Compound ID |
Compound Name |
Compound Formula |
CP0466905
|
US9012651, 223
Show/Hide
|
C18H24F4N2O
|
1
|
1 |
IC50 = 80 nM
|
|
|
CP0479325
|
US9012651, 247
Show/Hide
|
C17H19F3N2O
|
1
|
1 |
IC50 = 80 nM
|
|
|
CP0546074
|
US9012651, 97
Show/Hide
|
C20H25F2N3O
|
1
|
1 |
IC50 = 110 nM
|
|
|
CP0481157
|
US9012651, 294
Show/Hide
|
C17H19ClF2N2O
|
1
|
1 |
IC50 = 120 nM
|
|
|
CP0510275
|
US9012651, 273
Show/Hide
|
C24H30FN3O3
|
1
|
1 |
IC50 = 120 nM
|
|
|
CP0518952
|
US9012651, 94
Show/Hide
|
C19H23F2N3O
|
1
|
1 |
IC50 = 120 nM
|
|
|
CP0476959
|
US9012651, 289
Show/Hide
|
C19H21FN2O
|
1
|
1 |
IC50 = 130 nM
|
|
|
CP0479324
|
US9012651, 224
Show/Hide
|
C17H23F3N2O
|
1
|
1 |
IC50 = 140 nM
|
|
|
CP0520580
|
US9012651, 228
Show/Hide
|
C17H19F3N2O
|
1
|
1 |
IC50 = 140 nM
|
|
|
CP0526387
|
US9012651, 73
Show/Hide
|
C17H19F4N3O
|
1
|
1 |
IC50 = 140 nM
|
|
|
CP0546075
|
US9012651, 99
Show/Hide
|
C20H25F2N3O
|
1
|
1 |
IC50 = 140 nM
|
|
|
CP0423336
|
US9012651, 246
Show/Hide
|
C17H18F4N2O
|
1
|
1 |
IC50 = 160 nM
|
|
|
CP0441638
|
US9012651, 244
Show/Hide
|
C17H18F4N2O
|
1
|
1 |
IC50 = 160 nM
|
|
|
CP0478177
|
US9012651, 245
Show/Hide
|
C17H18F4N2O
|
1
|
1 |
IC50 = 160 nM
|
|
|
CP0516705
|
US9012651, 71
Show/Hide
|
C19H24FN3O
|
1
|
1 |
IC50 = 160 nM
|
|
|
CP0504004
|
US9012651, 290
Show/Hide
|
C16H18F4N2OS
|
1
|
1 |
IC50 = 170 nM
|
|
|
CP0510276
|
US9012651, 288
Show/Hide
|
C21H31FN2O
|
1
|
1 |
IC50 = 170 nM
|
|
|
CP0549875
|
US9012651, 264
Show/Hide
|
C19H21FN2O
|
1
|
1 |
IC50 = 170 nM
|
|
|
CP0469814
|
US9012651, 70
Show/Hide
|
C20H26FN3O
|
1
|
1 |
IC50 = 180 nM
|
|
|
CP0510274
|
US9012651, 267
Show/Hide
|
C18H20F4N2O
|
1
|
1 |
IC50 = 180 nM
|
|
|
CP0484031
|
US9012651, 61
Show/Hide
|
C22H32FN3O3S
|
1
|
1 |
IC50 = 190 nM
|
|
|
CP0520725
|
US9012651, 265
Show/Hide
|
C19H20F2N2O
|
1
|
1 |
IC50 = 190 nM
|
|
|
CP0570687
|
US9012651, 17
Show/Hide
|
C18H20F4N2O
|
1
|
1 |
IC50 = 200 nM
|
|
|
CP0520505
|
US9012651, 272
Show/Hide
|
C20H20F6N2O
|
1
|
1 |
IC50 = 220 nM
|
|
|
CP0548929
|
US9012651, 66
Show/Hide
|
C17H25F4N3O
|
1
|
1 |
IC50 = 220 nM
|
|
|
CP0490182
|
US9012651, 255
Show/Hide
|
C19H21FN2OS
|
1
|
1 |
IC50 = 230 nM
|
|
|
CP0501522
|
US9012651, 19
Show/Hide
|
C18H20F4N2O2
|
1
|
1 |
IC50 = 230 nM
|
|
|
CP0549982
|
US9012651, 280
Show/Hide
|
C18H22F2N2O
|
1
|
1 |
IC50 = 250 nM
|
|
|
CP0488714
|
US9012651, 283
Show/Hide
|
C18H21F3N2O2
|
1
|
1 |
IC50 = 260 nM
|
|
|
CP0508947
|
US9012651, 274
Show/Hide
|
C19H22FN3O
|
1
|
1 |
IC50 = 260 nM
|
|
|
CP0512637
|
US9012651, 103
Show/Hide
|
C21H25F4N3O
|
1
|
1 |
IC50 = 260 nM
|
|
|
CP0547614
|
US9012651, 93
Show/Hide
|
C19H23F2N3O
|
1
|
1 |
IC50 = 270 nM
|
|
|
CP0493271
|
US9012651, 292
Show/Hide
|
C17H19F4N3O
|
1
|
1 |
IC50 = 280 nM
|
|
|
CP0484029
|
US9012651, 47
Show/Hide
|
C18H19ClF4N2O
|
1
|
