| Compound ID |
Compound Name |
Compound Formula |
|
CP0295855
|
9-(trifluoromethyl)-5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide
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|
C16H9F3N2O2S
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0957416
|
1-(3,4-Difluoro-phenyl)-2-methyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene3,3-dioxide
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|
C17H13F2N3O2S
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0964022
|
1-[1-(4-Fluoro-phenyl)-2-methyl-3,3-dioxo-1,2,3,4-tetrahydro-3lambda6-thia-2,4,5-triaza-phenanthren-9-yl]-ethanone
Show/Hide
|
C19H16FN3O3S
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0924106
|
2-Amino-4-methyl-N-quinolin-8-yl-benzenesulfonamide
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|
C16H15N3O2S
|
1
|
| 1 |
IC50 = 300 nM
|
|
|
|
CP0942401
|
2,2,2-Trifluoro-N-[2-(quinolin-8-ylsulfamoyl)-phenyl]-acetamide
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|
C17H12F3N3O3S
|
1
|
| 1 |
IC50 = 307 nM
|
|
|
|
CP0957701
|
12-Chloro-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
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|
C15H9ClN2O2S
|
1
|
| 1 |
IC50 = 320 nM
|
|
|
|
CP0959877
|
1-(4-Fluoro-phenyl)-2-methyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene 3,3-dioxide
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|
C17H14FN3O2S
|
1
|
| 1 |
IC50 = 340 nM
|
|
|
|
CP0897764
|
8-Methyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
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|
C16H12N2O2S
|
1
|
| 1 |
IC50 = 360 nM
|
|
|
|
CP0969317
|
5-Methyl-pyridine-2-sulfonic acid quinolin-8-ylamide
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|
C15H13N3O2S
|
1
|
| 1 |
IC50 = 380 nM
|
|
|
|
CP0556224
|
3-cyano-N-quinolin-8-ylbenzenesulfonamide
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|
C16H11N3O2S
|
1
|
| 1 |
IC50 = 413 nM
|
|
|
|
CP0969310
|
N-Quinolin-8-yl-2-trifluoromethyl-benzenesulfonamide
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|
C16H11F3N2O2S
|
1
|
| 1 |
IC50 = 419 nM
|
|
|
|
CP0867129
|
12-Chloro-9-cyclopentyloxy-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
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|
C20H17ClN2O3S
|
1
|
| 1 |
IC50 = 420 nM
|
|
|
|
CP0870271
|
2-Phenyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene3,3-dioxide
Show/Hide
|
C16H13N3O2S
|
1
|
| 1 |
IC50 = 460 nM
|
|
|
|
CP0959871
|
Pyridine-2-sulfonic acid(5-trifluoromethyl-quinolin-8-yl)-amide
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|
C15H10F3N3O2S
|
1
|
| 1 |
IC50 = 460 nM
|
|
|
|
CP0867133
|
(6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-12-yl)-(2-methoxy-ethyl)-methyl-amine
Show/Hide
|
C19H19N3O3S
|
1
|
| 1 |
IC50 = 550 nM
|
|
|
|
CP0349446
|
2-amino-N-(6-methoxyquinolin-8-yl)-4-methylbenzenesulfonamide
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|
C17H17N3O3S
|
1
|
| 1 |
IC50 = 585 nM
|
|
|
|
CP0926142
|
12-Methyl-5H-6-thia-4,5-diaza-chrysene6,6-dioxide
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|
C16H12N2O2S
|
1
|
| 1 |
IC50 = 599 nM
|
|
|
|
CP0944903
|
2-Methyl-1-p-tolyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene 3,3-dioxide
Show/Hide
|
C18H17N3O2S
|
1
|
| 1 |
IC50 = 600 nM
|
|
|
|
CP0957689
|
N-(3-Methyl-quinolin-8-yl)-benzenesulfonamide
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|
C16H14N2O2S
|
1
|
| 1 |
IC50 = 610 nM
|
|
|
|
CP0961829
|
(12-Chloro-6,6-dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-9-yl)-(2-morpholin-4-yl-ethyl)-amine
Show/Hide
|
C21H21ClN4O3S
|
1
|
| 1 |
IC50 = 620 nM
|
|
|
|
CP0961022
|
4-Chloro-2-fluoro-N-(6-fluoro-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C15H9ClF2N2O2S
|
1
|
| 1 |
IC50 = 690 nM
|
|
|
|
CP0857281
|
1-(3-Fluoro-phenyl)-2-methyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene 3,3-dioxide
Show/Hide
|
C17H14FN3O2S
|
1
|
| 1 |
IC50 = 720 nM
|
|
|
|
CP0961025
|
N-Quinolin-8-yl-3-trifluoromethyl-benzenesulfonamide
Show/Hide
|
C16H11F3N2O2S
|
1
|
| 1 |
IC50 = 720 nM
|
|
|
|
CP0960142
|
2-Amino-N-quinolin-8-yl-4-trifluoromethyl-benzenesulfonamide
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|
C16H12F3N3O2S
|
1
|
| 1 |
IC50 = 760 nM
|
|
|
|
CP0192225
|
9-chloro-5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide
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|
C15H9ClN2O2S
|
1
|
| 1 |
IC50 = 770 nM
|
|
|
|
CP0960146
|
N-(6-Fluoro-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C15H11FN2O2S
|
1
|
| 1 |
IC50 = 780 nM
|
|
|
|
CP0415356
|
2-cyano-N-quinolin-8-ylbenzenesulfonamide
Show/Hide
|
C16H11N3O2S
|
1
|
| 1 |
IC50 = 815 nM
|
|
|
|
CP0959870
|
2,4,6-Trichloro-N-quinolin-8-yl-benzenesulfonamide
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|
C15H9Cl3N2O2S
|
1
|
| 1 |
IC50 = 857 nM
|
|
|
|
CP0926143
|
2-Methyl-1-phenyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene3,3-dioxide
Show/Hide
|
C17H15N3O2S
|
1
|
| 1 |
IC50 = 870 nM
|
|
|
|
CP0969309
|
4-Chloro-2-fluoro-N-quinolin-8-yl-benzenesulfonamide
Show/Hide
|
C15H10ClFN2O2S
|
1
|
| 1 |
IC50 = 873 nM
|
|
|
|
CP0949358
|
(6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-9-yl)-dimethyl-amine
Show/Hide
|
C17H15N3O2S
|
1
|
| 1 |
IC50 = 910 nM
|
|
|
|
CP0869078
|
4-Fluoro-2-nitro-N-quinolin-8-yl-benzenesulfonamide
Show/Hide
|
C15H10FN3O4S
|
1
|
| 1 |
IC50 = 920 nM
|
|
|
|
CP0867134
|
12-Methoxy-9-trifluoromethyl-5H-6-thia-4,5-diaza-chrysene6,6-dioxide
Show/Hide
|
C17H11F3N2O3S
|
1
|
| 1 |
IC50 = 960 nM
|
|
|
|
CP0960153
|
2-Methyl-1-(6-trifluoromethyl-pyridin-3-yl)-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene3,3-dioxide
Show/Hide
|
C17H13F3N4O2S
|
1
|
| 1 |
IC50 = 960 nM
|
|
|
|
CP0869089
|
1-Methoxy-9-trifluoromethyl-5H-6-thia-4,5-diaza-chrysene6,6-dioxide
Show/Hide
|
C17H11F3N2O3S
|
1
|
| 1 |
IC50 = 979 nM
