| Compound ID |
Compound Name |
Compound Formula |
|
CP0046376
|
PF-2545920
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|
C25H20N4O
|
2
|
| 1 |
IC50 = 0.5012 nM
|
|
|
| 2 |
IC50 = 0.6457 nM
|
|
|
|
CP0880529
|
2-[4-[1-(2-[18F]-fluoroethyl)-4-pyridin-4-yl-1H-pyrazol-3-yl]-phenoxymethyl]-quinoline
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|
C26H21FN4O
|
1
|
| 1 |
IC50 = 0.5012 nM
|
|
|
|
CP0168595
|
2-[[4-[1-(2-fluoroethyl)-4-pyridin-4-ylpyrazol-3-yl]phenoxy]methyl]-3,5-dimethylpyridine
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|
C24H23FN4O
|
1
|
| 1 |
IC50 = 1.585 nM
|
|
|
|
CP0399327
|
2-[[4-[1-(2-fluoroethyl)-4-pyridin-4-ylpyrazol-3-yl]phenoxy]methyl]-6-methylpyridine
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|
C23H21FN4O
|
1
|
| 1 |
IC50 = 2.512 nM
|
|
|
|
CP0105098
|
2-[[4-[1-(2-fluoroethyl)-4-pyridin-4-ylpyrazol-3-yl]phenoxy]methyl]-5-methoxypyridine
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|
C23H21FN4O2
|
1
|
| 1 |
IC50 = 3.162 nM
|
|
|
|
CP0452191
|
2-[[4-[1-(2-fluoroethyl)-4-pyridin-4-ylpyrazol-3-yl]phenoxy]methyl]-6-methoxypyridine
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|
C23H21FN4O2
|
1
|
| 1 |
IC50 = 3.162 nM
|
|
|
|
CP0419876
|
2-[[4-[1-(2-fluoroethyl)-4-pyridin-4-ylpyrazol-3-yl]phenoxy]methyl]-3-methoxypyridine
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|
C23H21FN4O2
|
1
|
| 1 |
IC50 = 3.981 nM
|
|
|
|
CP0500207
|
2-[[4-[1-(2-fluoroethyl)-4-pyridin-4-ylpyrazol-3-yl]phenoxy]methyl]-3,4,5-trimethylpyridine
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|
C25H25FN4O
|
1
|
| 1 |
IC50 = 3.981 nM
|
|
|
|
CP0390230
|
7-methoxy-4-pyridin-3-yl-6-(2-quinolin-2-ylethoxy)quinazoline
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|
C25H20N4O2
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0400548
|
3-methoxy-2-[[4-[4-pyridin-4-yl-1-(2,2,2-trifluoroethyl)pyrazol-3-yl]phenoxy]methyl]pyridine
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|
C23H19F3N4O2
|
1
|
| 1 |
IC50 = 5.012 nM
|
|
|
|
CP0466842
|
5-methoxy-2-[[4-[4-pyridin-4-yl-1-(2,2,2-trifluoroethyl)pyrazol-3-yl]phenoxy]methyl]pyridine
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|
C23H19F3N4O2
|
1
|
| 1 |
IC50 = 5.012 nM
|
|
|
|
CP0046541
|
7-methoxy-6-[3-(1-methylbenzimidazol-2-yl)propoxy]-4-(3-phenylpiperidin-1-yl)quinazoline
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|
C31H33N5O2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0399328
|
2-bromo-6-[[4-[1-(2-fluoroethyl)-4-pyridin-4-ylpyrazol-3-yl]phenoxy]methyl]pyridine
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|
C22H18BrFN4O
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0419877
|
5-bromo-2-[[4-[1-(2-fluoroethyl)-4-pyridin-4-ylpyrazol-3-yl]phenoxy]methyl]pyridine
Show/Hide
|
C22H18BrFN4O
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0503248
|
7-methoxy-4-(3-phenylpiperidin-1-yl)-6-(2-quinolin-2-ylethoxy)quinazoline
Show/Hide
|
C31H30N4O2
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0520746
|
7-methoxy-3-methyl-6-(2-quinolin-2-ylethoxy)quinazolin-4-one
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|
C21H19N3O3
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0391027
|
2-[[4-[1-(3-fluoropropyl)-4-pyridin-4-ylpyrazol-3-yl]phenoxy]methyl]-3-methoxypyridine
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|
C24H23FN4O2
|
1
|
| 1 |
IC50 = 12.59 nM
|
|
|
|
CP0529500
|
7-methoxy-N,N-dimethyl-6-(2-quinolin-2-ylethoxy)quinazolin-4-amine
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|
C22H22N4O2
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0500206
|
3-fluoro-2-[[4-[1-(2-fluoroethyl)-4-pyridin-4-ylpyrazol-3-yl]phenoxy]methyl]pyridine
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|
C22H18F2N4O
|
1
|
| 1 |
IC50 = 15.85 nM
|
|
|
|
CP0506049
|
2-[[4-[1-(3-fluoropropyl)-4-pyridin-4-ylpyrazol-3-yl]phenoxy]methyl]-5-methoxypyridine
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|
C24H23FN4O2
|
1
|
| 1 |
IC50 = 15.85 nM
|
|
|
|
CP0233769
|
6-methoxy-7-(2-quinolin-2-ylethoxy)quinazoline
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|
C20H17N3O2
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0481488
|
1-[[1-(2-chlorophenyl)-4-methyl-[1,2,4]triazolo[4,3-a]quinoxalin-8-yl]methyl]pyrrolidin-3-ol
Show/Hide
|
C21H20ClN5O
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0482193
|
1-(2,6-dichlorophenyl)-N-ethyl-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline-8-carboxamide
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|
C19H15Cl2N5O
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0565855
|
1-(2-chlorophenyl)-N-[2-(diethylamino)ethyl]-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline-8-carboxamide
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|
C23H25ClN6O
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0452189
|
2-[[4-[1-(3-fluoropropyl)-4-pyridin-4-ylpyrazol-3-yl]phenoxy]methyl]-6-methylpyridine
Show/Hide
|
C24H23FN4O
|
1
|
| 1 |
IC50 = 19.95 nM
|
|
|
|
CP0490371
|
2-ethoxy-6-[[4-[1-(2-fluoroethyl)-4-pyridin-4-ylpyrazol-3-yl]phenoxy]methyl]pyridine
Show/Hide
|
C24H23FN4O2
|
1
|
| 1 |
IC50 = 19.95 nM
|
|
|
|
CP0414049
|
N-ethyl-4-methyl-1-pyridin-4-yl-[1,2,4]triazolo[4,3-a]quinoxaline-8-carboxamide
Show/Hide
|
C18H16N6O
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0425611
|
1-(2-chlorophenyl)-4-methyl-N-(pyridin-2-ylmethyl)-[1,2,4]triazolo[4,3-a]quinoxaline-8-carboxamide
Show/Hide
|
C23H17ClN6O
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0453340
|
1-[[1-(2-chlorophenyl)-4-methyl-[1,2,4]triazolo[4,3-a]quinoxalin-8-yl]methyl]piperidin-3-ol
Show/Hide
|
C22H22ClN5O
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0400550
|
6-[[4-[1-(2-fluoroethyl)-4-pyridin-4-ylpyrazol-3-yl]phenoxy]methyl]pyridine-2-carbonitrile
Show/Hide
|
C23H18FN5O
|
1
|
| 1 |
IC50 = 31.62 nM
|
|
|
|
CP0400551
|
3-bromo-2-[[4-[1-(2-fluoroethyl)-4-pyridin-4-ylpyrazol-3-yl]phenoxy]methyl]-6-methoxypyridine
Show/Hide
|
C23H20BrFN4O2
|
1
|
| 1 |
IC50 = 31.62 nM
|
|
|
|
CP0440262
|
2-cyclopropyl-6-[[4-[1-(2-fluoroethyl)-4-pyridin-4-ylpyrazol-3-yl]phenoxy]methyl]pyridine
Show/Hide
|
C25H23FN4O
|
1
|
| 1 |
IC50 = 31.62 nM
|
|
|
|
CP0452190
|
5-cyclopropyl-2-[[4-[1-(2-fluoroethyl)-4-pyridin-4-ylpyrazol-3-yl]phenoxy]methyl]pyridine
Show/Hide
|
C25H23FN4O
|
1
|
| 1 |
IC50 = 31.62 nM
|
|
|
|
CP0414199
|
4-[[1-(2-chlorophenyl)-4-methyl-[1,2,4]triazolo[4,3-a]quinoxalin-8-yl]methyl]morpholine
Show/Hide
|
C21H20ClN5O
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0435545
|
ethyl 1-(2-chlorophenyl)-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline-8-carboxylate
Show/Hide
|
C19H15ClN4O2
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0477195
|
N-ethyl-1-(2-methoxypyridin-3-yl)-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline-8-carboxamide
Show/Hide
|
C19H18N6O2
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0385742
|
1-(2-chlorophenyl)-8-[(4-methoxypiperidin-1-yl)methyl]-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline
Show/Hide
|
C23H24ClN5O
|
1
|
| 1 |
IC50 = 39 nM
|
|
|
|
CP0385743
|
1-(2-chlorophenyl)-4-methyl-N-(2-morpholin-4-ylethyl)-[1,2,4]triazolo[4,3-a]quinoxaline-8-carboxamide
Show/Hide
|
C23H23ClN6O2
|
1
|
| 1 |
IC50 = 39 nM
|
|
|
|
CP0425609
|
N-ethyl-4-methyl-1-pyridin-2-yl-[1,2,4]triazolo[4,3-a]quinoxaline-8-carboxamide