1 |
IC50 = 290 nM
|
|
|
CP0519531
|
US9012651, 80
Show/Hide
|
C19H20F4N2O
|
1
|
1 |
IC50 = 290 nM
|
|
|
CP0520723
|
US9012651, 258
Show/Hide
|
C18H26F4N2O
|
1
|
1 |
IC50 = 290 nM
|
|
|
CP0549979
|
US9012651, 238
Show/Hide
|
C19H20F2N2O
|
1
|
1 |
IC50 = 290 nM
|
|
|
CP0425574
|
US9012651, 260
Show/Hide
|
C20H23FN4O
|
1
|
1 |
IC50 = 300 nM
|
|
|
CP0469815
|
US9012651, 86
Show/Hide
|
C17H18F4N2O
|
1
|
1 |
IC50 = 300 nM
|
|
|
CP0443729
|
US9012651, 216
Show/Hide
|
C18H26F4N2O
|
1
|
1 |
IC50 = 310 nM
|
|
|
CP0525186
|
US9012651, 27
Show/Hide
|
C17H20F2N2O
|
1
|
1 |
IC50 = 320 nM
|
|
|
CP0548928
|
US9012651, 65
Show/Hide
|
C17H25F4N3O
|
1
|
1 |
IC50 = 320 nM
|
|
|
CP0563964
|
US9012651, 98
Show/Hide
|
C20H25F2N3O
|
1
|
1 |
IC50 = 320 nM
|
|
|
CP0483687
|
US9012651, 48
Show/Hide
|
C22H30FN3O3S
|
1
|
1 |
IC50 = 330 nM
|
|
|
CP0526392
|
US9012651, 96
Show/Hide
|
C20H23F4N3O
|
1
|
1 |
IC50 = 330 nM
|
|
|
CP0490183
|
US9012651, 257
Show/Hide
|
C18H26F4N2O
|
1
|
1 |
IC50 = 340 nM
|
|
|
CP0518602
|
US9012651, 95
Show/Hide
|
C19H23ClFN3O
|
1
|
1 |
IC50 = 340 nM
|
|
|
CP0443730
|
US9012651, 217
Show/Hide
|
C21H27FN2O
|
1
|
1 |
IC50 = 350 nM
|
|
|
CP0493231
|
US9012651, 249
Show/Hide
|
C20H24FN3O
|
1
|
1 |
IC50 = 350 nM
|
|
|
CP0570663
|
US9012651, 102
Show/Hide
|
C21H25F4N3O
|
1
|
1 |
IC50 = 350 nM
|
|
|
CP0553591
|
US9012651, 129
Show/Hide
|
C18H29FN2O
|
1
|
1 |
IC50 = 360 nM
|
|
|
CP0510273
|
US9012651, 229
Show/Hide
|
C19H21FN2OS
|
1
|
1 |
IC50 = 370 nM
|
|
|
CP0520137
|
US9012651, 239
Show/Hide
|
C19H23F3N2O
|
1
|
1 |
IC50 = 370 nM
|
|
|
CP0520726
|
US9012651, 282
Show/Hide
|
C18H19F5N2O
|
1
|
1 |
IC50 = 370 nM
|
|
|
CP0441637
|
US9012651, 243
Show/Hide
|
C16H21FN2OS
|
1
|
1 |
IC50 = 380 nM
|
|
|
CP0493230
|
US9012651, 233
Show/Hide
|
C19H22F2N2O
|
1
|
1 |
IC50 = 380 nM
|
|
|
CP0518950
|
US9012651, 42
Show/Hide
|
C17H20ClFN2O
|
1
|
1 |
IC50 = 390 nM
|
|
|
CP0549876
|
US9012651, 266
Show/Hide
|
C18H20ClFN2O
|
1
|
1 |
IC50 = 390 nM
|
|
|
CP0567817
|
US9012651, 281
Show/Hide
|
C18H19F5N2O
|
1
|
1 |
IC50 = 390 nM
|
|
|
CP0520503
|
US9012651, 29
Show/Hide
|
C18H18F4N2O
|
1
|
1 |
IC50 = 410 nM
|
|
|
CP0560092
|
US9012651, 242
Show/Hide
|
C15H18ClFN2OS
|
1
|
1 |
IC50 = 410 nM
|
|
|
CP0425575
|
US9012651, 268
Show/Hide
|
C19H20F4N2O
|
1
|
1 |
IC50 = 420 nM
|
|
|
CP0520582
|
US9012651, 256
Show/Hide
|
C19H21FN2O2
|
1
|
1 |
IC50 = 420 nM
|
|
|
CP0546073
|
US9012651, 67
Show/Hide
|
C16H23F4N3O
|
1
|
1 |
IC50 = 420 nM
|
|
|
CP0450817
|
US9012651, 269
Show/Hide
|
C18H20FN3O
|
1
|
1 |
IC50 = 440 nM
|
|
|
CP0462622
|
US9012651, 131
Show/Hide
|
C17H19F4N3O
|
1
|
1 |
IC50 = 460 nM
|
|
|
CP0469812
|
US9012651, 43
Show/Hide
|
C19H26FN3O
|
1
|
1 |
IC50 = 460 nM
|
|
|
CP0548926
|
US9012651, 53
Show/Hide
|
C19H22F4N2O2
|
1
|
1 |
IC50 = 460 nM
|
|
|