|
|
|
|
CP0963392
|
3-Chloro-N-quinolin-8-yl-benzenesulfonamide
Show/Hide
|
C15H11ClN2O2S
|
1
|
| 1 |
IC50 = 985 nM
|
|
|
|
CP0966697
|
N-(5-Fluoro-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C15H11FN2O2S
|
1
|
| 1 |
IC50 = 988 nM
|
|
|
|
CP0567337
|
2,4-dichloro-N-quinolin-8-ylbenzenesulfonamide
Show/Hide
|
C15H10Cl2N2O2S
|
1
|
| 1 |
IC50 = 989 nM
|
|
|
|
CP0866765
|
12-Chloro-6,6-dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysene-9-carboxylicacidcyclopentylester
Show/Hide
|
C21H17ClN2O4S
|
1
|
| 1 |
IC50 = 990 nM
|
|
|
|
CP0969316
|
12-Methoxy-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C16H12N2O3S
|
1
|
| 1 |
IC50 = 990 nM
|
|
|
|
CP0866757
|
2-Amino-N-(6-methoxy-quinolin-8-yl)-4-trifluoromethyl-benzenesulfonamide
Show/Hide
|
C17H14F3N3O3S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0866934
|
2,6-Difluoro-N-(6-fluoro-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C15H9F3N2O2S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0969308
|
N-Quinolin-8-yl-4-trifluoromethyl-benzenesulfonamide
Show/Hide
|
C16H11F3N2O2S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0963395
|
N-(5-Trifluoromethyl-quinolin-8-yl)-benzene sulfonamide
Show/Hide
|
C16H11F3N2O2S
|
1
|
| 1 |
IC50 = 1050 nM
|
|
|
|
CP0957707
|
1-(2,4-Dimethoxy-phenyl)-2-methyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene3,3-dioxide
Show/Hide
|
C19H19N3O4S
|
1
|
| 1 |
IC50 = 1070 nM
|
|
|
|
CP0944900
|
Pyridine-2-sulfonic acid(6-trifluoromethoxy-quinolin-8-yl)-amide
Show/Hide
|
C15H10F3N3O3S
|
1
|
| 1 |
IC50 = 1090 nM
|
|
|
|
CP0869085
|
N-(5-Methyl-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C16H14N2O2S
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0961011
|
1-(12-Chloro-6,6-dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-9-yl)-piperidin-4-ol
Show/Hide
|
C20H18ClN3O3S
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0930452
|
12-Morpholin-4-yl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C19H17N3O3S
|
1
|
| 1 |
IC50 = 1140 nM
|
|
|
|
CP0959874
|
2,6-Difluoro-N-quinolin-8-yl-benzenesulfonamide
Show/Hide
|
C15H10F2N2O2S
|
1
|
| 1 |
IC50 = 1140 nM
|
|
|
|
CP0957417
|
2-Methyl-1-(4-trifluoromethoxy-phenyl)-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene3,3-dioxide
Show/Hide
|
C18H14F3N3O3S
|
1
|
| 1 |
IC50 = 1150 nM
|
|
|
|
CP0966518
|
9-Trifluoromethoxy-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C16H9F3N2O3S
|
1
|
| 1 |
IC50 = 1170 nM
|
|
|
|
CP0964034
|
N-Quinolin-8-yl-3-trifluoromethoxy-benzenesulfonamide
Show/Hide
|
C16H11F3N2O3S
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0869081
|
2-Amino-N-(5-chloro-quinolin-8-yl)-4-methyl-benzenesulfonamide
Show/Hide
|
C16H14ClN3O2S
|
1
|
| 1 |
IC50 = 1220 nM
|
|
|
|
CP0959875
|
4-Chloro-2-fluoro-N-(3-methyl-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C16H12ClFN2O2S
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0845858
|
2-Methyl-1-(4-trifluoromethyl-phenyl)-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene 3,3-dioxide
Show/Hide
|
C18H14F3N3O2S
|
1
|
| 1 |
IC50 = 1370 nM
|
|
|
|
CP0969311
|
N-[2-(Quinolin-8-ylsulfamoyl)-phenyl]-acetamide
Show/Hide
|
C17H15N3O3S
|
1
|
| 1 |
IC50 = 1370 nM
|
|
|
|
CP0968263
|
4-Chloro-N-(5-chloro-quinolin-8-yl)-2-fluoro-benzenesulfonamide
Show/Hide
|
C15H9Cl2FN2O2S
|
1
|
| 1 |
IC50 = 1380 nM
|
|
|
|
CP0930849
|
12-Fluoro-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C15H9FN2O2S
|
1
|
| 1 |
IC50 = 1390 nM
|
|
|
|
CP0957691
|
Pyridine-3-sulfonic acid(3-methyl-quinolin-8-yl)-amide
Show/Hide
|
C15H13N3O2S
|
1
|
| 1 |
IC50 = 1390 nM
|
|
|
|
CP0869079
|
3-(Quinolin-8-ylsulfamoyl)-benzoic acid methyl ester
Show/Hide
|
C17H14N2O4S
|
1
|
| 1 |
IC50 = 1420 nM
|
|
|
|
CP0957418
|
1-(3-Fluoro-4-methoxy-phenyl)-2-methyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene 3,3-dioxide
Show/Hide
|
C18H16FN3O3S
|
1
|
| 1 |
IC50 = 1480 nM
|
|
|
|
CP0423082
|
3-methoxy-N-quinolin-8-ylbenzenesulfonamide
Show/Hide
|
C16H14N2O3S
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0959876
|
3-Fluoro-2-methyl-N-quinolin-8-yl-benzenesulfonamide
Show/Hide
|
C16H13FN2O2S
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0960148
|
N-(5-Chloro-6-fluoro-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C15H10ClFN2O2S
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0964040
|
1-(4-Fluoro-2-methyl-phenyl)-2-methyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene 3,3-dioxide
Show/Hide
|
C18H16FN3O2S
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0294411
|
9-fluoro-5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide
Show/Hide
|
C15H9FN2O2S
|
1
|
| 1 |
IC50 = 1560 nM
|
|
|
|
CP0964024
|
12-Piperidin-1-yl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C20H19N3O2S
|
1
|
| 1 |
IC50 = 1560 nM
|
|
|
|
CP0924107
|
1-(5-Fluoro-pyridin-2-yl)-2-methyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene3,3-dioxide
Show/Hide
|
C16H13FN4O2S
|
1
|
| 1 |
IC50 = 1570 nM
|
|
|
|
CP0311125
|
9-methoxy-5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide
Show/Hide
|
C16H12N2O3S
|
1
|
| 1 |
IC50 = 1580 nM
|
|
|
|
CP0957706
|
1-(3-Fluoro-pyridin-4-yl)-2-methyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene3,3-dioxide
Show/Hide
|
C16H13FN4O2S
|
1
|
| 1 |
IC50 = 1600 nM
|
|
|
|
CP0845857
|
8-Fluoro-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C15H9FN2O2S
|
1
|
| 1 |
IC50 = 1620 nM
|
|
|
|
CP0964016
|
12-Chloro-9-morpholin-4-yl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C19H16ClN3O3S
|
1
|
| 1 |
IC50 = 1620 nM
|
|
|
|
CP0944898
|
N-(5-Chloro-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C15H11ClN2O2S
|
1
|
| 1 |
IC50 = 1670 nM
|
|
|
|
CP0942402
|
3-Chloro-2-fluoro-N-quinolin-8-yl-benzenesulfonamide
Show/Hide
|
C15H10ClFN2O2S
|
1
|
| 1 |
IC50 = 1710 nM
|
|
|
|
CP0969314
|
