| Compound ID |
Compound Name |
Compound Formula |
|
CP0076890
|
(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide
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|
C18H17ClN6O4S
|
1
|
| 1 |
Ki = 1.55 nM
|
|
|
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CP0393494
|
methyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate
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|
C20H18ClN5O4S
|
1
|
| 1 |
Ki = 5.38 nM
|
|
|
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CP0393511
|
propyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate
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|
C22H22ClN5O4S
|
1
|
| 1 |
Ki = 5.78 nM
|
|
|
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CP0076892
|
(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide
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|
C20H21ClN6O4S
|
1
|
| 1 |
Ki = 6.25 nM
|
|
|
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CP0393809
|
ethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate
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|
C21H20BrN5O4S
|
1
|
| 1 |
Ki = 6.42 nM
|
|
|
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CP0393808
|
benzyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate
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|
C26H22ClN5O4S
|
1
|
| 1 |
Ki = 7.31 nM
|
|
|
|
CP0126419
|
methyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate
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|
C20H18BrN5O4S
|
1
|
| 1 |
Ki = 8.56 nM
|
|
|
|
CP0393806
|
(1S,2R,3S,4R,5S)-4-[6-[2-(5-chlorothiophen-2-yl)ethynyl]-4-(methylamino)imidazo[4,5-c]pyridin-1-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide
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|
C21H20ClN5O3S
|
1
|
| 1 |
Ki = 9.33 nM
|
|
|
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CP0076893
|
methyl (2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate
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|
C18H16ClN5O5S
|
1
|
| 1 |
Ki = 11.5 nM
|
|
|
|
CP0405283
|
ethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate
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|
C21H20ClN5O4S
|
1
|
| 1 |
Ki = 14.5 nM
|
|
|
|
CP0391668
|
butyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate
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|
C23H24ClN5O4S
|
1
|
| 1 |
Ki = 17.5 nM
|
|
|
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CP0393807
|
3-methylbutyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate
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|
C24H26ClN5O4S
|
1
|
| 1 |
Ki = 24.4 nM
|
|
|
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CP0463333
|
propan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate
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|
C22H22ClN5O4S
|
1
|
| 1 |
Ki = 42.9 nM
|
|
|
|
CP0416965
|
(1S,2R,3S,4R,5S)-N-(2-aminoethyl)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxamide
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|
C21H22ClN7O3S
|
1
|
| 1 |
Ki = 156 nM
|
|
|
|
CP0103702
|
ethyl (1S,2R,3S,4R,5S)-4-[6-[2-(5-chlorothiophen-2-yl)ethynyl]-4-(methylamino)imidazo[4,5-c]pyridin-1-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate
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|
C22H21ClN4O4S
|
1
|
| 1 |
Ki = 169 nM
|
|
|
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CP0393810
|
3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate
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|
C28H26ClN5O4S
|
1
|
| 1 |
Ki = 255 nM
|
|
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CP0463334
|
2-phenylethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate
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|
C27H24ClN5O4S
|
1
|
| 1 |
Ki = 262 nM
|
|
|
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CP0393805
|
(1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid
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|
C19H16ClN5O4S
|
1
|
| 1 |
Ki = 684 nM
|
|
|
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CP0455571
|
2-cyclohexylethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate
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|
C27H30ClN5O4S
|
1
|
| 1 |
Ki = 770 nM
|
|
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