| Compound ID |
Compound Name |
Compound Formula |
|
CP0041613
|
Anapriline
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|
C16H21NO2
|
2
|
| 1 |
EC50 > 5011.87 nM
|
|
|
| 2 |
IC50 > 5011.87 nM
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CP0066236
|
1-(dimethylamino)-3-[(2-methyl-1H-1,2-benzazaborinin-8-yl)oxy]propan-2-ol
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|
C14H21BN2O2
|
2
|
| 1 |
EC50 > 5011.87 nM
|
|
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| 2 |
IC50 > 5011.87 nM
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CP0366351
|
1-(dimethylamino)-3-[(2-methyl-1H-1,2-benzazaborinin-5-yl)oxy]propan-2-ol
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|
C14H21BN2O2
|
2
|
| 1 |
EC50 > 5011.87 nM
|
|
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| 2 |
IC50 > 5011.87 nM
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|
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CP0195952
|
(2S,4R)-1-((R)-5-chloro-1-(2,4-dimethoxyphenylsulfonyl)-3-(2-methoxyphenyl)-2-oxoindolin-3-yl)-4-hydroxy-N,N-dimethylpyrrolidine-2-carboxamide
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|
C30H32ClN3O8S
|
1
|
| 1 |
Ki = 22 nM
|
|
|
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CP0457764
|
1-(2-(1-(2,4-dimethoxyphenylsulfonyl)-1,2,3,4-tetrahydroquinolin-2-yl)ethylsulfonyl)-N-(thiophen-3-ylmethyl)piperidin-4-amine
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|
C29H37N3O6S3
|
1
|
| 1 |
Ki = 33 nM
|
|
|
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CP0401557
|
N-(cyclohexylmethyl)-1-[2-[1-(2,4-dimethoxyphenyl)sulfonyl-3,4-dihydro-2H-quinolin-2-yl]ethylsulfonyl]piperidin-4-amine
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|
C31H45N3O6S2
|
1
|
| 1 |
Ki = 188 nM
|
|
|
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CP0453825
|
N-benzyl-1-[2-[1-(2,4-dimethoxyphenyl)sulfonyl-3,4-dihydro-2H-quinolin-2-yl]ethylsulfonyl]piperidin-4-amine
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|
C31H39N3O6S2
|
1
|
| 1 |
Ki = 192 nM
|
|
|
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CP0874438
|
N-(cyclohexylmethyl)-1-(2-(1-(2,4-dimethoxyphenylsulfonyl)-1,2,3,4-tetrahydroquinolin-2-yl)ethylsulfonyl)piperidin-4-amine hydrobromide
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|
C31H46BrN3O6S2
|
1
|
| 1 |
Ki = 314 nM
|
|
|
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CP0390542
|
1-(2-(1-(2,4-dimethoxyphenylsulfonyl)-1,2,3,4-tetrahydroquinolin-2-yl)ethylsulfonyl)-N-(4-fluorobenzyl)piperidin-4-amine
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|
C31H38FN3O6S2
|
1
|
| 1 |
Ki = 395 nM
|
|
|
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CP0439177
|
1-(2-(1-(2,4-dimethoxyphenylsulfonyl)-1,2,3,4-tetrahydroquinolin-2-yl)ethylsulfonyl)-N-phenethylpiperidin-4-amine
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|
C32H41N3O6S2
|
1
|
| 1 |
Ki = 486 nM
|
|
|
|
CP0374019
|
1-(2-(1-(2,4-dimethoxyphenylsulfonyl)-1,2,3,4-tetrahydroquinolin-2-yl)ethylsulfonyl)-N-((tetrahydro-2H-pyran-4-yl)methyl)piperidin-4-amine
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|
C30H43N3O7S2
|
1
|
| 1 |
Ki = 553 nM
|
|
|
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CP0430021
|
N-cyclobutyl-1-[2-[1-(2,4-dimethoxyphenyl)sulfonyl-3,4-dihydro-2H-quinolin-2-yl]ethylsulfonyl]piperidin-4-amine
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|
C28H39N3O6S2
|
1
|
| 1 |
Ki = 709 nM
|
|
|
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CP0390541
|
1-(2-(1-(2,4-dimethoxyphenylsulfonyl)-1,2,3,4-tetrahydroquinolin-2-yl)ethylsulfonyl)-N-(thiophen-2-ylmethyl)piperidin-4-amine
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|
C29H37N3O6S3
|
1
|
| 1 |
Ki = 720 nM
|
|
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CP0397362
|
1-(2-(1-(2,4-dimethoxyphenylsulfonyl)-1,2,3,4-tetrahydroquinolin-2-yl)ethylsulfonyl)-N-isopentylpiperidin-4-amine
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|
C29H43N3O6S2
|
1
|
| 1 |
Ki = 947 nM
|
|
|
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CP0845382
|
N-(cyclohexylmethyl)-1-(2-(1-(2,4-dimethoxyphenylsulfonyl)-1,2,3,4-tetrahydroquinolin-2-yl)ethylsulfonyl)piperidin-4-amine hydrochloride
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|
C31H46ClN3O6S2
|
1
|
| 1 |
Ki = 1129 nM
|
|
|
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CP0534465
|
