| Compound ID |
Compound Name |
Compound Formula |
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CP0463365
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(2R)-N'-(3,5-difluorophenyl)-2-methyl-N-[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]butanediamide
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C23H24F2N4O3
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
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CP0001342
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benzyl N-[(2S)-4-methyl-1-[[(2S)-4-methyl-1-[[3-[[(2S)-4-methyl-2-[[(2S)-4-methyl-2-(phenylmethoxycarbonylamino)pentanoyl]amino]pentanoyl]amino]-2-oxopropyl]amino]-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]carbamate
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|
C43H64N6O9
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
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CP0013350
|
N-[(2S,3S)-3-amino-2-hydroxy-3-phenylpropyl]-3-tert-butyl-N-cyclobutylbenzenesulfonamide
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|
C23H32N2O3S
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
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CP0013376
|
N-[(2S,3S)-3-amino-2-hydroxy-3-[4-(trifluoromethoxy)phenyl]propyl]-4-tert-butyl-N-cyclobutylbenzenesulfonamide
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|
C24H31F3N2O4S
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
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CP0000571
|
(2S)-2-((S)-2-(3,5-difluorophenyl)-2-hydroxyacetamido)-N-((7S)-5-methyl-6-oxo-6,7-dihydro-5H-dibenzo[b,d]azepin-7-yl)propanamide
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|
C26H23F2N3O4
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
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CP0014645
|
N-[(2S,3S)-3-amino-2-hydroxy-3-phenylpropyl]-N-cyclobutyl-5,5,8,8-tetramethyl-6,7-dihydronaphthalene-2-sulfonamide
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|
C27H38N2O3S
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
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CP0007975
|
N-[(2S,3S)-3-amino-2-hydroxy-3-phenylpropyl]-3,4-dichloro-N-cycloheptylbenzenesulfonamide
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|
C22H28Cl2N2O3S
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
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CP0013293
|
N-[(2S,3S)-3-amino-2-hydroxy-3-phenylpropyl]-4-tert-butyl-N-cyclobutylbenzenesulfonamide
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|
C23H32N2O3S
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
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CP0430084
|
(2R)-2-methyl-N'-(2-methylphenyl)-N-[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]butanediamide
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|
C24H28N4O3
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
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CP0328884
|
(2R)-N'-(5-fluoro-2-methylpyridin-3-yl)-2-methyl-N-[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]butanediamide
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|
C23H26FN5O3
|
1
|
| 1 |
IC50 = 44 nM
|
|
|
|
CP0495110
|
(2R)-2-methyl-N'-(3-methylphenyl)-N-[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]butanediamide
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|
C24H28N4O3
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0408802
|
(2R)-N'-(5-fluoro-2-methylpyridin-3-yl)-N-[(6S)-10-fluoro-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]-2-methylbutanediamide
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|
C23H25F2N5O3
|
1
|
| 1 |
IC50 = 76 nM
|
|
|
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CP0460550
|
(2S)-2-cyclopropyl-N-[(6S)-5,11-dioxospiro[3,6-dihydro-1H-pyrazolo[1,2-b][2,3]benzodiazepine-2,1'-cyclopropane]-6-yl]-N'-(5-fluoro-2-methylpyridin-3-yl)butanediamide
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|
C27H28FN5O4
|
1
|
| 1 |
IC50 = 77 nM
|
|
|
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CP0013292
|
