Compound ID |
Compound Name |
Compound Formula |
CP0781525
|
1-[[1-[(2S,3R,5R)-2-(hydroxymethyl)-5-(5-methyl-2,4-dioxo-pyrimidin-1-yl)tetrahydrofuran-3-yl]triazol-4-yl]methyl]-3-(3-sulfamoylphenyl)urea
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|
C20H24N8O7S
|
1
|
1 |
IC50 = 2200 nM
|
|
|
CP0913154
|
[1-[(2S,3R,5R)-2-(hydroxymethyl)-5-(5-methyl-2,4-dioxo-pyrimidin-1-yl)tetrahydrofuran-3-yl]triazol-4-yl]methyl 4-sulfamoylbenzoate
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|
C20H22N6O8S
|
1
|
1 |
IC50 = 9500 nM
|
|
|
CP0964507
|
4-[[1-[(2S,3R,5R)-2-(hydroxymethyl)-5-(5-methyl-2,4-dioxo-pyrimidin-1-yl)tetrahydrofuran-3-yl]triazol-4-yl]methoxy]benzenesulfonamide
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|
C19H22N6O7S
|
1
|
1 |
IC50 = 18400 nM
|
|
|
CP0781526
|
1-[(2R,4R,5S)-5-(hydroxymethyl)-4-[4-[(2-oxochromen-6-yl)oxymethyl]triazol-1-yl]tetrahydrofuran-2-yl]-5-methyl-pyrimidine-2,4-dione
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|
C22H21N5O7
|
1
|
1 |
IC50 = 28600 nM
|
|
|
CP0917647
|
1-[(2R,4R,5S)-4-[4-[(2,2-dioxo-1,2$l^6-benzoxathiin-6-yl)oxymethyl]triazol-1-yl]-5-(hydroxymethyl)tetrahydrofuran-2-yl]-5-methyl-pyrimidine-2,4-dione
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|
C21H21N5O8S
|
1
|
1 |
IC50 = 65000 nM
|
|
|