| Compound ID |
Compound Name |
Compound Formula |
|
CP0087426
|
21-methyl-3,13,21-triazapentacyclo[11.8.0.02,10.04,9.015,20]henicosa-2(10),4,6,8,15,17,19-heptaen-14-one
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|
C19H17N3O
|
1
|
| 1 |
EC50 > 20000 nM
|
|
|
|
CP0955774
|
(S)-4-Methoxy-14-methyl-7,8,13b,14-tetrahydroindolo-[2',3':3,4]pyrido[2,1-b]quinazolin-5(13H)-one
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|
C20H19N3O2
|
1
|
| 1 |
EC50 > 20000 nM
|
|
|
|
CP0959864
|
4-Methoxyevodiamine
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|
C20H19N3O2
|
1
|
| 1 |
EC50 > 20000 nM
|
|
|
|
CP0385143
|
2-[4-[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenoxy]piperidin-1-yl]-N-hydroxypyrimidine-5-carboxamide
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|
C26H30N8O5
|
1
|
| 1 |
IC50 = 0.13 nM
|
|
|
|
CP0411277
|
(3S)-3-(5-ethylthiophen-2-yl)-2-(5-pyridin-2-ylpyrimidin-2-yl)-3,4-dihydro-1H-pyrrolo[3,4-b]quinolin-9-one
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|
C26H21N5OS
|
1
|
| 1 |
IC50 = 1.2 nM
|
|
|
|
CP0391810
|
(3S)-3-(5-ethylfuran-2-yl)-2-(5-pyridin-2-ylpyrimidin-2-yl)-3,4-dihydro-1H-pyrrolo[3,4-b]quinolin-9-one
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|
C26H21N5O2
|
1
|
| 1 |
IC50 = 1.5 nM
|
|
|
|
CP0175962
|
3-(5-ethylfuran-2-yl)-2-(5-pyridin-2-ylpyrimidin-2-yl)-3,4-dihydro-1H-pyrrolo[3,4-b]quinolin-9-one
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|
C26H21N5O2
|
1
|
| 1 |
IC50 = 2.3 nM
|
|
|
|
CP0007669
|
3-[[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]-N-hydroxycyclobutane-1-carboxamide
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|
C22H27N5O4
|
1
|
| 1 |
IC50 = 2.6 nM
|
|
|
|
CP0457227
|
3-(5-ethylthiophen-2-yl)-2-pyrimidin-2-yl-3,4-dihydro-1H-pyrrolo[3,4-b]quinolin-9-one
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|
C21H18N4OS
|
1
|
| 1 |
IC50 = 3.7 nM
|
|
|
|
CP0383136
|
(3R)-3-(5-ethylfuran-2-yl)-2-(5-pyridin-2-ylpyrimidin-2-yl)-3,4-dihydro-1H-pyrrolo[3,4-b]quinolin-9-one
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|
C26H21N5O2
|
1
|
| 1 |
IC50 = 3.8 nM
|
|
|
|
CP0117113
|
3-(5-ethylthiophen-2-yl)-2-(5-pyridin-2-ylpyrimidin-2-yl)-3,4-dihydro-1H-pyrrolo[3,4-b]quinolin-9-one
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|
C26H21N5OS
|
1
|
| 1 |
IC50 = 4.8 nM
|
|
|
|
CP0383137
|
3-(5-ethylfuran-2-yl)-2-pyrimidin-2-yl-3,4-dihydro-1H-pyrrolo[3,4-b]quinolin-9-one
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|
C21H18N4O2
|
1
|
| 1 |
IC50 = 6.2 nM
|
|
|
|
CP0392075
|
(10R,15R)-13-ethyl-10-(5-ethylfuran-2-yl)-8,11,13-triazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(9),2,4,6-tetraene-12,14-dione
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|
C21H21N3O3
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0440103
|
(10S,15S)-13-ethyl-10-(3-methylthiophen-2-yl)-8,11,13-triazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(9),2,4,6-tetraene-12,14-dione
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|
C20H19N3O2S
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0384486
|
N-[3-(4,5-diethyl-6-oxo-1H-pyrimidin-2-yl)-4-propoxyphenyl]-2-(4-methylpiperazin-1-yl)acetamide
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|
C24H35N5O3
|
1
|
| 1 |
IC50 = 19.8 nM
|
|
|
|
CP0411276
|
(3R)-3-(5-ethylthiophen-2-yl)-2-(5-pyridin-2-ylpyrimidin-2-yl)-3,4-dihydro-1H-pyrrolo[3,4-b]quinolin-9-one
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|
C26H21N5OS
|
1
|
| 1 |
IC50 = 34.1 nM
|
|
|
|
CP0010658
|
5-[2-ethoxy-5-(4-methyl-1-piperazinylsulfonyl)phenyl]-1-methyl-3-n-propyl-1,6-dihydro-7H-pyrazolo[4,3-d]pyrimidin-7-one
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|
C22H30N6O4S
|
1
|
| 1 |
IC50 = 36.42 nM
|
|
|
|
CP0157969
|
(10S,15S)-13-ethyl-10-(5-ethylthiophen-2-yl)-8,11,13-triazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(9),2,4,6-tetraene-12,14-dione
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|
C21H21N3O2S
|
1
|
| 1 |
IC50 = 56 nM
|
|
|
|
CP0157968
|
(10S,15S)-13-ethyl-10-(5-methylfuran-2-yl)-8,11,13-triazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(9),2,4,6-tetraene-12,14-dione
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|
C20H19N3O3
|
1
|
| 1 |
IC50 = 62 nM
|
|
|
|
CP0392073
|
(10S,15S)-13-butyl-10-(5-ethylthiophen-2-yl)-8,11,13-triazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(9),2,4,6-tetraene-12,14-dione
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|
C23H25N3O2S
|
1
|
| 1 |
IC50 = 107 nM
|
|
|
|
CP0257911
|
