Brief Information of the Cell Line and Protein
Cell Line ID: CL000025 , HEK-293T
Synonyms
Hek293T
HEK-293T
HEK 293T
HEK-293-T
HEK 293 T
293-T
293 T
293T
Human Embryonic Kidney 293T
293tsA1609neo
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0063
Protein ID: PT02149 , Transient receptor potential cation channel subfamily A member 1
Gene Name TRPA1
Organism Homo sapiens, Human
Protein Classification Ion channel
Uniprot ID O75762
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000025  Protein ID: PT02149
 
Compound ID Compound Name Compound Formula
CP0041478
3-isothiocyanatoprop-1-ene
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C4H5NS
 1
1
EC50 = 500 nM
   TI
   LI
   LO
   TS
CP0126907
methyl (1S,15S,17S,18S)-17-ethyl-7-methoxy-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2(10),4(9),5,7-tetraene-1-carboxylate
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C22H28N2O3
 1
1
EC50 = 8000 nM
   TI
   LI
   LO
   TS
CP0578580
US11136336, Example 15
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C20H16ClN5O4S
 1
1
IC50 = 9 nM
   TI
   LI
   LO
   TS
CP0557799
US11136336, Example 11
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C20H18ClN5O4S
 1
1
IC50 = 10 nM
   TI
   LI
   LO
   TS
CP0568398
3-({3-[(2S)-2-(4-chlorophenyl)-2-hydroxyethyl]-1,2,4-oxadiazol-5-yl}methyl)-5-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
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C19H16ClN5O4S
 1
1
IC50 = 13 nM
   TI
   LI
   LO
   TS
CP0552408
US11136336, Example 12
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C21H18ClF2N5O4S
 1
1
IC50 = 15 nM
   TI
   LI
   LO
   TS
CP0534366
US11136336, Example 16
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C18H13Cl2N5O4S
 1
1
IC50 = 16 nM
   TI
   LI
   LO
   TS
CP0552407
US11136336, Example 3
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C21H17N5O5S
 1
1
IC50 = 19 nM
   TI
   LI
   LO
   TS
CP0494206
US11136336, Example 13
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C23H24ClN5O5S
 1
1
IC50 = 37 nM
   TI
   LI
   LO
   TS
CP0572639
US11136336, Example 6
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C19H15F2N5O4S
 1
1
IC50 = 48 nM
   TI
   LI
   LO
   TS
CP0575314
US11136336, Example 8
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C20H17N5O6S
 1
1
IC50 = 56 nM
   TI
   LI
   LO
   TS
CP0562992
US11136336, Example 9
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C21H19N5O6S
 1
1
IC50 = 78 nM
   TI
   LI
   LO
   TS
CP0539936
N-[(1R)-2-amino-2-oxo-1-phenylethyl]-N-[(1R)-6-chloro-4-fluoro-2,3-dihydro-1H-inden-1-yl]-2-methylpyridine-3-carboxamide
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C24H21ClFN3O2
 1
1
IC50 > 30000 nM
   TI
   LI
   LO
   TS