Brief Information of the Cell Line and Protein
Cell Line ID: CL000025 , HEK-293T
 Cell Line Info 
Synonyms
Hek293T
HEK-293T
HEK 293T
HEK-293-T
HEK 293 T
293-T
293 T
293T
Human Embryonic Kidney 293T
293tsA1609neo
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0063
Protein ID: PT00903 , C-C chemokine receptor type 5
 Protein Info 
Gene Name CCR5
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P51681
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000025
 Cell Line Info 
 Protein ID: PT00903
 Protein Info 
 
Compound ID Compound Name Compound Formula
CP0666580
 Compound Info 
Dimethyl-(tetrahydro-pyran-4-yl)-{4-[(3-p-tolyl-8,9-dihydro-7H-benzocycloheptene-6-carbonyl)-amino]-benzyl}-ammonium chloride(TAK-779)
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C33H39ClN2O2
  1
1
EC50 = 7 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0478193
 Compound Info 
N-[4-[[methyl(oxan-4-yl)amino]methyl]phenyl]-2-(2-methylpropyl)-1-oxo-3H-2-benzazepine-4-carboxamide
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C28H35N3O3
  1
1
EC50 = 2470 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0116643
 Compound Info 
N-[4-[[methyl(oxan-4-yl)amino]methyl]phenyl]-2-(2-methylpropyl)-8-nitro-1-oxo-3H-2-benzazepine-4-carboxamide
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C28H34N4O5
  1
1
EC50 > 10 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0210291
 Compound Info 
8-acetamido-N-[4-[[methyl(oxan-4-yl)amino]methyl]phenyl]-2-(2-methylpropyl)-1-oxo-3H-2-benzazepine-4-carboxamide
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C30H38N4O4
  1
1
EC50 > 10 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0231889
 Compound Info 
N-[4-[[methyl(oxan-4-yl)amino]methyl]phenyl]-8-(4-methylphenyl)-2-(2-methylpropyl)-1-oxo-3H-2-benzazepine-4-carboxamide
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C35H41N3O3
  1
1
EC50 > 10 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0330352
 Compound Info 
8-(methanesulfonamido)-N-[4-[[methyl(oxan-4-yl)amino]methyl]phenyl]-2-(2-methylpropyl)-1-oxo-3H-2-benzazepine-4-carboxamide
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C29H38N4O5S
  1
1
EC50 > 10 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0355485
 Compound Info 
2-(2-methylpropyl)-1-oxo-N-[4-(1,3-thiazol-2-ylsulfamoyl)phenyl]-3H-2-benzazepine-4-carboxamide
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C24H24N4O4S2
  1
1
EC50 > 10 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0355486
 Compound Info 
N-[4-[[methyl(oxan-4-yl)amino]methyl]phenyl]-7-(4-methylphenyl)-2-(2-methylpropyl)-1-oxo-3H-2-benzazepine-4-carboxamide
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C35H41N3O3
  1
1
EC50 > 10 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0481532
 Compound Info 
N-[4-[[methyl(oxan-4-yl)amino]methyl]phenyl]-2-(2-methylpropyl)-6-nitro-1-oxo-3H-2-benzazepine-4-carboxamide
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C28H34N4O5
  1
1
EC50 > 10 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS