| Compound ID |
Compound Name |
Compound Formula |
|
CP0199989
|
5,5,5-trifluoro-1-[4-[3-(1,3-thiazol-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]pentan-1-one
Show/Hide
|
C15H17F3N4O2S
|
1
|
| 1 |
EC50 = 60 nM
|
|
|
|
CP0079444
|
4,4,4-trifluoro-1-(4-(3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl)piperidin-1-yl)butan-1-one
Show/Hide
|
C15H16F3N3O2S
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0282421
|
4,4,4-trifluoro-1-[4-[3-(6-methoxy-1,3-benzothiazol-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]butan-1-one
Show/Hide
|
C19H19F3N4O3S
|
1
|
| 1 |
EC50 = 200 nM
|
|
|
|
CP0114261
|
N-[4-(1,3-benzothiazol-2-yl)phenyl]-2-(3-methoxyphenoxy)acetamide
Show/Hide
|
C22H18N2O3S
|
1
|
| 1 |
EC50 = 210 nM
|
|
|
|
CP0339516
|
N-[4-(1,3-benzothiazol-2-yl)phenyl]-2-(3-cyanophenoxy)acetamide
Show/Hide
|
C22H15N3O2S
|
1
|
| 1 |
EC50 = 340 nM
|
|
|
|
CP0290722
|
4,4,4-Trifluoro-1-[(R)-3-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)-pyrrolidin-1-yl]-butan-1-one
Show/Hide
|
C14H14F3N3O2S
|
1
|
| 1 |
EC50 = 400 nM
|
|
|
|
CP0079442
|
4,4,4-trifluoro-1-[4-[3-(1,3-thiazol-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]butan-1-one
Show/Hide
|
C14H15F3N4O2S
|
1
|
| 1 |
EC50 = 500 nM
|
|
|
|
CP0248346
|
4,4,4-trifluoro-1-[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]butan-1-one
Show/Hide
|
C17H18F3N3O2
|
1
|
| 1 |
EC50 = 500 nM
|
|
|
|
CP0456763
|
1-[4-(3-cyclopentyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]-4,4,4-trifluorobutan-1-one
Show/Hide
|
C16H22F3N3O2
|
1
|
| 1 |
EC50 = 800 nM
|
|
|
|
CP0502837
|
4,4,4-trifluoro-1-[4-(4-thiophen-2-yl-1,3-thiazol-2-yl)piperidin-1-yl]butan-1-one
Show/Hide
|
C16H17F3N2OS2
|
1
|
| 1 |
EC50 = 800 nM
|
|
|
|
CP0473250
|
4,4,4-trifluoro-1-[4-[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]butan-1-one
Show/Hide
|
C17H17F4N3O2
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0520621
|
4,4,4-trifluoro-1-[4-(5-thiophen-2-yl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]butan-1-one
Show/Hide
|
C15H16F3N3O2S
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0502866
|
1-[4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-4,4,4-trifluorobutan-1-one
Show/Hide
|
C17H17ClF3N3O2
|
1
|
| 1 |
EC50 = 1100 nM
|
|
|
|
CP0456759
|
4,4,4-trifluoro-1-[4-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]butan-1-one
Show/Hide
|
C18H20F3N3O2
|
1
|
| 1 |
EC50 = 1200 nM
|
|
|
|
CP0456758
|
4,4,4-trifluoro-1-[4-[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]butan-1-one
Show/Hide
|
C16H18F3N3O2S
|
1
|
| 1 |
EC50 = 1300 nM
|
|
|
|
CP0368776
|
N-(4-chlorophenyl)-2-(3-methoxyphenoxy)acetamide
Show/Hide
|
C15H14ClNO3
|
1
|
| 1 |
EC50 = 1600 nM
|
|
|
|
CP0524704
|
4,4,4-trifluoro-1-[4-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]butan-1-one
Show/Hide
|
C18H20F3N3O2
|
1
|
| 1 |
EC50 = 2200 nM
|
|
|
|
CP0087646
|
2-(2-fluorophenoxy)-N-(2-methylquinolin-6-yl)acetamide
Show/Hide
|
C18H15FN2O2
|
1
|
| 1 |
EC50 = 2200 nM
|
|
|
|
CP0456761
|
4,4,4-trifluoro-1-[4-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]butan-1-one
Show/Hide
|
C18H20F3N3O2
|
1
|
| 1 |
EC50 = 2300 nM
|
|
|
|
CP0499338
|
4,4,4-trifluoro-1-[4-[3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]piperidin-1-yl]butan-1-one
Show/Hide
|
C18H17F6N3O2
|
1
|
| 1 |
EC50 = 2500 nM
|
|
|
|
CP0533602
|
4,4,4-trifluoro-1-[4-[3-(1,3-thiazol-5-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]butan-1-one
Show/Hide
|
C14H15F3N4O2S
|
1
|
| 1 |
EC50 = 2500 nM
|
|
|
|
CP0513095
|
4,4,4-trifluoro-1-[4-(4-phenyl-1,3-thiazol-2-yl)piperidin-1-yl]butan-1-one
Show/Hide
|
C18H19F3N2OS
|
1
|
| 1 |
EC50 = 3200 nM
|
|
|
|
CP0499339
|
1-[4-(3-cyclohexyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]-4,4,4-trifluorobutan-1-one
Show/Hide
|
C17H24F3N3O2
|
1
|
| 1 |
EC50 = 4000 nM
|
|
|
|
CP0502838
|
4,4,4-trifluoro-1-[4-(3-phenyl-1,2-oxazol-5-yl)piperidin-1-yl]butan-1-one
Show/Hide
|
C18H19F3N2O2
|
1
|
| 1 |
EC50 = 4000 nM
|
|
|
|
CP0533603
|
4,4,4-trifluoro-1-[4-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]butan-1-one
Show/Hide
|
C16H17F3N4O2
|
1
|
| 1 |
EC50 = 4300 nM
|
|
|
|
CP0508909
|
1-[4-[3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-4,4,4-trifluorobutan-1-one
Show/Hide
|
C17H17ClF3N3O2
|
1
|
| 1 |
EC50 = 6300 nM
|
|
|
|
CP0533608
|
4,4,4-trifluoro-1-[(3R)-3-[3-(1,3-thiazol-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]butan-1-one
Show/Hide
|
C13H13F3N4O2S
|
1
|
| 1 |
EC50 = 6300 nM
|
|
|
|
CP0473251
|
4,4,4-trifluoro-1-[4-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]butan-1-one
Show/Hide
|
C17H17F4N3O2
|
1
|
| 1 |
EC50 = 7900 nM
|
|
|
|
CP0508908
|
4,4,4-trifluoro-1-[4-(3-pyrimidin-2-yl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]butan-1-one
Show/Hide
|
C15H16F3N5O2
|
1
|
| 1 |
EC50 = 9000 nM
|
|
|
|
CP0533604
|
4,4,4-trifluoro-1-[4-(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]butan-1-one
Show/Hide
|
C16H17F3N4O2
|
1
|
| 1 |
EC50 = 9300 nM
|
|
|
|
CP0392833
|
1-[4-[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-4,4,4-trifluorobutan-1-one
Show/Hide
|
C21H26F3N3O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0454690
|
4,4,4-trifluoro-1-[4-[3-(4-hydroxyphenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]butan-1-one
Show/Hide
|
C17H18F3N3O3
|
1
|
| 1 |
EC50 = 10000 nM
|
|
|
|
CP0502865
|
4,4,4-trifluoro-1-[4-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]butan-1-one
Show/Hide
|
C16H17F3N4O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0508910
|
1-[4-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-4,4,4-trifluorobutan-1-one
Show/Hide
|
C17H17ClF3N3O2
|
1
|
| 1 |
EC50 = 10000 nM
|
|
|
|
CP0522167
|
4,4,4-trifluoro-1-[4-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]butan-1-one
Show/Hide
|
C17H17F4N3O2
|
1
|
| 1 |
EC50 = 10000 nM
|
|
|
|
CP0522168
|
1-[4-[3-[4-(dimethylamino)phenyl]-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-4,4,4-trifluorobutan-1-one
Show/Hide
|
C19H23F3N4O2
|
1
|
| 1 |
EC50 = 10000 nM
|
|
|
|
CP0523537
|
4,4,4-trifluoro-1-[4-[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]piperidin-1-yl]butan-1-one
Show/Hide
|
C18H17F6N3O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0523721
|
4,4,4-trifluoro-1-[4-[3-[2-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]piperidin-1-yl]butan-1-one
Show/Hide
|
C18H17F6N3O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0533605
|
4,4,4-trifluoro-1-[4-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]butan-1-one
Show/Hide
|
C18H20F3N3O3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0533606
|
4,4,4-trifluoro-1-[4-[3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]butan-1-one
Show/Hide
|
C18H20F3N3O3
|
1
|
| 1 |
EC50 = 10000 nM
|
|
|
|
CP0533607
|
4,4,4-trifluoro-1-[4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]butan-1-one
Show/Hide
|
C18H20F3N3O3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0248881
|
2-(2-methylphenoxy)-N-[2-(4-methylphenyl)benzotriazol-5-yl]acetamide
Show/Hide
|
C22H20N4O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0339513
|
N-[4-(1,3-benzothiazol-2-yl)phenyl]-2-(3-methoxyphenyl)sulfanylacetamide
Show/Hide
|
C22H18N2O2S2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0523720
|
4,4,4-trifluoro-1-[4-(3-pyrazin-2-yl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]butan-1-one
Show/Hide
|
C15H16F3N5O2
|
1
|
| 1 |
EC50 = 20000 nM
|
|
|
|
CP0392834
|
4,4,4-trifluoro-1-[4-(5-phenyl-1,3,4-oxadiazol-2-yl)piperidin-1-yl]butan-1-one
Show/Hide
|
C17H18F3N3O2
|
1
|
| 1 |
EC50 > 5000 nM
|
|
|
|
CP0456764
|
4,4,4-trifluoro-1-[4-(3-thiophen-2-yl-1H-pyrazol-5-yl)piperidin-1-yl]butan-1-one
Show/Hide
|
C16H18F3N3OS
|
1
|
| 1 |
EC50 > 5000 nM
|
|
|
|
CP0854333
|
3-Phenyl-1-[1-(4,4,4-trifluorobutanoyl)piperidin-4-yl]-4,5-dihydro-1H-pyrazol-5-one
Show/Hide
|
C18H20F3N3O2
|
1
|
| 1 |
EC50 > 5000 nM
|
|
|
