Brief Information of the Cell Line and Protein
Cell Line ID: CL000006 , HEK293
Synonyms
Hek293
HEK-293
HEK/293
HEK 293
HEK;293
293
293 HEK
293 Ad5
Graham 293
Graham-293
Human Embryonic Kidney 293
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0045
Protein ID: PT05750 , Protein Wnt-3a
Gene Name WNT3A
Organism Mus musculus, Mouse
Protein Classification Secreted protein
Uniprot ID P27467
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000006  Protein ID: PT05750
 
Compound ID Compound Name Compound Formula
CP0666603
4-((1R,2R,6S,7R)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-N-quinolin-8-yl-benzamide
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C25H19N3O3
 1
1
IC50 = 77 nM
   TI
   LI
   LO
   TS
CP0053018
2-(4-(Trifluoromethyl)phenyl)-7,8-dihydro-5H-thiopyrano-[4,3-d]pyrimidin-4-ol
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C14H11F3N2OS
 1
1
IC50 = 78 nM
   TI
   LI
   LO
   TS
CP0056588
3-(3,4-dimethoxyphenyl)-5-[[4-(4-methoxyphenyl)-5-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,2,4-oxadiazole
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C21H21N5O4S
 1
1
IC50 = 126 nM
   TI
   LI
   LO
   TS
CP0070829
3-(4-methoxyphenyl)-5-[[4-(4-methoxyphenyl)-5-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,2,4-oxadiazole
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C20H19N5O3S
 1
1
IC50 = 215 nM
   TI
   LI
   LO
   TS
CP0056599
3-(4-methoxyphenyl)-5-[[4-(4-methoxyphenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,2,4-oxadiazole
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C24H20N6O3S
 1
1
IC50 = 341 nM
   TI
   LI
   LO
   TS
CP0064177
5-[[4-(4-methoxyphenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]sulfanylmethyl]-3-(4-methylphenyl)-1,2,4-oxadiazole
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C24H20N6O2S
 1
1
IC50 = 548 nM
   TI
   LI
   LO
   TS
CP0056596
5-[[4-(4-ethoxyphenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]sulfanylmethyl]-3-(4-methoxyphenyl)-1,2,4-oxadiazole
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C25H22N6O3S
 1
1
IC50 = 919 nM
   TI
   LI
   LO
   TS
CP0550531
5-[[4-(4-methoxyphenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]sulfanylmethyl]-3-phenyl-1,2,4-oxadiazole
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C23H18N6O2S
 1
1
IC50 = 1060 nM
   TI
   LI
   LO
   TS
CP0380973
CHEMBL1459534
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C21H18N2O6
 1
1
IC50 = 1170 nM
   TI
   LI
   LO
   TS