| Compound ID |
Compound Name |
Compound Formula |
|
CP0564578
|
2-[2-(2,4-difluorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazole-8-carboxamide
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|
C20H13F2N5O2S
|
1
|
| 1 |
IC50 = 1.7 nM
|
|
|
|
CP0550417
|
N-[6-[4-(2-chlorophenyl)-1,2,4-triazol-3-yl]isoquinolin-3-yl]-2-fluorocyclopropane-1-carboxamide
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|
C21H15ClFN5O
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0570964
|
N-[4-[(7R)-4-oxo-7-propan-2-yl-6,7-dihydro-5H-pyrazolo[1,5-a]pyrazin-2-yl]pyridin-2-yl]cyclopropanecarboxamide
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|
C18H21N5O2
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0576970
|
N-(4-imidazo[1,2-a]pyridin-7-ylpyridin-2-yl)cyclopropanecarboxamide
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|
C16H14N4O
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0543610
|
(R)-2-((R)-3-methylmorpholino)-6-(trifluoromethyl)-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5H)-one
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|
C12H15F3N4O2
|
1
|
| 1 |
IC50 = 37 nM
|
|
|
|
CP0571364
|
(R)-7-(tert-butyl)-2-((R)-3-methylmorpholino)-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5H)-one
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|
C15H24N4O2
|
1
|
| 1 |
IC50 = 43 nM
|
|
|
|
CP0571798
|
N-[5-methyl-4-[(7R)-4-oxo-7-propan-2-yl-6,7-dihydro-5H-pyrazolo[1,5-a]pyrazin-2-yl]pyridin-2-yl]cyclopropanecarboxamide
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|
C19H23N5O2
|
1
|
| 1 |
IC50 = 48 nM
|
|
|
|
CP0577592
|
N-[4-(benzimidazol-1-yl)pyridin-2-yl]cyclopropanecarboxamide
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|
C16H14N4O
|
1
|
| 1 |
IC50 = 53 nM
|
|
|
|
CP0569807
|
(R)-7-isopropyl-2-((R)-3-methylmorpholino)-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5H)-one
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|
C14H22N4O2
|
1
|
| 1 |
IC50 = 78 nM
|
|
|
|
CP0577891
|
(5aS,8aR)-2-((R)-3-methylmorpholino)-5,5a,6,7,8,8a-hexahydro-4H-cyclopenta[e]pyrazolo[1,5-a]pyrazin-4-one
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|
C14H20N4O2
|
1
|
| 1 |
IC50 = 83 nM
|
|
|
|
CP0580148
|
(R)-7'-cyclopropyl-2'-((R)-3-methylmorpholino)-7'H-spiro[cyclopropane-1,6'-pyrazolo[1,5-a]pyrazin]-4'(5'H)-one
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|
C16H22N4O2
|
1
|
| 1 |
IC50 = 84 nM
|
|
|
|
CP0577005
|
(S)-2-((R)-3-methylmorpholino)-7-(trifluoromethyl)-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5H)-one
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|
C12H15F3N4O2
|
1
|
| 1 |
IC50 = 92 nM
|
|
|
|
CP0564579
|
2-[2-(2,4-difluorophenyl)-1,2,4-triazol-3-yl]-4-methyl-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazole-8-carboxamide
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|
C21H15F2N5O2S
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0577004
|
N-[4-[(7R)-7-methyl-4-oxo-6,7-dihydro-5H-pyrazolo[1,5-a]pyrazin-2-yl]pyridin-2-yl]cyclopropanecarboxamide
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|
C16H17N5O2
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0550418
|
(S)-7-(2-hydroxypropan-2-yl)-2-((R)-3-methylmorpholino)-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5H)-one
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|
C14H22N4O3
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0578494
|
(6S,7R)-7-cyclopropyl-6-methyl-2-((R)-3-methylmorpholino)-6,7- dihydropyrazolo[1,5-a]pyrazin-4(5H)-one
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|
C15H22N4O2
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0571362
|
(7R)-7-cyclopropyl-2-[(3R)-3-methylmorpholin-4-yl]-6,7-dihydro-5H-pyrazolo[1,5-a]pyrazin-4-one
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|
C14H20N4O2
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0571363
|
(R)-7-cyclobutyl-2-((R)-3-methylmorpholino)-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5H)-one
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|
C15H22N4O2
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0576945
|
2-[[2-(cyclopropanecarbonylamino)pyridin-4-yl]amino]benzamide
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|
C16H16N4O2
|
1
|
| 1 |
IC50 = 320 nM
|
|
|
|
CP0578672
|
(R)-7-cyclopentyl-2-((R)-3-methylmorpholino)-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5H)-one
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|
C16H24N4O2
|
1
|
| 1 |
IC50 = 350 nM
|
|
|
|
CP0578822
|
N-[4-(1-methyl-2-oxopyridin-4-yl)pyridin-2-yl]cyclopropanecarboxamide
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|
C15H15N3O2
|
1
|
| 1 |
IC50 = 470 nM
|
|
|
|
CP0577609
|
(6S,7R)-6,7-dicyclopropyl-2-((R)-3-methylmorpholino)-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5H)-one
Show/Hide
|
C17H24N4O2
|
1
|
| 1 |
IC50 = 560 nM
|
|
|
|
CP0564576
|
(7R)-2-morpholin-4-yl-7-propan-2-yl-6,7-dihydro-5H-pyrazolo[1,5-a]pyrazin-4-one
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|
C13H20N4O2
|
1
|
| 1 |
IC50 = 710 nM
|
|
|
|
CP0564577
|
(R)-7-cyclopropyl-6,6-dimethyl-2-((R)-3-methylmorpholino)-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5H)-one
Show/Hide
|
C16H24N4O2
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
