| Compound ID |
Compound Name |
Compound Formula |
|
CP0506945
|
US8940771, 48
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|
C21H24F3N5O2S
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0563214
|
US8940771, 119
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|
C19H22F3N5O2S
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0542016
|
US8940771, 46
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|
C20H22F3N5O2S
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0554263
|
US8940771, 3
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|
C17H22N6O2S
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0554851
|
US8940771, 7
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|
C18H23N5O2S
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0551331
|
US8940771, 49
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|
C20H22N6O2S
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0542017
|
US8940771, 129
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|
C19H22ClN5O2S
|
1
|
| 1 |
IC50 = 24 nM
|
|
|
|
CP0557585
|
US8940771, 117
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|
C19H23N5O2S
|
1
|
| 1 |
IC50 = 26 nM
|
|
|
|
CP0506805
|
US8940771, 124
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|
C25H29N5O3S
|
1
|
| 1 |
IC50 = 28 nM
|
|
|
|
CP0530606
|
US8940771, 65
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|
C19H26N6O3S
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0565280
|
US8940771, 40
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|
C19H23N5O2S
|
1
|
| 1 |
IC50 = 37 nM
|
|
|
|
CP0529231
|
US8940771, 253
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|
C20H24F3N5O2S
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0557587
|
US8940771, 66
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|
C18H23FN6O2S
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0537003
|
US8940771, 107
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|
C21H31N7O2S
|
1
|
| 1 |
IC50 = 44 nM
|
|
|
|
CP0478460
|
US8940771, 11
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|
C18H22N6O2S
|
1
|
| 1 |
IC50 = 48 nM
|
|
|
|
CP0553843
|
US8940771, 112
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|
C20H28N6O3S
|
1
|
| 1 |
IC50 = 49 nM
|
|
|
|
CP0520698
|
US8940771, 122
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|
C19H26N6O2S
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0426467
|
US8940771, 111
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|
C19H26N6O2S
|
1
|
| 1 |
IC50 = 52 nM
|
|
|
|
CP0400587
|
US8940771, 110
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|
C19H24N6O2S
|
1
|
| 1 |
IC50 = 71 nM
|
|
|
|
CP0529232
|
US8940771, 59
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|
C19H21F2N5O2S
|
1
|
| 1 |
IC50 = 71 nM
|
|
|
|
CP0563213
|
US8940771, 88
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|
C19H25N7O2S
|
1
|
| 1 |
IC50 = 76 nM
|
|
|
|
CP0557586
|
US8940771, 101
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|
C20H29N7O3S
|
1
|
| 1 |
IC50 = 99 nM
|
|
|
|
CP0521202
|
US8940771, 74
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|
C16H20N6O2S2
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0521255
|
US8940771, 114
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|
C19H24F2N6O2S
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0536925
|
US8940771, 98
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|
C24H29N7O2S
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0519145
|
US8940771, 1
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|
C23H27N5O4S2
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0506946
|
US8940771, 54
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|
C26H29N5O3S
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0537004
|
US8940771, 102
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|
C19H22N8O2S
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0400586
|
US8940771, 80
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|
C20H30N8O2S
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0526547
|
4-[[5-(4-amino-6-methyl-1,3,5-triazin-2-yl)-6-[[6-chloro-5-(dimethylsulfamoylamino)pyridin-3-yl]amino]pyridin-3-yl]methyl]morpholine
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|
C21H27ClN10O3S
|
1
|
| 1 |
Ki = 1.9 nM
|
|
|
|
CP0371423
|
N-[5-[[3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-5-(oxan-4-yl)pyridin-2-yl]amino]-2-chloropyridin-3-yl]methanesulfonamide
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|
C20H23ClN8O3S
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0523492
|
