Brief Information of the Cell Line and Protein
Cell Line ID: CL000025 , HEK-293T
Synonyms
Hek293T
HEK-293T
HEK 293T
HEK-293-T
HEK 293 T
293-T
293 T
293T
Human Embryonic Kidney 293T
293tsA1609neo
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0063
Protein ID: PT01007 , Alpha-1B adrenergic receptor
Gene Name ADRA1B
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P35368
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000025  Protein ID: PT01007
 
Compound ID Compound Name Compound Formula
CP0129619
N-[3-[2-[[(6S)-2-amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl]-propylamino]ethyl]-3-hydroxycyclobutyl]naphthalene-2-carboxamide
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C27H34N4O2S
 1
1
Ki = 666 nM
   TI
   LI
   LO
   TS
CP0244206
7-[4-imidazo[1,2-a]pyridin-5-yl-3-(trifluoromethyl)phenoxy]thieno[2,3-c]pyridine
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C21H12F3N3OS
 1
1
Ki = 4800 nM
   TI
   LI
   LO
   TS
CP0369306
4-[4-imidazo[1,2-a]pyridin-5-yl-3-(trifluoromethyl)phenoxy]furo[3,2-c]pyridine
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C21H12F3N3O2
 1
1
Ki = 7400 nM
   TI
   LI
   LO
   TS
CP0064188
4-[4-(6-methylimidazo[1,2-a]pyrazin-5-yl)-3-(trifluoromethyl)phenoxy]furo[3,2-c]pyridine
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C21H13F3N4O2
 1
1
Ki = 8800 nM
   TI
   LI
   LO
   TS
CP0064183
4-[3-methyl-4-(6-methylimidazo[1,2-a]pyrazin-5-yl)phenoxy]furo[3,2-c]pyridine
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C21H16N4O2
 1
1
Ki = 9200 nM
   TI
   LI
   LO
   TS
CP0054519
(1R,12R,13S,17R,21S)-12-ethyl-18-propyl-7-(trifluoromethyl)-10,18-diazapentacyclo[11.7.1.02,11.04,9.017,21]henicosa-2(11),3,5,7,9-pentaene
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C25H31F3N2
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0085414
(3aS,6R,6aS,9aR,9bR)-6-benzyl-1-methyl-3,3a,4,6,6a,7,8,9,9a,9b-decahydro-2H-benzo[de]quinolin-5-one
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C20H27NO
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0387083
(3aS,9bS)-3a-methyl-5-phenyl-2,3,4,9b-tetrahydro-1H-pyrrolo[2,3-c]quinoline
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C18H20N2
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0391120
(1S,2R)-1-ethyl-7-methoxy-2-methyl-3,4-dihydro-1H-naphthalen-2-amine
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C14H21NO
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0391121
(3S,4S)-4-ethyl-3,6-dimethyl-2,4-dihydrochromen-3-amine
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C13H19NO
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0391154
(3aS,9bS)-7,9-dimethoxy-3a-methyl-2,3,4,9b-tetrahydro-1H-chromeno[3,4-b]pyrrole
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C14H19NO3
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0411059
(3S,4S)-4-ethyl-3-methyl-1-phenyl-2,4-dihydroquinolin-3-amine
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C18H22N2
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0156479
(+)-N-methyl-laurotetanine
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C20H23NO4
 1
1
Ki > 950 nM
   TI
   LI
   LO
   TS