Brief Information of the Cell Line and Protein
Cell Line ID: CL000025 , HEK-293T
Synonyms
Hek293T
HEK-293T
HEK 293T
HEK-293-T
HEK 293 T
293-T
293 T
293T
Human Embryonic Kidney 293T
293tsA1609neo
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0063
Protein ID: PT01427 , Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
Gene Name PKMYT1
Organism Homo sapiens, Human
Protein Classification Kinase
Uniprot ID Q99640
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000025  Protein ID: PT01427
 
Compound ID Compound Name Compound Formula
CP0546952
2-amino-1-(3-hydroxy-2,6-dimethylphenyl)-5-methylpyrrolo[2,3-b]pyridine-3-carboxamide
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C17H18N4O2
 1
1
IC50 = 1 nM
   TI
   LI
   LO
   TS
CP0577047
2-amino-5-chloro-1-(3-hydroxy-2,6-dimethylphenyl)pyrrolo[2,3-b]pyridine-3-carboxamide
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C16H15ClN4O2
 1
1
IC50 = 1 nM
   TI
   LI
   LO
   TS
CP0578487
6-amino-2-cyclopropyl-5-(3-hydroxy-2,6-dimethylphenyl)pyrrolo[2,3-b]pyrazine-7-carboxamide
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C18H19N5O2
 1
1
IC50 = 1 nM
   TI
   LI
   LO
   TS
CP0574498
2-amino-1-(3-hydroxy-2,6-dimethylphenyl)-5,6-dimethylpyrrolo[2,3-b]pyridine-3-carboxamide
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C18H20N4O2
 1
1
IC50 = 2 nM
   TI
   LI
   LO
   TS
CP0574500
2-amino-5-cyclopropyl-1-(3-hydroxy-2,6-dimethylphenyl)pyrrolo[2,3-b]pyridine-3-carboxamide
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C19H20N4O2
 1
1
IC50 = 3 nM
   TI
   LI
   LO
   TS
CP0548461
6-amino-5-(3-hydroxy-2,6-dimethylphenyl)-2,3-dimethylpyrrolo[2,3-b]pyrazine-7-carboxamide
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C17H19N5O2
 1
1
IC50 = 5 nM
   TI
   LI
   LO
   TS
CP0574502
2-amino-5-bromo-1-(3-hydroxy-2,6-dimethylphenyl)pyrrolo[2,3-b]quinoxaline-3-carboxamide
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C19H16BrN5O2
 1
1
IC50 = 9 nM
   TI
   LI
   LO
   TS
CP0571617
6-amino-5-(3-hydroxy-2,6-dimethylphenyl)pyrrolo[2,3-b]pyrazine-7-carboxamide
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C15H15N5O2
 1
1
IC50 = 12 nM
   TI
   LI
   LO
   TS
CP0577566
6-amino-5-(3-hydroxy-2,6-dimethylphenyl)-2-(2-hydroxypropan-2-yl)pyrrolo[2,3-b]pyrazine-7-carboxamide
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C18H21N5O3
 1
1
IC50 = 23 nM
   TI
   LI
   LO
   TS