| Compound ID |
Compound Name |
Compound Formula |
|
CP0549830
|
1-(4-bromophenyl)-3-[2-oxo-1-(1-pyrimidin-2-ylpiperidin-4-yl)pyrrolidin-3-yl]urea
Show/Hide
|
C20H23BrN6O2
|
2
|
| 1 |
EC50 = 8 nM
|
|
|
| 2 |
EC50 = 385 nM
|
|
|
|
CP0545821
|
1-[(3S,4R)-4-(2,6-difluoro-4-methoxyphenyl)-2-oxopyrrolidin-3-yl]-3-phenylurea
Show/Hide
|
C18H17F2N3O3
|
1
|
| 1 |
EC50 = 130 nM
|
|
|
|
CP0494974
|
1-(4-bromophenyl)-3-[1-(1,3-dimethylpyrazol-4-yl)-2-oxopyrrolidin-3-yl]urea
Show/Hide
|
C16H18BrN5O2
|
2
|
| 1 |
EC50 = 142 nM
|
|
|
| 2 |
EC50 = 740 nM
|
|
|
|
CP0532499
|
1-(4-bromophenyl)-3-(2-oxo-1-piperidin-4-ylpyrrolidin-3-yl)urea
Show/Hide
|
C16H21BrN4O2
|
2
|
| 1 |
EC50 = 230 nM
|
|
|
| 2 |
EC50 = 1030 nM
|
|
|
|
CP0494973
|
1-[1-[(1-benzylpiperidin-4-yl)methyl]-2-oxopyrrolidin-3-yl]-3-(4-bromophenyl)urea
Show/Hide
|
C24H29BrN4O2
|
2
|
| 1 |
EC50 = 250 nM
|
|
|
| 2 |
EC50 = 2250 nM
|
|
|
|
CP0568771
|
1-(4-bromophenyl)-3-[2-oxo-1-(piperidin-4-ylmethyl)pyrrolidin-3-yl]urea
Show/Hide
|
C17H23BrN4O2
|
2
|
| 1 |
EC50 = 270 nM
|
|
|
| 2 |
EC50 = 3290 nM
|
|
|
|
CP0568770
|
1-(4-bromophenyl)-3-[1-(3,5-dimethyl-1-phenylpyrazol-4-yl)-2-oxopyrrolidin-3-yl]urea
Show/Hide
|
C22H22BrN5O2
|
2
|
| 1 |
EC50 = 280 nM
|
|
|
| 2 |
EC50 = 400 nM
|
|
|
|
CP0544015
|
1-(4-bromophenyl)-3-(2-oxo-1-phenylpyrrolidin-3-yl)urea
Show/Hide
|
C17H16BrN3O2
|
2
|
| 1 |
EC50 = 300 nM
|
|
|
| 2 |
EC50 = 430 nM
|
|
|
|
CP0574204
|
1-[1-(1-benzylpiperidin-4-yl)-2-oxopyrrolidin-3-yl]-3-(4-bromophenyl)urea
Show/Hide
|
C23H27BrN4O2
|
2
|
| 1 |
EC50 = 350 nM
|
|
|
| 2 |
EC50 = 2870 nM
|
|
|
|
CP0532500
|
tert-butyl 4-[[3-[(4-bromophenyl)carbamoylamino]-2-oxopyrrolidin-1-yl]methyl]piperidine-1-carboxylate
Show/Hide
|
C22H31BrN4O4
|
2
|
| 1 |
EC50 = 400 nM
|
|
|
| 2 |
EC50 = 2160 nM
|
|
|
|
CP0567577
|
tert-butyl 3-[3-[(4-bromophenyl)carbamoylamino]-2-oxopyrrolidin-1-yl]azetidine-1-carboxylate
Show/Hide
|
C19H25BrN4O4
|
2
|
| 1 |
EC50 = 410 nM
|
|
|
| 2 |
EC50 = 2350 nM
|
|
|
|
CP0572629
|
N-(azetidin-3-yl)-2-[(4-bromophenyl)carbamoylamino]-2-cyclopentylacetamide
Show/Hide
|
C17H23BrN4O2
|
1
|
| 1 |
EC50 = 500 nM
|
|
|
|
CP0573212
|
1-(4-bromophenyl)-3-[1-(4-fluorophenyl)-2-oxopyrrolidin-3-yl]urea
Show/Hide
|
C17H15BrFN3O2
|
2
|
| 1 |
EC50 = 510 nM
|
|
|
| 2 |
