Brief Information of the Cell Line and Protein
Cell Line ID: CL000017 , HeLa
Synonyms
HELA
Hela
He La
He-La
HeLa-CCL2
Henrietta Lacks cells
Helacyton gartleri
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0030
Protein ID: PT00941 , 5-hydroxytryptamine receptor 7
Gene Name HTR7
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P34969
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000017  Protein ID: PT00941
 
Compound ID Compound Name Compound Formula
CP0238957
1-[2-(4-methoxyphenyl)phenyl]piperazine
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C17H20N2O
 1
1
IC50 = 438 nM
   TI
   LI
   LO
   TS
CP0194931
1-(2-phenylphenyl)piperazine
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C16H18N2
 1
1
IC50 = 531 nM
   TI
   LI
   LO
   TS
CP0379542
5-(4-Methylpiperazin-1-yl)-3-(1-naphthalenesulfonyl)-1H-indazole
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C22H22N4O2S
 1
1
Ki = 579 nM
   TI
   LI
   LO
   TS
CP0379544
5-(4-methylpiperazin-1-yl)-3-(phenylsulfonyl)-1H-indazole
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C18H20N4O2S
 1
1
Ki = 753 nM
   TI
   LI
   LO
   TS
CP0379545
3-(Naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
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C21H20N4O2S
 1
1
Ki = 1563 nM
   TI
   LI
   LO
   TS
CP0379546
1-methyl-3-(naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
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C22H22N4O2S
 1
1
Ki > 5000 nM
   TI
   LI
   LO
   TS
CP0379601
1-isopropyl-3-(naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
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C24H26N4O2S
 1
1
Ki > 5000 nM
   TI
   LI
   LO
   TS
CP0406091
1-benzyl-3-(naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
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C28H26N4O2S
 1
1
Ki > 5000 nM
   TI
   LI
   LO
   TS
CP0479094
1-isobutyl-3-(naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
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C25H28N4O2S
 1
1
Ki > 5000 nM
   TI
   LI
   LO
   TS