| Compound ID |
Compound Name |
Compound Formula |
|
CP0421772
|
methyl 7-[2-[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]ethoxy]-2-oxochromene-3-carboxylate
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|
C24H21NO6
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0421773
|
methyl 7-[2-[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]ethoxy]-2-oxochromene-3-carboxylate
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|
C24H21NO6
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0434889
|
methyl 7-[2-[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]ethoxy]-2-oxo-3,4-dihydrochromene-3-carboxylate
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|
C24H23NO6
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0434893
|
methyl 7-[2-[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]ethoxy]-2-oxo-3,4-dihydrochromene-3-carboxylate
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|
C24H23NO7
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0491338
|
methyl 7-[2-[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]ethoxy]-2-oxo-3,4-dihydrochromene-3-carboxylate
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|
C23H20FNO6
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0502422
|
methyl 7-[2-[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]ethoxy]-2-oxochromene-3-carboxylate
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|
C24H21NO7
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0502423
|
methyl 7-[2-[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]ethoxy]-2-oxo-3,4-dihydrochromene-3-carboxylate
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|
C24H23NO6
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0005387
|
Avandamet
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|
C18H19N3O3S
|
2
|
| 1 |
EC50 = 20 nM
|
|
|
| 2 |
EC50 = 50 nM
|
|
|
|
CP0434894
|
methyl 7-[2-[2-(3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]ethoxy]-2-oxo-3,4-dihydrochromene-3-carboxylate
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|
C24H23NO7
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0434891
|
7-[2-(5-Methyl-2-phenyl-oxazol-4-yl)-ethoxy]-2-oxo-chroman-3-carboxylic acid methyl ester
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|
C23H21NO6
|
1
|
| 1 |
EC50 = 130 nM
|
|
|
|
CP0491337
|
methyl 7-[2-[5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl]ethoxy]-2-oxo-3,4-dihydrochromene-3-carboxylate
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|
C24H20F3NO6
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
|
CP0421777
|
methyl 7-[2-[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]ethoxy]-2-oxo-3,4-dihydrochromene-3-carboxylate
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|
C23H20FNO6
|
1
|
| 1 |
EC50 = 170 nM
|
|
|
|
CP0491370
|
methyl 7-[2-[2-(4-tert-butylphenyl)-5-methyl-1,3-oxazol-4-yl]ethoxy]-2-oxo-3,4-dihydrochromene-3-carboxylate
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|
C27H29NO6
|
1
|
| 1 |
EC50 = 250 nM
|
|
|
|
CP0421776
|
methyl 7-[2-[2-(3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]ethoxy]-2-oxochromene-3-carboxylate
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|
C24H21NO7
|
1
|
| 1 |
EC50 = 350 nM
|
|
|
|
CP0417458
|
methyl 7-[2-[5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl]ethoxy]-2-oxochromene-3-carboxylate
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|
C24H18F3NO6
|
1
|
| 1 |
EC50 = 420 nM
|
|
|
|
CP0507965
|
methyl 7-[2-[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]ethoxy]-2-oxochromene-3-carboxylate
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|
C23H18FNO6
|
1
|
| 1 |
EC50 = 960 nM
|
|
|
|
CP0491339
|
methyl 7-[2-[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]ethoxy]-2-oxo-3,4-dihydrochromene-3-carboxylate
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|
