Brief Information of the Compound and Protein
Compound Name
2-(2-methylpropyl)-1-oxo-N-[4-(1,3-thiazol-2-ylsulfamoyl)phenyl]-3H-2-benzazepine-4-carboxamide
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PubChem ID
CID: 137648323
Canonical SMILES
CC(C)CN1CC(=Cc2ccccc2C1=O)C(=O)Nc1ccc(cc1)S(=O)(=O)Nc1nccs1
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Compound Formula C24H24N4O4S2
Compound Structure
Protein Name
C-C chemokine receptor type 5
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Chemokine receptor
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CC chemokine receptor
Uniprot ID
P51681
Gene Name
CCR5
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000025 HEK-293T Homo sapiens (Human)  1
1
EC50 > 10 nM
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