Brief Information of the Compound and Protein
Compound Name
(R)-6-butyl-5-(2,6-dimethoxyphenyl)-4-hydroxy-3-(3-phenylpyrrolidine-1-carbonyl)pyridin-2(1H)-one
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PubChem ID
CID: 129032236
Canonical SMILES
CCCCc1[nH]c(=O)c(C(=O)N2CC[C@H](c3ccccc3)C2)c(O)c1-c1c(OC)cccc1OC
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Compound Formula C28H32N2O5
Compound Structure
Protein Name
Apelin receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Neuropeptide receptor
Uniprot ID
P35414
Gene Name
APLNR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000025 HEK-293T Homo sapiens (Human)  1
1
EC50 = 1 nM
   TI
   LI
   LO
   TS
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 1 nM
   TI
   LI
   LO
   TS