Show/Hide
|
C18H16N6O
|
1
|
| 1 |
IC50 = 39 nM
|
|
|
|
CP0435544
|
N-ethyl-4-methyl-1-pyridin-3-yl-[1,2,4]triazolo[4,3-a]quinoxaline-8-carboxamide
Show/Hide
|
C18H16N6O
|
1
|
| 1 |
IC50 = 39 nM
|
|
|
|
CP0481487
|
1-[[1-(2-chlorophenyl)-4-methyl-[1,2,4]triazolo[4,3-a]quinoxalin-8-yl]methyl]piperidin-4-ol
Show/Hide
|
C22H22ClN5O
|
1
|
| 1 |
IC50 = 39 nM
|
|
|
|
CP0482195
|
1-(2-chlorophenyl)-4-methyl-N-(2-pyrrolidin-1-ylethyl)-[1,2,4]triazolo[4,3-a]quinoxaline-8-carboxamide
Show/Hide
|
C23H23ClN6O
|
1
|
| 1 |
IC50 = 39 nM
|
|
|
|
CP0480454
|
4-[2-methyl-3-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]imidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
|
C16H17F3N6O
|
1
|
| 1 |
IC50 = 46.77 nM
|
|
|
|
CP0425610
|
[1-[[1-(2-chlorophenyl)-4-methyl-[1,2,4]triazolo[4,3-a]quinoxalin-8-yl]methyl]piperidin-3-yl]methanol
Show/Hide
|
C23H24ClN5O
|
1
|
| 1 |
IC50 = 47 nM
|
|
|
|
CP0481490
|
N-ethyl-4-methyl-1-(2-methylpyridin-3-yl)-[1,2,4]triazolo[4,3-a]quinoxaline-8-carboxamide
Show/Hide
|
C19H18N6O
|
1
|
| 1 |
IC50 = 47 nM
|
|
|
|
CP0482192
|
N-[[1-(2-chlorophenyl)-4-methyl-[1,2,4]triazolo[4,3-a]quinoxalin-8-yl]methyl]ethanamine
Show/Hide
|
C19H18ClN5
|
1
|
| 1 |
IC50 = 47 nM
|
|
|
|
CP0385740
|
N-ethyl-4-methyl-1-phenyl-[1,2,4]triazolo[4,3-a]quinoxaline-8-carboxamide
Show/Hide
|
C19H17N5O
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0440871
|
N-[[1-(2-chlorophenyl)-4-methyl-[1,2,4]triazolo[4,3-a]quinoxalin-8-yl]methyl]-1-phenylmethanamine
Show/Hide
|
C24H20ClN5
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0447959
|
N-ethyl-1-(5-methoxypyridin-3-yl)-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline-8-carboxamide
Show/Hide
|
C19H18N6O2
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0433377
|
N-benzyl-1-(2-chlorophenyl)-N,4-dimethyl-[1,2,4]triazolo[4,3-a]quinoxaline-8-carboxamide
Show/Hide
|
C25H20ClN5O
|
1
|
| 1 |
IC50 = 51 nM
|
|
|
|
CP0482191
|
1-(2-chlorophenyl)-4-methyl-N-(oxan-4-yl)-[1,2,4]triazolo[4,3-a]quinoxalin-8-amine
Show/Hide
|
C21H20ClN5O
|
1
|
| 1 |
IC50 = 51 nM
|
|
|
|
CP0482330
|
N-ethyl-1-(2-methoxyphenyl)-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline-8-carboxamide
Show/Hide
|
C20H19N5O2
|
1
|
| 1 |
IC50 = 51 nM
|
|
|
|
CP0381821
|
1-(2-chlorophenyl)-4-methyl-N-(2-phenylethyl)-[1,2,4]triazolo[4,3-a]quinoxaline-8-carboxamide
Show/Hide
|
C25H20ClN5O
|
1
|
| 1 |
IC50 = 52 nM
|
|
|
|
CP0450414
|
N-ethyl-1-(2-fluorophenyl)-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline-8-carboxamide
Show/Hide
|
C19H16FN5O
|
1
|
| 1 |
IC50 = 52 nM
|
|
|
|
CP0481489
|
4-[[1-(2-chlorophenyl)-4-methyl-[1,2,4]triazolo[4,3-a]quinoxalin-8-yl]amino]cyclohexan-1-ol
Show/Hide
|
C22H22ClN5O
|
1
|
| 1 |
IC50 = 52 nM
|
|
|
|
CP0411633
|
4-[2-cyclopropyl-3-[1-(2-methoxyethyl)pyrazol-4-yl]imidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
|
C19H24N6O2
|
1
|
| 1 |
IC50 = 53.7 nM
|
|
|
|
CP0542605
|
(1-methylsulfonylindol-5-yl)-[(3S)-3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]methanone
Show/Hide
|
C20H20N6O3S
|
1
|
| 1 |
IC50 = 54 nM
|
|
|
|
CP0526575
|
4-[3-[1-[(2S)-2-methoxypropyl]pyrazol-4-yl]-2-methylimidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
|
C18H24N6O2
|
1
|
| 1 |
IC50 = 60.26 nM
|
|
|
|
CP0480453
|
4-[3-[1-(cyclopropylmethyl)pyrazol-4-yl]-2-methylimidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
|
C18H22N6O
|
1
|
| 1 |
IC50 = 64.57 nM
|
|
|
|
CP0411635
|
4-[3-[1-(2-methoxy-2-methylpropyl)pyrazol-4-yl]-2-methylimidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
|
C19H26N6O2
|
1
|
| 1 |
IC50 = 66.07 nM
|
|
|
|
CP0425613
|
N-benzyl-1-(2-chlorophenyl)-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline-8-carboxamide
Show/Hide
|
C24H18ClN5O
|
1
|
| 1 |
IC50 = 74 nM
|
|
|
|
CP0450415
|
1-(2-chlorophenyl)-N-ethyl-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline-8-carboxamide
Show/Hide
|
C19H16ClN5O
|
1
|
| 1 |
IC50 = 74 nM
|
|
|
|
CP0450478
|
1-(2-chlorophenyl)-4-methyl-8-[(4-methylpiperazin-1-yl)methyl]-[1,2,4]triazolo[4,3-a]quinoxaline
Show/Hide
|
C22H23ClN6
|
1
|
| 1 |
IC50 = 74 nM
|
|
|
|
CP0490370
|
6-[[4-[1-(2-fluoroethyl)-4-pyridin-4-ylpyrazol-3-yl]phenoxy]methyl]pyridine-3-carbonitrile
Show/Hide
|
C23H18FN5O
|
1
|
| 1 |
IC50 = 79.43 nM
|
|
|
|
CP0382733
|
3-[1-(2-methoxyethyl)pyrazol-4-yl]-8-morpholin-4-ylimidazo[1,2-a]pyrazine-2-carbonitrile
Show/Hide
|
C17H19N7O2
|
1
|
| 1 |
IC50 = 85.11 nM
|
|
|
|
CP0481902
|
4-[2-cyclopropyl-3-[6-(2-methoxyethyl)pyridin-3-yl]imidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
|
C21H25N5O2
|
1
|
| 1 |
IC50 = 97.72 nM
|
|
|
|
CP0400549
|
2-[[4-[1-(2-fluoroethyl)-4-pyridin-4-ylpyrazol-3-yl]phenoxy]methyl]-5-(trifluoromethyl)pyridine
Show/Hide
|
C23H18F4N4O
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0517900
|
2-[[4-[1-(2-fluoroethyl)-4-pyridin-4-ylpyrazol-3-yl]phenoxy]methyl]-6-(trifluoromethyl)pyridine
Show/Hide
|
C23H18F4N4O
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0535017
|
[3-(2,5-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]-(4,5,6,7-tetrahydro-1-benzothiophen-2-yl)methanone
Show/Hide
|
C21H25N5OS
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0535019
|
1-[5-[3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidine-1-carbonyl]indol-1-yl]ethanone
Show/Hide
|
C21H20N6O2
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0549711
|
4-[2-methyl-3-[1-(pyridin-4-ylmethyl)pyrazol-4-yl]imidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
|
C20H21N7O
|
1
|
| 1 |
IC50 = 102.33 nM
|
|
|
|
CP0511167
|
4-[2-methyl-3-[2-(2-methylpropyl)-1,3-thiazol-5-yl]imidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
|
C18H23N5OS
|
1
|
| 1 |
IC50 = 104.71 nM
|
|
|
|
CP0398225
|
4-[[1-(2-chloro-5-methoxyphenyl)-4-methyl-[1,2,4]triazolo[4,3-a]quinoxalin-8-yl]methyl]morpholine
Show/Hide
|
C22H22ClN5O2
|
1
|
| 1 |
IC50 = 106 nM
|
|
|
|
CP0498444
|
(1-methylsulfonylindol-5-yl)-[3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]methanone
Show/Hide
|
C20H20N6O3S
|
1
|
| 1 |
IC50 = 107 nM
|
|
|
|
CP0435370
|
4-[3-[1-(2-fluoroethyl)pyrazol-4-yl]-2-methylimidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
|
C16H19FN6O
|
1
|
| 1 |
IC50 = 112.2 nM
|
|
|
|
CP0556577
|
4-[2-methyl-3-(1-propan-2-ylpyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
|
C17H22N6O
|
1
|
| 1 |
IC50 = 112.2 nM
|
|
|
|
CP0409221
|
N-ethyl-4-methyl-1-(4-methylpyridin-3-yl)-[1,2,4]triazolo[4,3-a]quinoxaline-8-carboxamide
Show/Hide
|
C19H18N6O
|
1
|
| 1 |
IC50 = 113 nM
|
|
|
|
CP0538446
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1-[1-(2-chlorophenyl)-4-methyl-[1,2,4]triazolo[4,3-a]quinoxalin-8-yl]-N,N-dimethylmethanamine
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C19H18ClN5
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1
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| 1 |
IC50 = 113 nM
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CP0386831
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4-[3-[6-(ethoxymethyl)pyridin-3-yl]-2-methylimidazo[1,2-a]pyrazin-8-yl]morpholine
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C19H23N5O2
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1
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| 1 |
IC50 = 117.49 nM
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CP0508481
