Compound ID |
Compound Name |
Compound Formula |
CP0076794
|
US10028961, Compound 101
Show/Hide
|
C14H13ClF6N6
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0233887
|
US10028961, Compound 160
Show/Hide
|
C20H22F7N7
|
3
|
1 |
IC50 = 50 nM
|
|
|
2 |
IC50 < 50 nM
|
|
|
3 |
IC50 = 100 nM
|
|
|
CP0387391
|
US10028961, Compound 158
Show/Hide
|
C20H15F8N7
|
3
|
1 |
IC50 = 50 nM
|
|
|
2 |
IC50 < 50 nM
|
|
|
3 |
IC50 = 100 nM
|
|
|
CP0393570
|
US10946023, Compound 168
Show/Hide
|
C22H17F5N8
|
2
|
1 |
IC50 < 50 nM
|
|
|
2 |
IC50 = 50 nM
|
|
|
CP0394782
|
US10028961, Compound 410
Show/Hide
|
C18H18F7N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0401744
|
US10028961, Compound 133
Show/Hide
|
C23H19F5N8
|
3
|
1 |
IC50 = 50 nM
|
|
|
2 |
IC50 < 50 nM
|
|
|
3 |
IC50 = 100 nM
|
|
|
CP0401756
|
US10946023, Compound 174
Show/Hide
|
C21H18F5N9
|
2
|
1 |
IC50 < 50 nM
|
|
|
2 |
IC50 = 50 nM
|
|
|
CP0412011
|
US10028961, Compound 389
Show/Hide
|
C20H16F8N8
|
3
|
1 |
IC50 = 50 nM
|
|
|
2 |
IC50 < 50 nM
|
|
|
3 |
IC50 = 100 nM
|
|
|
CP0412014
|
US10028961, Compound 161
Show/Hide
|
C16H14F7N7
|
2
|
1 |
IC50 < 50 nM
|
|
|
2 |
IC50 = 50 nM
|
|
|
CP0412024
|
US10028961, Compound 401
Show/Hide
|
C21H16F5N9
|
2
|
1 |
IC50 < 50 nM
|
|
|
2 |
IC50 = 100 nM
|
|
|
CP0412025
|
US10028961, Compound 137
Show/Hide
|
C23H19F5N8
|
2
|
1 |
IC50 < 50 nM
|
|
|
2 |
IC50 = 100 nM
|
|
|
CP0429242
|
US10028961, Compound 393
Show/Hide
|
C18H14F8N8
|
3
|
1 |
IC50 = 50 nM
|
|
|
2 |
IC50 < 50 nM
|
|
|
3 |
IC50 = 100 nM
|
|
|
CP0429886
|
US10028961, Compound 391
Show/Hide
|
C19H14F8N8
|
3
|
1 |
IC50 = 50 nM
|
|
|
2 |
IC50 < 50 nM
|
|
|
3 |
IC50 = 100 nM
|
|
|
CP0450645
|
US10028961, Compound 414
Show/Hide
|
C20H24F3N5
|
3
|
1 |
IC50 = 50 nM
|
|
|
2 |
IC50 < 50 nM
|
|
|
3 |
IC50 = 100 nM
|
|
|
CP0450659
|
US10028961, Compound 106
Show/Hide
|
C17H12F7N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0450660
|
US10028961, Compound 350
Show/Hide
|
C21H18F5N9
|
2
|
1 |
IC50 < 50 nM
|
|
|
2 |
IC50 = 50 nM
|
|
|
CP0387382
|
US10028961, Compound 129
Show/Hide
|
C17H18ClF4N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0387386
|
US10028961, Compound 109
Show/Hide
|
C18H14ClF4N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0387394
|
US10028961, Compound 230
Show/Hide
|
C24H22F6N6
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0387418
|
US10028961, Compound 184
Show/Hide
|
C25H25F5N6
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0387419
|
US10028961, Compound 188
Show/Hide
|
C22H20F5N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0387420
|
US10028961, Compound 227
Show/Hide
|
C22H22F5N9
|
3
|
1 |
IC50 < 50 nM
|
|
|
2 |
IC50 = 50 nM
|
|
|
3 |
IC50 = 100 nM
|
|
|
CP0393560
|
US10028961, Compound 86
Show/Hide
|
C17H21FN6O
|
2
|
1 |
IC50 = 50 nM
|
|
|
2 |
IC50 >= 1000 nM
|
|
|
CP0394783
|
US10028961, Compound 222
Show/Hide
|
C23H23F5N8
|
3
|
1 |
IC50 < 50 nM
|
|
|
2 |
IC50 = 50 nM
|
|
|
3 |
IC50 = 100 nM
|
|
|
CP0401745
|
US10028961, Compound 139
Show/Hide
|
C19H14F6N6
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0401748
|
US10028961, Compound 148
Show/Hide
|
C17H17F7N6S
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0401752
|
US10028961, Compound 166
Show/Hide
|
C24H23F5N6O
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0401759
|
US10946023, Compound 189
Show/Hide
|
C24H21F5N8
|
2
|
1 |
IC50 < 50 nM
|
|
|
2 |
IC50 = 100 nM
|
|
|
CP0401762
|
US10028961, Compound 208
Show/Hide
|
C24H23F5N6
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0401764
|
US10028961, Compound 218
Show/Hide
|
C22H26F6N6
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0401765