C29H25NO6
|
1
|
| 1 |
EC50 = 1120 nM
|
|
|
|
CP0421785
|
methyl 7-[2-[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]ethoxy]-2-oxochromene-3-carboxylate
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|
C29H23NO6
|
1
|
| 1 |
EC50 = 1260 nM
|
|
|
|
CP0491340
|
methyl 7-[2-[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]ethoxy]-2-oxochromene-3-carboxylate
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|
C23H18FNO6
|
1
|
| 1 |
EC50 = 1620 nM
|
|
|
|
CP0387527
|
methyl 7-[2-[2-(4-tert-butylphenyl)-5-methyl-1,3-oxazol-4-yl]ethoxy]-2-oxochromene-3-carboxylate
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|
C27H27NO6
|
1
|
| 1 |
EC50 = 1740 nM
|
|
|
|
CP0404977
|
3-{4-[2-Amino-6-(4-(naphthalen-1-ylmethyl)-piperazin-1-yl)-pyrimidin-4-yloxy]-phenyl}-2-methyl-2-phenoxypropionic acid
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|
C35H35N5O4
|
1
|
| 1 |
EC50 = 3500 nM
|
|
|
|
CP0499088
|
methyl 7-[2-[5-methyl-2-(3-nitrophenyl)-1,3-oxazol-4-yl]ethoxy]-2-oxochromene-3-carboxylate
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|
C23H18N2O8
|
1
|
| 1 |
EC50 = 3550 nM
|
|
|
|
CP0375697
|
3-{4-{2-Amino-6-[4-(3-methyl-benzyl)-piperazin-1-yl]-pyrimidin-4-yloxy}-phenyl}-2-methyl-2-phenoxy-propionic acid
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|
C32H35N5O4
|
1
|
| 1 |
EC50 = 4460 nM
|
|
|
|
CP0429893
|
3-{4-{2-Amino-6-[4-(3-chloro-phenyl)-piperazin-1-yl]-pyrimidin-4-yloxy}-phenyl}-2-methyl-2-phenoxy-propionic acid
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|
C30H30ClN5O4
|
1
|
| 1 |
EC50 = 4470 nM
|
|
|
|
CP0375698
|
3-{4-{2-Amino-6-[4-(3-trifluoromethyl-benzyl)-piperazin-1-yl]-pyrimidin-4-yloxy}-phenyl}-2-methyl-2-phenoxy-propionic acid
Show/Hide
|
C32H32F3N5O4
|
1
|
| 1 |
EC50 = 4790 nM
|
|
|
|
CP0404978
|
3-{4-[2-Amino-6-(4-phenyl-piperazin-1-yl)-pyrimidin-4-yloxy]-phenyl}-2-methyl-2-phenoxy-propionic acid
Show/Hide
|
C30H31N5O4
|
1
|
| 1 |
EC50 = 4940 nM
|
|
|
|
CP0429892
|
3-{4-[2-Amino-6-(4-furan-2-ylmethyl-piperazin-1-yl)-pyrimidin-4-yloxy]-phenyl}-2-methyl-2-phenoxy-propionic acid
Show/Hide
|
C29H31N5O5
|
1
|
| 1 |
EC50 = 5010 nM
|
|
|
|
CP0375695
|
3-{4-[2-Amino-6-(4-cyclohexylmethyl-piperazin-1-yl)-pyrimidin-4-yloxy]-phenyl}-2-methyl-2-phenoxy-propionic acid
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|
C31H39N5O4
|
1
|
| 1 |
EC50 = 5540 nM
|
|
|
|
CP0439276
|
3-{4-[2-Amino-6-(4-pyrimidin-2-yl-piperazin-1-yl)-pyrimidin-4-yloxy]-phenyl}-2-methyl-2-phenoxy-propionic acid
Show/Hide
|
C28H29N7O4
|
1
|
| 1 |
EC50 = 6130 nM
|
|
|
|
CP0506141
|
3-{4-{2-Amino-6-[4-(4-tert-butyl-benzyl)-piperazin-1-yl]-pyrimidin-4-yloxy}-phenyl}-2-methyl-2-phenoxy-propionic acid
Show/Hide
|
C35H41N5O4
|
1
|
| 1 |
EC50 = 6360 nM
|
|
|
|
CP0375696
|
3-{4-[2-Amino-6-(4-benzyl-piperazin-1-yl)-pyrimidin-4-yloxy]-phenyl}-2-methyl-2-phenoxy-propionic acid
Show/Hide
|
C31H33N5O4
|
1
|
| 1 |
EC50 = 6620 nM
|
|
|
|
CP0474559
|
3-{4-[2-Amino-6-(4-benzoyl-piperazin-1-yl)-pyrimidin-4-yloxy]-phenyl}-2-methyl-2-phenoxy-propionic acid
Show/Hide
|
C31H31N5O5
|
1
|
| 1 |
EC50 >= 50000 nM
|
|
|
|
CP0503927
|
3-{4-{2-Amino-6-[4-(4-propyl-benzoyl)-piperazin-1-yl]-pyrimidin-4-yloxy}-phenyl}-2-methyl-2-phenoxy-propionic acid
Show/Hide
|
C34H37N5O5
|
1
|
| 1 |
EC50 >= 50000 nM
|
|
|
|
CP0857631
|
3-{4-{2-Amino-6-[4-(2-methoxy-benzoyl)-piperazin-1-yl]-pyrimidin-4-yloxy}-phenyl}-2-methyl-2-phenoxy-propionic acid
Show/Hide
|
C32H33N5O6
|
1
|
| 1 |
EC50 >= 50000 nM
|
|
|
|
CP0874379
|
3-{4-[2-Amino-6-(4-pyridin-2-ylmethyl-piperazin-1-yl)-pyrimidin-4-yloxy]-phenyl}-2-methyl-2-phenoxy-propionic acid
Show/Hide
|
C30H32N6O4
|
1
|
| 1 |
EC50 >= 50000 nM
|
|
|
|
CP0893219
|
3-(4-(2-Amino-6-(4-(furan-2-carbonyl)piperazin-1-yl)pyrimidin-4-yloxy)phenyl)-2-methyl-2-phenoxypropanoic acid
Show/Hide
|
C29H29N5O6
|
1
|
| 1 |
EC50 >= 50000 nM
|
|
|