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5-(2-methyl-8-morpholin-4-ylimidazo[1,2-a]pyrazin-3-yl)-N-propan-2-ylpyridin-2-amine
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C19H24N6O
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1
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| 1 |
IC50 = 125.89 nM
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CP0379404
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4-[2-methyl-3-(6-propan-2-ylpyridin-3-yl)imidazo[1,2-a]pyrazin-8-yl]morpholine
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C19H23N5O
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1
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| 1 |
IC50 = 134.9 nM
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CP0522983
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4-[3-[6-(2-ethoxyethyl)pyridin-3-yl]-2-methylimidazo[1,2-a]pyrazin-8-yl]morpholine
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C20H25N5O2
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1
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| 1 |
IC50 = 134.9 nM
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CP0410122
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4-[3-[1-[(2-chlorophenyl)methyl]pyrazol-4-yl]-2-methylimidazo[1,2-a]pyrazin-8-yl]morpholine
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C21H21ClN6O
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1
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| 1 |
IC50 = 138.04 nM
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CP0056799
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4-[3-[1-(2-methoxyethyl)pyrazol-4-yl]-2-methylimidazo[1,2-a]pyrazin-8-yl]morpholine
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C17H22N6O2
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1
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| 1 |
IC50 = 141.25 nM
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CP0414691
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4-[3-[6-(2-methoxy-2-methylpropyl)pyridin-3-yl]-2-methylimidazo[1,2-a]pyrazin-8-yl]morpholine
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C21H27N5O2
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1
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| 1 |
IC50 = 141.25 nM
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CP0391671
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4-[2-methyl-3-[1-(2-methylpropyl)pyrazol-4-yl]imidazo[1,2-a]pyrazin-8-yl]morpholine
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C18H24N6O
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1
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| 1 |
IC50 = 144.54 nM
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CP0352707
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6,7-dimethoxy-4-(3-phenylpiperidin-1-yl)quinazoline
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C21H23N3O2
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1
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| 1 |
IC50 = 146 nM
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CP0474693
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4-[2-ethyl-3-[1-(2-methoxyethyl)pyrazol-4-yl]imidazo[1,2-a]pyrazin-8-yl]morpholine
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C18H24N6O2
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1
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| 1 |
IC50 = 154.88 nM
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CP0379800
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4-[3-[6-(3-methoxypropyl)pyridin-3-yl]-2-methylimidazo[1,2-a]pyrazin-8-yl]morpholine
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C20H25N5O2
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1
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| 1 |
IC50 = 154.88 nM
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CP0048656
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4-[3-(3,4,5-trimethoxyphenyl)imidazo[1,2-a]pyrazin-8-yl]morpholine
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C19H22N4O4
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1
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| 1 |
IC50 = 158.49 nM
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CP0379804
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4-[2-methyl-3-[6-(2-propan-2-yloxyethyl)pyridin-3-yl]imidazo[1,2-a]pyrazin-8-yl]morpholine
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C21H27N5O2
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1
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| 1 |
IC50 = 169.82 nM
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CP0428851
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4-[3-[6-(2-methoxyethyl)pyridin-3-yl]-2-methylimidazo[1,2-a]pyrazin-8-yl]morpholine
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C19H23N5O2
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1
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| 1 |
IC50 = 181.97 nM
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CP0488686
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4-[2-methyl-3-[6-(2-methylpropyl)pyridin-3-yl]imidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
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C20H25N5O
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1
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| 1 |
IC50 = 181.97 nM
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CP0379802
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4-[3-(6-ethylpyridin-3-yl)-2-methylimidazo[1,2-a]pyrazin-8-yl]morpholine
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C18H21N5O
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1
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| 1 |
IC50 = 190.55 nM
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CP0414692
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2-[5-(2-methyl-8-morpholin-4-ylimidazo[1,2-a]pyrazin-3-yl)pyridin-2-yl]ethanol
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C18H21N5O2
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1
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| 1 |
IC50 = 194.98 nM
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CP0488687
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4-[3-[2-(2-methoxyethyl)pyridin-4-yl]-2-methylimidazo[1,2-a]pyrazin-8-yl]morpholine
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C19H23N5O2
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1
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| 1 |
IC50 = 194.98 nM
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CP0508483
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4-[3-[6-(2-methoxyethoxy)pyridin-3-yl]-2-methylimidazo[1,2-a]pyrazin-8-yl]morpholine
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C19H23N5O3
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1
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| 1 |
IC50 = 199.53 nM
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CP0398570
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4-[2-methyl-3-(6-pyrrolidin-1-ylpyridin-3-yl)imidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
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C20H24N6O
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1