|
US10028961, Compound 223
Show/Hide
|
C19H21F7N6S
|
3
|
1 |
IC50 < 50 nM
|
|
|
2 |
IC50 = 50 nM
|
|
|
3 |
IC50 = 100 nM
|
|
|
CP0401768
|
US10028961, Compound 252
Show/Hide
|
C19H19F7N6O
|
3
|
1 |
IC50 = 50 nM
|
|
|
2 |
IC50 = 100 nM
|
|
|
3 |
IC50 >= 1000 nM
|
|
|
CP0401786
|
US10028961, Compound 253
Show/Hide
|
C19H15F5N8
|
2
|
1 |
IC50 = 50 nM
|
|
|
2 |
IC50 = 100 nM
|
|
|
CP0412020
|
US10946023, Compound 226
Show/Hide
|
C20H14F6N8
|
3
|
1 |
IC50 < 50 nM
|
|
|
2 |
IC50 = 50 nM
|
|
|
3 |
IC50 = 100 nM
|
|
|
CP0412032
|
US10028961, Compound 59
Show/Hide
|
C20H22F5N7O2
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0412033
|
US10028961, Compound 63
Show/Hide
|
C19H25F3N6O2
|
1
|
1 |
IC50 = 50 nM
|
|
|
CP0412689
|
US10028961, Compound 190
Show/Hide
|
C19H13F8N7
|
3
|
1 |
IC50 < 50 nM
|
|
|
2 |
IC50 = 100 nM
|
|
|
3 |
IC50 >= 1000 nM
|
|
|
CP0446178
|
US10028961, Compound 114
Show/Hide
|
C13H11F9N6S
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0446197
|
US10028961, Compound 231
Show/Hide
|
C21H19F5N8
|
3
|
1 |
IC50 < 50 nM
|
|
|
2 |
IC50 = 50 nM
|
|
|
3 |
IC50 = 100 nM
|
|
|
CP0446203
|
US10028961, Compound 228
Show/Hide
|
C22H23F7N6
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0446216
|
US10028961, Compound 198
Show/Hide
|
C19H24F2N6
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0446217
|
US10946023, Compound 229
Show/Hide
|
C25H21F5N8
|
3
|
1 |
IC50 < 50 nM
|
|
|
2 |
IC50 = 50 nM
|
|
|
3 |
IC50 = 100 nM
|
|
|
CP0450639
|
US10028961, Compound 20
Show/Hide
|
C22H23F3N6
|
2
|
1 |
IC50 < 50 nM
|
|
|
2 |
IC50 = 50 nM
|
|
|
CP0457659
|
US10028961, Compound 117
Show/Hide
|
C20H18F3N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0457660
|
US10028961, Compound 150
Show/Hide
|
C23H20F6N6
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0471533
|
US10028961, Compound 28
Show/Hide
|
C22H22F4N6
|
2
|
1 |
IC50 < 50 nM
|
|
|
2 |
IC50 = 50 nM
|
|
|
CP0473729
|
US10028961, Compound 204
Show/Hide
|
C21H17F5N8
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0477112
|
US10028961, Compound 250
Show/Hide
|
C20H17F5N8
|
2
|
1 |
IC50 = 50 nM
|
|
|
2 |
IC50 = 100 nM
|
|
|
CP0484637
|
US10028961, Compound 416
Show/Hide
|
C20H24F3N5
|
3
|
1 |
IC50 < 50 nM
|
|
|
2 |
IC50 = 100 nM
|
|
|
3 |
IC50 >= 1000 nM
|
|
|
CP0513507
|
US10028961, Compound 241
Show/Hide
|
C20H27F3N6O
|
2
|
1 |
IC50 < 50 nM
|
|
|
2 |
IC50 = 100 nM
|
|
|
CP0517753
|
US10028961, Compound 225
Show/Hide
|
C23H20BrF5N6
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0530691
|
US10028961, Compound 219
Show/Hide
|
C24H24F5N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0530692
|
US10028961, Compound 254
Show/Hide
|
C23H19Br2F5N6
|
1
|
1 |
IC50 = 50 nM
|
|
|
CP0539508
|
US10172864, Compound 418
Show/Hide
|
C18H19ClF5N5
|
1
|
1 |
IC50 = 50 nM
|
|
|
CP0539512
|
US10028961, Compound 135
Show/Hide
|
C23H23F3N6
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0558586
|
US10028961, Compound 60
Show/Hide
|
C23H23F3N6
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0558589
|
US10028961, Compound 233
Show/Hide
|
C19H25F3N6O
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0559099
|
US10028961, Compound 36
Show/Hide
|
C21H23F3N6
|
2
|
1 |
IC50 < 50 nM
|
|
|
2 |
IC50 = 50 nM
|
|
|
CP0561693
|
US10028961, Compound 240
Show/Hide
|
C20H26N6
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0571860
|
US10028961, Compound 206
Show/Hide
|
C23H25F3N6
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0575456
|
US10028961, Compound 64
Show/Hide
|
C19H24ClN5
|
1
|
1 |
IC50 = 50 nM
|
|
|
CP0851745
|
