| Compound ID |
Compound Name |
Compound Formula |
|
CP0550348
|
tert-butyl N-[3-[6-carbamoyl-3-[(E)-4-[5-carbamoyl-2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]-7-methoxybenzimidazol-1-yl]but-2-enyl]-2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]benzimidazol-4-yl]oxypropyl]carbamate
Show/Hide
|
C43H53N13O8
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0550242
|
4-[5-[3-[[2-(3-carboxy-3-methylbutanoyl)-4-fluoro-6-methoxy-1-benzothiophen-5-yl]oxy]propoxy]-4-fluoro-6-methoxy-1-benzothiophen-2-yl]-2,2-dimethyl-4-oxobutanoic acid
Show/Hide
|
C33H34F2O10S2
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0444686
|
9-[(1R,6R,8R,9R,10R,15R,17R,18R)-17-(6-aminopurin-9-yl)-9,18-difluoro-3-hydroxy-12-oxo-12-sulfanyl-3-sulfanylidene-2,4,7,11,13,16-hexaoxa-3lambda5,12lambda5-diphosphatricyclo[13.3.0.06,10]octadecan-8-yl]-1H-purin-6-one
Show/Hide
|
C20H21F2N9O9P2S2
|
2
|
| 1 |
EC50 = 300 nM
|
|
|
| 2 |
EC50 = 1600 nM
|
|
|
|
CP0248590
|
benzyl N-[3-[5-carbamoyl-2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]-7-methoxybenzimidazol-1-yl]propyl]carbamate
Show/Hide
|
C27H31N7O5
|
1
|
| 1 |
EC50 = 872 nM
|
|
|
|
CP0534593
|
9-[(1R,6R,8R,9R,10R,15R,17R,18R)-17-(6-aminopurin-9-yl)-9,18-difluoro-3,12-dihydroxy-3,12-dioxo-2,4,7,11,13,16-hexaoxa-3lambda5,12lambda5-diphosphatricyclo[13.3.0.06,10]octadecan-8-yl]-1H-purin-6-one
Show/Hide
|
C20H21F2N9O11P2
|
2
|
| 1 |
EC50 = 1100 nM
|
|
|
| 2 |
EC50 = 15400 nM
|
|
|
|
CP0243314
|
benzyl N-[3-[5-carbamoyl-2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]-7-(3-morpholin-4-ylpropoxy)benzimidazol-1-yl]propyl]carbamate
Show/Hide
|
C33H42N8O6
|
1
|
| 1 |
EC50 = 1140 nM
|
|
|
|
CP0069029
|
tert-butyl N-[3-[5-carbamoyl-2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]-7-methoxybenzimidazol-1-yl]propyl]carbamate
Show/Hide
|
C24H33N7O5
|
1
|
| 1 |
EC50 = 1240 nM
|
|
|
|
CP0532334
|
9-[(1R,6R,8R,10S,15R,17R,18R)-17-(6-aminopurin-9-yl)-18-fluoro-3,12-dihydroxy-3,12-dioxo-2,4,7,11,13,16-hexaoxa-3lambda5,12lambda5-diphosphatricyclo[13.3.0.06,10]octadecan-8-yl]-1H-purin-6-one
Show/Hide
|
C20H22FN9O11P2
|
2
|
| 1 |
EC50 = 1400 nM
|
|
|
| 2 |
EC50 = 25500 nM
|
|
|
|
CP0176927
|
9-[(1S,6R,8R,9R,10S,15R,17R,18R)-17-(6-aminopurin-9-yl)-9,12,18-trihydroxy-3-oxo-3-sulfanyl-12-sulfanylidene-2,4,7,11,13,16-hexaoxa-3lambda5,12lambda5-diphosphatricyclo[13.3.0.06,10]octadecan-8-yl]-1H-purin-6-one
Show/Hide
|
C20H23N9O11P2S2
|
2
|
| 1 |
EC50 = 1600 nM
|
|
|
| 2 |
EC50 = 7800 nM
|
|
|
|
CP0551716
|
benzyl N-[3-[5-carbamoyl-7-(3-methoxypropoxy)-2-(pyridine-2-carbonylamino)benzimidazol-1-yl]propyl]carbamate
Show/Hide
|
C29H32N6O6
|
1
|
| 1 |
EC50 = 1900 nM
|
|
|
|
CP0444685
|
9-[(1S,6R,8R,9R,10R,15R,17R)-17-(6-aminopurin-9-yl)-9-fluoro-12-hydroxy-3-oxo-3-sulfanyl-12-sulfanylidene-2,4,7,11,13,16-hexaoxa-3lambda5,12lambda5-diphosphatricyclo[13.3.0.06,10]octadecan-8-yl]-1H-purin-6-one
Show/Hide
|
C20H22FN9O9P2S2
|
2
|
| 1 |
EC50 = 1900 nM
|
|
|
| 2 |
EC50 = 9900 nM
|
|
|
|
CP0569706
|
4,5-difluoro-2-[(6-imidazol-1-ylpyridazine-3-carbonyl)amino]benzoic acid
Show/Hide
|
C15H9F2N5O3
|
1
|
| 1 |
EC50 = 2100 nM
|
|
|
|
CP0543189
|
2-[[6-(1,2-dihydroimidazol-3-yl)pyridazine-3-carbonyl]amino]-4,5-difluorobenzoic acid
Show/Hide
|
C15H11F2N5O3
|
1
|
| 1 |
EC50 = 2100 nM
|
|
|
|
CP0551714
|