4-Chloro-2-fluoro-N-(6-methoxy-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C16H12ClFN2O3S
|
1
|
| 1 |
IC50 = 1750 nM
|
|
|
|
CP0963394
|
Pyridine-3-sulfonicacid(5-chloro-quinolin-8-yl)-amide
Show/Hide
|
C14H10ClN3O2S
|
1
|
| 1 |
IC50 = 1780 nM
|
|
|
|
CP0864581
|
SID26755436
Show/Hide
|
C16H13N3O5S
|
1
|
| 1 |
IC50 = 1810 nM
|
|
|
|
CP0957705
|
1-(2-Methoxy-phenyl)-2-methyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene3,3-dioxide
Show/Hide
|
C18H17N3O3S
|
1
|
| 1 |
IC50 = 1870 nM
|
|
|
|
CP0389645
|
N-quinolin-8-ylpyridine-2-sulfonamide
Show/Hide
|
C14H11N3O2S
|
1
|
| 1 |
IC50 = 1890 nM
|
|
|
|
CP0968267
|
Pyrazine-2-sulfonic acid quinolin-8-ylamide
Show/Hide
|
C13H10N4O2S
|
1
|
| 1 |
IC50 = 1910 nM
|
|
|
|
CP0952471
|
(12-Chloro-6,6-dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-9-yl)-(2-methoxy-ethyl)-amine
Show/Hide
|
C18H16ClN3O3S
|
1
|
| 1 |
IC50 = 1980 nM
|
|
|
|
CP0961830
|
6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysene-1-carboxylic acid(2-piperidin-1-yl-ethyl)-amide
Show/Hide
|
C23H24N4O3S
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0930465
|
1-(6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-9-yl)-pyrrolidin-3-ol
Show/Hide
|
C19H17N3O3S
|
1
|
| 1 |
IC50 = 2010 nM
|
|
|
|
CP0866933
|
Quinoline-3-sulfonic acid quinolin-8-ylamide
Show/Hide
|
C18H13N3O2S
|
1
|
| 1 |
IC50 = 2060 nM
|
|
|
|
CP0861219
|
3-Methyl-N-quinolin-8-yl-benzenesulfonamide
Show/Hide
|
C16H14N2O2S
|
1
|
| 1 |
IC50 = 2090 nM
|
|
|
|
CP0942407
|
6-Cyano-pyridine-3-sulfonic acid(6-trifluoromethoxy-quinolin-8-yl)-amide
Show/Hide
|
C16H9F3N4O3S
|
1
|
| 1 |
IC50 = 2110 nM
|
|
|
|
CP0969463
|
8-Methoxy-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C16H12N2O3S
|
1
|
| 1 |
IC50 = 2110 nM
|
|
|
|
CP0861220
|
N-(6-Methyl-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C16H14N2O2S
|
1
|
| 1 |
IC50 = 2180 nM
|
|
|
|
CP0930464
|
(12-Chloro-6,6-dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-9-yl)-diethyl-amine
Show/Hide
|
C19H18ClN3O2S
|
1
|
| 1 |
IC50 = 2190 nM
|
|
|
|
CP0952644
|
1-Ethyl-2-methyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene 3,3-dioxide
Show/Hide
|
C13H15N3O2S
|
1
|
| 1 |
IC50 = 2220 nM
|
|
|
|
CP0897765
|
1-(4-Methoxy-phenyl)-2-methyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene3,3-dioxide
Show/Hide
|
C18H17N3O3S
|
1
|
| 1 |
IC50 = 2240 nM
|
|
|
|
CP0866754
|
N-phenyl(quinolin-8-ylamino)sulfonamide
Show/Hide
|
C15H13N3O2S
|
1
|
| 1 |
IC50 = 2300 nM
|
|
|
|
CP0964038
|
8-Trifluoromethyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C16H9F3N2O2S
|
1
|
| 1 |
IC50 = 2340 nM
|
|
|
|
CP0942406
|
Pyridine-2-sulfonic acid(6-fluoro-quinolin-8-yl)-amide
Show/Hide
|
C14H10FN3O2S
|
1
|
| 1 |
IC50 = 2370 nM
|
|
|
|
CP0952643
|
1-[1-(4-Fluoro-phenyl)-2-methyl-3,3-dioxo-1,2,3,4-tetrahydro-3lambda6-thia-2,4,5-triaza-phenanthren-9-yl]-ethanol
Show/Hide
|
C19H18FN3O3S
|
1
|
| 1 |
IC50 = 2370 nM
|
|
|
|
CP0957698
|
N-Quinolin-8-yl-2-trifluoromethoxy-benzenesulfonamide
Show/Hide
|
C16H11F3N2O3S
|
1
|
| 1 |
IC50 = 2500 nM
|
|
|
|
CP0960149
|
6-Cyano-pyridine-3-sulfonic acid(5-trifluoromethyl-quinolin-8-yl)-amide
Show/Hide
|
C16H9F3N4O2S
|
1
|
| 1 |
IC50 = 2600 nM
|
|
|
|
CP0957654
|
[2-Fluoro-5-(2-methyl-3,3-dioxo-1,2,3,4-tetrahydro-3lambda6-thia-2,4,5-triaza-phenanthren-1-yl)-phenyl]-morpholin-4-yl-methanone
Show/Hide
|
C22H21FN4O4S
|
1
|
| 1 |
IC50 = 2620 nM
|
|
|
|
CP0952472
|
(12-Chloro-6,6-dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-9-yl)-morpholin-4-yl-methanone
Show/Hide
|
C20H16ClN3O4S
|
1
|
| 1 |
IC50 = 2740 nM
|
|
|
|
CP0930468
|
[2-(6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-12-yloxy)-ethyl]-dimethyl-amine
Show/Hide
|
C19H19N3O3S
|
1
|
| 1 |
IC50 = 2760 nM
|
|
|
|
CP0962715
|
1-(4-Fluoro-phenyl)-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene 3,3-dioxide
Show/Hide
|
C16H12FN3O2S
|
1
|
| 1 |
IC50 = 2780 nM
|
|
|
|
CP0968264
|
Pyridine-3-sulfonicacid(6-methoxy-quinolin-8-yl)-amide
Show/Hide
|
C15H13N3O3S
|
1
|
| 1 |
IC50 = 2800 nM
|
|
|
|
CP0957414
|
6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysene-9-carbonitrile
Show/Hide
|
C16H9N3O2S
|
1
|
| 1 |
IC50 = 2830 nM
|
|
|
|
CP0959850
|
(6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-12-yl)-(2-methoxy-ethyl)-amine
Show/Hide
|
C18H17N3O3S
|
1
|
| 1 |
IC50 = 2830 nM
|
|
|
|
CP0041688
|
2-nitro-N-(8-quinolinyl)benzenesulfonamide
Show/Hide
|
C15H11N3O4S
|
1
|
| 1 |
IC50 = 2900 nM
|
|
|
|
CP0211410
|
5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide
Show/Hide
|
C15H10N2O2S
|
1
|
| 1 |
IC50 = 2900 nM
|
|
|
|
CP0861209
|
6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysene-1-carboxylicacidmethylester
Show/Hide
|
C17H12N2O4S
|
1
|
| 1 |
IC50 = 2940 nM
|
|
|
|
CP0869080
|
2-Amino-N-(3-methyl-quinolin-8-yl)-4-trifluoromethyl-benzenesulfonamide
Show/Hide
|
C17H14F3N3O2S
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0295856
|
9-methyl-5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide
Show/Hide
|
C16H12N2O2S
|
1
|
| 1 |
IC50 = 3200 nM
|
|
|
|
CP0513264
|
4-chloro-N-quinolin-8-ylbenzenesulfonamide
Show/Hide
|
C15H11ClN2O2S
|
1
|
| 1 |
IC50 = 3200 nM
|
|
|
|
CP0926553
|
9-Fluoro-8-methyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C16H11FN2O2S
|
1
|
| 1 |
IC50 = 3240 nM
|
|
|
|
CP0942403
|
Quinolin-8-yl-sulfamic acid phenyl ester
Show/Hide
|
C15H12N2O3S
|
1
|
| 1 |
IC50 = 3250 nM
|
|
|
|
CP0962719
|
1-Pyrazol-1-yl-5H-6-thia-4,5-diaza-chrysene6,6-dioxide
Show/Hide
|
C18H12N4O2S
|
1
|
| 1 |
IC50 = 3530 nM
|
|
|
|
CP0949359
|
12-Chloro-6,6-dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-9-ylamine
Show/Hide
|
C15H10ClN3O2S
|
1
|
| 1 |
IC50 = 3570 nM
|
|
|
|
CP0556225
|
N-quinolin-8-ylpyridine-3-sulfonamide
Show/Hide
|
C14H11N3O2S
|
1
|
| 1 |
IC50 = 3640 nM
|
|
|
|
CP0869084
|
6-Trifluoromethyl-pyridine-3-sulfonic acid quinolin-8-ylamide
Show/Hide
|
