| Compound ID |
Compound Name |
Compound Formula |
|
CP0510803
|
(3S)-3-[[5-(3,3-dimethyl-2-oxobutoxy)-1-(2-fluorophenyl)pyrazole-3-carbonyl]amino]-3-(2-methylphenyl)propanoic acid
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|
C26H28FN3O5
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0193752
|
(3S)-3-[[1-(2-fluorophenyl)-5-[(2R)-2-hydroxy-3,3-dimethylbutoxy]pyrazole-3-carbonyl]amino]-3-(2-methylphenyl)propanoic acid
Show/Hide
|
C26H30FN3O5
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0507599
|
(3S)-3-[[1-(2-fluorophenyl)-5-[(2S)-2-hydroxy-3,3-dimethylbutoxy]pyrazole-3-carbonyl]amino]-3-(2-methylphenyl)propanoic acid
Show/Hide
|
C26H30FN3O5
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0114192
|
(3S)-3-[[5-(cyclopropylmethoxy)-1-(2-fluorophenyl)pyrazole-3-carbonyl]amino]-3-(2-methylphenyl)propanoic acid
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|
C24H24FN3O4
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0252596
|
(3S)-3-[[5-ethoxy-1-(2-fluorophenyl)pyrazole-3-carbonyl]amino]-3-(2-methylphenyl)propanoic acid
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|
C22H22FN3O4
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0507315
|
3-[[2-(2-fluorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-[4-(4-fluorophenyl)phenyl]propanoic acid
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|
C25H19F2N3O4
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0087655
|
(3S)-3-[[1-(2-fluorophenyl)-5-methoxypyrazole-3-carbonyl]amino]-3-(2-methylphenyl)propanoic acid
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|
C21H20FN3O4
|
1
|
| 1 |
IC50 = 26 nM
|
|
|
|
CP0453563
|
(3S)-3-[[4-fluoro-1-(2-fluorophenyl)-5-methoxypyrazole-3-carbonyl]amino]-3-(2-methylphenyl)propanoic acid
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|
C21H19F2N3O4
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0193987
|
(3S)-3-[[2-(2-fluorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-(2-methylphenyl)propanoic acid
Show/Hide
|
C20H18FN3O4
|
1
|
| 1 |
IC50 = 38 nM
|
|
|
|
CP0139037
|
(3S)-3-(2,4-dichlorophenyl)-3-[[1-(2-fluorophenyl)-5-[(2R)-2-hydroxy-3,3-dimethylbutoxy]pyrazole-3-carbonyl]amino]propanoic acid
Show/Hide
|
C25H26Cl2FN3O5
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0493571
|
(3S)-3-[[2-(2-chlorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-(2-methylphenyl)propanoic acid
Show/Hide
|
C20H18ClN3O4
|
1
|
| 1 |
IC50 = 57 nM
|
|
|
|
CP0492156
|
(3S)-3-[[2-(3-fluorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-(2-methylphenyl)propanoic acid
Show/Hide
|
C20H18FN3O4
|
1
|
| 1 |
IC50 = 59 nM
|
|
|
|
CP0445558
|
(3S)-3-(2,4-dichlorophenyl)-3-[[5-(3,3-dimethyl-2-oxobutoxy)-1-(2-fluorophenyl)pyrazole-3-carbonyl]amino]propanoic acid
Show/Hide
|
C25H24Cl2FN3O5
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0513948
|
(3S)-3-(2,4-dichlorophenyl)-3-[[1-(2-fluorophenyl)-5-[(2S)-2-hydroxy-3,3-dimethylbutoxy]pyrazole-3-carbonyl]amino]propanoic acid
Show/Hide
|
C25H26Cl2FN3O5
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0525546
|
(3S)-3-(2-methylphenyl)-3-[(3-oxo-2-phenyl-1H-pyrazole-5-carbonyl)amino]propanoic acid
Show/Hide
|
C20H19N3O4
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0525548
