| Compound ID |
Compound Name |
Compound Formula |
|
CP0494228
|
5-(2,6-dimethoxyphenyl)-6-(ethoxymethyl)-4-hydroxy-3-[5-[(5-methylpyridin-2-yl)methyl]-1,3,4-oxadiazol-2-yl]-1H-pyridin-2-one
Show/Hide
|
C25H26N4O6
|
1
|
| 1 |
EC50 = 0.023 nM
|
|
|
|
CP0494226
|
2-butyl-5-[(3R)-3-(5-chloropyridin-2-yl)pyrrolidine-1-carbonyl]-3-(2,6-dimethoxyphenyl)-6-hydroxypyrimidin-4-one
Show/Hide
|
C26H29ClN4O5
|
1
|
| 1 |
EC50 = 0.027 nM
|
|
|
|
CP0546421
|
2-butyl-5-[(3S)-3-(5-chloropyridin-2-yl)pyrrolidine-1-carbonyl]-3-(2,6-dimethoxyphenyl)-6-hydroxypyrimidin-4-one
Show/Hide
|
C26H29ClN4O5
|
1
|
| 1 |
EC50 = 0.032 nM
|
|
|
|
CP0235875
|
(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-1-[2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-1-[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-5-oxopyrrolidine-2-carbonyl]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]pentanoyl]amino]-4-methylpentanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]hexanoyl]amino]acetyl]pyrrolidine-2-carbonyl]amino]-4-methylsulfanylbutanoyl]pyrrolidine-2-carbonyl]amino]-3-phenylpropanoic acid
Show/Hide
|
C69H108N22O16S
|
2
|
| 1 |
EC50 = 0.05 nM
|
|
|
| 2 |
EC50 = 54 nM
|
|
|
|
CP0487481
|
2-butyl-3-(2,6-dimethoxyphenyl)-6-hydroxy-5-[(3R)-3-phenylpyrrolidine-1-carbonyl]pyrimidin-4-one
Show/Hide
|
C27H31N3O5
|
1
|
| 1 |
EC50 = 0.22 nM
|
|
|
|
CP0487479
|
(2S,3R)-N-(4-(2,6-dimethoxyphenyl)-5-(5-methyl-3-pyridinyl)-4H-1,2,4-triazol-3-yl)-3-(5-methyl-2-pyrazinyl)-2-butanesulfonamide
Show/Hide
|
C25H29N7O4S
|
1
|
| 1 |
EC50 = 0.23 nM
|
|
|
|
CP0546419
|
2-butyl-3-(2,6-dimethoxyphenyl)-6-hydroxy-5-[(3S)-3-phenylpyrrolidine-1-carbonyl]pyrimidin-4-one
Show/Hide
|
C27H31N3O5
|
1
|
| 1 |
EC50 = 0.26 nM
|
|
|
|
CP0555754
|
3-(2,6-dimethoxyphenyl)-2-(ethoxymethyl)-6-hydroxy-5-[(3R)-3-phenylpyrrolidine-1-carbonyl]pyrimidin-4-one
Show/Hide
|
C26H29N3O6
|
1
|
| 1 |
EC50 = 0.44 nM
|
|
|
|
CP0955645
|
(R)-2-((S)-1-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanoyl)pyrrolidine-2-carboxamido)-3-(4-(benzyloxy)phenyl)propanoic acid
Show/Hide
|
C77H116N22O17
|
2
|
| 1 |
EC50 = 0.5 nM
|
|
|
| 2 |
EC50 = 11 nM
|
|
|
|
CP0902553
|
(R)-2-((S)-1-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanoyl)pyrrolidine-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
Show/Hide
|
C71H110N22O16
|
2
|
| 1 |
EC50 = 1 nM
|
|
|
| 2 |
EC50 = 23 nM
|
|
|
|
CP0902559
|
(2S,3R)-2-((S)-1-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanoyl)pyrrolidine-2-carboxamido)-3-phenylbutanoic acid