C15H10F3N3O2S
|
1
|
| 1 |
IC50 = 3690 nM
|
|
|
|
CP0960154
|
1-(3-Chloro-4-fluoro-phenyl)-2-methyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene3,3-dioxide
Show/Hide
|
C17H13ClFN3O2S
|
1
|
| 1 |
IC50 = 3700 nM
|
|
|
|
CP0848498
|
6-Cyano-pyridine-3-sulfonicacid(6-fluoro-quinolin-8-yl)-amide
Show/Hide
|
C15H9FN4O2S
|
1
|
| 1 |
IC50 = 3750 nM
|
|
|
|
CP0926552
|
11-Fluoro-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C15H9FN2O2S
|
1
|
| 1 |
IC50 = 3750 nM
|
|
|
|
CP0964036
|
Pyridine-3-sulfonic acid(6-trifluoromethoxy-quinolin-8-yl)-amide
Show/Hide
|
C15H10F3N3O3S
|
1
|
| 1 |
IC50 = 3840 nM
|
|
|
|
CP0957704
|
7-Methyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C16H12N2O2S
|
1
|
| 1 |
IC50 = 3880 nM
|
|
|
|
CP0962720
|
12-Chloro-6,6-dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysene-9-carboxylic acid(2-methoxy-ethyl)-amide
Show/Hide
|
C19H16ClN3O4S
|
1
|
| 1 |
IC50 = 3900 nM
|
|
|
|
CP0952863
|
2-Amino-4-fluoro-N-quinolin-8-yl-benzenesulfonamide
Show/Hide
|
C15H12FN3O2S
|
1
|
| 1 |
IC50 = 3940 nM
|
|
|
|
CP0926144
|
5-Trifluoromethyl-pyridine-3-sulfonic acid quinolin-8-ylamide
Show/Hide
|
C15H10F3N3O2S
|
1
|
| 1 |
IC50 = 3980 nM
|
|
|
|
CP0968265
|
3-Chloro-2-methyl-N-quinolin-8-yl-benzenesulfonamide
Show/Hide
|
C16H13ClN2O2S
|
1
|
| 1 |
IC50 = 4000 nM
|
|
|
|
CP0964035
|
8,9-Dimethyl-5H-6-thia-4,5-diaza-chrysene6,6-dioxide
Show/Hide
|
C17H14N2O2S
|
1
|
| 1 |
IC50 = 4020 nM
|
|
|
|
CP0867130
|
12-Chloro-6,6-dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysene-9-carboxylicaciddimethylamide
Show/Hide
|
C18H14ClN3O3S
|
1
|
| 1 |
IC50 = 4060 nM
|
|
|
|
CP0960152
|
6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysene-9-carboxylic acid methyl ester
Show/Hide
|
C17H12N2O4S
|
1
|
| 1 |
IC50 = 4180 nM
|
|
|
|
CP0900936
|
12-Fluoro-9-trifluoromethyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C16H8F4N2O2S
|
1
|
| 1 |
IC50 = 4190 nM
|
|
|
|
CP0952864
|
6-Cyano-pyridine-3-sulfonic acid quinolin-8-ylamide
Show/Hide
|
C15H10N4O2S
|
1
|
| 1 |
IC50 = 4260 nM
|
|
|
|
CP0930453
|
12-Pyrrolidin-1-yl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C19H17N3O2S
|
1
|
| 1 |
IC50 = 4360 nM
|
|
|
|
CP0962717
|
1-(4-Fluoro-3-piperazin-1-ylmethyl-phenyl)-2-methyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene 3,3-dioxide
Show/Hide
|
C22H24FN5O2S
|
1
|
| 1 |
IC50 = 4490 nM
|
|
|
|
CP0929054
|
Thiazole-2-sulfonic acid quinolin-8-ylamide
Show/Hide
|
C12H9N3O2S2
|
1
|
| 1 |
IC50 = 4580 nM
|
|
|
|
CP0031043
|
N-quinolin-8-ylbenzenesulfonamide
Show/Hide
|
C15H12N2O2S
|
1
|
| 1 |
IC50 = 4590 nM
|
|
|
|
CP0962716
|
1,2-Dimethyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene 3,3-dioxide
Show/Hide
|
C12H13N3O2S
|
1
|
| 1 |
IC50 = 4690 nM
|
|
|
|
CP0964018
|
6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysene-1-carboxylic acid methylamide
Show/Hide
|
C17H13N3O3S
|
1
|
| 1 |
IC50 = 4770 nM
|
|
|
|
CP0867132
|
N-(6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-12-yl)-N,N',N'-trimethyl-ethane-1,2-diamine
Show/Hide
|
C20H22N4O2S
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
|
CP0923931
|
2-Fluoro-5-(2-methyl-3,3-dioxo-1,2,3,4-tetrahydro-3lambda6-thia-2,4,5-triaza-phenanthren-1-yl)-benzoicacid
Show/Hide
|
C19H16FN3O3S
|
1
|
| 1 |
IC50 = 5430 nM
|
|
|
|
CP0968266
|
Pyridine-3-sulfonicacid(6-fluoro-quinolin-8-yl)-amide
Show/Hide
|
C14H10FN3O2S
|
1
|
| 1 |
IC50 = 5870 nM
|
|
|
|
CP0944902
|
11H-12-Thia-1,10,11-triaza-chrysene12,12-dioxide
Show/Hide
|
C14H9N3O2S
|
1
|
| 1 |
IC50 = 6150 nM
|
|
|
|
CP0947220
|
8-Benzene sulfonyl amino-quinoline-4-carboxylic acid methylamide
Show/Hide
|
C17H15N3O3S
|
1
|
| 1 |
IC50 = 6240 nM
|
|
|
|
CP0952868
|
12-Chloro-9-trifluoromethyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C16H8ClF3N2O2S
|
1
|
| 1 |
IC50 = 6250 nM
|
|
|
|
CP0960140
|
SID103061986
Show/Hide
|
C16H14N2O3S
|
1
|
| 1 |
IC50 = 6400 nM
|
|
|
|
CP0869380
|
2-Methyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene 3,3-dioxide
Show/Hide
|
C11H11N3O2S
|
1
|
| 1 |
IC50 = 6500 nM
|
|
|
|
CP0102947
|
5-bromo-N-quinolin-8-ylthiophene-2-sulfonamide
Show/Hide
|
C13H9BrN2O2S2
|
1
|
| 1 |
IC50 = 6800 nM
|
|
|
|
CP0857294
|
2,3-Dichloro-N-quinolin-8-yl-benzenesulfonamide
Show/Hide
|
C15H10Cl2N2O2S
|
1
|
| 1 |
IC50 = 7090 nM
|
|
|
|
CP0964015
|
N'-[2-Fluoro-5-(2-methyl-3,3-dioxo-1,2,3,4-tetrahydro-3lambda6-thia-2,4,5-triaza-phenanthren-1-yl)-benzyl]-N,N-dimethyl-ethane-1,2-diamine
Show/Hide
|
C22H26FN5O2S
|
1
|
| 1 |
IC50 = 7410 nM
|
|
|
|
CP0962718
|
N-(2-Dimethylamino-ethyl)-2-fluoro-5-(2-methyl-3,3-dioxo-1,2,3,4-tetrahydro-3lambda6-thia-2,4,5-triaza-phenanthren-1-yl)-benzamide
Show/Hide
|
C22H24FN5O3S
|
1
|
| 1 |
IC50 = 7460 nM
|
|
|
|
CP0961663
|
N-(5,6-Difluoro-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C15H10F2N2O2S
|
1
|
| 1 |
IC50 = 8000 nM
|
|
|
|
CP0969306
|
2-Chloro-N-quinolin-8-yl-benzenesulfonamide
Show/Hide
|
C15H11ClN2O2S
|
1
|
| 1 |
IC50 = 8000 nM
|
|
|
|
CP0957415
|
9-Chloro-12-trifluoromethyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C16H8ClF3N2O2S
|
1
|
| 1 |
IC50 = 8510 nM
|
|
|
|
CP0926570
|
[2-Fluoro-5-(2-methyl-3,3-dioxo-1,2,3,4-tetrahydro-3lambda6-thia-2,4,5-triaza-phenanthren-1-yl)-benzyl]-(2-morpholin-4-yl-ethyl)-amine
Show/Hide
|
C24H28FN5O3S
|
1
|
| 1 |
IC50 = 8560 nM
|
|
|
|
CP0961662
|
N-(6-Trifluoromethoxy-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C16H11F3N2O3S
|
1
|
| 1 |
IC50 = 9000 nM
|
|
|
|
CP0961012
|
N'-(6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-12-yl)-N,N-dimethyl-ethane-1,2-diamine
Show/Hide
|
C19H20N4O2S
|
1
|
| 1 |
IC50 = 9980 nM
|
|
|
|
CP0959873
|
N-[2-(Quinolin-8-ylsulfamoyl)-5-trifluoromethyl-phenyl]-isobutyramide
Show/Hide
|
C20H18F3N3O3S
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0962722
|
8-Benzene sulfonyl amino-quinoline-4-carboxylic acid amide
Show/Hide