CP0563962
|
US9012651, 83
Show/Hide
|
C18H20F4N2O
|
1
|
1 |
IC50 = 460 nM
|
|
|
CP0472337
|
US9012651, 128
Show/Hide
|
C19H24F2N2O
|
1
|
1 |
IC50 = 480 nM
|
|
|
CP0526385
|
US9012651, 64
Show/Hide
|
C20H24FN3O
|
1
|
1 |
IC50 = 480 nM
|
|
|
CP0549983
|
US9012651, 220
Show/Hide
|
C16H25FN2O
|
1
|
1 |
IC50 = 480 nM
|
|
|
CP0565671
|
US9012651, 49
Show/Hide
|
C21H28FN3O
|
1
|
1 |
IC50 = 480 nM
|
|
|
CP0518603
|
US9012651, 101
Show/Hide
|
C20H25ClFN3O
|
1
|
1 |
IC50 = 500 nM
|
|
|
CP0525190
|
US9012651, 57
Show/Hide
|
C19H26FN3O2
|
1
|
1 |
IC50 = 500 nM
|
|
|
CP0573329
|
US9012651, 51
Show/Hide
|
C21H30FN3O3S
|
1
|
1 |
IC50 = 500 nM
|
|
|
CP0422564
|
US9012651, 240
Show/Hide
|
C19H27FN2O
|
1
|
1 |
IC50 = 510 nM
|
|
|
CP0462620
|
US9012651, 115
Show/Hide
|
C17H19F4N3O
|
1
|
1 |
IC50 = 510 nM
|
|
|
CP0563963
|
US9012651, 89
Show/Hide
|
C18H21F4N3O
|
1
|
1 |
IC50 = 510 nM
|
|
|
CP0519532
|
US9012651, 85
Show/Hide
|
C19H22F4N2O
|
1
|
1 |
IC50 = 520 nM
|
|
|
CP0520727
|
US9012651, 286
Show/Hide
|
C19H21ClN2O
|
1
|
1 |
IC50 = 520 nM
|
|
|
CP0556154
|
US9012651, 284
Show/Hide
|
C19H20F2N2O
|
1
|
1 |
IC50 = 520 nM
|
|
|
CP0567812
|
US9012651, 259
Show/Hide
|
C31H36FN3O4
|
1
|
1 |
IC50 = 520 nM
|
|
|
CP0549409
|
US9012651, 203
Show/Hide
|
C17H25F3N2O
|
1
|
1 |
IC50 = 530 nM
|
|
|
CP0539058
|
US9012651, 77
Show/Hide
|
C17H18F4N2O
|
1
|
1 |
IC50 = 540 nM
|
|
|
CP0565673
|
US9012651, 108
Show/Hide
|
C18H21F4N3O
|
1
|
1 |
IC50 = 540 nM
|
|
|
CP0520728
|
US9012651, 293
Show/Hide
|
C19H19F7N2O
|
1
|
1 |
IC50 = 550 nM
|
|
|
CP0567814
|
US9012651, 270
Show/Hide
|
C19H20F6N2O
|
1
|
1 |
IC50 = 550 nM
|
|
|
CP0539356
|
US9012651, 88
Show/Hide
|
C20H23F4N3O
|
1
|
1 |
IC50 = 570 nM
|
|
|
CP0423337
|
US9012651, 251
Show/Hide
|
C15H19FN2O2
|
1
|
1 |
IC50 = 580 nM
|
|
|
CP0554244
|
US9012651, 271
Show/Hide
|
C20H20F6N2O
|
1
|
1 |
IC50 = 580 nM
|
|
|
CP0470312
|
US9012651, 68
Show/Hide
|
C18H21F4N3O2
|
1
|
1 |
IC50 = 590 nM
|
|
|
CP0559179
|
US9012651, 226
Show/Hide
|
C20H30N2OSi
|
1
|
1 |
IC50 = 600 nM
|
|
|
CP0519534
|
US9012651, 110
Show/Hide
|
C17H19ClF3N3O
|
1
|
1 |
IC50 = 630 nM
|
|
|
CP0563961
|
US9012651, 59
Show/Hide
|
C19H22F4N2O3S
|
1
|
1 |
IC50 = 630 nM
|
|
|
CP0567815
|
US9012651, 277
Show/Hide
|
C24H34FN3O2
|
1
|
1 |
IC50 = 650 nM
|
|
|
CP0570689
|
US9012651, 25
Show/Hide
|
C20H26F2N2O2
|
1
|
1 |
IC50 = 650 nM
|
|
|
CP0429121
|
US9012651, 219
Show/Hide
|
C21H34FN3O3
|
1
|
1 |
IC50 = 660 nM
|
|
|
CP0518957
|
US9012651, 207
Show/Hide
|
C17H20F3N3O3S
|
1
|
1 |
IC50 = 680 nM
|
|
|
CP0526389
|
US9012651, 81
Show/Hide
|
C20H22F4N2O
|
1
|
1 |
IC50 = 680 nM
|
|
|
CP0484024
|
US9012651, 23
Show/Hide
|
C20H26F2N2O2
|
1
|
1 |
IC50 = 700 nM
|
|
|
CP0509048
|
US9012651, 253
Show/Hide
|
C21H29FN4O2
|
1
|
1 |
IC50 = 700 nM
|
|
|
CP0526390
|
US9012651, 84
