TS
CP0373143
N-(2,6-dimethylphenyl)-5-(furan-2-yl)-N-methylfuran-2-carboxamide
   Show/Hide
C18H17NO3
 1
1
IC50 = 130 nM
   TI
   LI
   LO
   TS
CP0424622
5-(2,5-dichlorophenyl)-N-(2-methoxy-6-methyl-phenyl)-2-furamide
   Show/Hide
C19H15Cl2NO3
 1
1
IC50 = 163 nM
   TI
   LI
   LO
   TS
CP0487484
5-(2,5-dichlorophenyl)-N-(2,5-dimethylphenyl)-2-furamide
   Show/Hide
C19H15Cl2NO2
 1
1
IC50 = 165 nM
   TI
   LI
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   TS
CP0459159
5-[2,5-bis(chloranyl)phenyl]-N-(2-chloranyl-6-methyl-phenyl)furan-2-carboxamide
   Show/Hide
C18H12Cl3NO2
 1
1
IC50 = 169 nM
   TI
   LI
   LO
   TS
CP0530966
5-(2,5-dimethylphenyl)-N-(2,6-dimethylphenyl)-3-methylfuran-2-carboxamide
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C22H23NO2
 1
1
IC50 = 173 nM
   TI
   LI
   LO
   TS
CP0455494
4-(2,5-dimethylphenyl)-N-(2,6-dimethylphenyl)furan-2-carboxamide
   Show/Hide
C21H21NO2
 1
1
IC50 = 211 nM
   TI
   LI
   LO
   TS
CP0503194
5-(2,5-dimethylphenyl)-N-(2,6-dimethylphenyl)furan-3-carboxamide
   Show/Hide
C21H21NO2
 1
1
IC50 = 233 nM
   TI
   LI
   LO
   TS
CP0385591
5-(2,5-dichlorophenyl)-N-(2-methyl-1-naphthalenyl)-2-furancarboxamide
   Show/Hide
C22H15Cl2NO2
 1
1
IC50 = 253 nM
   TI
   LI
   LO
   TS
CP0390703
5-(2-chlorophenyl)-N-(2,6-dimethylphenyl)-N-methylfuran-2-carboxamide
   Show/Hide
C20H18ClNO2
 1
1
IC50 = 269 nM
   TI
   LI
   LO
   TS
CP0378116
N-(2,6-dimethylphenyl)-5-(4-methyl-3-thienyl)-2-furamide
   Show/Hide
C18H17NO2S
 1
1
IC50 = 286 nM
   TI
   LI
   LO
   TS
CP0439056
5-(2,5-dichlorophenyl)-N-(2,6-dimethyl-3-methylsulfonylphenyl)-2-furancarboxamide
   Show/Hide
C20H17Cl2NO4S
 1
1
IC50 = 302 nM
   TI
   LI
   LO
   TS
CP0472583
5-(2,5-difluorophenyl)-N-(2,6-dimethylphenyl)-2-furamide
   Show/Hide
C19H15F2NO2
 1
1
IC50 = 308 nM
   TI
   LI
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   TS
CP0456357
5-(2,5-dichlorophenyl)-N-(4-((dimethylamino)methyl)-2,6-dimethylphenyl)furan-2-carboxamide
   Show/Hide
C22H22Cl2N2O2
 1
1
IC50 = 348 nM
   TI
   LI
   LO
   TS
CP0437509
5-(2,5-dichlorophenyl)-N-(2,6-dimethoxyphenyl)-2-furamide
   Show/Hide
C19H15Cl2NO4
 1
1
IC50 = 417 nM
   TI
   LI
   LO
   TS
CP0520934
N-(2,6-dimethylphenyl)-5-thiophen-3-ylfuran-2-carboxamide
   Show/Hide
C17H15NO2S
 1
1
IC50 = 448 nM
   TI
   LI
   LO
   TS
CP0397767
5-(3-chlorophenyl)-N-(2,6-dimethylphenyl)-2-furamide
   Show/Hide
C19H16ClNO2
 1
1
IC50 = 497 nM
   TI
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   TS
CP0512507
5-(2,5-dimethoxyphenyl)-N-(2,6-dimethylphenyl)-N-methylfuran-2-carboxamide
   Show/Hide
C22H23NO4
 1
1
IC50 = 513 nM
   TI
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   TS
CP0505020
5-(5-chlorothiophen-2-yl)-N-(2,6-dimethylphenyl)furan-2-carboxamide
   Show/Hide
C17H14ClNO2S
 1
1
IC50 = 515 nM
   TI
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   LO
   TS
CP0460398
5-(2,5-dichlorophenyl)-N-(2-(hydroxymethyl)-6-methylphenyl)furan-2-carboxamide
   Show/Hide
C19H15Cl2NO3
 1
1
IC50 = 573 nM
   TI
   LI
   LO
   TS
CP0512773
N-(2,6-dimethylphenyl)-5-phenylfuran-2-carboxamide
   Show/Hide
C19H17NO2
 1
1
IC50 = 575 nM
   TI
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CP0502791
5-(2,5-dichlorophenyl)-N-(4-methoxy-2-methylphenyl)furan-2-carboxamide
   Show/Hide
C19H15Cl2NO3
 1
1
IC50 = 589 nM
   TI
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   LO
   TS
CP0488296
5-(2,5-dimethylphenyl)-N-(2,6-dimethylphenyl)-4-methylfuran-2-carboxamide
   Show/Hide
C22H23NO2
 1
1
IC50 = 911 nM
   TI
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   TS
CP0378114
5-(2,5-dichlorophenyl)-N-(5-methoxy-2-methylphenyl)furan-2-carboxamide
   Show/Hide
C19H15Cl2NO3
 1
1
IC50 = 931 nM
   TI
   LI
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   TS
CP0456913
5-(2,4-dichlorophenyl)-N-(2,6-dimethylphenyl)-2-furamide
   Show/Hide
C19H15Cl2NO2
 1
1
IC50 = 2000 nM
   TI
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CP0530967
3-(2,5-dimethylphenyl)-N-(2,6-dimethylphenyl)-4-methylbenzamide
   Show/Hide
C24H25NO
 1
1
IC50 = 2400 nM
   TI
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CP0449291
5-(2,5-dimethylphenyl)-N-(2,6-dimethylphenyl)-1-methylpyrrole-2-carboxamide
   Show/Hide
C22H24N2O
 1
1
IC50 = 6300 nM
   TI
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CP0479452
5-(2,5-dichlorophenyl)-N-(2,6-difluorophenyl)furan-2-carboxamide
   Show/Hide
C17H9Cl2F2NO2
 1
1
IC50 = 6400 nM
   TI
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   TS
CP0479454
5-(2,5-dichlorophenyl)-N-mesityl-N-methylfuran-2-carboxamide
   Show/Hide
C21H19Cl2NO2
 1
1
IC50 = 8100 nM
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   TS