|
C16H13N3O3S
|
1
|
| 1 |
IC50 = 10400 nM
|
|
|
|
CP0909203
|
9-Chloro-1-(4-fluoro-phenyl)-2-methyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene3,3-dioxide
Show/Hide
|
C17H13ClFN3O2S
|
1
|
| 1 |
IC50 = 12500 nM
|
|
|
|
CP0957419
|
6-Trifluoromethyl-pyridine-3-sulfonic acid(6-trifluoromethoxy-quinolin-8-yl)-amide
Show/Hide
|
C16H9F6N3O3S
|
1
|
| 1 |
IC50 = 12500 nM
|
|
|
|
CP0960150
|
1-Chloro-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C15H9ClN2O2S
|
1
|
| 1 |
IC50 = 12500 nM
|
|
|
|
CP0952473
|
12-Bromo-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C15H9BrN2O2S
|
1
|
| 1 |
IC50 = 12600 nM
|
|
|
|
CP0964023
|
6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysene-9-carboxylicacidmethylamide
Show/Hide
|
C17H13N3O3S
|
1
|
| 1 |
IC50 = 13200 nM
|
|
|
|
CP0930466
|
2-(12-Chloro-6,6-dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-9-ylamino)-propane-1,3-diol
Show/Hide
|
C18H16ClN3O4S
|
1
|
| 1 |
IC50 = 13400 nM
|
|
|
|
CP0969462
|
12-Trifluoromethyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C16H9F3N2O2S
|
1
|
| 1 |
IC50 = 14100 nM
|
|
|
|
CP0962721
|
(12-Chloro-6,6-dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-9-yl)-(3-hydroxy-pyrrolidin-1-yl)-methanone
Show/Hide
|
C20H16ClN3O4S
|
1
|
| 1 |
IC50 = 15000 nM
|
|
|
|
CP0969318
|
6-Methyl-pyridine-2-sulfonic acid quinolin-8-ylamide
Show/Hide
|
C15H13N3O2S
|
1
|
| 1 |
IC50 = 15400 nM
|
|
|
|
CP0232467
|
2-amino-N-quinolin-8-ylbenzenesulfonamide
Show/Hide
|
C15H13N3O2S
|
1
|
| 1 |
IC50 = 20800 nM
|
|
|
|
CP0949360
|
6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysene-1-carboxylicaciddimethylamide
Show/Hide
|
C18H15N3O3S
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1
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| 1 |
IC50 = 21000 nM
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CP0961831
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(6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-12-yl)-(2-morpholin-4-yl-ethyl)-amine
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C21H22N4O3S
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1
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| 1 |
IC50 = 22000 nM
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CP0866755
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N-[2-(Quinolin-8-ylsulfamoyl)-phenyl]-isobutyramide
Show/Hide
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C19H19N3O3S
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1
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| 1 |
IC50 = 24600 nM
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CP0848499
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8,12-Dichloro-9-fluoro-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
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C15H7Cl2FN2O2S
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1
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| 1 |
IC50 = 25000 nM
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CP0852827
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2,2,2-Trifluoro-N-[2-(quinolin-8-ylsulfamoyl)-5-trifluoromethyl-phenyl]-acetamide
Show/Hide
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C18H11F6N3O3S
|
1
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| 1 |
IC50 = 25000 nM
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CP0861208
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3-Chloro-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
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C15H9ClN2O2S
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1
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| 1 |
IC50 = 25000 nM
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CP0863749
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(6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-1-yl)-methyl-amine
Show/Hide
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C16H13N3O2S
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1
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| 1 |
IC50 = 25000 nM
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CP0866764
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12-Chloro-9-ethoxy-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
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C17H13ClN2O3S
|
1
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| 1 |
IC50 = 25000 nM
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CP0867131
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(12-Chloro-6,6-dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-9-yl)-(4-hydroxy-piperidin-1-yl)-methanone
Show/Hide
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C21H18ClN3O4S
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1
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| 1 |
IC50 = 25000 nM
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CP0869091
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1-Trifluoromethyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
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C16H9F3N2O2S
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1
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| 1 |
IC50 = 25000 nM
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CP0869381
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1-Methyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene 3,3-dioxide
Show/Hide
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C11H11N3O2S
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1
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| 1 |
IC50 = 25000 nM
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CP0869382
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(6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-1-yl)-diethyl-amine