Show/Hide
|
C71H112N22O16
|
2
|
| 1 |
EC50 = 1 nM
|
|
|
| 2 |
EC50 = 108 nM
|
|
|
|
CP0959379
|
(R)-6-butyl-5-(2,6-dimethoxyphenyl)-4-hydroxy-3-(3-phenylpyrrolidine-1-carbonyl)pyridin-2(1H)-one
Show/Hide
|
C28H32N2O5
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0153773
|
(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-1-[2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-1-[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-2,5-diamino-5-oxopentanoyl]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]pentanoyl]amino]-4-methylpentanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]hexanoyl]amino]acetyl]pyrrolidine-2-carbonyl]amino]-4-methylsulfanylbutanoyl]pyrrolidine-2-carbonyl]amino]-3-phenylpropanoic acid
Show/Hide
|
C69H111N23O16S
|
2
|
| 1 |
EC50 = 1.1 nM
|
|
|
| 2 |
EC50 = 43 nM
|
|
|
|
CP0910681
|
(R)-2-((S)-1-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanoyl)pyrrolidine-2-carboxamido)-3-(biphenyl-3-yl)propanoic acid
Show/Hide
|
C76H114N22O16
|
2
|
| 1 |
EC50 = 1.4 nM
|
|
|
| 2 |
EC50 = 24 nM
|
|
|
|
CP0902547
|
2-((S)-1-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanoyl)pyrrolidine-2-carboxamido)-2-benzyl-3-phenylpropanoic acid
Show/Hide
|
C77H116N22O16
|
2
|
| 1 |
EC50 = 1.5 nM
|
|
|
| 2 |
EC50 = 10 nM
|
|
|
|
CP0902551
|
(R)-2-((R)-2-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanamido)-3-(naphthalen-1-yl)propanoyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
Show/Hide
|
C79H114N22O16
|
2
|
| 1 |
EC50 = 1.6 nM
|
|
|
| 2 |
EC50 = 15 nM
|
|
|
|
CP0953669
|
(S)-6-butyl-5-(2,6-dimethoxyphenyl)-4-hydroxy-3-(3-phenylpyrrolidine-1-carbonyl)pyridin-2(1H)-one
Show/Hide
|
C28H32N2O5
|
1
|
| 1 |
EC50 = 1.8 nM
|
|
|
|
CP0943092
|
(R)-2-((S)-1-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanoyl)pyrrolidine-2-carboxamido)-3-(biphenyl-4-yl)propanoic acid
Show/Hide
|
C76H114N22O16
|
2
|
| 1 |
EC50 = 2.1 nM
|
|
|
| 2 |
EC50 = 21 nM
|
|
|
|
CP0955646
|
(S)-2-((S)-1-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanoyl)pyrrolidine-2-carboxamido)-3-methyl-3-phenylbutanoic acid
Show/Hide
|
C72H114N22O16
|
2
|
| 1 |
EC50 = 2.4 nM
|
|
|
| 2 |
EC50 = 67 nM
|
|
|
|
CP0765197
|
(R)-2-((S)-4-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanamido)-3-oxo-4,5-dihydroazepino[3,4-b]indol-2(1H,3H,10H)-yl)-3-phenylpropanoic acid
Show/Hide
|
C77H113N23O16
|
2
|
| 1 |
EC50 = 2.5 nM
|
|
|
| 2 |
EC50 = 11 nM
|
|
|
|
CP0943236
|
