| Compound ID |
Compound Name |
Compound Formula |
|
CP0398974
|
N-[(5-chloro-2-nitrophenyl)methyl]-N,1-dimethylpiperidin-4-amine
Show/Hide
|
C14H20ClN3O2
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
|
CP0511679
|
4-chloro-2-[[methyl-[1-(2-phenylethyl)piperidin-4-yl]amino]methyl]benzonitrile
Show/Hide
|
C22H26ClN3
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
|
CP0153439
|
(S)-2-Amino-5-(2-methyl-isothioureido)-pentanoic acid
Show/Hide
|
C7H15N3O2S
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0905339
|
N-(1-(2-(Pyrrolidin-1-yl)ethyl)indolin-5-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C19H26Cl2N4S
|
1
|
| 1 |
IC50 = 410 nM
|
|
|
|
CP0462455
|
4-chloro-2-[[(1-ethylpiperidin-4-yl)-methylamino]methyl]benzonitrile
Show/Hide
|
C16H22ClN3
|
1
|
| 1 |
IC50 = 450 nM
|
|
|
|
CP0404972
|
4-chloro-2-[[methyl-[1-(3-methylbutyl)piperidin-4-yl]amino]methyl]benzonitrile
Show/Hide
|
C19H28ClN3
|
1
|
| 1 |
IC50 = 540 nM
|
|
|
|
CP0490417
|
4-chloro-2-[[piperidin-4-yl(propan-2-yl)amino]methyl]benzonitrile
Show/Hide
|
C16H22ClN3
|
1
|
| 1 |
IC50 = 570 nM
|
|
|
|
CP0857490
|
(S)-2-amino-5-(3-methylguanidino)pentanoic acid dihydrochloride
Show/Hide
|
C7H18Cl2N4O2
|
1
|
| 1 |
IC50 = 650 nM
|
|
|
|
CP0418062
|
methyl (2S)-2-amino-5-[(N'-methylcarbamimidoyl)amino]pentanoate
Show/Hide
|
C8H18N4O2
|
1
|
| 1 |
IC50 = 650 nM
|
|
|
|
CP0052287
|
(2S)-5-{[(Z)-amino(imino)methyl]amino}-2-(methylamino)pentanoic acid
Show/Hide
|
C7H16N4O2
|
1
|
| 1 |
IC50 = 650 nM
|
|
|
|
CP0053263
|
(2S)-2-azaniumyl-5-[(N'-methylcarbamimidoyl)amino]pentanoate
Show/Hide
|
C7H16N4O2
|
1
|
| 1 |
IC50 = 650 nM
|
|
|
|
CP0382299
|
2-[[(1-butylpiperidin-4-yl)-methylamino]methyl]-4-chlorobenzonitrile
Show/Hide
|
C18H26ClN3
|
1
|
| 1 |
IC50 = 680 nM
|
|
|
|
CP0747739
|
L-nitro arginine methyl ester
Show/Hide
|
C7H16ClN5O4
|
1
|
| 1 |
IC50 = 680 nM
|
|
|
|
CP0444367
|
4-chloro-2-[[methyl-(1-methylpiperidin-4-yl)amino]methyl]benzonitrile
Show/Hide
|
C15H20ClN3
|
1
|
| 1 |
IC50 = 770 nM
|
|
|
|
CP0895048
|
N-(1-(2-(Pyrrolidin-1-yl)acetyl)indolin-5-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C19H24Cl2N4OS
|
1
|
| 1 |
IC50 = 770 nM
|
|
|
|
CP0454333
|
4-bromo-2-[[methyl-(1-methylpiperidin-4-yl)amino]methyl]benzonitrile
Show/Hide
|
C15H20BrN3
|
1
|
| 1 |
IC50 = 810 nM
|
|
|
|
CP0433268
|
N-[(2-bromo-5-chlorophenyl)methyl]-N,1-dimethylpiperidin-4-amine
Show/Hide
|
C14H20BrClN2
|
1
|
| 1 |
IC50 = 820 nM
|
|
|
|
CP0490416
|
4-chloro-2-[[[1-(cyclopropylmethyl)piperidin-4-yl]-methylamino]methyl]benzonitrile
Show/Hide
|
C18H24ClN3
|
1
|
| 1 |
IC50 = 860 nM
|
|
|
|
CP0483667
|
4-chloro-2-[[methyl(piperidin-3-yl)amino]methyl]benzonitrile
Show/Hide
|
C14H18ClN3
|
1
|
| 1 |
IC50 = 983 nM
|
|
|
|
CP0382255
|
4-chloro-2-[[ethyl(piperidin-4-yl)amino]methyl]benzonitrile
Show/Hide
|
C15H20ClN3
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0382280
|
4-chloro-2-[[methyl-(1-propylpiperidin-4-yl)amino]methyl]benzonitrile