Show/Hide
|
C21H24F4N2O
|
1
|
1 |
IC50 = 700 nM
|
|
|
CP0539059
|
US9012651, 107
Show/Hide
|
C19H22F4N2O
|
1
|
1 |
IC50 = 700 nM
|
|
|
CP0544920
|
US9012651, 79
Show/Hide
|
C18H18F4N2O
|
1
|
1 |
IC50 = 700 nM
|
|
|
CP0499870
|
US9012651, 222
Show/Hide
|
C20H32FN3O3
|
1
|
1 |
IC50 = 710 nM
|
|
|
CP0509079
|
US9012651, 287
Show/Hide
|
C21H24FN3OS
|
1
|
1 |
IC50 = 730 nM
|
|
|
CP0472336
|
US9012651, 126
Show/Hide
|
C17H25FN2O
|
1
|
1 |
IC50 = 740 nM
|
|
|
CP0480068
|
US9012651, 24
Show/Hide
|
C20H27FN2O2
|
1
|
1 |
IC50 = 750 nM
|
|
|
CP0567813
|
US9012651, 261
Show/Hide
|
C17H24FN5O
|
1
|
1 |
IC50 = 750 nM
|
|
|
CP0548927
|
US9012651, 54
Show/Hide
|
C21H28FN3O4S
|
1
|
1 |
IC50 = 760 nM
|
|
|
CP0512643
|
US9012651, 201
Show/Hide
|
C19H31FN2O
|
1
|
1 |
IC50 = 770 nM
|
|
|
CP0468036
|
US9012651, 202
Show/Hide
|
C19H31FN2O
|
1
|
1 |
IC50 = 790 nM
|
|
|
CP0510272
|
US9012651, 213
Show/Hide
|
C21H35FN2O
|
1
|
1 |
IC50 = 790 nM
|
|
|
CP0567818
|
US9012651, 291
Show/Hide
|
C16H20F4N4O
|
1
|
1 |
IC50 = 790 nM
|
|
|
CP0484022
|
US9012651, 14
Show/Hide
|
C17H20F2N2O
|
1
|
1 |
IC50 = 810 nM
|
|
|
CP0520138
|
US9012651, 262
Show/Hide
|
C21H29ClN2O2
|
1
|
1 |
IC50 = 810 nM
|
|
|
CP0525189
|
US9012651, 44
Show/Hide
|
C21H28FN3O2
|
1
|
1 |
IC50 = 830 nM
|
|
|
CP0573326
|
US9012651, 12
Show/Hide
|
C18H24N2O2
|
1
|
1 |
IC50 = 910 nM
|
|
|
CP0539060
|
US9012651, 124
Show/Hide
|
C19H23FN2O
|
1
|
1 |
IC50 = 920 nM
|
|
|
CP0567816
|
US9012651, 279
Show/Hide
|
C18H19F2N3O
|
1
|
1 |
IC50 = 940 nM
|
|
|
CP0484025
|
US9012651, 28
Show/Hide
|
C17H19F4N3O
|
1
|
1 |
IC50 = 950 nM
|
|
|
CP0519529
|
US9012651, 36
Show/Hide
|
C16H19F2N3O
|
1
|
1 |
IC50 = 950 nM
|
|
|
CP0472335
|
US9012651, 92
Show/Hide
|
C16H24F3N3O
|
1
|
1 |
IC50 = 960 nM
|
|
|
CP0423334
|
US9012651, 236
Show/Hide
|
C20H29FN2O
|
1
|
1 |
IC50 = 980 nM
|
|
|
CP0503638
|
US9012651, 285
Show/Hide
|
C19H21FN2O
|
1
|
1 |
IC50 = 990 nM
|
|
|
CP0526405
|
US9012651, 200
Show/Hide
|
C18H29FN2O
|
1
|
1 |
IC50 = 1030 nM
|
|
|
CP0484033
|
US9012651, 111
Show/Hide
|
C18H22F3N3O
|
1
|
1 |
IC50 = 1070 nM
|
|
|
CP0518601
|
US9012651, 60
Show/Hide
|
C21H28FN3O3S
|
1
|
1 |
IC50 = 1080 nM
|
|
|
CP0509047
|
US9012651, 235
Show/Hide
|
C20H23FN2O2
|
1
|
1 |
IC50 = 1110 nM
|
|
|
CP0565669
|
US9012651, 16
Show/Hide
|
C18H20F4N2O
|
1
|
1 |
IC50 = 1110 nM
|
|
|
CP0512632
|
US9012651, 13
Show/Hide
|
C17H20F2N2O
|
1
|
1 |
IC50 = 1120 nM
|
|
|
CP0570688
|
US9012651, 18
Show/Hide
|
C18H20F4N2O2
|
1
|
1 |
IC50 = 1120 nM
|
|
|
CP0484027
|
US9012651, 37
Show/Hide
|
C19H22F2N2O2
|
1
|
1 |
IC50 = 1190 nM
|
|
|
CP0516707
|
US9012651, 206
Show/Hide
|
C19H31FN2O
|
1
|
1 |
IC50 = 1230 nM
|
|
|
CP0526393
|
US9012651, 106
Show/Hide
|
C19H23F4N3O
|
1
|
1 |
IC50 = 1260 nM
|
|
|
CP0548925
|
US9012651, 22
Show/Hide
|
C19H19F7N2O