|
3-(5-fluoro-2-methylphenyl)-3-[[2-(2-fluorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]propanoic acid
Show/Hide
|
C20H17F2N3O4
|
1
|
| 1 |
IC50 = 76 nM
|
|
|
|
CP0445560
|
(3S)-3-[[2-(4-fluorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-(2-methylphenyl)propanoic acid
Show/Hide
|
C20H18FN3O4
|
1
|
| 1 |
IC50 = 87 nM
|
|
|
|
CP0248778
|
3-(2,3-dichlorophenyl)-3-[(3-oxo-2-phenyl-1H-pyrazole-5-carbonyl)amino]propanoic acid
Show/Hide
|
C19H15Cl2N3O4
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0397483
|
(3S)-3-[(4-methoxy-1-phenylpyrazole-3-carbonyl)amino]-3-(2-methylphenyl)propanoic acid
Show/Hide
|
C21H21N3O4
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0445559
|
(3S)-3-[[2-(3-chlorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-(2-methylphenyl)propanoic acid
Show/Hide
|
C20H18ClN3O4
|
1
|
| 1 |
IC50 = 102 nM
|
|
|
|
CP0492157
|
(3S)-3-[(4-hydroxy-1-phenylpyrazole-3-carbonyl)amino]-3-(2-methylphenyl)propanoic acid
Show/Hide
|
C20H19N3O4
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0492158
|
(3S)-3-[[4-chloro-1-(2-fluorophenyl)-5-methoxypyrazole-3-carbonyl]amino]-3-(2-methylphenyl)propanoic acid
Show/Hide
|
C21H19ClFN3O4
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0492155
|
3-(2,3-dichlorophenyl)-3-[[2-(2,4-difluorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]propanoic acid
Show/Hide
|
C19H13Cl2F2N3O4
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0397482
|
3-[(3-oxo-2-phenyl-1H-pyrazole-5-carbonyl)amino]-3-(4-phenoxyphenyl)propanoic acid
Show/Hide
|
C25H21N3O5
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0453312
|
3-[[2-(2-fluorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-phenylpropanoic acid
Show/Hide
|
C19H16FN3O4
|
1
|
| 1 |
IC50 = 226 nM
|
|
|
|
CP0513951
|
(3S)-3-[[2-(2-fluorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-(3-methylphenyl)propanoic acid
Show/Hide
|
C20H18FN3O4
|
1
|
| 1 |
IC50 = 252 nM
|
|
|
|
CP0527235
|
(3S)-3-[[2-(2-fluorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-(4-methylphenyl)propanoic acid
Show/Hide
|
C20H18FN3O4
|
1
|
| 1 |
IC50 = 274 nM
|
|
|
|
CP0513950
|
(3S)-3-[[2-(2-fluorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-(2-methoxyphenyl)propanoic acid
Show/Hide
|
C20H18FN3O5
|
1
|
| 1 |
IC50 = 357 nM
|
|
|
|
CP0482385
|
(3S)-3-[[2-(2-fluorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-[2-(trifluoromethyl)phenyl]propanoic acid
Show/Hide
|
C20H15F4N3O4
|
1
|
| 1 |
IC50 = 375 nM
|
|
|
|
CP0525547
|
3-[[2-(2,5-dimethylphenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-(4-phenylphenyl)propanoic acid
Show/Hide
|
C27H25N3O4
|
1
|
| 1 |
IC50 = 803 nM
|
|
|
|
CP0482384
|
3-[[2-(2,5-dimethylphenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-(4-fluorophenyl)propanoic acid
Show/Hide
|
C21H20FN3O4
|
1
|
| 1 |
IC50 = 5380 nM
|
|
|
|
CP0513949
|
(3R)-3-(2-methylphenyl)-3-[(3-oxo-2-phenyl-1H-pyrazole-5-carbonyl)amino]propanoic acid
Show/Hide
|
C20H19N3O4
|
1
|
| 1 |
IC50 = 7800 nM
|
|
|
|
CP0252589
|
3-[[2-(4-chlorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-(2,5-dichlorophenyl)propanoic acid
Show/Hide
|
C19H14Cl3N3O4
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
