| Compound ID |
Compound Name |
Compound Formula |
|
CP0539985
|
US10300060, Example 15-96
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|
C24H18F4N6O4S
|
1
|
| 1 |
IC50 = 0.4 nM
|
|
|
|
CP0490938
|
US10300060, Example 15-104
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|
C24H18ClF3N6O4S
|
1
|
| 1 |
IC50 = 0.5 nM
|
|
|
|
CP0536138
|
US10300060, Example 21-65
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|
C30H21F3N8O2
|
1
|
| 1 |
IC50 = 0.7 nM
|
|
|
|
CP0493160
|
US10300060, Example 15-98
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|
C25H18F6N6O4S
|
1
|
| 1 |
IC50 = 0.8 nM
|
|
|
|
CP0409416
|
US9242977, 85-226
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|
C25H23F3N6O4S2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0404975
|
US10300060, Example 21-1
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|
C32H24F3N9O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0404976
|
US10300060, Example 22-34
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|
C31H23F3N8O3
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0406935
|
US10300060, Example 9-2
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|
C26H18ClF3N8O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0406936
|
US10300060, Example 15-4
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|
C26H18ClF3N8O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0445193
|
US10300060, Example 21-37
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|
C31H24F3N9O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0451937
|
US10300060, Example 8-4
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|
C23H15Cl2F3N6O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0477830
|
US10300060, Example 11
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|
C29H20ClF3N6O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0477831
|
US10300060, Example 14-5
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|
C25H17F4N9O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0484449
|
US10300060, Example 21-2
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|
C31H25F3N10O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0491135
|
US10300060, Example 23-12
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|
C29H19F3N8O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0500950
|
US10300060, Example 14-6
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|
C28H19F4N7O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0512369
|
US10300060, Example 21-9
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|
C30H21F3N8O3
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0517479
|
US10300060, Example 15-87
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|
C27H17ClF6N8O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0526120
|
US10300060, Example 8-1
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|
C26H19ClF3N9O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0539986
|
US10300060, Example 21-13
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|
C29H19F3N8O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0567650
|
US10300060, Example 21-51
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|
C30H25F3N10O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0569378
|
US10300060, Example 23-11
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|
C30H20F3N7O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0569410
|
US10300060, Example 23-3
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|
C28H19F3N8O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0575850
|
US10300060, Example 23-10
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|
C29H19F3N8O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0576941
|
US10300060, Example 22-8
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|
C30H21F3N8O3
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0576942
|
US10300060, Example 22-9
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|
C28H20F3N9O3
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0577338
|
US10300060, Example 7
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|
C26H18ClF3N8O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0129156
|
US9242977, 85-117
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|
C24H20ClF3N6O2S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0323802
|
US9242977, 65-1
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|
C33H34N8O3S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0409415
|
US9242977, 85-184
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|
C28H22F6N8O2S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0414641
|
US9242977, 71
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|
C33H32N10O3S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0419634
|
US10300060, Example 21-70
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|
C32H25F3N8O2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0419639
|
US10300060, Example 15-71
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|
C26H17Cl2F3N8O2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0445195
|
US10300060, Example 23-7
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|
C30H20F3N7O2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0469617
|
US10300060, Example 13-1
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|
C27H20ClF3N8O2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0512368
|
US10300060, Example 15-6
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|
C23H15Cl2F3N6O2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0517478
|
US10300060, Example 15-77
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|
C24H15ClF6N6O2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0565477
|
US10300060, Example 15-63
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|
C26H17Cl2F3N8O2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0567649
|
US10300060, Example 15-58
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|
C29H20F4N6O2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0570747
|
US10300060, Example 8-2
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|
C27H17ClF6N8O2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0251769
|
US9242977, 57
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|
C31H24F3N7O3S
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0469616
|
US10300060, Example 9-1
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|
C27H19ClF3N7O2
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0507884
|
US10300060, Example 15-5
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|
C23H15ClF4N6O2
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0578207
|
US10300060, Example 21-73
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|
C33H27F3N8O2
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0264758
|
US9242977, 54
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|
C30H22F3N7O3S
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0302038
|
US9242977, 66-19
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|
C33H32N8O4S
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0326832
|
US9242977, 23
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|
C29H24F3N7O2S
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0414646
|
US9242977, 85-209
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|
C23H20F2N6O2S
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0507782
|
US9242977, 85-225
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|
C26H26F3N7O4S2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0419632
|
US10300060, Example 21-67
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|
C33H27F3N8O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0517477
|
US10300060, Example 15-55
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|
C29H20ClF3N6O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0517480
|
US10300060, Example 15-105
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|
C26H21F6N7O4S
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0565476
|
US10300060, Example 15-52
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|
C28H17F9N8O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0578208
|
US10300060, Example 21-75
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|
C33H27F3N8O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0107004
|
US9242977, 34
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|
C31H27F3N6O2S
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0251770
|
US9242977, 66-27
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|
C33H32N8O5S
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0319106
|
US9242977, 48
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|
C28H22F3N7O3S
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0302039
|
US9242977, 72-1
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|
C29H23F3N8O3S
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0319107
|
US9242977, 50
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|
C30H20F6N8O3S
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0117061
|
US9242977, 66-28
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|
C33H33N9O4S
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0227337
|
US9242977, 72-3
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|
C30H26F2N8O3S
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0228183
|
US9242977, 66-72
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|
C31H31N9O5S2
|
1
|
| 1 |
IC50 = 32 nM
|
|
|
|
CP0515510
|
US9242977, 72-7
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|
C30H26N8O3S
|
1
|
| 1 |
IC50 = 33 nM
|
|
|
|
CP0319108
|
US9242977, 59
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|
C34H30F3N7O3S
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0562354
|
US9242977, 9
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|
C31H22F6N8O3S
|
1
|
| 1 |
IC50 = 93 nM
|
|
|