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| 1 |
IC50 = 218.78 nM
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CP0498445
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[3-(5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]-(4,5,6,7-tetrahydro-1-benzothiophen-2-yl)methanone
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C20H23N5OS
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1
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| 1 |
IC50 = 229 nM
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CP0411634
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4-[2-methyl-3-[1-(quinolin-2-ylmethyl)pyrazol-4-yl]imidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
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C24H23N7O
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1
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| 1 |
IC50 = 234.42 nM
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CP0549710
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4-[3-(1-ethylpyrazol-4-yl)-2-methylimidazo[1,2-a]pyrazin-8-yl]morpholine
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C16H20N6O
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1
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| 1 |
IC50 = 234.42 nM
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CP0499785
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4-[3-[6-[(3S)-3-methoxypyrrolidin-1-yl]pyridin-3-yl]-2-methylimidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
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C21H26N6O2
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1
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| 1 |
IC50 = 234.42 nM
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CP0411783
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4-[2-methyl-3-(6-propan-2-yloxypyridin-3-yl)imidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
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C19H23N5O2
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1
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| 1 |
IC50 = 245.47 nM
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CP0296762
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7-methoxy-4-(3-phenylpiperidin-1-yl)-6-(2-pyridin-2-ylethoxy)quinazoline
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C27H28N4O2
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1
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| 1 |
IC50 = 247 nM
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CP0549709
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4-[2-methoxy-3-[1-(2-methoxyethyl)pyrazol-4-yl]imidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
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C17H22N6O3
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1
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| 1 |
IC50 = 257.04 nM
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CP0523066
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4-[3-[5-(2-methoxyethyl)pyridin-2-yl]-2-methylimidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
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C19H23N5O2
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1
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| 1 |
IC50 = 257.04 nM
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CP0419391
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4-[[1-(2-chloro-5-ethoxyphenyl)-4-methyl-[1,2,4]triazolo[4,3-a]quinoxalin-8-yl]methyl]morpholine
Show/Hide
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C23H24ClN5O2
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1
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| 1 |
IC50 = 266 nM
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CP0573430
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4-[[1-(5-methoxypyridin-3-yl)-4-methyl-[1,2,4]triazolo[4,3-a]quinoxalin-8-yl]methyl]morpholine
Show/Hide
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C21H22N6O2
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1
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| 1 |
IC50 = 271 nM
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CP0488685
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4-[2-methoxy-3-[6-(2-methoxyethyl)pyridin-3-yl]imidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
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C19H23N5O3
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1
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| 1 |
IC50 = 275.42 nM
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CP0516962
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4-[2-methyl-3-(6-piperazin-1-ylpyridin-3-yl)imidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
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C20H25N7O
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1
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| 1 |
IC50 = 275.42 nM
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CP0386714
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4-[3-[6-(2-methoxyethyl)pyridin-3-yl]-2-(trifluoromethyl)imidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
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C19H20F3N5O2
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1
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| 1 |
IC50 = 281.84 nM
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CP0532944
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4,5,6,7-tetrahydro-1-benzothiophen-2-yl-[(3S)-3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]methanone
Show/Hide
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C19H21N5OS
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1
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| 1 |
IC50 = 288 nM
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CP0511166
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4-[2-methyl-3-[2-(2-methylpropyl)-1,3-oxazol-4-yl]imidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
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C18H23N5O2
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1
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| 1 |
IC50 = 302 nM
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CP0490041
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4-[3-[1-(2-methoxyethyl)pyrazol-4-yl]-2-(trifluoromethyl)imidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
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C17H19F3N6O2
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1
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| 1 |
IC50 = 309.03 nM
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CP0516963
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4-[2-methyl-3-(6-methylpyridin-3-yl)imidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
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C17H19N5O
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1
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| 1 |
IC50 = 309.03 nM
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CP0482864
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4-[[1-(2-chloro-5-propoxyphenyl)-4-methyl-[1,2,4]triazolo[4,3-a]quinoxalin-8-yl]methyl]morpholine
Show/Hide