Show/Hide
|
C17H24ClN3
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0433267
|
4-chloro-2-[[methyl(piperidin-4-yl)amino]methyl]benzonitrile
Show/Hide
|
C14H18ClN3
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0444370
|
N-[[5-chloro-2-(trifluoromethyl)phenyl]methyl]-N,1-dimethylpiperidin-4-amine
Show/Hide
|
C15H20ClF3N2
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
|
CP0870593
|
N-(1-(1-(2-Hydroxyethyl)piperidin-4-yl)indolin-5-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H28Cl2N4OS
|
1
|
| 1 |
IC50 = 1580 nM
|
|
|
|
CP0454332
|
4-chloro-2-[[piperidin-4-yl(propyl)amino]methyl]benzonitrile
Show/Hide
|
C16H22ClN3
|
1
|
| 1 |
IC50 = 1700 nM
|
|
|
|
CP0919242
|
(S)-N-(1-(2-(1-methylpyrrolidin-2-yl)ethyl)-1H-indol-5-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H26Cl2N4S
|
1
|
| 1 |
IC50 = 1920 nM
|
|
|
|
CP0462462
|
4-chloro-2-[[cyclopropylmethyl(piperidin-4-yl)amino]methyl]benzonitrile
Show/Hide
|
C17H22ClN3
|
1
|
| 1 |
IC50 = 2100 nM
|
|
|
|
CP0044041
|
(L-N6-1-iminoethyl)lysine
Show/Hide
|
C8H17N3O2
|
1
|
| 1 |
IC50 = 2500 nM
|
|
|
|
CP0887882
|
N-(1-(4-(dimethylamino)butyl)-1H-indol-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C19H26Cl2N4S
|
1
|
| 1 |
IC50 = 2530 nM
|
|
|
|
CP0910864
|
N-{1-[3-(Adamantan-1-ylamino)-propyl]-1H-indol-5-yl}-thiophene-2-carboxamidine dihydrochloride
Show/Hide
|
C26H34Cl2N4S
|
1
|
| 1 |
IC50 = 3150 nM
|
|
|
|
CP0454913
|
N'-[1-[2-(2-hydroxyethylamino)ethyl]-2,3-dihydroindol-6-yl]thiophene-2-carboximidamide
Show/Hide
|
C17H22N4OS
|
1
|
| 1 |
IC50 = 3360 nM
|
|
|
|
CP0893901
|
(R)-N-(1-(2-(1-methylpyrrolidin-2-yl)ethyl)-1H-indol-5-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H26Cl2N4S
|
1
|
| 1 |
IC50 = 3370 nM
|
|
|
|
CP0919195
|
N-(1-(2-(dimethylamino)ethyl)-1H-indol-5-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C17H22Cl2N4S
|
1
|
| 1 |
IC50 = 3700 nM
|
|
|
|
CP0852924
|
N-(1-(2-(piperidin-1-yl)ethyl)-1H-indol-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H26Cl2N4S
|
1
|
| 1 |
IC50 = 3800 nM
|
|
|
|
CP0404973
|
4-chloro-2-[[methyl(pyrrolidin-3-yl)amino]methyl]benzonitrile
Show/Hide
|
C13H16ClN3
|
1
|
| 1 |
IC50 = 4000 nM
|
|
|
|
CP0899695
|
N-(1-(2-(dimethylamino)ethyl)indolin-5-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C17H24Cl2N4S
|
1
|
| 1 |
IC50 = 4070 nM
|
|
|
|
CP0382298
|
2-[[(1-benzylpiperidin-4-yl)-methylamino]methyl]-4-chlorobenzonitrile
Show/Hide
|
C21H24ClN3
|
1
|
| 1 |
IC50 = 4300 nM
|
|
|
|
CP0505110
|
2-[[azepan-4-yl(methyl)amino]methyl]-4-chlorobenzonitrile
Show/Hide
|
C15H20ClN3
|
1
|
| 1 |
IC50 = 4400 nM
|
|
|
|
CP0918473
|
rac-N-(1-(2-(1-methylpyrrolidin-2-yl)ethyl)-1H-indol-5-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H26Cl2N4S
|
1
|
| 1 |
IC50 = 4490 nM
|
|
|
|
CP0899694
|
N-(1-(1-Methylpiperidin-4-yl)indolin-5-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C19H26Cl2N4S
|
1
|
| 1 |
IC50 = 4670 nM
|
|
|
|
CP0040036
|
(S)-5-Acetimidoylamino-2-amino-pent