2-(4-(3,5-difluorophenylamino)-6-(3-(trifluoromethyl)-1H-pyrazol-1-yl)-1,3,5-triazin-2-ylamino)-1,1-difluoroethanol
Show/Hide
|
C15H10F7N7O
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0859577
|
(R)-N2-(1-cyclopropylethyl)-N4-(4,4-dimethylcyclohexyl)-6-(6-(trifluoromethyl)pyridin-2-yl)-1,3,5-triazine-2,4-diamine
Show/Hide
|
C22H29F3N6
|
2
|
1 |
IC50 < 50 nM
|
|
|
2 |
IC50 = 50 nM
|
|
|
CP0393543
|
US10028961, Compound 125
Show/Hide
|
C21H17F7N6
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0401850
|
US10028961, Compound 261
Show/Hide
|
C22H18F5N9
|
3
|
1 |
IC50 = 50 nM
|
|
|
2 |
IC50 = 100 nM
|
|
|
3 |
IC50 >= 1000 nM
|
|
|
CP0450675
|
US10028961, Compound 256
Show/Hide
|
C16H14F7N7
|
3
|
1 |
IC50 = 50 nM
|
|
|
2 |
IC50 = 100 nM
|
|
|
3 |
IC50 >= 1000 nM
|
|
|
CP0457662
|
US10028961, Compound 268
Show/Hide
|
C18H22F3N7
|
3
|
1 |
IC50 < 50 nM
|
|
|
2 |
IC50 = 100 nM
|
|
|
3 |
IC50 >= 1000 nM
|
|
|
CP0548469
|
US10028961, Compound 58
Show/Hide
|
C21H23F5N6
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0387380
|
US10028961, Compound 404
Show/Hide
|
C13H11F9N6S
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0387396
|
US10028961, Compound 372
Show/Hide
|
C23H20F4N8
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0387397
|
US10028961, Compound 378
Show/Hide
|
C22H18F5N9
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0387398
|
US10028961, Compound 386
Show/Hide
|
C14H12F9N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0394779
|
US10946023, Compound 392
Show/Hide
|
C19H15F6N9
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0394780
|
US10028961, Compound 402
Show/Hide
|
C17H18F6N6S
|
1
|
1 |
IC50 = 50 nM
|
|
|
CP0401864
|
US10028961, Compound 344
Show/Hide
|
C14H12F9N7
|
1
|
1 |
IC50 = 50 nM
|
|
|
CP0401865
|
US10028961, Compound 355
Show/Hide
|
C21H18F7N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0405662
|
US10028961, Compound 370
Show/Hide
|
C19H21F6N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0405664
|
US10028961, Compound 409
Show/Hide
|
C16H15F6N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0405670
|
US10028961, Compound 349
Show/Hide
|
C19H15F6N9
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0405696
|
US10028961, Compound 390
Show/Hide
|
C18H12F8N8
|
1
|
1 |
IC50 = 50 nM
|
|
|
CP0405697
|
US10946023, Compound 394
Show/Hide
|
C23H20F5N9
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0412023
|
US10028961, Compound 400
Show/Hide
|
C16H11F9N8
|
2
|
1 |
IC50 < 50 nM
|
|
|
2 |
IC50 = 100 nM
|
|
|
CP0412686
|
US10028961, Compound 360
Show/Hide
|
C21H18F7N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0429884
|
US10028961, Compound 338
Show/Hide
|
C23H21F4N9
|
1
|
1 |
IC50 = 50 nM
|
|
|
CP0446210
|
US10028961, Compound 356
Show/Hide
|
C16H11F9N8
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0446221
|
US10028961, Compound 354
Show/Hide
|
C17H15F7N6
|
1
|
1 |
IC50 = 50 nM
|
|
|
CP0446222
|
US10028961, Compound 357
Show/Hide
|
C20H24F6N6S
|
1
|
1 |
IC50 = 50 nM
|
|
|
CP0446223
|
US10028961, Compound 381
Show/Hide
|
C18H14F5N9
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0446224
|
US10028961, Compound 384
Show/Hide
|
C24H22F4N8
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0450646
|
US10028961, Compound 352
Show/Hide
|
C21H16F6N8
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0450647
|
US10028961, Compound 365
Show/Hide
|
C19H13F8N7
|
1
|
1 |
IC50 = 50 nM
|
|
|
CP0450650
|
US10028961, Compound 403
Show/Hide
|
C15H14F6N6S
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0450962
|
US10028961, Compound 377
Show/Hide
|
C20H15F6N9
