Brief Information of the Compound and Protein
Compound Name
(2R)-N-[(6S)-5,11-dioxo-1,2,3,6-tetrahydropyrazolo[1,2-b][2,3]benzodiazepin-6-yl]-N'-(5-fluoro-2-methylpyridin-3-yl)-2-methylbutanediamide
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PubChem ID
CID: 137649442
Canonical SMILES
C[C@H](CC(=O)Nc1cc(F)cnc1C)C(=O)N[C@H]1c2ccccc2C(=O)N2CCCN2C1=O
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Compound Formula C23H24FN5O4
Compound Structure
Protein Name
Signal peptide peptidase-like 2A
Protein Classification
Enzyme
>
Hydrolase
Uniprot ID
Q8TCT8
Gene Name
SPPL2A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 870 nM
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