EC50 = 1970 nM
|
|
|
|
CP0544334
|
tert-butyl 4-[3-[(4-bromophenyl)carbamoylamino]-2-oxopyrrolidin-1-yl]piperidine-1-carboxylate
Show/Hide
|
C21H29BrN4O4
|
2
|
| 1 |
EC50 = 730 nM
|
|
|
| 2 |
EC50 = 6300 nM
|
|
|
|
CP0557848
|
2-[(4-bromophenyl)carbamoylamino]-2-cyclopentyl-N-pyridin-3-ylacetamide
Show/Hide
|
C19H21BrN4O2
|
1
|
| 1 |
EC50 = 740 nM
|
|
|
|
CP0494972
|
1-(4-bromophenyl)-3-[2-oxo-1-(1-propan-2-ylpyrazol-4-yl)pyrrolidin-3-yl]urea
Show/Hide
|
C17H20BrN5O2
|
1
|
| 1 |
EC50 = 884 nM
|
|
|
|
CP0578433
|
2-[(4-bromophenyl)carbamoylamino]-2-cyclopentyl-N-(oxolan-2-ylmethyl)acetamide
Show/Hide
|
C19H26BrN3O3
|
1
|
| 1 |
EC50 = 940 nM
|
|
|
|
CP0571851
|
1-[(4-bromophenyl)carbamoylamino]-N-pyridin-3-ylcyclopentane-1-carboxamide
Show/Hide
|
C18H19BrN4O2
|
1
|
| 1 |
EC50 = 1300 nM
|
|
|
|
CP0560516
|
(2S)-2-[(4-bromophenyl)carbamoylamino]-3-cyclopropyl-N-pyridin-3-ylpropanamide
Show/Hide
|
C18H19BrN4O2
|
1
|
| 1 |
EC50 = 1350 nM
|
|
|
|
CP0486346
|
2-[(4-bromophenyl)carbamoylamino]-2-cyclopentyl-N-pyridazin-3-ylacetamide
Show/Hide
|
C18H20BrN5O2
|
1
|
| 1 |
EC50 = 1410 nM
|
|
|
|
CP0513802
|
1-[(4-bromophenyl)carbamoylamino]-N-(1,3-dimethylpyrazol-4-yl)cyclopentane-1-carboxamide
Show/Hide
|
C18H22BrN5O2
|
1
|
| 1 |
EC50 = 1850 nM
|
|
|
|
CP0577733
|
2-[(4-bromophenyl)carbamoylamino]-2-cyclopentyl-N-(1,3-dimethylpyrazol-4-yl)acetamide
Show/Hide
|
C19H24BrN5O2
|
1
|
| 1 |
EC50 = 1900 nM
|
|
|
|
CP0574643
|
2-[(4-bromophenyl)carbamoylamino]-3-cyclohexyl-N-pyridin-3-ylpropanamide
Show/Hide
|
C21H25BrN4O2
|
1
|
| 1 |
EC50 = 2150 nM
|
|
|
|
CP0513791
|
1-[(4-bromophenyl)carbamoylamino]-N-(6-chloropyridin-3-yl)cyclopentane-1-carboxamide
Show/Hide
|
C18H18BrClN4O2
|
1
|
| 1 |
EC50 = 2580 nM
|
|
|
|
CP0549831
|
1-(4-bromophenyl)-3-[2-oxo-1-(1-pyridin-4-ylpyrazol-4-yl)pyrrolidin-3-yl]urea
Show/Hide
|
C19H17BrN6O2
|
1
|
| 1 |
EC50 = 3760 nM
|
|
|
|
CP0553343
|
1-[(4-bromophenyl)carbamoylamino]-N-(1-propan-2-ylpyrazol-4-yl)cyclopentane-1-carboxamide
Show/Hide
|
C19H24BrN5O2
|
1
|
| 1 |
EC50 = 4150 nM
|
|
|
|
CP0560497
|
2-[(4-bromophenyl)carbamoylamino]-2-(oxan-4-yl)-N-pyridin-3-ylacetamide
Show/Hide
|
C19H21BrN4O3
|
1
|
| 1 |
EC50 = 4170 nM
|
|
|
|
CP0565446
|
(2S)-2-[(4-bromophenyl)carbamoylamino]-4-methyl-N-pyridin-3-ylpentanamide