|
1
|
1 |
IC50 = 1280 nM
|
|
|
CP0509077
|
US9012651, 275
Show/Hide
|
C24H32FN3O2
|
1
|
1 |
IC50 = 1330 nM
|
|
|
CP0518596
|
US9012651, 20
Show/Hide
|
C17H19Cl2FN2O
|
1
|
1 |
IC50 = 1390 nM
|
|
|
CP0525188
|
US9012651, 34
Show/Hide
|
C16H20ClN3O
|
1
|
1 |
IC50 = 1390 nM
|
|
|
CP0573328
|
US9012651, 40
Show/Hide
|
C19H23FN2O2
|
1
|
1 |
IC50 = 1400 nM
|
|
|
CP0483688
|
US9012651, 52
Show/Hide
|
C25H34FN3O2
|
1
|
1 |
IC50 = 1420 nM
|
|
|
CP0484037
|
US9012651, 127
Show/Hide
|
C19H25FN2O
|
1
|
1 |
IC50 = 1440 nM
|
|
|
CP0549980
|
US9012651, 248
Show/Hide
|
C20H24FN3O
|
1
|
1 |
IC50 = 1440 nM
|
|
|
CP0539363
|
US9012651, 209
Show/Hide
|
C16H18F3N3O3S
|
1
|
1 |
IC50 = 1470 nM
|
|
|
CP0563960
|
US9012651, 58
Show/Hide
|
C26H30FN3O2
|
1
|
1 |
IC50 = 1490 nM
|
|
|
CP0554243
|
US9012651, 234
Show/Hide
|
C18H20FN3OS
|
1
|
1 |
IC50 = 1520 nM
|
|
|
CP0524581
|
US9012651, 231
Show/Hide
|
C15H23F3N4O
|
1
|
1 |
IC50 = 1530 nM
|
|
|
CP0563972
|
US9012651, 199
Show/Hide
|
C18H27FN2O
|
1
|
1 |
IC50 = 1590 nM
|
|
|
CP0462618
|
US9012651, 76
Show/Hide
|
C18H19F4N3O2
|
1
|
1 |
IC50 = 1600 nM
|
|
|
CP0564358
|
US9012651, 125
Show/Hide
|
C19H22F2N2O
|
1
|
1 |
IC50 = 1630 nM
|
|
|
CP0484032
|
US9012651, 82
Show/Hide
|
C16H16F4N2O
|
1
|
1 |
IC50 = 1640 nM
|
|
|
CP0573327
|
US9012651, 39
Show/Hide
|
C19H26FN3O3S
|
1
|
1 |
IC50 = 1700 nM
|
|
|
CP0469813
|
US9012651, 63
Show/Hide
|
C20H24FN3O
|
1
|
1 |
IC50 = 1740 nM
|
|
|
CP0484030
|
US9012651, 50
Show/Hide
|
C20H28FN3O3S
|
1
|
1 |
IC50 = 1770 nM
|
|
|
CP0501523
|
US9012651, 56
Show/Hide
|
C24H34FN3O2
|
1
|
1 |
IC50 = 1780 nM
|
|
|
CP0509046
|
US9012651, 227
Show/Hide
|
C21H34N2OSSi
|
1
|
1 |
IC50 = 1800 nM
|
|
|
CP0501521
|
US9012651, 15
Show/Hide
|
C17H20ClFN2O
|
1
|
1 |
IC50 = 1840 nM
|
|
|
CP0478176
|
US9012651, 241
Show/Hide
|
C23H29FN2O
|
1
|
1 |
IC50 = 1860 nM
|
|
|
CP0526396
|
US9012651, 148
Show/Hide
|
C16H18F3N3O
|
1
|
1 |
IC50 = 1870 nM
|
|
|
CP0523913
|
US9012651, 11
Show/Hide
|
C16H27N3O
|
1
|
1 |
IC50 = 1940 nM
|
|
|
CP0484028
|
US9012651, 46
Show/Hide
|
C24H32FN3O2
|
1
|
1 |
IC50 = 2020 nM
|
|
|
CP0468040
|
US9012651, 55
Show/Hide
|
C20H27FN4O2
|
1
|
1 |
IC50 = 2160 nM
|
|
|
CP0523915
|
US9012651, 31
Show/Hide
|
C17H19F4N3O
|
1
|
1 |
IC50 = 2190 nM
|
|
|
CP0484034
|
US9012651, 114
Show/Hide
|
C17H20F4N4O2
|
1
|
1 |
IC50 = 2330 nM
|
|
|
CP0525187
|
US9012651, 33
Show/Hide
|
C17H20F3N3O
|
1
|
1 |
IC50 = 2360 nM
|
|
|
CP0526386
|
US9012651, 72
Show/Hide
|
C20H22FN3O
|
1
|
1 |
IC50 = 2390 nM
|
|
|
CP0468037
|
US9012651, 205
Show/Hide
|
C21H34FN3O3
|
1
|
1 |
IC50 = 2460 nM
|
|
|
CP0518958
|
US9012651, 212
Show/Hide
|
C16H18F3N3O4S
|
1
|
1 |
IC50 = 2530 nM
|
|
|
CP0503996
|
US9012651, 130
Show/Hide
|
C26H22F4N4O2
|
1
|
1 |
IC50 = 2550 nM
|
|
|
CP0518951
|
US9012651, 90
Show/Hide
|