benzyl N-[3-[5-carbamoyl-7-methoxy-2-(pyridazine-3-carbonylamino)benzimidazol-1-yl]propyl]carbamate
Show/Hide
|
C25H25N7O5
|
1
|
| 1 |
EC50 = 2200 nM
|
|
|
|
CP0444689
|
9-[(1S,6R,8R,9R,10R,15R,17R)-17-(6-aminopurin-9-yl)-9-fluoro-3,12-dihydroxy-3,12-dioxo-2,4,7,11,13,16-hexaoxa-3lambda5,12lambda5-diphosphatricyclo[13.3.0.06,10]octadecan-8-yl]-1H-purin-6-one
Show/Hide
|
C20H22FN9O11P2
|
2
|
| 1 |
EC50 = 2300 nM
|
|
|
| 2 |
EC50 = 32300 nM
|
|
|
|
CP0466828
|
tert-butyl N-[4-[5-carbamoyl-7-methoxy-2-(pyridazine-3-carbonylamino)benzimidazol-1-yl]butyl]carbamate
Show/Hide
|
C23H29N7O5
|
1
|
| 1 |
EC50 = 2850 nM
|
|
|
|
CP0466829
|
tert-butyl N-[4-[5-carbamoyl-7-methoxy-2-(pyridine-2-carbonylamino)benzimidazol-1-yl]butyl]carbamate
Show/Hide
|
C24H30N6O5
|
1
|
| 1 |
EC50 = 3000 nM
|
|
|
|
CP0158278
|
2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]-1-propylbenzimidazole-5-carboxamide
Show/Hide
|
C18H22N6O2
|
1
|
| 1 |
EC50 = 3300 nM
|
|
|
|
CP0176928
|
9-[(1S,6R,8R,9R,10S,15R,17R,18R)-17-(6-aminopurin-9-yl)-3,9,12,18-tetrahydroxy-3,12-dioxo-2,4,7,11,13,16-hexaoxa-3lambda5,12lambda5-diphosphatricyclo[13.3.0.06,10]octadecan-8-yl]-1H-purin-6-one
Show/Hide
|
C20H23N9O13P2
|
2
|
| 1 |
EC50 = 5100 nM
|
|
|
| 2 |
EC50 = 15900 nM
|
|
|
|
CP0158277
|
2-amino-9-[(1R,6R,8R,9R,10S,15R,17R,18R)-8-(6-aminopurin-9-yl)-3,9,12,18-tetrahydroxy-3,12-dioxo-2,4,7,11,13,16-hexaoxa-3lambda5,12lambda5-diphosphatricyclo[13.2.1.06,10]octadecan-17-yl]-1H-purin-6-one
Show/Hide
|
C20H24N10O13P2
|
3
|
| 1 |
EC50 = 7200 nM
|
|
|
| 2 |
EC50 = 38600 nM
|
|
|
| 3 |
EC50 = 39100 nM
|
|
|
|
CP0455790
|
benzyl N-[3-[5-carbamoyl-7-methoxy-2-(pyridine-2-carbonylamino)benzimidazol-1-yl]propyl]carbamate
Show/Hide
|
C26H26N6O5
|
1
|
| 1 |
EC50 = 8280 nM
|
|
|
|
CP0444687
|
9-[(1S,6R,8R,10S,15R,17R)-17-(6-aminopurin-9-yl)-3,12-dihydroxy-3,12-dioxo-2,4,7,11,13,16-hexaoxa-3lambda5,12lambda5-diphosphatricyclo[13.3.0.06,10]octadecan-8-yl]-1H-purin-6-one
Show/Hide
|
C20H23N9O11P2
|
2
|
| 1 |
EC50 = 10000 nM
|
|
|
| 2 |
EC50 = 62300 nM
|
|
|
|
CP0220338
|
9-[(1R,6R,8R,9R,10S,15R,17R,18R)-8-(6-aminopurin-9-yl)-3,9,12,18-tetrahydroxy-3,12-dioxo-2,4,7,11,13,16-hexaoxa-3lambda5,12lambda5-diphosphatricyclo[13.2.1.06,10]octadecan-17-yl]-1H-purin-6-one
Show/Hide
|
C20H23N9O13P2
|
2
|
| 1 |
EC50 = 12500 nM
|
|
|
| 2 |
EC50 = 54300 nM
|
|
|
|
CP0537187
|
9-[(1R,6R,8R,9R,10S,15R,17R,18R)-17-(6-aminopurin-9-yl)-3,9,12,18-tetrahydroxy-3,12-dioxo-2,4,7,11,13,16-hexaoxa-3lambda5,12lambda5-diphosphatricyclo[13.2.1.06,10]octadecan-8-yl]-1H-purin-6-one
Show/Hide
|
C20H23N9O13P2
|
2
|
| 1 |
EC50 = 15100 nM
|
|
|
| 2 |
EC50 = 60600 nM
|
|
|
|
CP0444688
|
9-[(1R,6R,8R,9R,14R,16R,17R,18R)-16-(6-aminopurin-9-yl)-3,11,17,18-tetrahydroxy-3,11-dioxo-2,4,7,10,12,15-hexaoxa-3lambda5,11lambda5-diphosphatricyclo[12.2.1.16,9]octadecan-8-yl]-1H-purin-6-one
Show/Hide
|
C20H23N9O13P2
|
1
|
| 1 |
EC50 = 17900 nM
|
|
|
|
CP0563788
|
methyl 2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]-7-methoxy-1-[3-(phenylmethoxycarbonylamino)propyl]benzimidazole-5-carboxylate
Show/Hide
|
C28H32N6O6
|
1
|
| 1 |
EC50 = 20700 nM
|
|
|
|
CP0387061
|
1-[3-(2,2-dimethylpropanoylamino)propyl]-2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]-7-methoxybenzimidazole-5-carboxamide
Show/Hide
|
C24H33N7O4
|
1
|
| 1 |
EC50 = 27500 nM
|
|
|
|
CP0387063
|