(S)-2-((S)-1-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanoyl)pyrrolidine-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
Show/Hide
|
C71H110N22O16
|
2
|
| 1 |
EC50 = 2.5 nM
|
|
|
| 2 |
EC50 = 88 nM
|
|
|
|
CP0910683
|
(R)-2-((S)-1-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanoyl)pyrrolidine-2-carboxamido)-3-(4-(benzyloxy)phenyl)-2-methylpropanoic acid
Show/Hide
|
C78H118N22O17
|
2
|
| 1 |
EC50 = 2.7 nM
|
|
|
| 2 |
EC50 = 4.4 nM
|
|
|
|
CP0902560
|
2-((R)-2-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanamido)-3-(naphthalen-1-yl)propanamido)-2-benzyl-3-phenylpropanoic acid
Show/Hide
|
C85H120N22O16
|
2
|
| 1 |
EC50 = 2.8 nM
|
|
|
| 2 |
EC50 = 3.8 nM
|
|
|
|
CP0915429
|
(R)-2-((S)-1-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanoyl)pyrrolidine-2-carbonyl)-7-(benzyloxy)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
Show/Hide
|
C78H116N22O17
|
2
|
| 1 |
EC50 = 3.4 nM
|
|
|
| 2 |
EC50 = 22 nM
|
|
|
|
CP0902550
|
(S)-2-((R)-2-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanamido)-3-(1H-indol-3-yl)propanamido)-3-phenylpropanoic acid
Show/Hide
|
C76H113N23O16
|
2
|
| 1 |
EC50 = 3.8 nM
|
|
|
| 2 |
EC50 = 17 nM
|
|
|
|
CP0902555
|
(R)-2-((S)-1-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanoyl)pyrrolidine-2-carboxamido)-3-(3-(benzyloxy)phenyl)propanoic acid
Show/Hide
|
C77H116N22O17
|
2
|
| 1 |
EC50 = 3.8 nM
|
|
|
| 2 |
EC50 = 45 nM
|
|
|
|
CP0902552
|
2-((R)-2-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanamido)-3-(naphthalen-1-yl)propanoyl)-4,4-dimethyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
Show/Hide
|
C81H118N22O16
|
2
|
| 1 |
EC50 = 4.1 nM
|
|
|
| 2 |
EC50 = 10 nM
|
|
|
|
CP0954798
|
(S)-2-((R)-2-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanamido)-3-(naphthalen-1-yl)propanoyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
Show/Hide
|
C79H114N22O16
|
2
|
| 1 |
EC50 = 4.2 nM
|
|
|
| 2 |
EC50 = 28 nM
|
|
|
|
CP0910682
|
2-((R)-2-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanamido)-3-(naphthalen-1-yl)propanoyl)-4-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
Show/Hide
|
C80H116N22O16
|
2
|
| 1 |
EC50 = 4.3 nM
|
|
|
| 2 |
EC50 = 111 nM
|
|
|
|
CP0943072
|
(R)-2-((R)-2-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanamido)-3-(naphthalen-2-yl)propanoyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
Show/Hide
|
C79H114N22O16
|
1
|
| 1 |
EC50 = 4.3 nM
|
|
|
|
CP0910677
|
(S)-2-((R)-2-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanamido)-3-(naphthalen-1-yl)propanamido)-3-phenylpropanoic acid
