Brief Information of the Cell Line and Protein
Cell Line ID: CL000027 , tsA201
Synonyms
tsA-201
HEK293-TSA
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_2737
Protein ID: PT02526 , Sodium- and chloride-dependent GABA transporter 3
Gene Name SLC6A11
Organism Homo sapiens, Human
Protein Classification Transporter
Uniprot ID P48066
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000027  Protein ID: PT02526
 
Compound ID Compound Name Compound Formula
CP0000066
4-amino-n-[2,3-3H]butyric acid
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C4H9NO2
 1
1
IC50 = 1000 nM
   TI
   LI
   LO
   TS
CP0552300
CHEBI:18383
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C3H8N2O2
 1
1
IC50 = 31622.78 nM
   TI
   LI
   LO
   TS
CP0417616
2,4-dichloro-N-[1-[(4-cyanophenyl)methyl]piperidin-4-yl]benzamide
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C20H19Cl2N3O
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
CP0417622
2,4-dichloro-N-[1-(quinolin-2-ylmethyl)piperidin-4-yl]benzamide
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C22H21Cl2N3O
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
CP0436977
2,4-dichloro-N-[1-(naphthalen-2-ylmethyl)piperidin-4-yl]benzamide
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C23H22Cl2N2O
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
CP0474990
2,4-dichloro-N-[1-[(2-cyanophenyl)methyl]piperidin-4-yl]benzamide
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C20H19Cl2N3O
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
CP0417613
2,4-dichloro-N-[1-[(4-nitrophenyl)methyl]piperidin-4-yl]benzamide
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C19H19Cl2N3O3
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0436978
2,4-dichloro-N-(1-phenacylpiperidin-4-yl)benzamide
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C20H20Cl2N2O2
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0461786
2,4-dichloro-N-[1-[(4-iodophenyl)methyl]piperidin-4-yl]benzamide
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C19H19Cl2IN2O
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0463253
methyl 4-[[4-[(2,4-dichlorobenzoyl)amino]piperidin-1-yl]methyl]benzoate
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C21H22Cl2N2O3
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0470479
2,4-dichloro-N-[1-[(2-nitrophenyl)methyl]piperidin-4-yl]benzamide
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C19H19Cl2N3O3
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0510358
2,4-dichloro-N-[1-[(E)-3-phenylprop-2-enyl]piperidin-4-yl]benzamide
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C21H22Cl2N2O
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0202964
N-(1-benzylpiperidin-4-yl)naphthalene-2-carboxamide
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C23H24N2O
 1
1
Ki > 100000 nM
   TI
   LI
   LO
   TS
CP0390469
N-(1-benzylpiperidin-4-yl)-2,4-dichlorobenzamide
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C19H20Cl2N2O
 1
1
Ki > 100000 nM
   TI
   LI
   LO
   TS
CP0461828
N-(1-benzylpiperidin-4-yl)-1,3-benzodioxole-5-carboxamide
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C20H22N2O3
 1
1
Ki > 100000 nM
   TI
   LI
   LO
   TS