C16H17F4N3O
|
1
|
1 |
IC50 = 2590 nM
|
|
|
CP0523912
|
US9012651, 8
Show/Hide
|
C18H21F3N2O
|
1
|
1 |
IC50 = 2600 nM
|
|
|
CP0570664
|
US9012651, 113
Show/Hide
|
C16H18F4N4O
|
1
|
1 |
IC50 = 2650 nM
|
|
|
CP0479326
|
US9012651, 278
Show/Hide
|
C16H19ClFN3O
|
1
|
1 |
IC50 = 2690 nM
|
|
|
CP0565672
|
US9012651, 105
Show/Hide
|
C20H24F4N2O
|
1
|
1 |
IC50 = 2760 nM
|
|
|
CP0570690
|
US9012651, 38
Show/Hide
|
C16H19ClFN3O
|
1
|
1 |
IC50 = 2850 nM
|
|
|
CP0466906
|
US9012651, 225
Show/Hide
|
C17H22N2O
|
1
|
1 |
IC50 = 2920 nM
|
|
|
CP0468035
|
US9012651, 184
Show/Hide
|
C16H19F3N4O
|
1
|
1 |
IC50 = 2940 nM
|
|
|
CP0565670
|
US9012651, 41
Show/Hide
|
C22H30FN3O2
|
1
|
1 |
IC50 = 2970 nM
|
|
|
CP0565667
|
US9012651, 4
Show/Hide
|
C19H21F3N2O
|
1
|
1 |
IC50 = 3000 nM
|
|
|
CP0539057
|
US9012651, 75
Show/Hide
|
C17H17F4N3O
|
1
|
1 |
IC50 = 3020 nM
|
|
|
CP0462623
|
US9012651, 138
Show/Hide
|
C16H18F3N3O
|
1
|
1 |
IC50 = 3050 nM
|
|
|
CP0469816
|
US9012651, 145
Show/Hide
|
C17H18F3N3O
|
1
|
1 |
IC50 = 3050 nM
|
|
|
CP0472334
|
US9012651, 87
Show/Hide
|
C17H19F4N3O
|
1
|
1 |
IC50 = 3100 nM
|
|
|
CP0519013
|
US9012651, 7
Show/Hide
|
C19H21F3N2O
|
1
|
1 |
IC50 = 3250 nM
|
|
|
CP0523914
|
US9012651, 21
Show/Hide
|
C17H19Cl2FN2O
|
1
|
1 |
IC50 = 3300 nM
|
|
|
CP0518600
|
US9012651, 45
Show/Hide
|
C23H30FN3O2
|
1
|
1 |
IC50 = 3470 nM
|
|
|
CP0512639
|
US9012651, 109
Show/Hide
|
C17H19F4N3O
|
1
|
1 |
IC50 = 3590 nM
|
|
|
CP0525191
|
US9012651, 74
Show/Hide
|
C17H18F4N2O2
|
1
|
1 |
IC50 = 3680 nM
|
|
|
CP0569110
|
US9012651, 6
Show/Hide
|
C19H21F3N2O
|
1
|
1 |
IC50 = 3700 nM
|
|
|
CP0480066
|
US9012651, 5
Show/Hide
|
C19H21F3N2O
|
1
|
1 |
IC50 = 3710 nM
|
|
|
CP0519530
|
US9012651, 69
Show/Hide
|
C17H20F3N3O
|
1
|
1 |
IC50 = 3720 nM
|
|
|
CP0565668
|
US9012651, 10
Show/Hide
|
C15H25N3O
|
1
|
1 |
IC50 = 3790 nM
|
|
|
CP0573325
|
US9012651, 2
Show/Hide
|
C19H23F3N2O
|
1
|
1 |
IC50 = 3810 nM
|
|
|
CP0484039
|
US9012651, 150
Show/Hide
|
C16H18F3N3O2
|
1
|
1 |
IC50 = 3820 nM
|
|
|
CP0518954
|
US9012651, 122
Show/Hide
|
C18H19F4N3O
|
1
|
1 |
IC50 = 3940 nM
|
|
|
CP0573330
|
US9012651, 62
Show/Hide
|
C22H28FN3O2S
|
1
|
1 |
IC50 = 4000 nM
|
|
|
CP0484021
|
US9012651, 1
Show/Hide
|
C19H21F3N2O
|
1
|
1 |
IC50 = 4020 nM
|
|
|
CP0568595
|
US9012651, 26
Show/Hide
|
C16H28N2O2
|
1
|
1 |
IC50 = 4060 nM
|
|
|
CP0462624
|
US9012651, 141
Show/Hide
|
C17H20F3N3O
|
1
|
1 |
IC50 = 4900 nM
|
|
|
CP0526401
|
US9012651, 172
Show/Hide
|
C18H20F3N3O
|
1
|
1 |
IC50 = 4930 nM
|
|
|
CP0539061
|
US9012651, 171
Show/Hide
|
C18H20F3N3O
|
1
|
1 |
IC50 = 5510 nM
|
|
|
CP0559178
|
US9012651, 215
Show/Hide
|
C19H29FN2O3
|
1
|
1 |
IC50 = 5670 nM
|
|
|
CP0508943
|
US9012651, 237
Show/Hide
|
C19H28N2OSi
|
1
|
1 |
IC50 = 5750 nM
|
|
|
CP0560091
|
US9012651, 170
Show/Hide
|