Show/Hide
|
C78H114N22O16
|
2
|
| 1 |
EC50 = 4.4 nM
|
|
|
| 2 |
EC50 = 9.2 nM
|
|
|
|
CP0915430
|
(S)-2-((2R,4S)-1-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanoyl)-4-(benzyloxy)pyrrolidine-2-carboxamido)-3-phenylpropanoic acid
Show/Hide
|
C77H116N22O17
|
2
|
| 1 |
EC50 = 5.6 nM
|
|
|
| 2 |
EC50 = 54 nM
|
|
|
|
CP0902549
|
(R)-2-((S)-1-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanoyl)pyrrolidine-2-carboxamido)-3-(4-(benzyloxy)-3-cyclopentylphenyl)propanoic acid
Show/Hide
|
C82H124N22O17
|
2
|
| 1 |
EC50 = 5.7 nM
|
|
|
| 2 |
EC50 = 53 nM
|
|
|
|
CP0902557
|
(R)-2-((R)-2-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanamido)-3-(naphthalen-1-yl)propanoyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid
Show/Hide
|
C81H115N23O16
|
2
|
| 1 |
EC50 = 6 nM
|
|
|
| 2 |
EC50 = 25 nM
|
|
|
|
CP0902558
|
2-((S)-4-((S)-1-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanoyl)pyrrolidine-2-carboxamido)-3-oxo-4,5-dihydroazepino[3,4-b]indol-2(1H,3H,10H)-yl)acetic acid
Show/Hide
|
C77H115N23O17
|
2
|
| 1 |
EC50 = 6.4 nM
|
|
|
| 2 |
EC50 = 74 nM
|
|
|
|
CP0910679
|
(2R,4S)-1-((S)-1-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanoyl)pyrrolidine-2-carbonyl)-4-(benzyloxy)pyrrolidine-2-carboxylic acid
Show/Hide
|
C73H114N22O17
|
2
|
| 1 |
EC50 = 6.4 nM
|
|
|
| 2 |
EC50 = 63 nM
|
|
|
|
CP0910678
|
2-((S)-4-((S)-1-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanoyl)pyrrolidine-2-carboxamido)-3-oxo-4,5-dihydro-1H-naphtho[2,3-c]azepin-2(3H)-yl)acetic acid
Show/Hide
|
C75H114N24O17
|
2
|
| 1 |
EC50 = 6.8 nM
|
|
|
| 2 |
EC50 = 481 nM
|
|
|
|
CP0902548
|
(R)-2-((S)-1-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanoyl)pyrrolidine-2-carboxamido)-3-(biphenyl-2-yl)propanoic acid
Show/Hide
|
C76H114N22O16
|
2
|
| 1 |
EC50 = 8.6 nM
|
|
|
| 2 |
EC50 = 142 nM
|
|
|
|
CP0546418
|
6-butyl-N-[2-(4-chlorophenyl)ethyl]-5-(2,6-dimethoxyphenyl)-4-hydroxy-N-methyl-2-oxo-1H-pyridine-3-carboxamide
Show/Hide
|
C27H31ClN2O5
|
1
|
| 1 |
EC50 = 9.3 nM
|
|
|
|
CP0943091
|
(S)-2-((R)-2-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanoyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamido)-3-phenylpropanoic acid
Show/Hide
|
C75H112N22O16
|
2
|
| 1 |
EC50 = 9.6 nM
|
|
|
| 2 |
EC50 = 67 nM
|
|
|
|
CP0910680
|
(R)-2-((R)-2-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanamido)-3-(naphthalen-1-yl)propanamido)-3-(3,5-dicyclopentyl-4-hydroxyphenyl)propanoic acid
Show/Hide
|
C88H130N22O17
|
2
|
| 1 |
EC50 = 10 nM
|
|
|
| 2 |
EC50 = 178 nM
