Brief Information of the Cell Line and Protein
Cell Line ID: CL000043 , U2OS
 Cell Line Info 
Synonyms
U-2 OS
U-2OS
U-2-OS
U2-OS
U20-S
U20S
2T
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0042
Protein ID: PT01298 , Cannabinoid receptor 1
 Protein Info 
Gene Name CNR1
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P21554
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000043
 Cell Line Info 
 Protein ID: PT01298
 Protein Info 
 
Compound ID Compound Name Compound Formula
CP0048192
 Compound Info 
2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohexyl)-5-(2-methyloctan-2-yl)phenol
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C24H40O3
  1
1
EC50 = 5.754 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0438382
 Compound Info 
AM4054
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C26H36O3
  1
1
EC50 = 96 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0449572
 Compound Info 
(6aR,10aR)-3-(1-adamantyl)-9-(hydroxymethyl)-6,6-dimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-1-ol
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C26H34O3
  1
1
EC50 = 230 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0425336
 Compound Info 
AM4089
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C26H30O3
  1
1
EC50 = 450 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0085444
 Compound Info 
(6aR,10aR)-3-Adamantan-1-yl-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol
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C26H34O2
  1
1
EC50 = 1530 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0050487
 Compound Info 
(11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphthalen-1-ylcarbonyl)-9-oxa-1-azatricyclo[6.3.1.0^{4,12}]dodeca-2,4(12),5,7-tetraene
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C27H26N2O3
  1
1
EC50 = 1760 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0396544
 Compound Info 
(E)-3-(2-methoxyphenyl)-N-[[4-[methyl(phenyl)sulfamoyl]phenyl]carbamothioyl]prop-2-enamide
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C24H23N3O4S2
  1
1
EC50 > 30000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0396545
 Compound Info 
MLS000569095
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C23H18FN5O2S2
  1
1
EC50 > 30000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0456697
 Compound Info 
3-[4-(2,3-dimethylphenyl)piperazin-1-yl]carbonyl-N,N-dimethyl-4-pyrrolidin-1-yl-benzenesulfonamide
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C25H34N4O3S
  1
1
EC50 > 30000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS