| Compound ID |
Compound Name |
Compound Formula |
|
CP0378207
|
(R)-N-(2-(3-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-3-oxoprop-1-enyl)-5-chloro-4-methoxyphenyl)acetamide
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|
C24H27ClFN3O3
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0448801
|
N-[5-chloro-2-[(E)-3-[3-[(4-fluorophenyl)methyl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-3-oxoprop-1-enyl]-4-methoxyphenyl]acetamide
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|
C25H27ClFN3O3
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0428267
|
N-[5-chloro-2-[(E)-3-[(2R,5S)-4-[(4-fluorophenyl)methyl]-2,5-dimethylpiperazin-1-yl]-3-oxoprop-1-enyl]phenyl]acetamide
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|
C24H27ClFN3O2
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0378206
|
(R)-1-(2-(3-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-3-oxoprop-1-enyl)-5-chlorophenyl)urea
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|
C22H24ClFN4O2
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0050382
|
(R)-N-(2-(3-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-3-oxoprop-1-enyl)-5-chlorophenyl)acetamide
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|
C23H25ClFN3O2
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0378208
|
N-[5-chloro-2-[(E)-3-[3-[(4-fluorophenyl)methyl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-3-oxoprop-1-enyl]phenyl]-2-(dimethylamino)acetamide
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|
C26H30ClFN4O2
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0442404
|
(R)-N-(6-(3-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-3-oxoprop-1-enyl)quinolin-7-yl)acetamide
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|
C26H27FN4O2
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0853916
|
BX 471
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|
C21H25Cl2FN4O3
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0378007
|
(R)-N-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethylamino)-5-chlorophenyl)acetamide
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|
C22H26ClFN4O2
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0428270
|
(R)-N-(3-(3-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-3-oxoprop-1-enyl)naphthalen-2-yl)acetamide
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|
C27H28FN3O2
|
1
|
| 1 |
IC50 = 80 nM
|
|
|
|
CP0392271
|
N-[5-chloro-2-[(E)-3-[(2S,5R)-4-[(4-fluorophenyl)methyl]-2,5-dimethylpiperazin-1-yl]-3-oxoprop-1-enyl]phenyl]acetamide
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|
C24H27ClFN3O2
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0428291
|
(R)-N-(2-(1-(4-fluorobenzyl)-3-methylpiperazine-4-carbonyl)-5-chlorobenzofuran-7-yl)acetamide
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|
C23H23ClFN3O3
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0378011
|
N-[6-[(E)-3-[3-[(4-fluorophenyl)methyl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-3-oxoprop-1-enyl]quinolin-7-yl]acetamide
Show/Hide
|
C27H27FN4O2
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0445798
|
N-[5-chloro-2-[(E)-3-[4-[(4-fluorophenyl)methyl]piperazin-1-yl]-3-oxoprop-1-enyl]phenyl]acetamide
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|
C22H23ClFN3O2
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0448800
|
N-[5-chloro-2-[(E)-3-[3-[(4-fluorophenyl)methyl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-3-oxoprop-1-enyl]phenyl]acetamide
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|
C24H25ClFN3O2
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0455658
|
N-[5-chloro-2-[(E)-3-[8-[(4-fluorophenyl)methyl]-3,8-diazabicyclo[3.2.1]octan-3-yl]-3-oxoprop-1-enyl]phenyl]acetamide
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|
C24H25ClFN3O2
|
1
|
| 1 |
IC50 = 300 nM
|
|
|
|
CP0378006
|
(R)-N-(2-(3-(4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-3-oxopropyl)-5-chlorophenyl)acetamide
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|
C23H27ClFN3O2
|
1
|
| 1 |
IC50 = 360 nM
|
|
|
|
CP0378209
|
(R)-N-(2-(1-(4-fluorobenzyl)-3-methylpiperazine-4-carbonyl)-5-chloro-1H-indol-7-yl)acetamide
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|
C23H24ClFN4O2
|
1
|
| 1 |
IC50 = 560 nM
|
|
|
|
CP0378008
|
4-(2-((R)-4-(4-fluorobenzyl)-2-methylpiperazin-1-yl)-2-oxoethyl)-7-chloro-6-methoxy-3,4-dihydroquinazolin-2(1H)-one
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|
C23H26ClFN4O3
|
1
|
| 1 |
IC50 = 800 nM
|
|
|
|
CP0378222
|
(R)-N-(2-(3-(4-(4-fluorobenzyl)-2-methyl-1,4-diazepan-1-yl)-3-oxoprop-1-enyl)-5-chlorophenyl)acetamide
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|
C24H27ClFN3O2
|
1
|
| 1 |
IC50 = 1600 nM
|
|
|
|
CP0428268
|
N-[5-chloro-2-[(E)-3-[(1R,4R)-5-[(4-fluorophenyl)methyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]-3-oxoprop-1-enyl]phenyl]acetamide
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|
C23H23ClFN3O2
|
1
|
| 1 |
IC50 = 1700 nM
|
|
|