2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]-7-methoxy-1-[3-(3-pyridin-3-ylpropanoylamino)propyl]benzimidazole-5-carboxamide
Show/Hide
|
C27H32N8O4
|
1
|
| 1 |
EC50 = 39500 nM
|
|
|
|
CP0387059
|
benzyl N-[3-[5-carbamoyl-2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]benzimidazol-1-yl]propyl]carbamate
Show/Hide
|
C26H29N7O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0387060
|
benzyl N-[3-[5-carbamoyl-7-methoxy-2-(3-phenylpropanoylamino)benzimidazol-1-yl]propyl]carbamate
Show/Hide
|
C29H31N5O5
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0387065
|
7-methoxy-2-(3-phenylpropanoylamino)-1-propylbenzimidazole-5-carboxamide
Show/Hide
|
C21H24N4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0387066
|
7-methoxy-2-[(2-methylpyrazole-3-carbonyl)amino]-1-propylbenzimidazole-5-carboxamide
Show/Hide
|
C17H20N6O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0432758
|
benzyl N-[3-[5-carbamoyl-7-(3-methoxypropoxy)-2-(pyridazine-3-carbonylamino)benzimidazol-1-yl]propyl]carbamate
Show/Hide
|
C28H31N7O6
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0432759
|
2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]-7-methoxy-1-[3-[3-(3,4,5-trimethoxyphenyl)propanoylamino]propyl]benzimidazole-5-carboxamide
Show/Hide
|
C31H39N7O7
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0434820
|
benzyl N-[3-[5-carbamoyl-7-(3-morpholin-4-ylpropoxy)-2-(pyridazine-3-carbonylamino)benzimidazol-1-yl]propyl]carbamate
Show/Hide
|
C31H36N8O6
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0434821
|
1-(3-aminopropyl)-2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]-7-methoxybenzimidazole-5-carboxamide
Show/Hide
|
C19H25N7O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0434822
|
1-(3-benzamidopropyl)-2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]-7-methoxybenzimidazole-5-carboxamide
Show/Hide
|
C26H29N7O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0455789
|
methyl 2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]-7-methoxy-1-propylbenzimidazole-5-carboxylate
Show/Hide
|
C20H25N5O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0455878
|
7-methoxy-2-[(1-methylindole-2-carbonyl)amino]-1-propylbenzimidazole-5-carboxamide
Show/Hide
|
C22H23N5O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0455880
|
benzyl N-[3-[5-carbamoyl-7-methoxy-2-[(1-methylindole-2-carbonyl)amino]benzimidazol-1-yl]propyl]carbamate
Show/Hide
|
C30H30N6O5
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0466827
|
methyl 2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]-3-[3-[(2-methylpropan-2-yl)oxycarbonylamino]propyl]imidazo[4,5-b]pyridine-6-carboxylate
Show/Hide
|
C23H31N7O5
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0466830
|
2-[(2-ethylpyrazole-3-carbonyl)amino]-7-methoxy-1-propylbenzimidazole-5-carboxamide
Show/Hide
|
C18H22N6O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0479159
|
tert-butyl N-[3-[6-carbamoyl-2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]imidazo[4,5-b]pyridin-3-yl]propyl]carbamate
Show/Hide
|
C22H30N8O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0479160
|
benzyl N-[3-[5-carbamoyl-7-methoxy-2-[(1-methylpyrrole-2-carbonyl)amino]benzimidazol-1-yl]propyl]carbamate
Show/Hide
|
C26H28N6O5
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0482212
|
benzyl N-[3-[2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]-7-methoxybenzimidazol-1-yl]propyl]carbamate