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C24H26ClN5O2
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1
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| 1 |
IC50 = 322 nM
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CP0433369
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ethyl 4-methyl-1-phenyl-[1,2,4]triazolo[4,3-a]quinoxaline-8-carboxylate
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C19H16N4O2
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1
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| 1 |
IC50 = 325 nM
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CP0419237
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4-[3-(6-cyclopropylpyridin-3-yl)-2-methylimidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
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C19H21N5O
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1
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| 1 |
IC50 = 338.84 nM
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CP0463133
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4-[3-[6-(2-methoxyethyl)pyridin-3-yl]-2-propan-2-ylimidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
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C21H27N5O2
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1
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| 1 |
IC50 = 338.84 nM
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CP0523084
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3-[6-(2-methoxyethyl)pyridin-3-yl]-2-methyl-8-pyridin-3-ylimidazo[1,2-a]pyrazine
Show/Hide
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C20H19N5O
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1
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| 1 |
IC50 = 338.84 nM
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CP0490043
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3-[1-(2-methoxyethyl)pyrazol-4-yl]-2-methyl-8-pyridin-4-ylimidazo[1,2-a]pyrazine
Show/Hide
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C18H18N6O
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1
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| 1 |
IC50 = 346.74 nM
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CP0480570
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3-[6-(2-methoxyethyl)pyridin-3-yl]-2-methyl-8-pyridin-4-ylimidazo[1,2-a]pyrazine
Show/Hide
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C20H19N5O
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1
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| 1 |
IC50 = 346.74 nM
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CP0398569
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4-[3-[6-(2-methoxyethyl)pyridin-3-yl]-2,6-dimethylimidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
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C20H25N5O2
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1
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| 1 |
IC50 = 407.38 nM
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CP0499784
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3-[6-(2-methoxyethyl)pyridin-3-yl]-2-methyl-8-pyrrolidin-1-ylimidazo[1,2-a]pyrazine
Show/Hide
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C19H23N5O
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1
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| 1 |
IC50 = 407.38 nM
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CP0550584
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1-benzofuran-5-yl-[3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]methanone
Show/Hide
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C19H17N5O2
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1
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| 1 |
IC50 = 447 nM
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CP0147040
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US11419874, Example 28
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C15H10ClN5
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1
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| 1 |
IC50 = 480 nM
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CP0490042
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3-[1-(2-methoxyethyl)pyrazol-4-yl]-2-methyl-8-pyrrolidin-1-ylimidazo[1,2-a]pyrazine
Show/Hide
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C17H22N6O
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1
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| 1 |
IC50 = 501.19 nM
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CP0484238
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[3-[5-methyl-2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]piperidin-1-yl]-(4,5,6,7-tetrahydro-1-benzothiophen-2-yl)methanone
Show/Hide
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C21H22F3N5OS
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1
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| 1 |
IC50 = 550 nM
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CP0486657
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[3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]-(3,4,5-trimethoxyphenyl)methanone
Show/Hide
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C20H23N5O4
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1
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| 1 |
IC50 = 551 nM
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CP0474694
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3-[1-(2-methoxyethyl)pyrazol-4-yl]-2-methyl-8-pyridin-3-ylimidazo[1,2-a]pyrazine
Show/Hide
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C18H18N6O
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1
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| 1 |
IC50 = 562.34 nM
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CP0553270
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4-[3-[1-(2-methoxyethyl)pyrrol-3-yl]-2-methylimidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
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C18H23N5O2
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1
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| 1 |
IC50 = 562.34 nM
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CP0540142
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(3,4-dimethoxyphenyl)-[3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]methanone
Show/Hide
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C19H21N5O3
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1
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| 1 |
IC50 = 589 nM
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CP0571414
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4-[3-[6-(2-methoxyethyl)pyridin-3-yl]-2-methyl-6-(trifluoromethyl)imidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
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C20H22F3N5O2
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1
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| 1 |
IC50 = 602.56 nM
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CP0542603
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[3-(5-propan-2-yl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]-(4,5,6,7-tetrahydro-1-benzothiophen-2-yl)methanone
