Brief Information of the Cell Line and Protein
Cell Line ID: CL000007 , HT-29
Synonyms
HT 29
HT29
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0320
Protein ID: PT00845 , RAC-alpha serine/threonine-protein kinase
Gene Name AKT1
Organism Homo sapiens, Human
Protein Classification Kinase
Uniprot ID P31749
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000007  Protein ID: PT00845
 
Compound ID Compound Name Compound Formula
CP0255330
US9320734, 415
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C17H19N5O7S2
 1
1
IC50 = 1000 nM
   TI
   LI
   LO
   TS
CP0323003
US9320734, 389
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C20H16ClN7O4S2
 1
1
IC50 = 5000 nM
   TI
   LI
   LO
   TS
CP0052017
4-Amino-N-[1,3,4]thiadiazol-2-yl-benzenesulfonamide
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C8H8N4O2S2
 1
1
IC50 = 20000 nM
   TI
   LI
   LO
   TS
CP0294317
US9320734, 316
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C21H16ClN7O4S
 1
1
IC50 = 24000 nM
   TI
   LI
   LO
   TS
CP0038251
N-[4-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfamoyl]phenyl]naphthalene-2-sulfonamide
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C19H16N4O4S3
 1
1
IC50 = 25000 nM
   TI
   LI
   LO
   TS
CP0564090
US9320734, 441
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C16H15NO4
 1
1
IC50 = 25000 nM
   TI
   LI
   LO
   TS
CP0419170
US9320734, 439
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C21H16N2O4
 1
1
IC50 = 50000 nM
   TI
   LI
   LO
   TS
CP0419171
US9320734, 450
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C14H16N4O5S
 1
1
IC50 = 50000 nM
   TI
   LI
   LO
   TS
CP0515145
US9320734, 444
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C16H16N4O5S
 1
1
IC50 = 50000 nM
   TI
   LI
   LO
   TS
CP0517510
US9320734, 456
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C14H14N6O6S4
 1
1
IC50 = 50000 nM
   TI
   LI
   LO
   TS
CP0555984
US9320734, 445
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C17H16N4O6S
 1
1
IC50 = 50000 nM
   TI
   LI
   LO
   TS
CP0095764
N-[4-(1,3,4-thiadiazol-2-ylsulfamoyl)phenyl]acetamide
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C10H10N4O3S2
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
CP0240356
2-[2-(2-methoxyethoxy)ethoxy]-N-[4-(1,3,4-thiadiazol-2-ylsulfamoyl)phenyl]acetamide
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C15H20N4O6S2
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
CP0402482
US9320734, 345
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C11H9N5O4S3
 1
1
IC50 = 50000 nM
   TI
   LI
   LO
   TS