N-[(2S,3S)-3-amino-2-hydroxy-3-phenylpropyl]-3,4-dichloro-N-cyclobutylbenzenesulfonamide
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|
C19H22Cl2N2O3S
|
1
|
| 1 |
IC50 = 88 nM
|
|
|
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CP0011744
|
N-[(2S,3S)-3-amino-2-hydroxy-3-phenylpropyl]-3,4-dichloro-N-(2-methylpropyl)benzenesulfonamide
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|
C19H24Cl2N2O3S
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
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CP0481546
|
(2S)-2-cyclopropyl-N-[(6S)-5,11-dioxo-1,2,3,6-tetrahydropyrazolo[1,2-b][2,3]benzodiazepin-6-yl]-N'-(5-fluoro-2-methylpyridin-3-yl)butanediamide
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|
C25H26FN5O4
|
1
|
| 1 |
IC50 = 225 nM
|
|
|
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CP0013349
|
N-[(2S,3S)-3-amino-2-hydroxy-3-phenylpropyl]-3,4-dichloro-N-propan-2-yloxybenzenesulfonamide
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|
C18H22Cl2N2O4S
|
1
|
| 1 |
IC50 = 350 nM
|
|
|
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CP0013291
|
N-[(2S,3S)-3-amino-2-hydroxy-3-phenylpropyl]-N-benzyl-3,4-dichlorobenzenesulfonamide
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|
C22H22Cl2N2O3S
|
1
|
| 1 |
IC50 = 620 nM
|
|
|
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CP0007976
|
N-[(2S,3S)-3-amino-2-hydroxy-3-phenylpropyl]-N-cyclobutyl-1,3-benzothiazole-5-sulfonamide
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|
C20H23N3O3S2
|
1
|
| 1 |
IC50 = 840 nM
|
|
|
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CP0512502
|
N-[(2S,3S)-3-amino-2-hydroxy-4-phenylbutyl]-3,4-dichloro-N-(2-methylpropyl)benzenesulfonamide
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|
C20H26Cl2N2O3S
|
1
|
| 1 |
IC50 = 860 nM
|
|
|
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CP0481547
|
(2R)-N-[(6S)-5,11-dioxo-1,2,3,6-tetrahydropyrazolo[1,2-b][2,3]benzodiazepin-6-yl]-N'-(5-fluoro-2-methylpyridin-3-yl)-2-methylbutanediamide
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|
C23H24FN5O4
|
1
|
| 1 |
IC50 = 870 nM
|
|
|
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CP0014400
|
N-[(2S,3S)-3-amino-2-hydroxy-3-phenylpropyl]-3,4-dichloro-N-(1-methylcyclobutyl)benzenesulfonamide
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|
C20H24Cl2N2O3S
|
1
|
| 1 |
IC50 = 900 nM
|
|
|
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CP0014314
|
N-[(2S,3S)-3-amino-2-hydroxy-3-phenylpropyl]-3,4-dichloro-N-(2-hydroxy-2-methylpropyl)benzenesulfonamide
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|
C19H24Cl2N2O4S
|
1
|
| 1 |
IC50 = 910 nM
|
|
|
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CP0478246
|
(2R)-2-methyl-N'-(2-methylpyridin-3-yl)-N-[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]butanediamide
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|
C23H27N5O3
|
1
|
| 1 |
IC50 = 1020 nM
|
|
|
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CP0481545
|
(2R)-2-methyl-N'-(4-methylphenyl)-N-[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]butanediamide
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|
C24H28N4O3
|
1
|
| 1 |
IC50 = 1390 nM
|
|
|
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CP0013374
|
N-[(2S,3S)-3-amino-2-hydroxy-3-phenylpropyl]-3,4-dichloro-N-(oxetan-3-yl)benzenesulfonamide
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|
C18H20Cl2N2O4S
|
1
|
| 1 |
IC50 = 1500 nM
|
|
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CP0463364
|
(2R)-2-methyl-N-[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]-N'-[2-(trifluoromethyl)phenyl]butanediamide
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|
C24H25F3N4O3
|
1
|
| 1 |
IC50 = 2850 nM
|
|
|
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CP0512501
|
benzyl N-[(2S,3S)-4-[(3,4-dichlorophenyl)sulfonyl-(2-methylpropyl)amino]-3-hydroxy-1-phenylbutan-2-yl]carbamate
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|
C28H32Cl2N2O5S
|
1
|
| 1 |
IC50 = 4300 nM
|
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