Show/Hide
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C22H27N5OS
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1
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| 1 |
IC50 = 603 nM
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CP0535023
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5-(difluoromethyl)-7-[1-[(3,4-dimethoxyphenyl)methyl]piperidin-3-yl]-[1,2,4]triazolo[1,5-a]pyrimidine
Show/Hide
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C20H23F2N5O2
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1
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| 1 |
IC50 = 661 nM
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CP0542604
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[3-[5-(difluoromethyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-1-yl]-(4,5,6,7-tetrahydro-1-benzothiophen-2-yl)methanone
Show/Hide
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C21H22F2N4OS
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1
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| 1 |
IC50 = 724 nM
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CP0532947
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7-[1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)piperidin-3-yl]-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonitrile
Show/Hide
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C20H20N6OS
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1
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| 1 |
IC50 = 759 nM
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CP0376865
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2-(2-isoquinolin-7-yloxyethyl)quinoline
Show/Hide
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C20H16N2O
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1
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| 1 |
IC50 = 809 nM
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CP0553921
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(4-methoxyphenyl)-[(3S)-3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]methanone
Show/Hide
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C18H19N5O2
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1
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| 1 |
IC50 = 871 nM
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CP0535021
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[3-[5-(difluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]piperidin-1-yl]-(4,5,6,7-tetrahydro-1-benzothiophen-2-yl)methanone
Show/Hide
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C20H21F2N5OS
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1
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| 1 |
IC50 = 912 nM
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CP0060511
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4-[3-[1-(2-methoxyethyl)pyrazol-4-yl]imidazo[1,2-a]pyrazin-8-yl]morpholine
Show/Hide
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C16H20N6O2
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1
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| 1 |
IC50 = 1000 nM
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CP0152286
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7-methoxy-4-(3-phenylpiperidin-1-yl)-6-propoxyquinazoline
Show/Hide
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C23H27N3O2
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1
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| 1 |
IC50 = 1040 nM
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CP0529994
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cyclopropyl-[(3S)-3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]methanone
Show/Hide
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C14H17N5O
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1
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| 1 |
IC50 = 1047 nM
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CP0491961
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[3-(7-methylimidazo[1,2-a]pyrimidin-5-yl)piperidin-1-yl]-(4,5,6,7-tetrahydro-1-benzothiophen-2-yl)methanone
Show/Hide
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C21H24N4OS
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1
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| 1 |
IC50 = 1096 nM
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CP0484243
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[3-(5-methoxy-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]-(4,5,6,7-tetrahydro-1-benzothiophen-2-yl)methanone
Show/Hide
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C20H23N5O2S
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1
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| 1 |
IC50 = 1148 nM
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CP0484309
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(3-methoxyphenyl)-[(3S)-3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]methanone
Show/Hide
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C18H19N5O2
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1
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| 1 |
IC50 = 1148 nM
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CP0542607
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2,3-dihydro-1,4-benzodioxin-6-yl-[(3S)-3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]methanone
Show/Hide
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C19H19N5O3
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1
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| 1 |
IC50 = 1148 nM
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CP0540143
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4,5,6,7-tetrahydro-1-benzothiophen-2-yl-[3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)azepan-1-yl]methanone
Show/Hide
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C20H23N5OS
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1
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| 1 |
IC50 = 1288 nM
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CP0508762
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4-[[1-(5-butoxy-2-chlorophenyl)-4-methyl-[1,2,4]triazolo[4,3-a]quinoxalin-8-yl]methyl]morpholine
Show/Hide
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C25H28ClN5O2
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1
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| 1 |
IC50 = 1622 nM
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CP0503247
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7-methoxy-6-(2-phenylethoxy)-4-(3-phenylpiperidin-1-yl)quinazoline
Show/Hide
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C28H29N3O2
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1
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| 1 |
IC50 = 1665 nM
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CP0521463
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4-[[1-(2-chloro-5-propan-2-yloxyphenyl)-4-methyl-[1,2,4]triazolo[4,3-a]quinoxalin-8-yl]methyl]morpholine
Show/Hide
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C24H26ClN5O2
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1
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| 1 |
IC50 = 1862 nM
