Brief Information of the Cell Line and Protein
Cell Line ID: CL000026 , CHO-K1
Synonyms
CHO K1
CHOK1
CHO cell clone K1
GM15452
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_0214
Protein ID: PT05453 , G-protein coupled receptor 55
Gene Name GPR55
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID Q9Y2T6
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000026  Protein ID: PT05453
 
Compound ID Compound Name Compound Formula
CP0516894
(E)-N-[[4-[[5-(hydroxymethyl)furan-2-yl]methyl-phenylsulfamoyl]phenyl]carbamothioyl]-3-(2-methoxyphenyl)prop-2-enamide
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C29H27N3O6S2
 1
1
EC50 = 100 nM
   TI
   LI
   LO
   TS
CP0402874
N-[[4-[2-hydroxyethyl(phenyl)sulfamoyl]phenyl]carbamothioyl]quinoline-7-carboxamide
   Show/Hide
C25H22N4O4S2
 1
1
EC50 = 200 nM
   TI
   LI
   LO
   TS
CP0512821
(E)-3-(2-methoxyphenyl)-N-[[4-[phenyl(pyridin-4-ylmethyl)sulfamoyl]phenyl]carbamothioyl]prop-2-enamide
   Show/Hide
C29H26N4O4S2
 1
1
EC50 = 300 nM
   TI
   LI
   LO
   TS
CP0512822
6-(2-hydroxyethyl)-N-[[4-[methyl(phenyl)sulfamoyl]phenyl]carbamothioyl]naphthalene-2-carboxamide
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C27H25N3O4S2
 1
1
EC50 = 300 nM
   TI
   LI
   LO
   TS
CP0396544
(E)-3-(2-methoxyphenyl)-N-[[4-[methyl(phenyl)sulfamoyl]phenyl]carbamothioyl]prop-2-enamide
   Show/Hide
C24H23N3O4S2
 1
1
EC50 = 400 nM
   TI
   LI
   LO
   TS
CP0389317
N-[[4-[(4-hydroxyphenyl)methyl-phenylsulfamoyl]phenyl]carbamothioyl]quinoline-7-carboxamide
   Show/Hide
C30H24N4O4S2
 1
1
EC50 = 500 nM
   TI
   LI
   LO
   TS
CP0516893
(E)-N-[[4-[(4-hydroxyphenyl)methyl-phenylsulfamoyl]phenyl]carbamothioyl]-3-(2-methoxyphenyl)prop-2-enamide
   Show/Hide
C30H27N3O5S2
 1
1
EC50 = 500 nM
   TI
   LI
   LO
   TS
CP0558995
(E)-3-(2-methoxyphenyl)-N-[[4-[methyl(pyridin-4-yl)sulfamoyl]phenyl]carbamothioyl]prop-2-enamide
   Show/Hide
C23H22N4O4S2
 1
1
EC50 = 500 nM
   TI
   LI
   LO
   TS
CP0396543
N-[[4-[[5-(hydroxymethyl)furan-2-yl]methyl-phenylsulfamoyl]phenyl]carbamothioyl]quinoline-7-carboxamide
   Show/Hide
C29H24N4O5S2
 1
1
EC50 = 600 nM
   TI
   LI
   LO
   TS
CP0456696
(E)-3-(2-methoxyphenyl)-N-[[4-(phenylsulfamoyl)phenyl]carbamothioyl]prop-2-enamide
   Show/Hide
C23H21N3O4S2
 1
1
EC50 = 600 nM
   TI
   LI
   LO
   TS
CP0530861
(E)-N-[[4-[2-hydroxyethyl(phenyl)sulfamoyl]phenyl]carbamothioyl]-3-(2-methoxyphenyl)prop-2-enamide
   Show/Hide
C25H25N3O5S2
 1
1
EC50 = 700 nM
   TI
   LI
   LO
   TS
CP0549790
N-[[4-[phenyl(pyridin-4-ylmethyl)sulfamoyl]phenyl]carbamothioyl]quinoline-7-carboxamide
   Show/Hide
C29H23N5O3S2
 1
1
EC50 = 900 nM
   TI
   LI
   LO
   TS
CP0396541
N-[[4-[methyl(phenyl)sulfamoyl]phenyl]carbamothioyl]quinoline-7-carboxamide
   Show/Hide
C24H20N4O3S2
 1
1
EC50 = 1000 nM
   TI
   LI
   LO
   TS
CP0396542