Show/Hide
|
C7H15N3O2
|
1
|
| 1 |
IC50 = 6000 nM
|
|
|
|
CP0858765
|
N-(1-(3-morpholinopropyl)-1H-indol-5-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H26Cl2N4OS
|
1
|
| 1 |
IC50 = 6000 nM
|
|
|
|
CP0913090
|
trans-N-(3-(4-(methylamino)cyclohexyl)-1H-indol-5-yl)thiophene-2-carboximidamide hydrochloride
Show/Hide
|
C20H25ClN4S
|
1
|
| 1 |
IC50 = 6240 nM
|
|
|
|
CP0940689
|
N-(1-(3-((1-ethylpyrrolidin-2-yl)methylamino)propyl)-1H-indol-5-yl)thiophene-2-carboximidamide trihydrochloride
Show/Hide
|
C23H32ClN5S
|
1
|
| 1 |
IC50 = 6330 nM
|
|
|
|
CP0846662
|
N-(1-(2-(1-methylpiperidin-2-yl)ethyl)-1H-indol-5-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C21H28Cl2N4S
|
1
|
| 1 |
IC50 = 6400 nM
|
|
|
|
CP0887630
|
N-(3-(1-methylpyrrolidin-3-yl)-1H-indol-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C18H22Cl2N4S
|
1
|
| 1 |
IC50 = 7100 nM
|
|
|
|
CP0403591
|
N'-[1-[2-[(3R)-3-hydroxypyrrolidin-1-yl]ethyl]-2,3-dihydroindol-6-yl]thiophene-2-carboximidamide
Show/Hide
|
C19H24N4OS
|
1
|
| 1 |
IC50 = 7120 nM
|
|
|
|
CP0476584
|
N'-(1-pyrrolidin-3-yl-2,3-dihydroindol-6-yl)thiophene-2-carboximidamide
Show/Hide
|
C17H20N4S
|
1
|
| 1 |
IC50 = 7170 nM
|
|
|
|
CP0861066
|
trans-(+/-)-N-(3-(3-(methylamino)cyclohexyl)-1H-indol-5-yl)thiophene-2-carboximidamide hydrochloride
Show/Hide
|
C20H25ClN4S
|
1
|
| 1 |
IC50 = 7760 nM
|
|
|
|
CP0904455
|
N-(1-(3-(cyclopropylamino)propyl)-1H-indol-5-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C19H24Cl2N4S
|
1
|
| 1 |
IC50 = 8720 nM
|
|
|
|
CP0846661
|
N-(1-(2-(piperidin-1-yl)ethyl)-1H-indol-5-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H26Cl2N4S
|
1
|
| 1 |
IC50 = 9200 nM
|
|
|
|
CP0875702
|
N-(1-(3-(Pyrrolidin-1-yl)propyl)-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C21H30Cl2N4S
|
1
|
| 1 |
IC50 = 9500 nM
|
|
|
|
CP0894570
|
N-(1-(3-(diethylamino)propyl)-1H-indol-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H28Cl2N4S
|
1
|
| 1 |
IC50 = 10200 nM
|
|
|
|
CP0893178
|
N-(3-(1-methylpiperidin-4-yl)-1H-indol-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C19H24Cl2N4S
|
1
|
| 1 |
IC50 = 10700 nM
|
|
|
|
CP0436023
|
(S)-2-(S)-Amino-3-methyl-5-(2-methyl-isothioureido)-pentanoic acid tert-butyl ester
Show/Hide
|
C12H25N3O2S
|
1
|
| 1 |
IC50 = 11000 nM
|
|
|
|
CP0870508
|
trans-(+/-)-N-(3-(3-(Ethylamino)cyclohexyl)-1H-indol-5-yl)thiophene-2-carboximidamide hydrochloride
Show/Hide
|
C21H27ClN4S
|
1
|
| 1 |
IC50 = 11000 nM
|
|
|
|
CP0894569
|
N-(1-(3-(pyrrolidin-1-yl)propyl)-1H-indol-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H26Cl2N4S
|
1
|
| 1 |
IC50 = 11200 nM
|
|
|
|
CP0858766
|
N-(1-(1-methylazepan-4-yl)-1H-indol-5-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H26Cl2N4S
|
1
|
| 1 |
IC50 = 11500 nM
|
|
|
|
CP0871043
|
N-(1-(3-(methylamino)propyl)-1H-indol-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C17H22Cl2N4S
|
1
|
| 1 |
IC50 = 11800 nM
|
|
|
|
CP0898981
|