C20H22F3N3O
|
1
|
1 |
IC50 = 6160 nM
|
|
|
CP0484036
|
US9012651, 121
Show/Hide
|
C16H17F4N3O2
|
1
|
1 |
IC50 = 6180 nM
|
|
|
CP0563968
|
US9012651, 147
Show/Hide
|
C18H22F3N3O
|
1
|
1 |
IC50 = 6430 nM
|
|
|
CP0564360
|
US9012651, 142
Show/Hide
|
C18H22F3N3O
|
1
|
1 |
IC50 = 7300 nM
|
|
|
CP0563967
|
US9012651, 137
Show/Hide
|
C15H16F3N3O
|
1
|
1 |
IC50 = 7830 nM
|
|
|
CP0520504
|
US9012651, 139
Show/Hide
|
C20H18F3N3O
|
1
|
1 |
IC50 = 8080 nM
|
|
|
CP0462615
|
US9012651, 190
Show/Hide
|
C15H17F3N4O
|
1
|
1 |
IC50 = 8150 nM
|
|
|
CP0475241
|
US9012651, 214
Show/Hide
|
C19H29FN2O3
|
1
|
1 |
IC50 = 8280 nM
|
|
|
CP0565675
|
US9012651, 123
Show/Hide
|
C18H19F4N3O
|
1
|
1 |
IC50 = 8550 nM
|
|
|
CP0539358
|
US9012651, 146
Show/Hide
|
C20H24F3N3O
|
1
|
1 |
IC50 = 8650 nM
|
|
|
CP0526397
|
US9012651, 153
Show/Hide
|
C21H20F3N3O2
|
1
|
1 |
IC50 = 9310 nM
|
|
|
CP0472338
|
US9012651, 133
Show/Hide
|
C18H20F3N3O
|
1
|
1 |
IC50 = 9320 nM
|
|
|
CP0469810
|
US9012651, 3
Show/Hide
|
C18H21F3N2O
|
1
|
1 |
IC50 = 9380 nM
|
|
|
CP0526388
|
US9012651, 78
Show/Hide
|
C16H17F4N3O
|
1
|
1 |
IC50 = 10200 nM
|
|
|
CP0493269
|
US9012651, 276
Show/Hide
|
C22H28FN3O2
|
1
|
1 |
IC50 = 10900 nM
|
|
|
CP0564359
|
US9012651, 134
Show/Hide
|
C19H22F3N3O
|
1
|
1 |
IC50 = 11000 nM
|
|
|
CP0469811
|
US9012651, 32
Show/Hide
|
C16H20FN3O
|
1
|
1 |
IC50 = 12000 nM
|
|
|
CP0526395
|
US9012651, 143
Show/Hide
|
C18H22F3N3O
|
1
|
1 |
IC50 = 12400 nM
|
|
|
CP0468038
|
US9012651, 208
Show/Hide
|
C19H22F3N3O3S
|
1
|
1 |
IC50 = 13500 nM
|
|
|
CP0565674
|
US9012651, 112
Show/Hide
|
C18H22F3N3O2
|
1
|
1 |
IC50 = 15300 nM
|
|
|
CP0484038
|
US9012651, 144
Show/Hide
|
C16H18F3N3O2
|
1
|
1 |
IC50 = 15600 nM
|
|
|
CP0468033
|
US9012651, 159
Show/Hide
|
C20H24F3N3O
|
1
|
1 |
IC50 = 17600 nM
|
|
|
CP0548931
|
US9012651, 210
Show/Hide
|
C16H18F3N3O4S
|
1
|
1 |
IC50 = 18500 nM
|
|
|
CP0423338
|
US9012651, 254
Show/Hide
|
C21H30FN5O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0462611
|
US9012651, 177
Show/Hide
|
C18H20F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0462614
|
US9012651, 187
Show/Hide
|
C15H17F3N4O2
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0462617
|
US9012651, 30
Show/Hide
|
C18H20F4N2O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0468034
|
US9012651, 164
Show/Hide
|
C21H20F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0472326
|
US9012651, 185
Show/Hide
|
C18H21F3N4O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0472327
|
US9012651, 189
Show/Hide
|
C16H19F3N4O2
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0472328
|
US9012651, 198
Show/Hide
|
C15H17F3N4O2
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0479352
|
US9012651, 120
Show/Hide
|
C16H16F4N4O2
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0484035