Show/Hide
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C19H19N3O2S
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1
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| 1 |
IC50 = 25000 nM
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CP0869384
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N-(5-Benzyloxy-quinolin-8-yl)-benzenesulfonamide
Show/Hide
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C22H18N2O3S
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1
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| 1 |
IC50 = 25000 nM
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CP0869385
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12-Chloro-9-methanesulfonyl-5H-6-thia-4,5-diaza-chrysene6,6-dioxide
Show/Hide
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C16H11ClN2O4S2
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1
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| 1 |
IC50 = 25000 nM
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CP0909202
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9-Bromo-1-(4-fluoro-phenyl)-2-methyl-1,4-dihydro-2H-3-thia-2,4,5-triaza-phenanthrene 3,3-dioxide
Show/Hide
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C17H13BrFN3O2S
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1
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| 1 |
IC50 = 25000 nM
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CP0909204
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N-[4-(2-Dimethylamino-ethylamino)-quinolin-8-yl]-benzenesulfonamide
Show/Hide
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C19H22N4O2S
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1
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| 1 |
IC50 = 25000 nM
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CP0909205
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6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-1-ylamine
Show/Hide
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C15H11N3O2S
|
1
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| 1 |
IC50 = 25000 nM
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CP0909206
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6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysene-1-carboxylic acid amide
Show/Hide
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C16H11N3O3S
|
1
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| 1 |
IC50 = 25000 nM
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CP0909246
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12-Chloro-6,6-dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysene-9-carboxylicacid(2-hydroxy-1-hydroxymethyl-ethyl)-amide
Show/Hide
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C19H16ClN3O5S
|
1
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| 1 |
IC50 = 25000 nM
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CP0926551
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9-Chloro-1-trifluoromethyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
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C16H8ClF3N2O2S
|
1
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| 1 |
IC50 = 25000 nM
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CP0930462
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N'-(6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-1-yl)-N,N-dimethyl-ethane-1,2-diamine
Show/Hide
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C19H20N4O2S
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1
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| 1 |
IC50 = 25000 nM
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CP0930467
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6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysene-9-carboxylicacidamide
Show/Hide
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C16H11N3O3S
|
1
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| 1 |
IC50 = 25000 nM
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CP0930469
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6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysene-12-carboxylic acid(2-dimethylamino-ethyl)-amide
Show/Hide
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C20H20N4O3S
|
1
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| 1 |
IC50 = 25000 nM
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CP0930470
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N-(5-Morpholin-4-yl-quinolin-8-yl)-benzenesulfonamide
Show/Hide
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C19H19N3O3S
|
1
|
| 1 |
IC50 = 25000 nM
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CP0930471
|
N-(4-Diethylamino-quinolin-8-yl)-benzenesulfonamide
Show/Hide
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C19H21N3O2S
|
1
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| 1 |
IC50 = 25000 nM
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CP0930891
|
N-(4-Methylamino-quinolin-8-yl)-benzenesulfonamide
Show/Hide
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C16H15N3O2S
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1
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| 1 |
IC50 = 25000 nM
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CP0944893
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{2-[4-(6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-12-yl)-piperazin-1-yl]-ethyl}-dimethyl-amine
Show/Hide
|
C23H27N5O2S
|
1
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| 1 |
IC50 = 25000 nM
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CP0944894
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6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysene-12-carboxylic acid(2-piperidin-1-yl-ethyl)-amide
Show/Hide
|
C23H24N4O3S