|
|
|
|
CP0943237
|
(S)-2-((S)-1-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanoyl)pyrrolidine-2-carboxamido)-3-(4-(benzyloxy)phenyl)-2-methylpropanoic acid
Show/Hide
|
C78H118N22O17
|
2
|
| 1 |
EC50 = 11 nM
|
|
|
| 2 |
EC50 = 19 nM
|
|
|
|
CP0902554
|
(R)-2-((S)-1-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanoyl)pyrrolidine-2-carboxamido)-3-(3,5-dicyclopentyl-4-hydroxyphenyl)propanoic acid
Show/Hide
|
C80H126N22O17
|
2
|
| 1 |
EC50 = 16 nM
|
|
|
| 2 |
EC50 = 111 nM
|
|
|
|
CP0902556
|
(S)-2-((2R,3R)-1-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanoyl)-3-phenylpyrrolidine-2-carboxamido)-3-phenylpropanoic acid
Show/Hide
|
C76H114N22O16
|
2
|
| 1 |
EC50 = 17 nM
|
|
|
| 2 |
EC50 = 48 nM
|
|
|
|
CP0902561
|
(R)-2-((S)-1-((S)-2-((S)-1-((6S,9S,12S,15S,18S)-15-((1H-imidazol-5-yl)methyl)-1-amino-18-(4-aminobutyl)-6-((S)-1-((S)-5-guanidino-2-((S)-5-oxopyrrolidine-2-carboxamido)pentanoyl)pyrrolidine-2-carboxamido)-12-(hydroxymethyl)-1-imino-9-isobutyl-7,10,13,16,19-pentaoxo-2,8,11,14,17,20-hexaazadocosane)pyrrolidine-2-carboxamido)hexanoyl)pyrrolidine-2-carboxamido)-3-(4-(benzyloxy)-3,5-dicyclopentylphenyl)propanoic acid
Show/Hide
|
C87H132N22O17
|
2
|
| 1 |
EC50 = 22 nM
|
|
|
| 2 |
EC50 = 141 nM
|
|
|
|
CP0953634
|
ELABELA
Show/Hide
|
C167H279N59O39S4
|
1
|
| 1 |
EC50 = 25 nM
|
|
|
|
CP0955254
|
(S)-2-((S)-2-((S)-1-((3S,6S,9S,12S,15S)-6-((1H-imidazol-5-yl)methyl)-1-((S)-1-((S)-2-aminohexanoyl)pyrrolidin-2-yl)-12-(3-guanidinopropyl)-9-(hydroxymethyl)-3-isobutyl-15-isopropyl-1,4,7,10,13-pentaoxo-2,5,8,11,14-pentaazahexadecane)pyrrolidine-2-carboxamido)-3-phenylpropanamido)-3-(naphthalen-1-yl)propanoic acid
Show/Hide
|
C64H91N15O12
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
|
CP0871209
|
(S)-2-((S)-2-((S)-1-((3S,6S,9S,12S,15S)-6-((1H-imidazol-5-yl)methyl)-1-((S)-1-((S)-2-aminohexanoyl)pyrrolidin-2-yl)-12-(3-guanidinopropyl)-9-(hydroxymethyl)-3-isobutyl-15-isopropyl-1,4,7,10,13-pentaoxo-2,5,8,11,14-pentaazahexadecane)pyrrolidine-2-carboxamido)-3-phenylpropanamido)-3-(naphthalen-2-yl)propanoic acid
Show/Hide
|
C64H91N15O12
|
1
|
| 1 |
EC50 = 37 nM
|
|
|
|
CP0955253
|
(S)-2-((S)-2-((S)-1-((3S,6S,9S,12S,15S)-6-((1H-imidazol-5-yl)methyl)-1-((S)-1-((S)-2-aminohexanoyl)pyrrolidin-2-yl)-12-(3-guanidinopropyl)-9-(hydroxymethyl)-3-isobutyl-15-isopropyl-1,4,7,10,13-pentaoxo-2,5,8,11,14-pentaazahexadecane)pyrrolidine-2-carboxamido)-3-phenylpropanamido)-3-phenylpropanoic acid
Show/Hide
|
C60H89N15O12
|
1
|
| 1 |
EC50 = 43 nM
|
|
|
|
