Brief Information of the Cell Line and Protein
Cell Line ID: CL000040 , THP-1
Synonyms
THP1
THP 1
THPI
THP-1(ATCC)
THP-1-O
O-THP-1
Tohoku Hospital Pediatrics-1
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0006
Protein ID: PT05434 , P2Y purinoceptor 14
Gene Name P2RY14
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID Q15391
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000040  Protein ID: PT05434
 
Compound ID Compound Name Compound Formula
CP0435758
3-[(4-methylbenzoyl)amino]-5-(4-piperidin-4-ylphenyl)benzoic acid
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C26H26N2O3
 1
1
IC50 = 1.77 nM
   TI
   LI
   LO
   TS
CP0032210
4-(4-piperidin-4-ylphenyl)-7-[4-(trifluoromethyl)phenyl]naphthalene-2-carboxylic acid
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C29H24F3NO2
 1
1
IC50 = 1.98 nM
   TI
   LI
   LO
   TS
CP0520379
3-(4-piperidin-4-ylphenyl)-5-(pyridine-4-carbonylamino)benzoic acid
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C24H23N3O3
 1
1
IC50 = 3.17 nM
   TI
   LI
   LO
   TS
CP0538507
3-(4-piperidin-4-ylphenyl)-5-(pyrazine-2-carbonylamino)benzoic acid
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C23H22N4O3
 1
1
IC50 = 4.35 nM
   TI
   LI
   LO
   TS
CP0435755
3-[(4-cyanobenzoyl)amino]-5-(4-piperidin-4-ylphenyl)benzoic acid
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C26H23N3O3
 1
1
IC50 = 4.54 nM
   TI
   LI
   LO
   TS
CP0473891
3-benzamido-5-(4-piperidin-4-ylphenyl)benzoic acid
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C25H24N2O3
 1
1
IC50 = 4.95 nM
   TI
   LI
   LO
   TS
CP0435756
3-[(4-nitrobenzoyl)amino]-5-(4-piperidin-4-ylphenyl)benzoic acid
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C25H23N3O5
 1
1
IC50 = 5.06 nM
   TI
   LI
   LO
   TS