| Compound ID |
Compound Name |
Compound Formula |
|
CP0002393
|
3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino)piperidin-1-yl)-3-oxopropanenitrile
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|
C16H20N6O
|
1
|
| 1 |
IC50 = 52 nM
|
|
|
|
CP0009734
|
4-amino-2-(4-morpholin-4-ylphenyl)thieno[3,2-c]pyridine-7-carboxamide
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|
C18H18N4O2S
|
1
|
| 1 |
IC50 = 66 nM
|
|
|
|
CP0392929
|
4-amino-2-[4-(2-cyanopropan-2-yl)phenyl]-N-methylthieno[3,2-c]pyridine-7-carboxamide
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|
C19H18N4OS
|
1
|
| 1 |
IC50 = 146 nM
|
|
|
|
CP0393021
|
4-amino-2-(4-tert-butylphenyl)-N-methylthieno[3,2-c]pyridine-7-carboxamide
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|
C19H21N3OS
|
1
|
| 1 |
IC50 = 202 nM
|
|
|
|
CP0441325
|
4-amino-N-methyl-2-[4-(trifluoromethoxy)phenyl]thieno[3,2-c]pyridine-7-carboxamide
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|
C16H12F3N3O2S
|
1
|
| 1 |
IC50 = 208 nM
|
|
|
|
CP0008918
|
4-amino-2-[4-(tert-butylsulfamoyl)phenyl]-N-methylthieno[3,2-c]pyridine-7-carboxamide
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|
C19H22N4O3S2
|
1
|
| 1 |
IC50 = 266 nM
|
|
|
|
CP0001805
|
4-amino-2-[4-(tert-butylsulfamoyl)phenyl]-N-(2-morpholin-4-ylethyl)thieno[3,2-c]pyridine-7-carboxamide
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|
C24H31N5O4S2
|
1
|
| 1 |
IC50 = 757 nM
|
|
|
|
CP0392981
|
4-amino-N-methyl-2-(4-methylphenyl)thieno[3,2-c]pyridine-7-carboxamide
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|
C16H15N3OS
|
1
|
| 1 |
IC50 = 888 nM
|
|
|
|
CP0388710
|
4-amino-2-[4-(tert-butylsulfamoyl)phenyl]-N-(2-hydroxyethyl)thieno[3,2-c]pyridine-7-carboxamide
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|
C20H24N4O4S2
|
1
|
| 1 |
IC50 = 932 nM
|
|
|
|
CP0392977
|
4-amino-N-methyl-2-phenylthieno[3,2-c]pyridine-7-carboxamide
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|
C15H13N3OS
|
1
|
| 1 |
IC50 = 937 nM
|
|
|
|
CP0417019
|
4-amino-N-ethyl-2-(4-morpholin-4-ylphenyl)thieno[3,2-c]pyridine-7-carboxamide
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|
C20H22N4O2S
|
1
|
| 1 |
IC50 = 1070 nM
|
|
|
|
CP0441323
|
4-amino-N-methyl-2-(4-morpholin-4-ylphenyl)thieno[3,2-c]pyridine-7-carboxamide
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|
C19H20N4O2S
|
1
|
| 1 |
IC50 = 1330 nM
|
|
|
|
CP0001781
|
4-amino-2-[4-(tert-butylsulfamoyl)phenyl]-N-(2-methoxyethyl)thieno[3,2-c]pyridine-7-carboxamide
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|
C21H26N4O4S2
|
1
|
| 1 |
IC50 = 1480 nM
|
|
|
|
CP0417018
|
4-amino-2-[4-(tert-butylsulfamoyl)phenyl]-N-(3-morpholin-4-ylpropyl)thieno[3,2-c]pyridine-7-carboxamide
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|
C25H33N5O4S2
|
1
|
| 1 |
IC50 = 1550 nM
|
|
|
|
CP0441326
|
4-amino-2-(4-morpholin-4-ylphenyl)-N-phenylthieno[3,2-c]pyridine-7-carboxamide
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|
C24H22N4O2S
|
1
|
| 1 |
IC50 = 1990 nM
|
|
|
|
CP0441324
|
4-amino-N-benzyl-2-(4-morpholin-4-ylphenyl)thieno[3,2-c]pyridine-7-carboxamide
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|
C25H24N4O2S
|
1
|
| 1 |
IC50 = 2600 nM
|
|
|
|
CP0417017
|
4-amino-2-[4-(tert-butylsulfamoyl)phenyl]-N-(2-piperidin-1-ylethyl)thieno[3,2-c]pyridine-7-carboxamide
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|
C25H33N5O3S2
|
1
|
| 1 |
IC50 = 2670 nM
|
|
|
|
CP0001071
|
4-amino-2-[4-(tert-butylsulfamoyl)phenyl]-N-[2-(dimethylamino)ethyl]thieno[3,2-c]pyridine-7-carboxamide
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|
C22H29N5O3S2
|
1
|
| 1 |
IC50 = 4100 nM
|
|
|
|
CP0427742
|
4-amino-N,N-dimethyl-2-(4-morpholin-4-ylphenyl)thieno[3,2-c]pyridine-7-carboxamide
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|
C20H22N4O2S
|
1
|
| 1 |
IC50 = 5150 nM
|
|
|
|
CP0452168
|
4-amino-N-tert-butyl-2-(4-morpholin-4-ylphenyl)thieno[3,2-c]pyridine-7-carboxamide
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|
C22H26N4O2S
|
1
|
| 1 |
IC50 = 6980 nM
|
|
|
|
CP0382724
|
3-(2,2-difluoro-10,12-dimethyl-1-aza-3-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-3,5,7,9,11-pentaen-4-yl)-N-[2-[2-[2-[2-[[(2S,3R,4R,6R)-3-methoxy-2-methyl-16-oxo-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-4-yl]amino]ethoxy]ethoxy]ethoxy]ethyl]propanamide
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|
C49H54BF2N7O7
|
1
|
| 1 |
Kd = 8 nM
|
|
|
|
CP0382649
|
3-(2,2-difluoro-10,12-dimethyl-1-aza-3-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-3,5,7,9,11-pentaen-4-yl)-N-[2-[2-[2-[2-[[(2S,3R,4R,6R)-3-methoxy-2-methyl-16-oxo-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-4-yl]-methylamino]ethoxy]ethoxy]ethoxy]ethyl]propanamide
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|
C50H56BF2N7O7
|
1
|
| 1 |
Kd = 49 nM
|
|
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