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0457665
|
US10028961, Compound 363
Show/Hide
|
C15H16F9N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0457666
|
US10028961, Compound 405
Show/Hide
|
C20H15F8N7
|
1
|
1 |
IC50 = 50 nM
|
|
|
CP0466620
|
US10028961, Compound 351
Show/Hide
|
C21H16F6N8
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0466622
|
US10028961, Compound 366
Show/Hide
|
C17H17F6N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0466623
|
US10028961, Compound 374
Show/Hide
|
C21H25F6N7
|
1
|
1 |
IC50 = 50 nM
|
|
|
CP0471768
|
US10028961, Compound 361
Show/Hide
|
C22H20F7N7
|
1
|
1 |
IC50 = 50 nM
|
|
|
CP0471769
|
US10028961, Compound 369
Show/Hide
|
C19H14F7N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0471770
|
US10946023, Compound 373
Show/Hide
|
C22H18F5N9
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0473720
|
US10028961, Compound 399
Show/Hide
|
C18H18F7N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0473721
|
US10028961, Compound 408
Show/Hide
|
C18H19F6N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0473724
|
US10028961, Compound 358
Show/Hide
|
C20H16F7N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0473725
|
US10028961, Compound 359
Show/Hide
|
C23H17F6N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0473726
|
US10028961, Compound 367
Show/Hide
|
C20H16F7N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0473731
|
US10028961, Compound 335
Show/Hide
|
C15H13F9N6
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0473733
|
US10028961, Compound 395
Show/Hide
|
C20H21F7N6
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0476928
|
US10028961, Compound 362
Show/Hide
|
C22H17F5N8
|
1
|
1 |
IC50 = 50 nM
|
|
|
CP0477102
|
US10028961, Compound 347
Show/Hide
|
C22H19F5N8
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0477103
|
US10028961, Compound 348
Show/Hide
|
C22H19F5N8
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0477105
|
US10028961, Compound 364
Show/Hide
|
C23H16ClF6N7
|
1
|
1 |
IC50 = 50 nM
|
|
|
CP0477106
|
US10028961, Compound 379
Show/Hide
|
C17H13F6N7S
|
1
|
1 |
IC50 = 50 nM
|
|
|
CP0477120
|
US10028961, Compound 337
Show/Hide
|
C20H16F5N9
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0477121
|
US10028961, Compound 345
Show/Hide
|
C16H16F9N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0477122
|
US10028961, Compound 353
Show/Hide
|
C18H13F8N7S
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0477123
|
US10028961, Compound 388
Show/Hide
|
C17H11F8N7S
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0477124
|
US10028961, Compound 406
Show/Hide
|
C18H18F7N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0484674
|
US10028961, Compound 346
Show/Hide
|
C17H17F9N6
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0484687
|
US10028961, Compound 385
Show/Hide
|
C24H20F5N9
|
1
|
1 |
IC50 = 50 nM
|
|
|
CP0513506
|
US10028961, Compound 339
Show/Hide
|
C16H16F9N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0533991
|
US10028961, Compound 336
Show/Hide
|
C20H16F5N9
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0539510
|
US10028961, Compound 371
Show/Hide
|
C23H16F7N7
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0387400
|
US10028961, Compound 298
Show/Hide
|
C18H17F5N8
|
2
|
1 |
IC50 = 100 nM
|
|
|
2 |
IC50 >= 1000 nM
|
|
|
CP0394778
|
US10028961, Compound 280
Show/Hide
|
C25H26F5N7
|
2
|
1 |
IC50 = 100 nM
|
|
|
2 |
IC50 >= 1000 nM
|
|
|
CP0401769
|
US10028961, Compound 259
Show/Hide
|
C22H21F3N8O
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0401772
|
US10028961, Compound 296
Show/Hide
|
C21H23F7N6O
|
2
|
1 |