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CP0389574
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7-methoxy-4-(3-phenylpiperidin-1-yl)-6-(2-pyridin-3-ylethoxy)quinazoline
Show/Hide
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C27H28N4O2
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1
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| 1 |
IC50 = 2338 nM
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CP0488089
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3-[2-chloro-5-(2,2,2-trifluoroethoxymethyl)phenyl]-7-methyl-2,4,5,8,12-pentazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7,10,12-hexaene
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C18H13ClF3N5O
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1
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| 1 |
IC50 = 2450 nM
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CP0553977
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[4-methyl-3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperazin-1-yl]-(4,5,6,7-tetrahydro-1-benzothiophen-2-yl)methanone
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C19H22N6OS
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1
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| 1 |
IC50 = 2455 nM
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CP0484310
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4,5,6,7-tetrahydro-1-benzothiophen-2-yl-[(2S)-2-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)morpholin-4-yl]methanone
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C18H19N5O2S
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1
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| 1 |
IC50 = 2630 nM
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CP0425612
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ethyl 4-methyl-1-phenyl-[1,2,4]triazolo[4,3-a]quinoxaline-7-carboxylate
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C19H16N4O2
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1
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| 1 |
IC50 = 2690 nM
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CP0535020
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4,5,6,7-tetrahydro-1-benzothiophen-2-yl-[3-[5-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]piperidin-1-yl]methanone
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C20H20F3N5OS
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1
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| 1 |
IC50 = 2692 nM
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CP0532945
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[(3S)-3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]-[4-(trifluoromethyl)phenyl]methanone
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C18H16F3N5O
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1
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| 1 |
IC50 = 3020 nM
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CP0484308
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2-(3,4-dimethoxyphenyl)-1-[(3S)-3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]ethanone
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C20H23N5O3
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1
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| 1 |
IC50 = 3162 nM
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CP0484314
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(1-methylsulfonylindol-5-yl)-[(3R)-3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]methanone
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C20H20N6O3S
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1
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| 1 |
IC50 = 3548 nM
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CP0414237
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3-(5-butoxypyridin-3-yl)-7-methyl-2,4,5,8,12-pentazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7,10,12-hexaene
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C18H18N6O
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1
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| 1 |
IC50 = 3800 nM
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CP0448309
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3-[2-chloro-5-(propoxymethyl)phenyl]-7-methyl-2,4,5,8,12-pentazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7,10,12-hexaene
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C19H18ClN5O
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1
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| 1 |
IC50 = 3890 nM
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CP0535016
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phenyl-[(3S)-3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]methanone
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C17H17N5O
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1
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| 1 |
IC50 = 4571 nM
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CP0090153
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4-[[1-(5-butoxypyridin-3-yl)-4-methyl-[1,2,4]triazolo[4,3-a]quinoxalin-8-yl]methyl]morpholine
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C24H28N6O2
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1
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| 1 |
IC50 = 4823 nM
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CP0498448
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(2-methoxyphenyl)-[(3S)-3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]methanone
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C18H19N5O2
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1
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| 1 |
IC50 = 5129 nM
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CP0486899
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3-(5-butoxy-2-chlorophenyl)-7-methyl-2,4,5,8,12-pentazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7,10,12-hexaene
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C19H18ClN5O
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1
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| 1 |
IC50 = 5500 nM
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CP0484239
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7-[(3S)-1-[(2-chloro-6-methylpyridin-4-yl)methyl]piperidin-3-yl]-5-(difluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidine
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C18H19ClF2N6
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1
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| 1 |
IC50 = 5623 nM
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CP0389452
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3-[2-chloro-5-(propan-2-yloxymethyl)phenyl]-7-methyl-2,4,5,8,12-pentazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7,10,12-hexaene
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C19H18ClN5O
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1
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| 1 |
IC50 = 6030 nM
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CP0482863
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4-[[4-methyl-1-(5-propoxypyridin-3-yl)-[1,2,4]triazolo[4,3-a]quinoxalin-8-yl]methyl]morpholine