CP0922756
|
(S)-1-((S)-2-((S)-1-((3S,6S,9S,12S,15S)-6-((1H-imidazol-5-yl)methyl)-1-((S)-1-((S)-2-aminohexanoyl)pyrrolidin-2-yl)-12-(3-guanidinopropyl)-9-(hydroxymethyl)-3-isobutyl-15-isopropyl-1,4,7,10,13-pentaoxo-2,5,8,11,14-pentaazahexadecane)pyrrolidine-2-carboxamido)-3-cyclohexylpropanoyl)pyrrolidine-2-carboxylic acid
Show/Hide
|
C56H93N15O12
|
1
|
| 1 |
EC50 = 54 nM
|
|
|
|
CP0944660
|
(S)-1-((S)-2-((S)-1-((3S,6S,9S,12S)-3-((1H-imidazol-5-yl)methyl)-1-(1-((S)-1-((S)-2-aminohexanoyl)pyrrolidine-2-carboxamido)cyclopentyl)-9-(3-guanidinopropyl)-6-(hydroxymethyl)-12-isopropyl-1,4,7,10-tetraoxo-2,5,8,11-tetraazatridecane)pyrrolidine-2-carboxamido)-3-phenylpropanoyl)pyrrolidine-2-carboxylic acid
Show/Hide
|
C56H85N15O12
|
1
|
| 1 |
EC50 = 70 nM
|
|
|
|
CP0953641
|
(S)-1-((S)-2-((S)-1-((3S,6S,9S,12S,15S)-6-((1H-imidazol-5-yl)methyl)-1-((S)-1-((S)-2-aminohexanoyl)pyrrolidin-2-yl)-12-(3-guanidinopropyl)-9-(hydroxymethyl)-3-isobutyl-15-isopropyl-3-methyl-1,4,7,10,13-pentaoxo-2,5,8,11,14-pentaazahexadecane)pyrrolidine-2-carboxamido)-3-phenylpropanoyl)pyrrolidine-2-carboxylic acid
Show/Hide
|
C57H89N15O12
|
1
|
| 1 |
EC50 = 74 nM
|
|
|
|
CP0953645
|
(S)-1-((S)-2-((S)-1-((3S,6S,9S,12S,15S)-6-((1H-imidazol-5-yl)methyl)-1-((S)-1-((S)-2-aminohexanoyl)pyrrolidin-2-yl)-3-(cyclohexylmethyl)-12-(3-guanidinopropyl)-9-(hydroxymethyl)-15-isopropyl-1,4,7,10,13-pentaoxo-2,5,8,11,14-pentaazahexadecane)pyrrolidine-2-carboxamido)-3-phenylpropanoyl)pyrrolidine-2-carboxylic acid
Show/Hide
|
C59H91N15O12
|
1
|
| 1 |
EC50 = 94 nM
|
|
|
|
CP0558216
|
N-benzyl-6-butyl-5-(2,6-dimethoxyphenyl)-4-hydroxy-2-oxo-N-propyl-1H-pyridine-3-carboxamide
Show/Hide
|
C28H34N2O5
|
1
|
| 1 |
EC50 = 120 nM
|
|
|
|
CP0957904
|
(S)-1-((S)-2-((S)-1-((3S,6S,9S,12S,15S)-6-((1H-imidazol-5-yl)methyl)-1-((S)-1-((S)-2-aminohexanoyl)pyrrolidin-2-yl)-12-(3-guanidinopropyl)-9-(hydroxymethyl)-3-isobutyl-15-isopropyl-1,4,7,10,13-pentaoxo-2,5,8,11,14-pentaazahexadecane)pyrrolidine-2-carboxamido)-4-phenylbutanoyl)pyrrolidine-2-carboxylic acid
Show/Hide
|
C57H89N15O12
|
1
|
| 1 |
EC50 = 128 nM
|
|
|
|
CP0922755
|
(S)-1-((S)-2-((S)-1-((3S,6S,9S,12S,15S)-6-((1H-imidazol-5-yl)methyl)-1-((S)-1-((S)-2-aminohexanoyl)pyrrolidin-2-yl)-3-sec-butyl-12-(3-guanidinopropyl)-9-(hydroxymethyl)-15-isopropyl-1,4,7,10,13-pentaoxo-2,5,8,11,14-pentaazahexadecane)pyrrolidine-2-carboxamido)-3-phenylpropanoyl)pyrrolidine-2-carboxylic acid
Show/Hide
|
C56H87N15O12
|
1
|
| 1 |
EC50 = 141 nM
|
|
|
|
CP0871172
|