N-(1-(quinuclidin-3-yl)-1H-indol-5-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H24Cl2N4S
|
1
|
| 1 |
IC50 = 12100 nM
|
|
|
|
CP0915579
|
N-(1-(3-(dimethylamino)propyl)-1H-indol-5-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C18H24Cl2N4S
|
1
|
| 1 |
IC50 = 12400 nM
|
|
|
|
CP0918474
|
N-(1-(2-(1-methylpyrrolidin-2-yl)ethyl)-1H-indol-5-yl)furan-2-carboximidamide dihydrochloride
Show/Hide
|
C20H26Cl2N4O
|
1
|
| 1 |
IC50 = 13900 nM
|
|
|
|
CP0666251
|
(R)-N-(1-(2-(1-Methylpyrrolidin-2-yl)ethyl)-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C21H30Cl2N4S
|
1
|
| 1 |
IC50 = 14300 nM
|
|
|
|
CP0888586
|
N-(1-(2-(dimethylamino)ethyl)-1H-indol-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C17H22Cl2N4S
|
1
|
| 1 |
IC50 = 15000 nM
|
|
|
|
CP0918475
|
N-(1-(1-methylpiperidin-4-yl)-1H-indol-5-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C19H24Cl2N4S
|
1
|
| 1 |
IC50 = 15800 nM
|
|
|
|
CP0877749
|
(R)-N-(1-(2-(1-methylpyrrolidin-2-yl)ethyl)-1H-indol-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H26Cl2N4S
|
1
|
| 1 |
IC50 = 16000 nM
|
|
|
|
CP0852925
|
N-(1-(3-morpholinopropyl)-1H-indol-6-yl)thiophene-3-carboximidamide dihydrochloride
Show/Hide
|
C20H26Cl2N4OS
|
1
|
| 1 |
IC50 = 17100 nM
|
|
|
|
CP0847605
|
cis-N-(3-(4-(dimethylamino)cyclohexyl)-1H-indol-5-yl)thiophene-2-carboximidamide hydrochloride
Show/Hide
|
C21H27ClN4S
|
1
|
| 1 |
IC50 = 17500 nM
|
|
|
|
CP0898980
|
N-(1-(8-methyl-8-azabicyclo[3.2.1]octan-3-yl)-1H-indol-5-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C21H26Cl2N4S
|
1
|
| 1 |
IC50 = 18900 nM
|
|
|
|
CP0915337
|
(+/-)-N-(1-(2-(1-methylpyrrolidin-2-yl)ethyl)-1H-indol-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H26Cl2N4S
|
1
|
| 1 |
IC50 = 19000 nM
|
|
|
|
CP0704704
|
cis-N-(3-(4-(ethylamino)cyclohexyl)-1H-indol-5-yl)thiophene-2-carboximidamide hydrochloride
Show/Hide
|
C21H27ClN4S
|
1
|
| 1 |
IC50 = 19000 nM
|
|
|
|
CP0871044
|
N-(1-(3-morpholinopropyl)-1H-indol-6-yl)furan-3-carboximidamide dihydrochloride
Show/Hide
|
C20H26Cl2N4O2
|
1
|
| 1 |
IC50 = 19100 nM
|
|
|
|
CP0867182
|
N-(1-(1-methylpiperidin-4-yl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C21H30Cl2N4S
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0403594
|
N'-[1-(thian-4-yl)-2,3-dihydroindol-6-yl]thiophene-2-carboximidamide
Show/Hide
|
C18H21N3S2
|
1
|
| 1 |
IC50 = 21500 nM
|
|
|
|
CP0859167
|
N-(1-(3-(Dimethylamino)propyl)-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C19H28Cl2N4S
|
1
|
| 1 |
IC50 = 22400 nM
|
|
|
|
CP0777464
|
N-(3-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)-1H-indol-5-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C19H22Cl2N4S
|
1
|
| 1 |
IC50 = 22400 nM
|
|
|
|
CP0917441
|
N-(1-(3-(Methylamino)propyl)-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C18H26Cl2N4S
|
1
|
| 1 |
IC50 = 22500 nM
|
|
|
|
CP0888604
|
N-(1-(4-(1H-imidazol-1-yl)butyl)-1H-indol-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H23Cl2N5S
|
1
|
| 1 |
