| Compound ID |
Compound Name |
Compound Formula |
|
CP0081974
|
US10034864, Example 1
Show/Hide
|
C11H13BrFN7O4S
|
1
|
| 1 |
IC50 = 9.63 nM
|
|
|
|
CP0565953
|
US11447477, Compound 8
Show/Hide
|
C14H17BrFN7O4S
|
1
|
| 1 |
IC50 = 19.88 nM
|
|
|
|
CP0563993
|
US11447477, Compound 9
Show/Hide
|
C14H17BrFN7O4S
|
1
|
| 1 |
IC50 = 42.58 nM
|
|
|
|
CP0258724
|
N'-(3-bromo-4-fluorophenyl)-N-hydroxy-4-[[(3S)-1-methylsulfonylpyrrolidin-3-yl]methylamino]-1,2,5-oxadiazole-3-carboximidamide
Show/Hide
|
C15H18BrFN6O4S
|
1
|
| 1 |
IC50 = 42.99 nM
|
|
|
|
CP0552669
|
N'-(3-bromo-4-fluorophenyl)-N-hydroxy-4-[[(3S)-1-methylsulfonylpiperidin-3-yl]methylamino]-1,2,5-oxadiazole-3-carboximidamide
Show/Hide
|
C16H20BrFN6O4S
|
1
|
| 1 |
IC50 = 49.83 nM
|
|
|
|
CP0563996
|
N'-(3-bromo-4-fluorophenyl)-N-hydroxy-4-[[(3R)-1-sulfamoylpiperidin-3-yl]methylamino]-1,2,5-oxadiazole-3-carboximidamide
Show/Hide
|
C15H19BrFN7O4S
|
1
|
| 1 |
IC50 = 57.76 nM
|
|
|
|
CP0542837
|
N'-(3-bromo-4-fluorophenyl)-N-hydroxy-4-[[(3S)-1-sulfamoylpiperidin-3-yl]methylamino]-1,2,5-oxadiazole-3-carboximidamide
Show/Hide
|
C15H19BrFN7O4S
|
1
|
| 1 |
IC50 = 68.59 nM
|
|
|
|
CP0552670
|
N'-(3-bromo-4-fluorophenyl)-N-hydroxy-4-[[(3R)-1-methylsulfonylpiperidin-3-yl]methylamino]-1,2,5-oxadiazole-3-carboximidamide
Show/Hide
|
C16H20BrFN6O4S
|
1
|
| 1 |
IC50 = 125.44 nM
|
|
|
|
CP0560224
|
N'-(3-bromo-4-fluorophenyl)-N-hydroxy-4-[[(1R,3R)-3-(sulfamoylamino)cyclohexyl]methylamino]-1,2,5-oxadiazole-3-carboximidamide
Show/Hide
|
C16H21BrFN7O4S
|
1
|
| 1 |
IC50 = 137.95 nM
|
|
|
|
CP0574184
|
N'-(3-bromo-4-fluorophenyl)-N-hydroxy-4-[2-(1-sulfamoylpiperidin-3-yl)ethylamino]-1,2,5-oxadiazole-3-carboximidamide
Show/Hide
|
C16H21BrFN7O4S
|
1
|
| 1 |
IC50 = 153.75 nM
|
|
|
|
CP0352136
|
N'-(3-bromo-4-fluorophenyl)-N-hydroxy-4-[[(2S)-1-sulfamoylpiperidin-2-yl]methylamino]-1,2,5-oxadiazole-3-carboximidamide
Show/Hide
|
C15H19BrFN7O4S
|
1
|
| 1 |
IC50 = 177.35 nM
|
|
|
|
CP0542835
|
N'-(3-bromo-4-fluorophenyl)-N-hydroxy-4-[[(2S)-1-methylsulfonylpyrrolidin-2-yl]methylamino]-1,2,5-oxadiazole-3-carboximidamide
Show/Hide
|
C15H18BrFN6O4S
|
1
|
| 1 |
IC50 = 186.2 nM
|
|
|
|
CP0542836
|
N'-(3-bromo-4-fluorophenyl)-N-hydroxy-4-[[(2R)-1-methylsulfonylpyrrolidin-2-yl]methylamino]-1,2,5-oxadiazole-3-carboximidamide
Show/Hide
|
C15H18BrFN6O4S
|
1
|
| 1 |
IC50 = 333.65 nM
|
|
|
|
CP0271852
|
N'-(3-bromo-4-fluorophenyl)-4-[(1-cyclopropylsulfonylpiperidin-3-yl)methylamino]-N-hydroxy-1,2,5-oxadiazole-3-carboximidamide
Show/Hide
|
C18H22BrFN6O4S
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0533459
|
N'-(3-bromo-4-fluorophenyl)-4-[[1-(difluoromethylsulfonyl)piperidin-3-yl]methylamino]-N-hydroxy-1,2,5-oxadiazole-3-carboximidamide
Show/Hide
|
C16H18BrF3N6O4S
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