|
1
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| 1 |
IC50 = 25000 nM
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CP0944901
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3,9-Dichloro-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C15H8Cl2N2O2S
|
1
|
| 1 |
IC50 = 25000 nM
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CP0952645
|
N-(4-Dimethylamino-quinolin-8-yl)-benzenesulfonamide
Show/Hide
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C17H17N3O2S
|
1
|
| 1 |
IC50 = 25000 nM
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CP0957700
|
6-Trifluoromethyl-pyridine-3-sulfonic acid(5-trifluoromethyl-quinolin-8-yl)-amide
Show/Hide
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C16H9F6N3O2S
|
1
|
| 1 |
IC50 = 25000 nM
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CP0959849
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6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysene-9-carboxylic acid
Show/Hide
|
C16H10N2O4S
|
1
|
| 1 |
IC50 = 25000 nM
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CP0961013
|
1-(6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-12-yl)-ethanol
Show/Hide
|
C17H14N2O3S
|
1
|
| 1 |
IC50 = 25000 nM
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CP0964017
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12-Chloro-6,6-dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysene-9-carboxylicacidpiperidin-4-ylester
Show/Hide
|
C21H18ClN3O4S
|
1
|
| 1 |
IC50 = 25000 nM
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CP0964019
|
(6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-12-yl)-morpholin-4-yl-methanone
Show/Hide
|
C20H17N3O4S
|
1
|
| 1 |
IC50 = 25000 nM
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CP0966513
|
(6,6-Dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysen-1-yl)-dimethyl-amine
Show/Hide
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C17H15N3O2S
|
1
|
| 1 |
IC50 = 25000 nM
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CP0966698
|
9-Chloro-6,6-dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysene-12-carbonitrile
Show/Hide
|
C16H8ClN3O2S
|
1
|
| 1 |
IC50 = 25000 nM
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CP0967194
|
{2-[1-(4-Fluoro-phenyl)-3,3-dioxo-3,4-dihydro-1H-3lambda6-thia-2,4,5-triaza-phenanthren-2-yl]-ethyl}-dimethyl-amine
Show/Hide
|
C20H21FN4O2S
|
1
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| 1 |
IC50 = 25000 nM
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CP0967195
|
12-Chloro-6,6-dioxo-5,6-dihydro-6lambda6-thia-4,5-diaza-chrysene-9-carboxylicacidpyrrolidin-3-ylester
Show/Hide
|
C20H16ClN3O4S
|
1
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| 1 |
IC50 = 25000 nM
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CP0969319
|
12-Chloro-8,9-difluoro-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C15H7ClF2N2O2S
|
1
|
| 1 |
IC50 = 25000 nM
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CP0969461
|
6-Trifluoromethyl-pyridine-3-sulfonicacid(6-fluoro-quinolin-8-yl)-amide
Show/Hide
|
C16H10F4N2O2S
|
1
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| 1 |
IC50 = 25000 nM
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CP0869090
|
1,4-Dihydro-2H-3-thia-2,4,5-triaza-phenanthrene3,3-dioxide
Show/Hide
|
C10H9N3O2S
|
1
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| 1 |
IC50 = 39500 nM
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CP0030614
|
4-methyl-N-(8-quinolinyl)benzenesulfonamide
Show/Hide
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C16H14N2O2S
|
1
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| 1 |
IC50 = 49900 nM
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CP0952865
|
8-Benzenesulfonylamino-quinoline-4-carboxylic acid methyl ester
Show/Hide
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C17H14N2O4S
|
1
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| 1 |
IC50 = 50000 nM
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CP0909247
|
2-(Quinolin-8-ylsulfamoyl)-benzoic acid methyl ester
Show/Hide
|
C17H14N2O4S
|
1
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| 1 |
IC50 = 58100 nM
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CP0969312
|
N-(5,7-Dichloro-quinolin-8-yl)-4-methyl-benzenesulfonamide
Show/Hide
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C16H12Cl2N2O2S
|
1
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| 1 |
IC50 = 79000 nM
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CP0052115
|
2-amino-N-(2-methylquinolin-8-yl)benzenesulfonamide
Show/Hide
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C16H15N3O2S
|
1
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| 1 |
IC50 = 100000 nM
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CP0336677
|
2-nitro-N-quinolin-8-yl-4-(trifluoromethyl)benzenesulfonamide
Show/Hide
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C16H10F3N3O4S
|
1
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| 1 |
IC50 = 100000 nM
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CP0378735
|
MLS001125540
Show/Hide
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C16H14N2O2S
|
1
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| 1 |
IC50 = 100000 nM
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CP0406533
|
4-methoxy-N-quinolin-8-ylbenzenesulfonamide
Show/Hide
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C16H14N2O3S
|
1
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| 1 |
IC50 = 100000 nM
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CP0406534
|
2-methoxy-N-quinolin-8-ylbenzenesulfonamide
Show/Hide
|
C16H14N2O3S
|
1
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| 1 |
IC50 = 100000 nM
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CP0857293
|
2-Amino-N-(5-chloro-quinolin-8-yl)-4-trifluoromethyl-benzenesulfonamide