(10S,15S)-13-ethyl-10-(5-ethylfuran-2-yl)-8,11,13-triazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(9),2,4,6-tetraene-12,14-dione
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|
C21H21N3O3
|
1
|
| 1 |
IC50 = 127 nM
|
|
|
|
CP0109248
|
(2S,8R)-2-(5-bromothiophen-2-yl)-6-methyl-3,6,17-triazatetracyclo[8.7.0.03,8.011,16]heptadeca-1(10),11,13,15-tetraene-4,7-dione
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|
C19H16BrN3O2S
|
1
|
| 1 |
IC50 = 136 nM
|
|
|
|
CP0392076
|
2-[5-(3,4-dimethoxyphenyl)pyrimidin-2-yl]-1-(5-ethylthiophen-2-yl)-3,9-dihydro-1H-pyrido[3,4-b]indol-4-one
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|
C29H26N4O3S
|
1
|
| 1 |
IC50 = 253 nM
|
|
|
|
CP0438006
|
2-[5-(3,4-dimethoxyphenyl)pyrimidin-2-yl]-1-(5-ethylfuran-2-yl)-3,9-dihydro-1H-pyrido[3,4-b]indol-4-one
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|
C29H26N4O4
|
1
|
| 1 |
IC50 = 288 nM
|
|
|
|
CP0000847
|
(2R,8R)-2-(2H-1,3-benzodioxol-5-yl)-6-methyl-3,6,17-triazatetracyclo[8.7.0.0^{3,8}.0^{11,16}]heptadeca-1(10),11(16),12,14-tetraene-4,7-dione
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|
C22H19N3O4
|
2
|
| 1 |
IC50 = 402 nM
|
|
|
| 2 |
IC50 > 10000 nM
|
|
|
|
CP0176508
|
[4-[3-(3-fluoro-4-methoxyphenyl)-5-(2-methylphenyl)-3,4-dihydropyrazol-2-yl]phenyl]-(4-methylpiperazin-1-yl)methanone
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|
C29H31FN4O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0365459
|
[4-[5-tert-butyl-3-(3,5-difluoro-4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]phenyl]-(4-methylpiperazin-1-yl)methanone
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|
C26H32F2N4O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0419692
|
N-(2-hydroxyethyl)-4-[3-(4-methoxyphenyl)-5-(2-methylphenyl)-3,4-dihydropyrazol-2-yl]benzamide
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|
C26H27N3O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0419693
|
[4-[5-tert-butyl-3-(2,3-difluoro-4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]phenyl]-(4-methylpiperazin-1-yl)methanone
Show/Hide
|
C26H32F2N4O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0444327
|
[4-[3-(4-methoxyphenyl)-5-(2-methylphenyl)-3,4-dihydropyrazol-2-yl]phenyl]-(4-methylpiperazin-1-yl)methanone
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|
C29H32N4O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0833740
|
(S)-4,9-Dimethoxy-14-methyl-7,8,13b,14-tetrahydroindolo-[2',3':3,4]pyrido[2,1-b]quinazolin-5(13H)-one
Show/Hide
|
C21H21N3O3
|
1
|
| 1 |
IC50 > 40000 nM
|
|
|
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CP0109250
|
(2S,8R)-6-methyl-2-(5-methylthiophen-2-yl)-3,6,17-triazatetracyclo[8.7.0.03,8.011,16]heptadeca-1(10),11,13,15-tetraene-4,7-dione
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|
C20H19N3O2S
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
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CP0144390
|
(2S,8R)-2-(5-ethylfuran-2-yl)-6-methyl-3,6,17-triazatetracyclo[8.7.0.03,8.011,16]heptadeca-1(10),11,13,15-tetraene-4,7-dione
Show/Hide
|
C21H21N3O3
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
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CP0164472
|
(10S,15R)-13-ethyl-10-(5-ethylthiophen-2-yl)-8,11,13-triazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(9),2,4,6-tetraene-12,14-dione
Show/Hide
|
C21H21N3O2S
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
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CP0168902
|
(10S,15R)-13-ethyl-10-(5-ethylfuran-2-yl)-8,11,13-triazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(9),2,4,6-tetraene-12,14-dione
Show/Hide
|
C21H21N3O3
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
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CP0268684
|
(2S,8R)-2-(5-ethylthiophen-2-yl)-6-methyl-3,6,17-triazatetracyclo[8.7.0.03,8.011,16]heptadeca-1(10),11,13,15-tetraene-4,7-dione
Show/Hide
|
C21H21N3O2S
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
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CP0392491
|
(2R,8S)-2-(5-ethylthiophen-2-yl)-6-methyl-3,6,17-triazatetracyclo[8.7.0.03,8.011,16]heptadeca-1(10),11,13,15-tetraene-4,7-dione
Show/Hide
|
C21H21N3O2S
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
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CP0432292
|
(10S,15R)-13-butyl-10-(5-ethylthiophen-2-yl)-8,11,13-triazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(9),2,4,6-tetraene-12,14-dione
Show/Hide
|
C23H25N3O2S
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