(E)-N-[[4-[(3-hydroxyphenyl)methyl-phenylsulfamoyl]phenyl]carbamothioyl]-3-(2-methoxyphenyl)prop-2-enamide
   Show/Hide
C30H27N3O5S2
 1
1
EC50 = 2000 nM
   TI
   LI
   LO
   TS
CP0402873
(E)-N-[[4-[(2-hydroxyphenyl)methyl-phenylsulfamoyl]phenyl]carbamothioyl]-3-(2-methoxyphenyl)prop-2-enamide
   Show/Hide
C30H27N3O5S2
 1
1
EC50 = 2000 nM
   TI
   LI
   LO
   TS
CP0430093
6-(hydroxymethyl)-N-[[4-[methyl(phenyl)sulfamoyl]phenyl]carbamothioyl]naphthalene-2-carboxamide
   Show/Hide
C26H23N3O4S2
 1
1
EC50 = 4000 nM
   TI
   LI
   LO
   TS
CP0512823
6-(2-hydroxyethyl)-N-[[4-[[5-(hydroxymethyl)furan-2-yl]methyl-phenylsulfamoyl]phenyl]carbamothioyl]naphthalene-2-carboxamide
   Show/Hide
C32H29N3O6S2
 1
1
EC50 = 6000 nM
   TI
   LI
   LO
   TS
CP0561102
6-(2-hydroxyethyl)-N-[[4-[2-hydroxyethyl(phenyl)sulfamoyl]phenyl]carbamothioyl]naphthalene-2-carboxamide
   Show/Hide
C28H27N3O5S2
 1
1
EC50 = 20000 nM
   TI
   LI
   LO
   TS
CP0529554
(E)-N-[[4-[(3,4-dimethyl-1,2-oxazol-5-yl)sulfamoyl]phenyl]carbamothioyl]-3-(2-methoxyphenyl)prop-2-enamide
   Show/Hide
C22H22N4O5S2
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0530859
N-[[4-[methyl(phenyl)sulfamoyl]phenyl]carbamothioyl]quinoline-3-carboxamide
   Show/Hide
C24H20N4O3S2
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0530860
(E)-N-[[4-(2-hydroxyethylsulfamoyl)phenyl]carbamothioyl]-3-(2-methoxyphenyl)prop-2-enamide
   Show/Hide
C19H21N3O5S2
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0541472
(E)-N-[[4-(2,3-dihydroxypropylsulfamoyl)phenyl]carbamothioyl]-3-(2-methoxyphenyl)prop-2-enamide
   Show/Hide
C20H23N3O6S2
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0384980
3-[1-(1-phenylcyclopropanecarbonyl)piperidin-4-yl]-5-pyridin-3-yl-1,3,4-oxadiazol-2-one
   Show/Hide
C22H22N4O3
 1
1
IC50 = 420 nM
   TI
   LI
   LO
   TS
CP0477753
3-[1-[1-(4-chlorophenyl)cyclopropanecarbonyl]-4-piperidyl]-5-phenyl-1,3,4-oxadiazol-2-one
   Show/Hide
C23H22ClN3O3
 1
1
IC50 = 640 nM
   TI
   LI
   LO
   TS
CP0464108
3-[1-[2,2-dimethyl-1-(4-methylphenyl)cyclopropanecarbonyl]piperidin-4-yl]-5-phenyl-1,3,4-oxadiazol-2-one
   Show/Hide
C26H29N3O3
 1
1
IC50 = 770 nM
   TI
   LI
   LO
   TS
CP0489065
3-[1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]piperidin-4-yl]-5-[4-(trifluoromethyl)phenyl]-1,3,4-oxadiazol-2-one
   Show/Hide
C25H24F3N3O4
 1
1
IC50 = 1800 nM
   TI
   LI
   LO
   TS
CP0489066
3-[1-[1-(2,4-dichlorophenyl)cyclopropanecarbonyl]piperidin-4-yl]-5-phenyl-1,3,4-oxadiazol-2-one
   Show/Hide
C23H21Cl2N3O3
 1
1
IC50 = 2500 nM
   TI
   LI
   LO
   TS
CP0489064
5-(4-methoxyphenyl)-3-[1-(1-phenylcyclopropanecarbonyl)piperidin-4-yl]-1,3,4-oxadiazol-2-one
   Show/Hide
C24H25N3O4
 1
1
IC50 = 7000 nM
   TI
   LI
   LO
   TS
CP0544723
3-[1-[oxo-(1-phenylcyclopropyl)methyl]-4-piperidinyl]-5-phenyl-1,3,4-oxadiazol-2-one
   Show/Hide
C23H23N3O3
 1
1
IC50 = 12000 nM
   TI
   LI
   LO
   TS