| Compound ID |
Compound Name |
Compound Formula |
|
CP0494228
|
5-(2,6-dimethoxyphenyl)-6-(ethoxymethyl)-4-hydroxy-3-[5-[(5-methylpyridin-2-yl)methyl]-1,3,4-oxadiazol-2-yl]-1H-pyridin-2-one
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|
C25H26N4O6
|
1
|
| 1 |
EC50 = 0.024 nM
|
|
|
|
CP0494226
|
2-butyl-5-[(3R)-3-(5-chloropyridin-2-yl)pyrrolidine-1-carbonyl]-3-(2,6-dimethoxyphenyl)-6-hydroxypyrimidin-4-one
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|
C26H29ClN4O5
|
1
|
| 1 |
EC50 = 0.035 nM
|
|
|
|
CP0546421
|
2-butyl-5-[(3S)-3-(5-chloropyridin-2-yl)pyrrolidine-1-carbonyl]-3-(2,6-dimethoxyphenyl)-6-hydroxypyrimidin-4-one
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|
C26H29ClN4O5
|
1
|
| 1 |
EC50 = 0.063 nM
|
|
|
|
CP0235875
|
(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-1-[2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-1-[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-5-oxopyrrolidine-2-carbonyl]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]pentanoyl]amino]-4-methylpentanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]hexanoyl]amino]acetyl]pyrrolidine-2-carbonyl]amino]-4-methylsulfanylbutanoyl]pyrrolidine-2-carbonyl]amino]-3-phenylpropanoic acid
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|
C69H108N22O16S
|
1
|
| 1 |
EC50 = 0.07 nM
|
|
|
|
CP0487481
|
2-butyl-3-(2,6-dimethoxyphenyl)-6-hydroxy-5-[(3R)-3-phenylpyrrolidine-1-carbonyl]pyrimidin-4-one
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|
C27H31N3O5
|
1
|
| 1 |
EC50 = 0.27 nM
|
|
|
|
CP0546419
|
2-butyl-3-(2,6-dimethoxyphenyl)-6-hydroxy-5-[(3S)-3-phenylpyrrolidine-1-carbonyl]pyrimidin-4-one
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|
C27H31N3O5
|
1
|
| 1 |
EC50 = 0.34 nM
|
|
|
|
CP0555754
|
3-(2,6-dimethoxyphenyl)-2-(ethoxymethyl)-6-hydroxy-5-[(3R)-3-phenylpyrrolidine-1-carbonyl]pyrimidin-4-one
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|
C26H29N3O6
|
1
|
| 1 |
EC50 = 0.61 nM
|
|
|
|
CP0959379
|
(R)-6-butyl-5-(2,6-dimethoxyphenyl)-4-hydroxy-3-(3-phenylpyrrolidine-1-carbonyl)pyridin-2(1H)-one
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|
C28H32N2O5
|
1
|
| 1 |
EC50 = 1.8 nM
|
|
|
|
CP0953669
|
(S)-6-butyl-5-(2,6-dimethoxyphenyl)-4-hydroxy-3-(3-phenylpyrrolidine-1-carbonyl)pyridin-2(1H)-one
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|
C28H32N2O5
|
1
|
| 1 |
EC50 = 3.1 nM
|
|
|
|
CP0546418
|
6-butyl-N-[2-(4-chlorophenyl)ethyl]-5-(2,6-dimethoxyphenyl)-4-hydroxy-N-methyl-2-oxo-1H-pyridine-3-carboxamide
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|
C27H31ClN2O5
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0558216
|
N-benzyl-6-butyl-5-(2,6-dimethoxyphenyl)-4-hydroxy-2-oxo-N-propyl-1H-pyridine-3-carboxamide
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|
C28H34N2O5
|
1
|
| 1 |
EC50 = 150 nM
|
|
|
|
CP0487480
|
6-butyl-5-(2,6-dimethoxyphenyl)-4-hydroxy-N,N-dimethyl-2-oxo-1H-pyridine-3-carboxamide
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|
C20H26N2O5
|
1
|
| 1 |
EC50 = 1200 nM
|
|
|
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CP0559788
|
N-benzyl-6-butyl-5-(2,6-dimethoxyphenyl)-4-hydroxy-2-oxo-1H-pyridine-3-carboxamide
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|
C25H28N2O5
|
1
|
| 1 |
EC50 = 4800 nM
|
|
|
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CP0565378
|
6-butyl-5-(2,6-dimethoxyphenyl)-N-ethyl-4-hydroxy-2-oxo-1H-pyridine-3-carboxamide
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|
C20H26N2O5
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
