Brief Information of the Cell Line and Protein
Cell Line ID: CL000007 , HT-29
Synonyms
HT 29
HT29
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0320
Protein ID: PT00955 , DNA-dependent protein kinase catalytic subunit
Gene Name PRKDC
Organism Homo sapiens, Human
Protein Classification Kinase
Uniprot ID P78527
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000007  Protein ID: PT00955
 
Compound ID Compound Name Compound Formula
CP0068243
(3R)-4-[2-(1H-indol-4-yl)-6-(1-methylsulfonylcyclopropyl)pyrimidin-4-yl]-3-methylmorpholine
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C21H24N4O3S
 1
1
IC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0068244
(3R)-3-methyl-4-[6-(1-methylsulfonylcyclopropyl)-2-(1H-pyrrolo[2,3-c]pyridin-4-yl)pyrimidin-4-yl]morpholine
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C20H23N5O3S
 1
1
IC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0068245
N-methyl-1-[4-[(3R)-3-methylmorpholin-4-yl]-6-(1-methylsulfonylcyclopropyl)pyrimidin-2-yl]benzimidazol-2-amine
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C21H26N6O3S
 1
1
IC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0669285
US8552004, 2.03
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C21H27N7O2S
 1
1
IC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0808811
CERALASERTIB
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C20H24N6O2S
 1
1
IC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0180776
6-[6-(methoxymethyl)pyridin-3-yl]-4-[[(1S)-1-(oxan-4-yl)ethyl]amino]quinoline-3-carboxamide
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C24H28N4O3
 1
1
IC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0180777
7-fluoro-6-[6-(methoxymethyl)pyridin-3-yl]-4-[[(1S)-1-(1-methylpyrazol-3-yl)ethyl]amino]quinoline-3-carboxamide
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C23H23FN6O2
 1
1
IC50 > 30000 nM
   TI
   LI
   LO
   TS