| Compound ID |
Compound Name |
Compound Formula |
|
CP0508188
|
16-methylsulfonyl-6-(trifluoromethyl)-2,4,8,14,16,25-hexazatetracyclo[18.3.1.13,7.010,15]pentacosa-1(23),3,5,7(25),10(15),11,13,20(24),21-nonaene
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C21H21F3N6O2S
|
1
|
| 1 |
IC50 = 0.67 nM
|
|
|
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CP0532758
|
4-[(18E)-16-methylsulfonyl-6-(trifluoromethyl)-2,4,8,14,16,25-hexazatetracyclo[18.3.1.13,7.010,15]pentacosa-1(24),3,5,7(25),10(15),11,13,18,20,22-decaen-21-yl]morpholine
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|
C25H26F3N7O3S
|
1
|
| 1 |
IC50 = 0.84 nM
|
|
|
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CP0508490
|
16-methylsulfonyl-26-(trifluoromethyl)-2,10,16,24,28,29-hexazapentacyclo[23.3.1.13,7.06,10.017,22]triaconta-1(28),3(30),4,6,17,19,21,25(29),26-nonaen-11-one
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|
C26H27F3N6O3S
|
1
|
| 1 |
IC50 = 0.9 nM
|
|
|
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CP0508489
|
4-[16-methylsulfonyl-6-(trifluoromethyl)-2,4,8,14,16,25-hexazatetracyclo[18.3.1.13,7.010,15]pentacosa-1(24),3,5,7(25),10(15),11,13,20,22-nonaen-21-yl]morpholine
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|
C25H28F3N7O3S
|
1
|
| 1 |
IC50 = 1.31 nM
|
|
|
|
CP0516060
|
24-methyl-16-methylsulfonyl-26-(trifluoromethyl)-2,10,16,24,28,29-hexazapentacyclo[23.3.1.13,7.06,10.017,22]triaconta-1(28),3(30),4,6,17,19,21,25(29),26-nonaen-11-one
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|
C27H29F3N6O3S
|
1
|
| 1 |
IC50 = 1.5 nM
|
|
|
|
CP0408956
|
4-[(18E)-8-methyl-16-methylsulfonyl-6-(trifluoromethyl)-2,4,8,14,16,25-hexazatetracyclo[18.3.1.13,7.010,15]pentacosa-1(24),3,5,7(25),10(15),11,13,18,20,22-decaen-21-yl]morpholine
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|
C26H28F3N7O3S
|
1
|
| 1 |
IC50 = 1.55 nM
|
|
|
|
CP0408955
|
16-ethylsulfonyl-26-(trifluoromethyl)-2,10,16,24,28,29-hexazapentacyclo[23.3.1.13,7.06,10.017,22]triaconta-1(28),3(30),4,6,17,19,21,25(29),26-nonaen-11-one
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|
C27H29F3N6O3S
|
1
|
| 1 |
IC50 = 1.9 nM
|
|
|
|
CP0511808
|
(18E)-16-methylsulfonyl-6-(trifluoromethyl)-2,4,8,14,16,25-hexazatetracyclo[18.3.1.13,7.010,15]pentacosa-1(23),3,5,7(25),10(15),11,13,18,20(24),21-decaene
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|
C21H19F3N6O2S
|
1
|
| 1 |
IC50 = 2.6 nM
|
|
|
|
CP0377487
|
4-[(18E)-8-methyl-16-methylsulfonyl-6-(trifluoromethyl)-2,4,8,13,16,25-hexazatetracyclo[18.3.1.13,7.010,15]pentacosa-1(24),3,5,7(25),10(15),11,13,18,20,22-decaen-21-yl]morpholine
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|
C26H28F3N7O3S
|
1
|
| 1 |
IC50 = 2.7 nM
|
|
|
|
CP0446131
|
16-methylsulfonyl-26-(trifluoromethyl)-2,10,16,18,24,28,29-heptazapentacyclo[23.3.1.13,7.06,10.017,22]triaconta-1(28),3(30),4,6,17(22),18,20,25(29),26-nonaen-11-one
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|
C25H26F3N7O3S
|
1
|
| 1 |
IC50 = 3.1 nM
|
|
|
|
CP0539694
|
16,16-dioxo-26-(trifluoromethyl)-16lambda6-thia-2,10,15,18,24,28,29-heptazapentacyclo[23.3.1.13,7.06,10.017,22]triaconta-1(28),3(30),4,6,17(22),18,20,25(29),26-nonaen-11-one
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|
C23H22F3N7O3S
|
1
|
| 1 |
IC50 = 3.5 nM
|
|
|
|
CP0153321
|
N-methyl-N-[3-[[[2-[(2-oxo-1,3-dihydroindol-5-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamide
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|
C21H20F3N7O3S
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0451767
|
N-[3-[[[2-(3-bromo-4-morpholin-4-ylanilino)-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-N-prop-2-enylmethanesulfonamide
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|
C25H27BrF3N7O3S
|
1
|
| 1 |
IC50 = 19.5 nM
|
|
|
|
CP0377488
|
18-methylsulfonyl-28-(trifluoromethyl)-2,10,18,20,26,30,31-heptazahexacyclo[25.3.1.13,7.112,16.06,10.019,24]tritriaconta-1(30),3(33),4,6,12,14,16(32),19(24),20,22,27(31),28-dodecaen-11-one
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|
C28H24F3N7O3S
|
1
|
| 1 |
IC50 = 26 nM
|
|
|
|
CP0451775
|
15-methylsulfonyl-25-(trifluoromethyl)-2,10,15,17,23,27,28-heptazapentacyclo[22.3.1.13,7.06,10.016,21]nonacosa-1(27),3(29),4,6,16(21),17,19,24(28),25-nonaen-11-one
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|
C24H24F3N7O3S
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0516061
|
N-[3-[[[2-(3-bromoanilino)-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-N-prop-2-enylmethanesulfonamide
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|
C21H20BrF3N6O2S
|
1
|
| 1 |
IC50 = 122 nM
|
|
|
|
CP0545412
|
5-[2-[[[2-(2,3-dihydro-1H-indol-5-ylamino)-5-(trifluoromethyl)pyrimidin-4-yl]-methylamino]methyl]-N-methylsulfonylanilino]pentanoic acid
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|
C27H31F3N6O4S
|
1
|
| 1 |
IC50 = 201 nM
|
|
|
|
CP0545411
|
5-[2-[[[2-(2,3-dihydro-1H-indol-5-ylamino)-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]-N-ethylsulfonylanilino]pentanoic acid
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|
C27H31F3N6O4S
|
1
|
| 1 |
IC50 = 256 nM
|
|
|
|
CP0454688
|
N-[4-[[[2-(3-bromo-4-morpholin-4-ylanilino)-5-(trifluoromethyl)pyrimidin-4-yl]-methylamino]methyl]pyridin-3-yl]-N-prop-2-enylmethanesulfonamide
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|
C26H29BrF3N7O3S
|
1
|
| 1 |
IC50 = 6625 nM
|
|
|