Show/Hide
|
C26H30N6O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0537021
|
N-(5-carbamoyl-7-methoxy-1-propylbenzimidazol-2-yl)isoquinoline-1-carboxamide
Show/Hide
|
C22H21N5O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0537025
|
7-methoxy-2-[(3-methylimidazole-4-carbonyl)amino]-1-propylbenzimidazole-5-carboxamide
Show/Hide
|
C17H20N6O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0537512
|
N-(5-carbamoyl-7-methoxy-1-propylbenzimidazol-2-yl)quinoline-2-carboxamide
Show/Hide
|
C22H21N5O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0537515
|
4-[3-[5-carbamoyl-2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]-7-methoxybenzimidazol-1-yl]propylamino]-4-oxobutanoic acid
Show/Hide
|
C23H29N7O6
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0537516
|
methyl 4-[3-[5-carbamoyl-2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]-7-methoxybenzimidazol-1-yl]propylamino]-4-oxobutanoate
Show/Hide
|
C24H31N7O6
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0551177
|
benzyl N-[3-[5-carbamoyl-2-(isoquinoline-1-carbonylamino)-7-methoxybenzimidazol-1-yl]propyl]carbamate
Show/Hide
|
C30H28N6O5
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0551178
|
7-methoxy-1-propyl-2-(pyridazine-3-carbonylamino)benzimidazole-5-carboxamide
Show/Hide
|
C17H18N6O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0551715
|
2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]-3-[3-[(2-methylpropan-2-yl)oxycarbonylamino]propyl]imidazo[4,5-b]pyridine-6-carboxylic acid
Show/Hide
|
C22H29N7O5
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0551717
|
benzyl N-[3-[5-carbamoyl-7-methoxy-2-[(1-methylpiperidine-4-carbonyl)amino]benzimidazol-1-yl]propyl]carbamate
Show/Hide
|
C27H34N6O5
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0552187
|
2-ethyl-N-(7-methoxy-1-propylbenzimidazol-2-yl)-5-methylpyrazole-3-carboxamide
Show/Hide
|
C18H23N5O2
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0552614
|
benzyl N-[3-[5-carbamoyl-2-[(2-ethylpyrazole-3-carbonyl)amino]-7-methoxybenzimidazol-1-yl]propyl]carbamate
Show/Hide
|
C26H29N7O5
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0552615
|
benzyl N-[3-[5-carbamoyl-7-(3-morpholin-4-ylpropoxy)-2-(pyridine-2-carbonylamino)benzimidazol-1-yl]propyl]carbamate
Show/Hide
|
C32H37N7O6
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0552616
|
benzyl N-[3-[5-carbamoyl-7-methoxy-2-(quinoline-2-carbonylamino)benzimidazol-1-yl]propyl]carbamate
Show/Hide
|
C30H28N6O5
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0561668
|
benzyl N-[3-[5-carbamoyl-7-methoxy-2-[(2-methylpyrazole-3-carbonyl)amino]benzimidazol-1-yl]propyl]carbamate
Show/Hide
|
C25H27N7O5
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0561669
|
7-methoxy-1-propyl-2-(pyridine-2-carbonylamino)benzimidazole-5-carboxamide
Show/Hide
|
C18H19N5O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0561672
|
benzyl N-[3-[5-carbamoyl-7-methoxy-2-[(3-methylimidazole-4-carbonyl)amino]benzimidazol-1-yl]propyl]carbamate
Show/Hide
|
C25H27N7O5
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0571477
|
benzyl N-[3-[5-carbamoyl-7-methoxy-2-[(1-methylpyrrolidine-2-carbonyl)amino]benzimidazol-1-yl]propyl]carbamate
Show/Hide
|
C26H32N6O5
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