Show/Hide
|
C16H11ClF3N3O2S
|
1
|
| 1 |
IC50 = 100000 nM
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CP0861221
|
N-(7-Ethyl-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C17H16N2O2S
|
1
|
| 1 |
IC50 = 100000 nM
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CP0861222
|
11-Methoxy-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C16H12N2O3S
|
1
|
| 1 |
IC50 = 100000 nM
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CP0866756
|
N-(5,7-Dichloro-quinolin-8-yl)-2,4,6-trimethyl-benzenesulfonamide
Show/Hide
|
C18H16Cl2N2O2S
|
1
|
| 1 |
IC50 = 100000 nM
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CP0869083
|
2-Amino-4-methyl-N-(3-methyl-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C17H17N3O2S
|
1
|
| 1 |
IC50 = 100000 nM
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CP0869088
|
N-(7-Chloro-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C15H11ClN2O2S
|
1
|
| 1 |
IC50 = 100000 nM
|
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CP0870270
|
N-(5-Chloro-6-methyl-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C16H13ClN2O2S
|
1
|
| 1 |
IC50 = 100000 nM
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CP0900935
|
N-(7-Hydroxy-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C15H12N2O3S
|
1
|
| 1 |
IC50 = 100000 nM
|
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CP0909207
|
1-Methoxy-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C16H12N2O3S
|
1
|
| 1 |
IC50 = 100000 nM
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CP0926141
|
N-(7-Methoxy-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C16H14N2O3S
|
1
|
| 1 |
IC50 = 100000 nM
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CP0942404
|
N-(2,6-difluorophenyl)[(6-methoxyquinolin-8-yl)amino]sulfonamide
Show/Hide
|
C16H13F2N3O3S
|
1
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| 1 |
IC50 = 100000 nM
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CP0944897
|
5-Methyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C16H12N2O2S
|
1
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| 1 |
IC50 = 100000 nM
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CP0944899
|
N-(4-Methoxy-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C16H14N2O3S
|
1
|
| 1 |
IC50 = 100000 nM
|
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CP0957690
|
2,4-Dichloro-N-(3-methyl-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C16H12Cl2N2O2S
|
1
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| 1 |
IC50 = 100000 nM
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CP0957692
|
N-(7-Isopropyl-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C18H18N2O2S
|
1
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| 1 |
IC50 = 100000 nM
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CP0957693
|
N-(3-chloro-2-methylphenyl)[(5-chloroquinolin-8-yl)amino]sulfonamide
Show/Hide
|
C16H13Cl2N3O2S
|
1
|
| 1 |
IC50 = 100000 nM
|
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CP0957697
|
N-(7-Methyl-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C16H14N2O2S
|
1
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| 1 |
IC50 = 100000 nM
|
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CP0959872
|
2-Amino-4-methoxy-N-(2-methyl-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C17H17N3O3S
|
1
|
| 1 |
IC50 = 100000 nM
|
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CP0960147
|
N-(5,6-Dimethyl-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C17H16N2O2S
|
1
|
| 1 |
IC50 = 100000 nM
|
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CP0961023
|
N-(2-Chloro-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C15H11ClN2O2S
|
1
|
| 1 |
IC50 = 100000 nM
|
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CP0961024
|
N-(5-Bromo-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C15H11BrN2O2S
|
1
|
| 1 |
IC50 = 100000 nM
|
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CP0961032
|
2,4-Dichloro-N-(6-methoxy-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C16H12Cl2N2O3S
|
1
|
| 1 |
IC50 = 100000 nM
|
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CP0961033
|
2-Chloro-6-methyl-N-quinolin-8-yl-benzenesulfonamide
Show/Hide
|
C16H13ClN2O2S
|
1
|
| 1 |
IC50 = 100000 nM
|
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CP0961034
|
N-(3-chloro-2-methylphenyl)[(6-methoxyquinolin-8-yl)amino]sulfonamide
Show/Hide
|
C17H16ClN3O3S
|
1
|
| 1 |
IC50 = 100000 nM
|
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|
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CP0961660
|
N-[2-(Quinolin-8-ylsulfamoyl)-5-trifluoromethyl-phenyl]-acetamide
Show/Hide
|
C18H14F3N3O3S
|
1
|
| 1 |
IC50 = 100000 nM
|
|
|
|
CP0963393
|
N-(6-Chloro-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C15H11ClN2O2S
|
1
|
| 1 |
IC50 = 100000 nM
|
|
|
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CP0963396
|
N-(6-Ethoxy-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C17H16N2O3S
|
1
|
| 1 |
IC50 = 100000 nM
|
|
|
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CP0964030
|
3-Methyl-5H-6-thia-4,5-diaza-chrysene 6,6-dioxide
Show/Hide
|
C16H12N2O2S
|
1
|
| 1 |
IC50 = 100000 nM
|
|
|
|
CP0969305
|
2-Methyl-N-quinolin-8-yl-benzenesulfonamide
Show/Hide
|
C16H14N2O2S
|
1
|
| 1 |
IC50 = 100000 nM
|
|
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CP0969307
|
SID26755381
Show/Hide
|
C16H15N3O3S
|
1
|
| 1 |
IC50 = 100000 nM
|
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CP0969313
|
2,4-Dichloro-N-(5-chloro-quinolin-8-yl)-benzenesulfonamide
Show/Hide
|
C15H9Cl3N2O2S
|
1
|
| 1 |
IC50 = 100000 nM
|
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CP0969315
|
2,6-Dichloro-N-quinolin-8-yl-benzenesulfonamide
Show/Hide
|
C15H10Cl2N2O2S
|
1
|
| 1 |
IC50 = 100000 nM
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