N-[5-[[3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-5-chloropyridin-2-yl]amino]-2-chloropyridin-3-yl]methanesulfonamide
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|
C15H14Cl2N8O2S
|
1
|
| 1 |
Ki = 3.5 nM
|
|
|
|
CP0057249
|
2-amino-4-[5-chloro-2-[[6-chloro-5-(dimethylsulfamoylamino)pyridin-3-yl]amino]pyridin-3-yl]-6-methyl-1,3,5-triazine
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|
C16H17Cl2N9O2S
|
1
|
| 1 |
Ki = 7.7 nM
|
|
|
|
CP0441821
|
N-[5-[[3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-5-chloropyridin-2-yl]amino]-2-chloropyridin-3-yl]morpholine-4-sulfonamide
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|
C18H19Cl2N9O3S
|
1
|
| 1 |
Ki = 8.6 nM
|
|
|
|
CP0218104
|
2-amino-4-[2-[[6-chloro-5-(dimethylsulfamoylamino)pyridin-3-yl]amino]-5-methoxypyridin-3-yl]-6-methyl-1,3,5-triazine
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|
C17H20ClN9O3S
|
1
|
| 1 |
Ki = 9.3 nM
|
|
|
|
CP0292752
|
N-[5-[[3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-5-(morpholin-4-ylmethyl)pyridin-2-yl]amino]-2-chloropyridin-3-yl]methanesulfonamide
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|
C20H24ClN9O3S
|
1
|
| 1 |
Ki = 9.7 nM
|
|
|
|
CP0131208
|
N-[5-[[3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-5-methoxypyridin-2-yl]amino]-2-chloropyridin-3-yl]methanesulfonamide
Show/Hide
|
C16H17ClN8O3S
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0174697
|
N-[5-[[3-(4-amino-6-methyl-1,3,5-triazin-2-yl)pyridin-2-yl]amino]-2-chloropyridin-3-yl]cyclopropanesulfonamide
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|
C17H17ClN8O2S
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0553313
|
2-amino-4-[2-[[6-chloro-5-(dimethylsulfamoylamino)pyridin-3-yl]amino]pyridin-3-yl]-6-methyl-1,3,5-triazine
Show/Hide
|
C16H18ClN9O2S
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0330470
|
N-[5-[[3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-5-methoxypyridin-2-yl]amino]-2-chloropyridin-3-yl]morpholine-4-sulfonamide
Show/Hide
|
C19H22ClN9O4S
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0441822
|
N-[5-[[3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-5-chloropyridin-2-yl]amino]-2-chloropyridin-3-yl]pyridine-3-sulfonamide
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|
C19H15Cl2N9O2S
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0093391
|
N-[5-[[3-(4-amino-6-methyl-1,3,5-triazin-2-yl)pyridin-2-yl]amino]-2-chloropyridin-3-yl]morpholine-4-sulfonamide
Show/Hide
|
C18H20ClN9O3S
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0395569
|
N-[5-[[3-(4-amino-6-methyl-1,3,5-triazin-2-yl)pyridin-2-yl]amino]-2-chloropyridin-3-yl]-4-fluorobenzenesulfonamide
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|
C20H16ClFN8O2S
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0279598
|
N-[5-[[3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-5-(2-methoxyethoxy)pyridin-2-yl]amino]-2-chloropyridin-3-yl]methanesulfonamide
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|
C18H21ClN8O4S
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0283801
|
N-[5-[[3-(4-amino-6-methyl-1,3,5-triazin-2-yl)pyridin-2-yl]amino]-2-chloropyridin-3-yl]methanesulfonamide
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|
C15H15ClN8O2S
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0501054
|
2-amino-4-[5-chloro-2-[[6-chloro-5-[[2-methoxyethyl(methyl)sulfamoyl]amino]pyridin-3-yl]amino]pyridin-3-yl]-6-methyl-1,3,5-triazine
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|
C18H21Cl2N9O3S
|
1
|
| 1 |
Ki = 29 nM
|
|
|
|
CP0499598
|
2-amino-4-[2-[[6-chloro-5-[[methyl(propan-2-yl)sulfamoyl]amino]pyridin-3-yl]amino]pyridin-3-yl]-6-methyl-1,3,5-triazine
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|
C18H22ClN9O2S
|
1
|
| 1 |
Ki = 43 nM
|
|
|
|
CP0093388
|
N-[5-[[3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-5-chloropyridin-2-yl]amino]-2-methoxypyridin-3-yl]methanesulfonamide
Show/Hide
|
C16H17ClN8O3S
|
1
|
| 1 |
Ki = 114 nM
|
|
|
|
CP0284209
|
N-[5-[[3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-5-chloropyridin-2-yl]amino]-2-methylpyridin-3-yl]methanesulfonamide
Show/Hide
|
C16H17ClN8O2S
|
1
|
| 1 |
Ki = 161 nM
|
|
|
|
CP0500925
|
N-[5-[[3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-5-chloropyridin-2-yl]amino]-2-chloropyridin-3-yl]-N-methylmethanesulfonamide
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|
C16H16Cl2N8O2S
|
1
|
| 1 |
Ki = 311 nM
|
|
|
|
CP0346732
|
5-N-[3-(4-amino-6-methyl-1,3,5-triazin-2-yl)pyridin-2-yl]-2-chloropyridine-3,5-diamine
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|
C14H13ClN8
|
1
|
| 1 |
Ki = 360 nM
|
|
|