IC50 = 23000 nM
|
|
|
|
CP0919240
|
N-(1-(3-(dimethylamino)propyl)-1H-indol-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C18H24Cl2N4S
|
1
|
| 1 |
IC50 = 23300 nM
|
|
|
|
CP0917822
|
(+/-)-N-(1-(Pyrrolidin-3-yl)-1,2,3,4-tetrahydroquinolin-6-yl)-thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C18H24Cl2N4S
|
1
|
| 1 |
IC50 = 23500 nM
|
|
|
|
CP0871802
|
(S)-N-(1-(2-(1-methylpyrrolidin-2-yl)ethyl)-1H-indol-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H26Cl2N4S
|
1
|
| 1 |
IC50 = 24000 nM
|
|
|
|
CP0859143
|
N-(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C19H24Cl2N4S
|
1
|
| 1 |
IC50 = 24200 nM
|
|
|
|
CP0859168
|
N-(1-(2-(Dimethylamino)ethyl)-8-fluoro-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C18H25Cl2FN4S
|
1
|
| 1 |
IC50 = 24300 nM
|
|
|
|
CP0873351
|
N-(1-(3-(Pyrrolidin-1-yl)propyl)-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C21H28Cl2N4OS
|
1
|
| 1 |
IC50 = 24500 nM
|
|
|
|
CP0851758
|
N-(2-Oxo-1-(2-(piperidin-1-yl)ethyl)-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C21H28Cl2N4OS
|
1
|
| 1 |
IC50 = 25200 nM
|
|
|
|
CP0704838
|
cis-N-(3-(4-(methylamino)cyclohexyl)-1H-indol-5-yl)thiophene-2-carboximidamide hydrochloride
Show/Hide
|
C20H25ClN4S
|
1
|
| 1 |
IC50 = 25400 nM
|
|
|
|
CP0902858
|
2-[[[[2-(1-Iminoethyl)amino]ethyl]thio]methyl]-D-valine dihydrochloride
Show/Hide
|
C9H22Cl2N4O2S
|
1
|
| 1 |
IC50 = 26000 nM
|
|
|
|
CP0734618
|
N-(3-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)-1H-indol-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C19H22Cl2N4S
|
1
|
| 1 |
IC50 = 26500 nM
|
|
|
|
CP0873352
|
(+/-)-N-(1-(1-Methylpyrrolidin-3-yl)-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C19H26Cl2N4S
|
1
|
| 1 |
IC50 = 27500 nM
|
|
|
|
CP0888580
|
N-(1-(3-morpholinopropyl)-1H-indol-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H26Cl2N4OS
|
1
|
| 1 |
IC50 = 28300 nM
|
|
|
|
CP0867649
|
N-(2-Oxo-1-(2-(pyrrolidin-1-yl)ethyl)-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H26Cl2N4OS
|
1
|
| 1 |
IC50 = 29800 nM
|
|
|
|
CP0917440
|
N-(1-(2-(Isopropylamino)ethyl)-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C19H28Cl2N4S
|
1
|
| 1 |
IC50 = 30200 nM
|
|
|
|
CP0871803
|
N-(1-(1-methylazepan-4-yl)-1H-indol-6-yl)furan-2-carboximidamide dihydrochloride
Show/Hide
|
C20H26Cl2N4O
|
1
|
| 1 |
IC50 = 30600 nM
|
|
|
|
CP0850822
|
(+/-)-N-(1-(2-(1-methylpyrrolidin-2-yl)ethyl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C22H32Cl2N4S
|
1
|
| 1 |
IC50 = 30800 nM
|
|
|
|
CP0667837
|
cis-(+/-)-N-(3-(3-(Ethylamino)cyclohexyl)-1H-indol-5-yl)thiophene-2-carboximidamide hydrochloride
Show/Hide
|
C21H27ClN4S
|
1
|
| 1 |
IC50 = 32000 nM
|
|
|
|
CP0913091
|
(+/-)-N-(3-(4-(methylamino)cyclohex-1-enyl)-1H-indol-5-yl)thiophene-2-carboximidamide hydrochloride
Show/Hide
|
C20H23ClN4S
|
1
|
| 1 |
IC50 = 32000 nM
|
|
|
|
CP0917442
|
N-(1-(2-(2-Hydroxyethylamino)ethyl)-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C18H26Cl2N4OS
