| Compound ID |
Compound Name |
Compound Formula |
|
CP0016691
|
N-(1-methylbenzimidazol-2-yl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamide
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|
C21H19N5O2
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0026929
|
N-(3-methyl-1,2-oxazol-5-yl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamide
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|
C17H16N4O3
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0060278
|
N-(1H-imidazol-2-yl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamide
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|
C16H15N5O2
|
1
|
| 1 |
IC50 = 290 nM
|
|
|
|
CP0340761
|
1-oxo-N-quinolin-3-yl-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamide
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|
C22H18N4O2
|
1
|
| 1 |
IC50 = 340 nM
|
|
|
|
CP0226208
|
N-(2-carbamoylphenyl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamide
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|
C20H18N4O3
|
1
|
| 1 |
IC50 = 560 nM
|
|
|
|
CP0094906
|
1-oxo-N-pyridin-4-yl-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamide
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|
C18H16N4O2
|
1
|
| 1 |
IC50 = 620 nM
|
|
|
|
CP0017602
|
N-(1-methylpyrazol-4-yl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamide
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|
C17H17N5O2
|
1
|
| 1 |
IC50 = 790 nM
|
|
|
|
CP0100105
|
(3S,4R)-3,4-dimethyl-1-oxo-N-pyridin-3-yl-3,4-dihydro-2H-pyrazino[1,2-a]indole-7-carboxamide
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|
C19H18N4O2
|
1
|
| 1 |
IC50 = 840 nM
|
|
|
|
CP0226449
|
1-oxo-N-(1-propan-2-ylpyrazolo[3,4-b]pyridin-5-yl)-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamide
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|
C22H22N6O2
|
1
|
| 1 |
IC50 = 840 nM
|
|
|
|
CP0169874
|
5-methyl-1-oxo-N-pyridin-3-yl-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamide
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|
C19H18N4O2
|
1
|
| 1 |
IC50 = 890 nM
|
|
|
|
CP0275549
|
1-oxo-N-quinolin-2-yl-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamide
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|
C22H18N4O2
|
1
|
| 1 |
IC50 = 1130 nM
|
|
|
|
CP0275545
|
4,4-dimethyl-1-oxo-N-pyridin-3-yl-2,3-dihydropyrazino[1,2-a]indole-7-carboxamide
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|
C19H18N4O2
|
1
|
| 1 |
IC50 = 1550 nM
|
|
|
|
CP0275544
|
4-methyl-1-oxo-N-pyridin-3-yl-3,4-dihydro-2H-pyrazino[1,2-a]indole-7-carboxamide
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|
C18H16N4O2
|
1
|
| 1 |
IC50 = 1630 nM
|
|
|
|
CP0283281
|
1-oxo-N-phenyl-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamide
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|
C19H17N3O2
|
1
|
| 1 |
IC50 = 1930 nM
|
|
|
|
CP0089165
|
indole-based 7-membered lactam, 23a
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|
C18H16N4O2
|
1
|
| 1 |
IC50 = 1940 nM
|
|
|
|
CP0275546
|
1-oxo-N-pyridin-2-yl-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamide
Show/Hide
|
C18H16N4O2
|
1
|
| 1 |
IC50 = 2630 nM
|
|
|
|
CP0089166
|
indole-based 7-membered lactam, 25d
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|
C19H18N4O2
|
1
|
| 1 |
IC50 = 4890 nM
|
|
|
|
CP0079200
|
N-(1H-benzimidazol-2-yl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamide
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|
C20H17N5O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0100107
|
1-oxo-N-(1H-pyrazol-4-yl)-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamide
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|
C16H15N5O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0285473
|
indole-based 6-membered lactam, 2
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|
C17H14N4O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0312274
|
N-(1,3-benzoxazol-2-yl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamide
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|
C20H16N4O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0392727
|
1-oxo-N-(pyridin-3-ylmethyl)-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamide
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|
C19H18N4O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
