Brief Information of the Cell Line and Protein
Cell Line ID: CL000006 , HEK293
Synonyms
Hek293
HEK-293
HEK/293
HEK 293
HEK;293
293
293 HEK
293 Ad5
Graham 293
Graham-293
Human Embryonic Kidney 293
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0045
Protein ID: PT07126 , Apolipoprotein L1
Gene Name APOL1
Organism Homo sapiens, Human
Protein Classification Unclassified protein
Uniprot ID O14791
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000006  Protein ID: PT07126
 
Compound ID Compound Name Compound Formula
CP0902820
3-[5,7-difluoro-2-(4-fluorophenyl)-1H-indol-3-yl]-N-[(3S,4S)-4-hydroxy-2-oxo-pyrrolidin-3-yl]propanamide
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C21H18F3N3O3
 1
1
IC50 < 250 nM
   TI
   LI
   LO
   TS
CP0902821
N-[(3S,4R)-4-hydroxy-2-oxo-pyrrolidin-3-yl]-3-[2-(4-methoxyphenyl)-1H-indol-3-yl]propanamide
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C22H23N3O4
 1
1
IC50 < 250 nM
   TI
   LI
   LO
   TS
CP0947392
3-[7-cyano-5-fluoro-2-(4-fluorophenyl)-1H-indol-3-yl]-N-[(3S,4R)-4-hydroxy-2-oxo-pyrrolidin-3-yl]propanamide
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C22H18F2N4O3
 1
1
IC50 < 250 nM
   TI
   LI
   LO
   TS
CP0950477
3-[2-(4-cyanophenyl)-5,7-difluoro-1H-indol-3-yl]-N-[(3S)-2-oxopyrrolidin-3-yl]propanamide
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C22H18F2N4O2
 1
1
IC50 < 250 nM
   TI
   LI
   LO
   TS
CP0957907
3-(7-fluoro-2-phenyl-1H-indol-3-yl)-N-[(3S,4R)-4-hydroxy-2-oxo-pyrrolidin-3-yl]propanamide
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C21H20FN3O3
 1
1
IC50 < 250 nM
   TI
   LI
   LO
   TS
CP0957908
3-(5,6-difluoro-2-phenyl-1H-indol-3-yl)-N-[(3S,4R)-4-hydroxy-2-oxo-pyrrolidin-3-yl]propanamide
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C21H19F2N3O3
 1
1
IC50 < 250 nM
   TI
   LI
   LO
   TS