Brief Information of the Cell Line and Protein
Cell Line ID: CL000006 , HEK293
Synonyms
Hek293
HEK-293
HEK/293
HEK 293
HEK;293
293
293 HEK
293 Ad5
Graham 293
Graham-293
Human Embryonic Kidney 293
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0045
Protein ID: PT05986 , Mas-related G-protein coupled receptor member X1
Gene Name MRGPRX1
Organism Rattus norvegicus, Rat
Protein Classification Membrane receptor
Uniprot ID Q8R4G1
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000006  Protein ID: PT05986
 
Compound ID Compound Name Compound Formula
CP0719182
(5S,8S,11S,14S,17S,20S,23S,26S,29S,32S)-26,29-bis((1H-indol-3-yl)methyl)-32-((S)-1-((S)-2-(2-((S)-2-amino-3-methylbutanamido)acetamido)-5-guanidinopentanoyl)pyrrolidine-2-carboxamido)-14-(3-amino-3-oxopropyl)-11-(4-aminobutyl)-20-(carboxymethyl)-8-(3-guanidinopropyl)-5,17-bis(4-hydroxybenzyl)-23-(2-(methylthio)ethyl)-4,7,10,13,16,19,22,25,28,31-decaoxo-3,6,9,12,15,18,21,24,27,30-decaazapentatriacontane-1,35-dioic acid
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C91H127N25O23S
 1
1
EC50 = 316.23 nM
   TI
   LI
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CP0536802
(2R)-2-amino-N-[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]-3-[4-(diaminomethylideneamino)phenyl]propanamide
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C19H24N6O2
 1
1
EC50 = 630.96 nM
   TI
   LI
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   TS
CP0551488
(2S)-2-[[2-amino-2-(1-carbamimidoylpiperidin-4-yl)acetyl]amino]-3-phenylpropanamide
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C17H26N6O2
 1
1
EC50 = 3981.07 nM
   TI
   LI
   LO
   TS
CP0179651
Adamantane-1-carboxylic acid [(S)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-4-guanidino-butyl]-amide
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C26H38N6O3
 1
1
EC50 = 6309.57 nM
   TI
   LI
   LO
   TS
CP0455916
(2S)-2-amino-N-[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]-5-(diaminomethylideneamino)pentanamide
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C15H24N6O2
 1
1
EC50 = 6309.57 nM
   TI
   LI
   LO
   TS
CP0379135
(2S)-2-amino-N-[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]-3-[4-(diaminomethylideneamino)phenyl]propanamide
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C19H24N6O2
 1
1
EC50 = 50118.72 nM
   TI
   LI
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   TS
CP0379134
(2S)-2-[[2-amino-2-[3-(diaminomethylideneamino)phenyl]acetyl]amino]-3-phenylpropanamide
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C18H22N6O2
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0379754
(2S,4S)-N-[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]-4-[(diaminomethylideneamino)methyl]pyrrolidine-2-carboxamide
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C16H24N6O2
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0520596
(2S,4S)-N-[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]-4-(diaminomethylideneamino)pyrrolidine-2-carboxamide
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C15H22N6O2
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0071244
4-(6-methoxypyridin-3-yl)-N-[2-methyl-3-[(6-oxo-4-piperazin-1-ylpyridazin-1-yl)methyl]phenyl]benzamide
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C29H30N6O3
 1
1
EC50 > 1995.26 nM
   TI
   LI
   LO
   TS