N-(cyclopropylmethyl)-1-[2-[1-(2,4-dimethoxyphenyl)sulfonyl-3,4-dihydro-2H-quinolin-2-yl]ethylsulfonyl]piperidin-4-amine
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|
C28H39N3O6S2
|
1
|
| 1 |
Ki = 1257 nM
|
|
|
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CP0430020
|
1-(2-(1-(2,4-dimethoxyphenylsulfonyl)-1,2,3,4-tetrahydroquinolin-2-yl)ethylsulfonyl)-N-propylpiperidin-4-amine
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|
C27H39N3O6S2
|
1
|
| 1 |
Ki = 1268 nM
|
|
|
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CP0401556
|
1-(2-(1-(2,4-dimethoxyphenylsulfonyl)-1,2,3,4-tetrahydroquinolin-2-yl)ethylsulfonyl)-N-(3-methoxybenzyl)piperidin-4-amine
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|
C32H41N3O7S2
|
1
|
| 1 |
Ki = 2600 nM
|
|
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CP0374012
|
2-(1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroquinolin-2-yl)-1-(4-(thiophen-2-ylmethylamino)piperidin-1-yl)ethanone
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|
C27H30ClN3O3S2
|
1
|
| 1 |
Ki = 3654 nM
|
|
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CP0374014
|
1-(3-(1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroquinolin-2-yl)propyl)-N-(thiophen-2-ylmethyl)piperidin-4-amine
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|
C28H34ClN3O2S2
|
1
|
| 1 |
Ki = 4617 nM
|
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CP0430019
|
1-(2-(1-(2,4-dimethoxyphenylsulfonyl)-1,2,3,4-tetrahydroquinolin-2-yl)ethylsulfonyl)-N-(1-phenylethyl)piperidin-4-amine
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|
C32H41N3O6S2
|
1
|
| 1 |
Ki = 4803 nM
|
|
|
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CP0390543
|
1-(2-(1-(2,4-dimethoxyphenylsulfonyl)-1,2,3,4-tetrahydroquinolin-2-yl)ethylsulfonyl)-N-(4-methoxybenzyl)piperidin-4-amine
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|
C32H41N3O7S2
|
1
|
| 1 |
Ki = 4926 nM
|
|
|
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CP0430006
|
1-(2-(1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroquinolin-2-yl)ethylsulfonyl)-N-(thiophen-2-ylmethyl)piperidin-4-amine
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|
C27H32ClN3O4S3
|
1
|
| 1 |
Ki = 4963 nM
|
|
|
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CP0439176
|
1-(3-(1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroquinolin-2-yl)propylsulfonyl)-N-(thiophen-2-ylmethyl)piperidin-4-amine
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|
C28H34ClN3O4S3
|
1
|
| 1 |
Ki = 5564 nM
|
|
|
|
CP0390537
|
(1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroquinolin-2-yl)methyl 4-(thiophen-2-ylmethylamino)piperidine-1-carboxylate
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|
C27H30ClN3O4S2
|
1
|
| 1 |
Ki = 6164 nM
|
|
|
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CP0390538
|
3-(1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroquinolin-2-yl)-1-(4-(thiophen-2-ylmethylamino)piperidin-1-yl)propan-1-one
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|
C28H32ClN3O3S2
|
1
|
| 1 |
Ki = 6888 nM
|
|
|
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CP0390540
|
1-((1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroquinolin-2-yl)methylsulfonyl)-N-(thiophen-2-ylmethyl)piperidin-4-amine
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|
C26H30ClN3O4S3
|
1
|
| 1 |
Ki = 8734 nM
|
|
|
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CP0430017
|
N-[[1-(4-chlorophenyl)sulfonyl-3,4-dihydro-2H-quinolin-2-yl]methyl]-N-methyl-4-(thiophen-2-ylmethylamino)piperidine-1-carboxamide
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|
C28H33ClN4O3S2
|
1
|
| 1 |
Ki = 8866 nM
|
|
|
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CP0374013
|
1-(2-(1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroquinolin-2-yl)ethyl)-N-(thiophen-2-ylmethyl)piperidin-4-amine
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|
C27H32ClN3O2S2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0430016
|
N-[[1-(4-chlorophenyl)sulfonyl-3,4-dihydro-2H-quinolin-2-yl]methyl]-4-(thiophen-2-ylmethylamino)piperidine-1-carboxamide
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|
C27H31ClN4O3S2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0390539
|
4-(1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroquinolin-2-yl)-1-(4-(thiophen-2-ylmethylamino)piperidin-1-yl)butan-1-one
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|
C29H34ClN3O3S2
|
1
|
| 1 |
Ki > 8000 nM
|
|
|