|
1
|
| 1 |
IC50 = 32900 nM
|
|
|
|
CP0853933
|
N-(1-(2-(Ethyl(methyl)amino)ethyl)-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C19H28Cl2N4S
|
1
|
| 1 |
IC50 = 33300 nM
|
|
|
|
CP0899149
|
N-(1-(3-morpholinopropyl)-1H-indol-6-yl)furan-2-carboximidamide dihydrochloride
Show/Hide
|
C20H26Cl2N4O2
|
1
|
| 1 |
IC50 = 34000 nM
|
|
|
|
CP0676501
|
N-(3-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)-1H-indol-5-yl)furan-2-carboximidamide dihydrochloride
Show/Hide
|
C19H22Cl2N4O
|
1
|
| 1 |
IC50 = 36100 nM
|
|
|
|
CP0868523
|
methyl 3-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)-1H-indol-5-ylcarbamimidothioate dihydrochloride
Show/Hide
|
C16H22Cl2N4S
|
1
|
| 1 |
IC50 = 36100 nM
|
|
|
|
CP0887881
|
N-(1-(1-methylazepan-4-yl)-1H-indol-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H26Cl2N4S
|
1
|
| 1 |
IC50 = 37700 nM
|
|
|
|
CP0853757
|
N-(1-(3-(2-Hydroxyethylamino)propyl)-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C19H28Cl2N4OS
|
1
|
| 1 |
IC50 = 39200 nM
|
|
|
|
CP0875724
|
(+/-)-N-(3-(4-(ethylamino)cyclohex-1-enyl)-1H-indol-5-yl)thiophene-2-carboximidamide hydrochloride
Show/Hide
|
C21H25ClN4S
|
1
|
| 1 |
IC50 = 40300 nM
|
|
|
|
CP0927411
|
N-(1-(2-(Methylamino)ethyl)-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C17H24Cl2N4S
|
1
|
| 1 |
IC50 = 40700 nM
|
|
|
|
CP0666250
|
N-(1-(2-(Dimethylamino)ethyl)-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C18H24Cl2N4OS
|
1
|
| 1 |
IC50 = 41100 nM
|
|
|
|
CP0853299
|
N-(1-(1-Methylpiperidin-4-yl)-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H28Cl2N4S
|
1
|
| 1 |
IC50 = 42700 nM
|
|
|
|
CP0896820
|
N-(3-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)-1H-indol-5-ylcarbamothioyl)benzamide dihydrochloride
Show/Hide
|
C22H24Cl2N4OS
|
1
|
| 1 |
IC50 = 43000 nM
|
|
|
|
CP0676856
|
(S)-N-(1-(2-(1-Methylpyrrolidin-2-yl)ethyl)-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C21H30Cl2N4S
|
1
|
| 1 |
IC50 = 45600 nM
|
|
|
|
CP0894438
|
N-(3-(1-azabicyclo[2.2.2]oct-2-en-3-yl)-1H-indol-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H22Cl2N4S
|
1
|
| 1 |
IC50 = 46200 nM
|
|
|
|
CP0948496
|
N-(1-(2-(Ethylamino)ethyl)-1,2,3,4-tetrahydroquinolin-6-yl)-thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C18H26Cl2N4S
|
1
|
| 1 |
IC50 = 46500 nM
|
|
|
|
CP0867192
|
N-(1-(2-(methylamino)ethyl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C18H26Cl2N4S
|
1
|
| 1 |
IC50 = 47100 nM
|
|
|
|
CP0895913
|
(+/-)-N-(1-(Piperidin-3-yl)indolin-5-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C18H24Cl2N4S
|
1
|
| 1 |
IC50 = 52200 nM
|
|
|
|
CP0867561
|
N-(1-(2-(piperidin-1-yl)ethyl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C22H32Cl2N4S
|
1
|
| 1 |
IC50 = 56300 nM
|
|
|
|
CP0676858
|
N-(1-(2-(Dimethylamino)ethyl)-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C18H26Cl2N4S
|
1
|
| 1 |
IC50 = 58700 nM
|
|
|
|
CP0867563
|
(+/-)-N-(1-(1-methylpyrrolidin-3-yl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H28Cl2N4S