IC50 = 100 nM
|
|
|
2 |
IC50 >= 1000 nM
|
|
|
CP0401774
|
US10028961, Compound 299
Show/Hide
|
C29H25F5N6
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0401852
|
US10028961, Compound 289
Show/Hide
|
C19H19F5N8
|
2
|
1 |
IC50 = 100 nM
|
|
|
2 |
IC50 >= 1000 nM
|
|
|
CP0446207
|
US10028961, Compound 288
Show/Hide
|
C19H17F3N8O
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0446220
|
US10028961, Compound 285
Show/Hide
|
C18H25N7
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0450708
|
US10028961, Compound 290
Show/Hide
|
C18H23ClN6O2
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0458085
|
US10028961, Compound 258
Show/Hide
|
C21H24F4N6
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0471467
|
US10028961, Compound 286
Show/Hide
|
C18H21F3N6O2
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0471510
|
US10028961, Compound 300
Show/Hide
|
C19H23F3N6
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0476931
|
US10028961, Compound 269
Show/Hide
|
C19H23N7
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0477100
|
US10028961, Compound 278
Show/Hide
|
C18H23ClN6
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0477113
|
US10028961, Compound 277
Show/Hide
|
C17H15F7N6O
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0481781
|
US10028961, Compound 301
Show/Hide
|
C15H16F4N6O
|
2
|
1 |
IC50 = 100 nM
|
|
|
2 |
IC50 >= 1000 nM
|
|
|
CP0541045
|
US10028961, Compound 282
Show/Hide
|
C21H26F4N6
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0558592
|
US10028961, Compound 284
Show/Hide
|
C17H17F3N6
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0559095
|
US10028961, Compound 294
Show/Hide
|
C19H26N6O
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0559574
|
US10028961, Compound 292
Show/Hide
|
C19H23F2N5
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0575446
|
US10028961, Compound 281
Show/Hide
|
C17H21F3N6O
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0575447
|
US10028961, Compound 295
Show/Hide
|
C20H27F3N6O2
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0859551
|
N2-(3,3-difluorocyclopentyl)-N4-(1H-indol-2-yl)-6-(6-(trifluoromethyl)pyridin-2-yl)-1,3,5-triazine-2,4-diamine
Show/Hide
|
C22H18F5N7
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0387390
|
US10028961, Compound 407
Show/Hide
|
C17H14F6N8
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0387408
|
US10946023, Compound 342
Show/Hide
|
C22H18F5N9
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0401867
|
US10028961, Compound 375
Show/Hide
|
C22H18F5N9
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0405663
|
US10028961, Compound 380
Show/Hide
|
C21H16F8N8
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0405665
|
US10028961, Compound 411
Show/Hide
|
C16H15F6N7
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0446209
|
US10946023, Compound 341
Show/Hide
|
C22H18F5N9
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0446212
|
US10028961, Compound 387
Show/Hide
|
C18H14F6N8
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0446225
|
US10028961, Compound 398
Show/Hide
|
C21H20F3N7O
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0473723
|
US10028961, Compound 343
Show/Hide
|
C19H14F8N8
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0477101
|
US10028961, Compound 340
Show/Hide
|
C19H14F8N8
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0477107
|
US10946023, Compound 383
Show/Hide
|
C24H16F6N8
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0517901
|
US10028961, Compound 412
Show/Hide
|
C18H19F6N7
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0534801
|