(S)-1-((S)-2-((S)-1-((3S,6S,9S,12S,15S)-6-((1H-imidazol-5-yl)methyl)-1-((S)-1-((S)-2-aminohexanoyl)pyrrolidin-2-yl)-12-(3-guanidinopropyl)-9-(hydroxymethyl)-3-isobutyl-15-isopropyl-1,4,7,10,13-pentaoxo-2,5,8,11,14-pentaazahexadecane)pyrrolidine-2-carboxamido)-3-(naphthalen-2-yl)propanoyl)pyrrolidine-2-carboxylic acid
Show/Hide
|
C60H89N15O12
|
1
|
| 1 |
EC50 = 152 nM
|
|
|
|
CP0953642
|
(R)-4-((S)-1-((3S,6S,9S,12S,15S)-6-((1H-imidazol-5-yl)methyl)-1-((S)-1-((S)-2-aminohexanoyl)pyrrolidin-2-yl)-12-(3-guanidinopropyl)-9-(hydroxymethyl)-3-isobutyl-15-isopropyl-1,4,7,10,13-pentaoxo-2,5,8,11,14-pentaazahexadecane)pyrrolidine-2-carboxamido)-5-phenylpentanoic acid
Show/Hide
|
C53H84N14O11
|
1
|
| 1 |
EC50 = 198 nM
|
|
|
|
CP0953635
|
(2S)-1-((S)-2-((S)-1-((3S,6S,9S,12S,15S)-6-((1H-imidazol-5-yl)methyl)-1-((S)-1-((S)-2-aminohexanoyl)pyrrolidin-2-yl)-12-(3-guanidinopropyl)-9-(hydroxymethyl)-3-isobutyl-15-isopropyl-1,4,7,10,13-pentaoxo-2,5,8,11,14-pentaazahexadecane)pyrrolidine-2-carboxamido)-3-phenylpropanoyl)octahydro-1H-indole-2-carboxylic acid
Show/Hide
|
C60H93N15O12
|
1
|
| 1 |
EC50 = 224 nM
|
|
|
|
CP0944656
|
(S)-1-((S)-2-((S)-1-((3S,6S,9S,12S,15S)-6-((1H-imidazol-5-yl)methyl)-1-((S)-1-((S)-2-aminohexanoyl)pyrrolidin-2-yl)-15-benzyl-12-(3-guanidinopropyl)-9-(hydroxymethyl)-3-isobutyl-1,4,7,10,13-pentaoxo-2,5,8,11,14-pentaazahexadecane)pyrrolidine-2-carboxamido)-3-phenylpropanoyl)pyrrolidine-2-carboxylic acid
Show/Hide
|
C60H87N15O12
|
1
|
| 1 |
EC50 = 314 nM
|
|
|
|
CP0944657
|
(S)-1-((S)-2-((S)-1-((3S,6S,9S,12S,15S)-6-((1H-imidazol-5-yl)methyl)-1-((S)-1-((S)-2-aminohexanoyl)pyrrolidin-2-yl)-12-(3-guanidinopropyl)-9-(hydroxymethyl)-3-isobutyl-15-isopropyl-1,4,7,10,13-pentaoxo-2,5,8,11,14-pentaazahexadecane)pyrrolidine-2-carboxamido)-3-phenylpropanoyl)pyrrolidine-2-carboxylic acid
Show/Hide
|
C56H87N15O12
|
1
|
| 1 |
EC50 = 371 nM
|
|
|
|
CP0955252
|
(S)-1-((S)-2-((S)-1-((3S,6S,9S,12S,15S)-6-((1H-imidazol-5-yl)methyl)-1-((S)-1-((S)-2-aminohexanoyl)pyrrolidin-2-yl)-3-benzyl-12-(3-guanidinopropyl)-9-(hydroxymethyl)-15-isopropyl-3-methyl-1,4,7,10,13-pentaoxo-2,5,8,11,14-pentaazahexadecane)pyrrolidine-2-carboxamido)-3-phenylpropanoyl)pyrrolidine-2-carboxylic acid
Show/Hide
|
C60H87N15O12
|
1
|
| 1 |
EC50 = 515 nM
|
|
|
|
CP0871210
|
(S)-2-((S)-2-((S)-1-((3S,6S,9S,12S,15S)-6-((1H-imidazol-5-yl)methyl)-1-((S)-1-((S)-2-aminohexanoyl)pyrrolidin-2-yl)-12-(3-guanidinopropyl)-9-(hydroxymethyl)-3-isobutyl-15-isopropyl-1,4,7,10,13-pentaoxo-2,5,8,11,14-pentaazahexadecane)pyrrolidine-2-carboxamido)-3-phenylpropanamido)-4-methylpentanoic acid