Show/Hide
|
C18H21BrN4O2
|
1
|
| 1 |
EC50 = 4260 nM
|
|
|
|
CP0557846
|
2-[(4-bromophenyl)carbamoylamino]-2-cyclopentyl-N-pyrimidin-5-ylacetamide
Show/Hide
|
C18H20BrN5O2
|
1
|
| 1 |
EC50 = 6330 nM
|
|
|
|
CP0513805
|
1-[(4-bromophenyl)carbamoylamino]-N-pyrimidin-5-ylcyclopentane-1-carboxamide
Show/Hide
|
C17H18BrN5O2
|
1
|
| 1 |
EC50 = 7270 nM
|
|
|
|
CP0513804
|
2-[(4-bromophenyl)carbamoylamino]-2-cyclopentyl-N-(1-propan-2-ylpyrazol-4-yl)acetamide
Show/Hide
|
C20H26BrN5O2
|
1
|
| 1 |
EC50 = 7450 nM
|
|
|
|
CP0553357
|
2-[(4-bromophenyl)carbamoylamino]-2-cyclopropyl-N-pyridin-3-ylacetamide
Show/Hide
|
C17H17BrN4O2
|
1
|
| 1 |
EC50 = 7800 nM
|
|
|
|
CP0513790
|
1-[(4-bromophenyl)carbamoylamino]-N-(5-methylpyridin-3-yl)cyclopentane-1-carboxamide
Show/Hide
|
C19H21BrN4O2
|
1
|
| 1 |
EC50 = 9800 nM
|
|
|
|
CP0569501
|
1-[(4-bromophenyl)carbamoylamino]-N-(6-methylpyridin-3-yl)cyclopentane-1-carboxamide
Show/Hide
|
C19H21BrN4O2
|
1
|
| 1 |
EC50 = 9900 nM
|
|
|
|
CP0557847
|
2-[(4-bromophenyl)carbamoylamino]-N-pyridin-3-ylacetamide
Show/Hide
|
C14H13BrN4O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0557849
|
1-[(4-bromophenyl)carbamoylamino]-N-pyridin-2-ylcyclopentane-1-carboxamide
Show/Hide
|
C18H19BrN4O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0560513
|
1-[(4-bromophenyl)carbamoylamino]-N-(2H-tetrazol-5-ylmethyl)cyclopentane-1-carboxamide
Show/Hide
|
C15H18BrN7O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0560517
|
2-[(4-bromophenyl)carbamoylamino]-2-cyclopentyl-N-(oxan-4-yl)acetamide
Show/Hide
|
C19H26BrN3O3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0569302
|
2-[(4-bromophenyl)carbamoylamino]-2-cyclopentyl-N-(oxetan-3-yl)acetamide
Show/Hide
|
C17H22BrN3O3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0572630
|
2-[(4-bromophenyl)carbamoylamino]-2-cyclopentyl-N-(1-methylpiperidin-4-yl)acetamide
Show/Hide
|
C20H29BrN4O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0578731
|
1-[(4-bromophenyl)carbamoylamino]-N-(1-methylpiperidin-4-yl)cyclopentane-1-carboxamide
Show/Hide
|
C19H27BrN4O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0568027
|
1-(4-cyanophenyl)-3-[1-(2-fluorophenyl)-2-oxopyrrolidin-3-yl]urea
Show/Hide
|
C18H15FN4O2
|
1
|
| 1 |
EC50 = 15000 nM
|
|
|