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C23H26N6O2
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1
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| 1 |
IC50 = 6131 nM
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CP0484312
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4-[(3S)-3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidine-1-carbonyl]benzonitrile
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C18H16N6O
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1
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| 1 |
IC50 = 6918 nM
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CP0532946
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7-[1-(1-benzofuran-5-ylmethyl)piperidin-3-yl]-5-(difluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidine
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C20H19F2N5O
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1
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| 1 |
IC50 = 7586 nM
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CP0547066
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4-[[1-[5-(2-methoxyethoxy)pyridin-3-yl]-4-methyl-[1,2,4]triazolo[4,3-a]quinoxalin-8-yl]methyl]morpholine
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C23H26N6O3
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1
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| 1 |
IC50 = 7762 nM
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CP0527831
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cyclohexyl-[3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]methanone
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C17H23N5O
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1
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| 1 |
IC50 = 7762 nM
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CP0484316
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5-(difluoromethyl)-7-[(3S)-1-[(2,6-dimethylpyridin-4-yl)methyl]piperidin-3-yl]-[1,2,4]triazolo[1,5-a]pyrimidine
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C19H22F2N6
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1
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| 1 |
IC50 = 8318 nM
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CP0448292
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3-[2-chloro-5-(trifluoromethoxy)phenyl]-7-methyl-2,4,5,8,12-pentazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7,10,12-hexaene
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C16H9ClF3N5O
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1
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| 1 |
IC50 = 8910 nM
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CP0488088
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3-[2-chloro-5-(2-methoxyethoxy)phenyl]-7-methyl-2,4,5,8,12-pentazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7,10,12-hexaene
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C18H16ClN5O2
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1
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| 1 |
IC50 = 9120 nM
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CP0482862
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4-[[4-methyl-1-(5-propan-2-yloxypyridin-3-yl)-[1,2,4]triazolo[4,3-a]quinoxalin-8-yl]methyl]morpholine
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C23H26N6O2
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1
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| 1 |
IC50 > 10000 nM
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CP0428749
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4-[4-chloro-3-(7-methyl-2,4,5,8,12-pentazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7,10,12-hexaen-3-yl)phenyl]morpholine
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C19H17ClN6O
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1
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| 1 |
IC50 > 10000 nM
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CP0529995
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4,5,6,7-tetrahydro-1-benzothiophen-2-yl-[3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperazin-1-yl]methanone
Show/Hide
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C18H20N6OS
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1
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| 1 |
IC50 > 10000 nM
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CP0910630
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(RS)-[3-(1H-Pyrrolo[2,3-b]pyridin-4-yl)-1-piperidyl]-(4,5,6,7-tetrahydrobenzothiophen-2-yl)methanone
Show/Hide
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C21H23N3OS
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1
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| 1 |
IC50 > 10000 nM
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CP0484242
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1-[4-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-2-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperazin-1-yl]ethanone
Show/Hide
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C20H22N6O2S
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1
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| 1 |
IC50 > 3020 nM
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CP0376864
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7-methoxy-4-(3-phenylpiperidin-1-yl)-6-(pyridin-3-ylmethoxy)quinazoline
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C26H26N4O2
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1
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| 1 |
IC50 > 3200 nM
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CP0431292
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7-methoxy-4-(3-phenylpiperidin-1-yl)-6-(quinolin-2-ylmethoxy)quinazoline
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C30H28N4O2
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1
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| 1 |
IC50 > 3200 nM
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CP0498870
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7-methoxy-4-(3-phenylpiperidin-1-yl)-6-(2-pyridin-4-ylethoxy)quinazoline
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C27H28N4O2
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1
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| 1 |
IC50 > 3200 nM
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CP0499347
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7-methoxy-4-(3-phenylpiperidin-1-yl)-6-(pyridin-2-ylmethoxy)quinazoline
Show/Hide
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C26H26N4O2
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1
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| 1 |
IC50 > 3200 nM
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CP0520756
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7-methoxy-4-(3-phenylpiperidin-1-yl)-6-(pyridin-4-ylmethoxy)quinazoline
Show/Hide
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C26H26N4O2
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1
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| 1 |
IC50 > 3200 nM
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