|
1
|
| 1 |
IC50 = 60500 nM
|
|
|
|
CP0912490
|
N-(1-(2-((2-Hydroxyethyl)(methyl)amino)ethyl)-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C19H28Cl2N4OS
|
1
|
| 1 |
IC50 = 63900 nM
|
|
|
|
CP0853298
|
N-(1-(2-(Diethylamino)ethyl)-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H30Cl2N4S
|
1
|
| 1 |
IC50 = 64400 nM
|
|
|
|
CP0868522
|
N-((3-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)-1H-indol-5-yl)methyl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H24Cl2N4S
|
1
|
| 1 |
IC50 = 64700 nM
|
|
|
|
CP0868524
|
5-methyl-N-(3-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)-1H-indol-5-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H24Cl2N4S
|
1
|
| 1 |
IC50 = 65300 nM
|
|
|
|
CP0867193
|
N-(1-(piperidin-4-yl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H28Cl2N4S
|
1
|
| 1 |
IC50 = 66200 nM
|
|
|
|
CP0873350
|
(+/-)-N-(1-(2-(1-Methylpyrrolidin-2-yl)ethyl)-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C21H28Cl2N4OS
|
1
|
| 1 |
IC50 = 68900 nM
|
|
|
|
CP0859166
|
N-(1-(2-(Diethylamino)ethyl)-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C20H28Cl2N4OS
|
1
|
| 1 |
IC50 = 73600 nM
|
|
|
|
CP0887415
|
(+/-)-N-(1-(pyrrolidin-3-yl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C19H26Cl2N4S
|
1
|
| 1 |
IC50 = 75000 nM
|
|
|
|
CP0746845
|
S-[2-[(1-Iminoethyl)aminolethyl]-2-methyl-L-cysteine dihydrochloride
Show/Hide
|
C7H18Cl2N4O2S
|
1
|
| 1 |
IC50 = 77000 nM
|
|
|
|
CP0873763
|
cis-(+/-)-N-(3-(3-(methylamino)cyclohexyl)-1H-indol-5-yl)thiophene-2-carboximidamide hydrochloride
Show/Hide
|
C20H25ClN4S
|
1
|
| 1 |
IC50 = 77600 nM
|
|
|
|
CP0902857
|
S-[2-[(1-Iminoethyl)amino]ethyl]-2-ethyl-L-cysteine dihydrochloride
Show/Hide
|
C8H20Cl2N4O2S
|
1
|
| 1 |
IC50 = 78000 nM
|
|
|
|
CP0864145
|
N-(1-(2-(pyrrolidin-1-yl)ethyl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C21H30Cl2N4S
|
1
|
| 1 |
IC50 = 82200 nM
|
|
|
|
CP0448315
|
N'-[1-(oxan-4-yl)-2,3-dihydroindol-6-yl]thiophene-2-carboximidamide
Show/Hide
|
C18H21N3OS
|
1
|
| 1 |
IC50 = 84800 nM
|
|
|
|
CP0896819
|
N-(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)furan-2-carboximidamide dihydrochloride
Show/Hide
|
C19H24Cl2N4O
|
1
|
| 1 |
IC50 = 97400 nM
|
|
|
|
CP0403595
|
N'-(1-piperidin-4-yl-2,3-dihydroindol-6-yl)thiophene-2-carboximidamide
Show/Hide
|
C18H22N4S
|
1
|
| 1 |
IC50 = 99000 nM
|
|
|
|
CP0688010
|
N-(1-(2-(dimethylamino)ethyl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-7-yl)thiophene-2-carboximidamide dihydrochloride
Show/Hide
|
C19H28Cl2N4S
|
1
|
| 1 |
IC50 = 99100 nM
|
|
|
|
CP0743881
|
S-[2-(1-Iminoethylamino)ethyl]-2-methyl-(D/L)-cysteine bistrifluoroacetate
Show/Hide
|
C11H18F6N4O6S
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0938036
|
(2R)-2-Amino-3[[2-[(1-iminoethyl)amino]ethyl]sulfinyl]-2-methylpropanoicacid dihydrochloride
Show/Hide
|
C7H18Cl2N4O3S
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
