| Compound ID |
Compound Name |
Compound Formula |
|
CP0528434
|
2-cyclopentyl-3-(4-methoxyphenyl)-10-methylpyrimido[4,5-b]quinoline-4,5-dione
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|
C24H23N3O3
|
1
|
| 1 |
EC50 = 25.4 nM
|
|
|
|
CP0479287
|
2-cyclopentyl-10-methyl-3-(4-methylphenyl)pyrimido[4,5-b]quinoline-4,5-dione
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|
C24H23N3O2
|
1
|
| 1 |
EC50 = 26.5 nM
|
|
|
|
CP0533055
|
2-cyclohexyl-10-methyl-3-(4-methylphenyl)pyrimido[4,5-b]quinoline-4,5-dione
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|
C25H25N3O2
|
1
|
| 1 |
EC50 = 27.4 nM
|
|
|
|
CP0479263
|
3-(3-chloro-4-methoxyphenyl)-2-cyclopentyl-10-methylpyrimido[4,5-b]quinoline-4,5-dione
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|
C24H22ClN3O3
|
1
|
| 1 |
EC50 = 27.5 nM
|
|
|
|
CP0314164
|
2-cyclohexyl-10-methyl-3-phenylpyrimido[4,5-b]quinoline-4,5-dione
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|
C24H23N3O2
|
1
|
| 1 |
EC50 = 28.8 nM
|
|
|
|
CP0479290
|
3-(4-methoxyphenyl)-10-methyl-2-(2-methylpropyl)pyrimido[4,5-b]quinoline-4,5-dione
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|
C23H23N3O3
|
1
|
| 1 |
EC50 = 33.7 nM
|
|
|
|
CP0479275
|
3-(4-chlorophenyl)-2-cyclopentyl-10-methylpyrimido[4,5-b]quinoline-4,5-dione
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|
C23H20ClN3O2
|
1
|
| 1 |
EC50 = 42.5 nM
|
|
|
|
CP0479269
|
3-(3-chlorophenyl)-2-cyclopentyl-10-methylpyrimido[4,5-b]quinoline-4,5-dione
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|
C23H20ClN3O2
|
1
|
| 1 |
EC50 = 43 nM
|
|
|
|
CP0479288
|
10-methyl-3-(4-methylphenyl)-2-(2-methylpropyl)pyrimido[4,5-b]quinoline-4,5-dione
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|
C23H23N3O2
|
1
|
| 1 |
EC50 = 43.9 nM
|
|
|
|
CP0479266
|
3-(4-chlorophenyl)-2-cyclohexyl-10-methylpyrimido[4,5-b]quinoline-4,5-dione
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|
C24H22ClN3O2
|
1
|
| 1 |
EC50 = 44.1 nM
|
|
|
|
CP0479268
|
2-(cyclohexylmethyl)-10-methyl-3-phenylpyrimido[4,5-b]quinoline-4,5-dione
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|
C25H25N3O2
|
1
|
| 1 |
EC50 = 49.1 nM
|
|
|
|
CP0479272
|
3-(4-chlorophenyl)-10-methyl-2-(2-methylpropyl)pyrimido[4,5-b]quinoline-4,5-dione
Show/Hide
|
C22H20ClN3O2
|
1
|
| 1 |
EC50 = 56.1 nM
|
|
|
|
CP0479264
|
3-(3-chloro-4-methoxyphenyl)-10-methyl-2-(2-methylpropyl)pyrimido[4,5-b]quinoline-4,5-dione
Show/Hide
|
C23H22ClN3O3
|
1
|
| 1 |
EC50 = 57.7 nM
|
|
|
|
CP0479286
|
3-(3-chloro-4-methoxyphenyl)-2-cyclohexyl-10-methylpyrimido[4,5-b]quinoline-4,5-dione
Show/Hide
|
C25H24ClN3O3
|
1
|
| 1 |
EC50 = 58.5 nM
|
|
|
|
CP0479274
|
2-cyclohexyl-3-(4-methoxyphenyl)-10-methylpyrimido[4,5-b]quinoline-4,5-dione
Show/Hide
|
C25H25N3O3
|
1
|
| 1 |
EC50 = 62.1 nM
|
|
|
|
CP0479271
|
3-(3-chlorophenyl)-10-methyl-2-(2-methylpropyl)pyrimido[4,5-b]quinoline-4,5-dione
Show/Hide
|
C22H20ClN3O2
|
1
|
| 1 |
EC50 = 63.1 nM
|
|
|
|
CP0533053
|
3-(4-chlorophenyl)-2-(cyclohexylmethyl)-10-methylpyrimido[4,5-b]quinoline-4,5-dione
Show/Hide
|
C25H24ClN3O2
|
1
|
| 1 |
EC50 = 73.5 nM
|
|
|
|
CP0479280
|
3-(3-chlorophenyl)-2-cyclohexyl-10-methylpyrimido[4,5-b]quinoline-4,5-dione
Show/Hide
|
C24H22ClN3O2
|
1
|
| 1 |
EC50 = 80.2 nM
|
|
|
|
CP0479270
|
2-cyclopentyl-10-methyl-3-phenylpyrimido[4,5-b]quinoline-4,5-dione
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|
C23H21N3O2
|
1
|
| 1 |
EC50 = 80.4 nM
|
|
|
|
CP0479276
|
2-cyclopentyl-10-methyl-3H-pyrimido[4,5-b]quinoline-4,5-dione
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|
C17H17N3O2
|
1
|
| 1 |
EC50 = 81.9 nM
|
|
|
|
CP0479277
|
3-(3-chloro-4-methoxyphenyl)-2-(cyclohexylmethyl)-10-methylpyrimido[4,5-b]quinoline-4,5-dione
Show/Hide
|
C26H26ClN3O3
|
1
|
| 1 |
EC50 = 94.4 nM
|
|
|
|
CP0479262
|
3-(3-chlorophenyl)-2-(cyclohexylmethyl)-10-methylpyrimido[4,5-b]quinoline-4,5-dione
Show/Hide
|
C25H24ClN3O2
|
1
|
| 1 |
EC50 = 94.8 nM
|
|
|
|
CP0479289
|
2-cyclopropyl-10-methyl-3-phenylpyrimido[4,5-b]quinoline-4,5-dione
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|
C21H17N3O2
|
1
|
| 1 |
EC50 = 95.1 nM
|
|
|
|
CP0479273
|
10-methyl-2-(2-methylpropyl)-3-phenylpyrimido[4,5-b]quinoline-4,5-dione
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|
C22H21N3O2
|
1
|
| 1 |
EC50 = 103 nM
|
|
|
|
CP0479278
|
2-(cyclohexylmethyl)-10-methyl-3-(4-methylphenyl)pyrimido[4,5-b]quinoline-4,5-dione
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|
C26H27N3O2
|
1
|
| 1 |
EC50 = 168 nM
|
|
|
|
CP0137322
|
1H-indol-2-yl-[4-[2-(4-methoxyphenoxy)ethyl]piperazin-1-yl]methanone
Show/Hide
|
C22H25N3O3
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