Show/Hide
|
C57H91N15O12
|
1
|
| 1 |
EC50 = 525 nM
|
|
|
|
CP0871208
|
(S)-3-((S)-1-((3S,6S,9S,12S,15S)-6-((1H-imidazol-5-yl)methyl)-1-((S)-1-((S)-2-aminohexanoyl)pyrrolidin-2-yl)-12-(3-guanidinopropyl)-9-(hydroxymethyl)-3-isobutyl-15-isopropyl-1,4,7,10,13-pentaoxo-2,5,8,11,14-pentaazahexadecane)pyrrolidine-2-carboxamido)-4-phenylbutanoic acid
Show/Hide
|
C52H82N14O11
|
1
|
| 1 |
EC50 = 740 nM
|
|
|
|
CP0953643
|
(S)-1-((S)-2-((S)-1-((3S,6S,9S,12S,15S)-6-((1H-imidazol-5-yl)methyl)-1-((S)-1-((S)-2-aminohexanoyl)pyrrolidin-2-yl)-3-tert-butyl-12-(3-guanidinopropyl)-9-(hydroxymethyl)-15-isopropyl-1,4,7,10,13-pentaoxo-2,5,8,11,14-pentaazahexadecane)pyrrolidine-2-carboxamido)-3-phenylpropanoyl)pyrrolidine-2-carboxylic acid
Show/Hide
|
C56H87N15O12
|
1
|
| 1 |
EC50 = 795 nM
|
|
|
|
CP0957089
|
(S)-1-((S)-2-((S)-1-((3S,6S,9S,12S,15S)-6-((1H-imidazol-5-yl)methyl)-1-((S)-1-((S)-2-aminohexanoyl)pyrrolidin-2-yl)-12-(3-guanidinopropyl)-9-(hydroxymethyl)-3-isobutyl-15-isopropyl-1,4,7,10,13-pentaoxo-2,5,8,11,14-pentaazahexadecane)pyrrolidine-2-carboxamido)-3-(naphthalen-1-yl)propanoyl)pyrrolidine-2-carboxylic acid
Show/Hide
|
C60H89N15O12
|
1
|
| 1 |
EC50 = 1040 nM
|
|
|
|
CP0487480
|
6-butyl-5-(2,6-dimethoxyphenyl)-4-hydroxy-N,N-dimethyl-2-oxo-1H-pyridine-3-carboxamide
Show/Hide
|
C20H26N2O5
|
1
|
| 1 |
EC50 = 1100 nM
|
|
|
|
CP0559788
|
N-benzyl-6-butyl-5-(2,6-dimethoxyphenyl)-4-hydroxy-2-oxo-1H-pyridine-3-carboxamide
Show/Hide
|
C25H28N2O5
|
1
|
| 1 |
EC50 = 1100 nM
|
|
|
|
CP0956057
|
(S)-2-((S)-2-((S)-1-((3S,6S,9S,12S,15S)-6-((1H-imidazol-5-yl)methyl)-1-((S)-1-((S)-2-aminohexanoyl)pyrrolidin-2-yl)-12-(3-guanidinopropyl)-9-(hydroxymethyl)-3-isobutyl-15-isopropyl-1,4,7,10,13-pentaoxo-2,5,8,11,14-pentaazahexadecane)pyrrolidine-2-carboxamido)-3-phenylpropanamido)-3-(4-(benzyloxy)phenyl)propanoic acid
Show/Hide
|
C67H95N15O13
|
1
|
| 1 |
EC50 = 1525 nM
|
|
|
|
CP0955245
|
(S)-1-((S)-2-((S)-1-((3S,6S,9S,12S,15S)-6-((1H-imidazol-5-yl)methyl)-1-((S)-1-((S)-2-amino-4-(methylthio)butanoyl)pyrrolidin-2-yl)-12-(3-guanidinopropyl)-9-(hydroxymethyl)-3-isobutyl-15-isopropyl-1,4,7,10,13-pentaoxo-2,5,8,11,14-pentaazahexadecane)pyrrolidine-2-carboxamido)-3-phenylpropanoyl)pyrrolidine-2-carboxylic acid
Show/Hide
|
C55H85N15O12S
|
1
|
| 1 |
EC50 = 2200 nM
|
|
|
|
CP0565378
|
6-butyl-5-(2,6-dimethoxyphenyl)-N-ethyl-4-hydroxy-2-oxo-1H-pyridine-3-carboxamide
Show/Hide
|
C20H26N2O5
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