US10028961, Compound 397
Show/Hide
|
C21H20F6N6O
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0494043
|
US10028961, Compound 420
Show/Hide
|
C20H24F3N5
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0393559
|
US10028961, Compound 66
Show/Hide
|
C19H24ClN5
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0401775
|
US10028961, Compound 303
Show/Hide
|
C19H24F3N7O
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0401776
|
US10028961, Compound 306
Show/Hide
|
C21H28F3N7O
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0401778
|
US10028961, Compound 318
Show/Hide
|
C21H23F7N6
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0401779
|
US10028961, Compound 327
Show/Hide
|
C18H24N6O
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0450676
|
US10028961, Compound 331
Show/Hide
|
C22H30F3N7
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0471468
|
US10028961, Compound 305
Show/Hide
|
C23H28F4N6
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0471469
|
US10028961, Compound 310
Show/Hide
|
C20H26N6O2
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0471470
|
US10028961, Compound 316
Show/Hide
|
C23H20F5N7
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0471511
|
US10028961, Compound 304
Show/Hide
|
C19H25F4N7
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0471513
|
US10028961, Compound 313
Show/Hide
|
C23H21F6N7
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0479118
|
US10028961, Compound 323
Show/Hide
|
C19H23F3N6
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0494045
|
US10028961, Compound 326
Show/Hide
|
C19H22F5N7
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0513527
|
US10028961, Compound 330
Show/Hide
|
C18H23F4N7
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0540896
|
US10028961, Compound 61
Show/Hide
|
C18H24N6
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0553618
|
US10028961, Compound 314
Show/Hide
|
C20H23ClF4N6
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0558593
|
US10028961, Compound 324
Show/Hide
|
C19H24F4N6O
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0559096
|
US10028961, Compound 322
Show/Hide
|
C20H24F3N5O
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0561698
|
US10028961, Compound 312
Show/Hide
|
C17H25N7
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0561736
|
US10028961, Compound 307
Show/Hide
|
C19H25N7O
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0563513
|
US10028961, Compound 320
Show/Hide
|
C20H24N6
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0564642
|
US10028961, Compound 67
Show/Hide
|
C18H24N6
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0575448
|
US10028961, Compound 329
Show/Hide
|
C19H24F4N6O
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0401781
|
US10028961, Compound 57
Show/Hide
|
C18H24N6
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0539506
|
US10028961, Compound 325
Show/Hide
|
C18H16F5N7O
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0552778
|
US10028961, Compound 54
Show/Hide
|
C18H20F5N7
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0446211
|
US10028961, Compound 376
Show/Hide
|
C22H18F5N9
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0471534
|
US10028961, Compound 78
Show/Hide
|
C20H26FN5O
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0450643
|
US10028961, Compound 47
Show/Hide
|
C17H19F3N6O2
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0450644
|
US10028961, Compound 48
Show/Hide
|
C19H24F3N7O
|
1
|
1 |
IC50 >= 1000 nM
|
|
|
CP0513504
|
US10028961, Compound 5
Show/Hide
|
C16H18F3N7O
|
1
|
1 |
IC50 >= 1000 nM
|
|
|