|
US9012651, 116
Show/Hide
|
C18H19F4N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0484040
|
US9012651, 162
Show/Hide
|
C21H20F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0484041
|
US9012651, 178
Show/Hide
|
C19H22F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0484042
|
US9012651, 181
Show/Hide
|
C16H18F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0484043
|
US9012651, 194
Show/Hide
|
C15H17F3N4O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0484044
|
US9012651, 196
Show/Hide
|
C16H17F3N4O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0493232
|
US9012651, 252
Show/Hide
|
C15H21FN4O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0512074
|
US9012651, 221
Show/Hide
|
C15H23FN2O2
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0518598
|
US9012651, 35
Show/Hide
|
C17H19F4N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0518953
|
US9012651, 117
Show/Hide
|
C17H18F4N4O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0518955
|
US9012651, 163
Show/Hide
|
C21H20F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0518956
|
US9012651, 173
Show/Hide
|
C17H18F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0520581
|
US9012651, 250
Show/Hide
|
C18H25FN4O3
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0523884
|
US9012651, 218
Show/Hide
|
C16H25FN2O2
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0526391
|
US9012651, 91
Show/Hide
|
C17H20F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
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CP0526394
|
US9012651, 140
Show/Hide
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C21H20F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0526398
|
US9012651, 154
Show/Hide
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C21H20F3N3O2
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0526399
|
US9012651, 158
Show/Hide
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C19H22F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0526400
|
US9012651, 165
Show/Hide
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C19H22F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0526402
|
US9012651, 188
Show/Hide
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C16H17F3N4O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0526403
|
US9012651, 191
Show/Hide
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C15H17F3N4O2
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0526404
|
US9012651, 195
Show/Hide
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C15H17F3N4O2
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0539357
|
US9012651, 136
Show/Hide
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C16H18F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0539359
|
US9012651, 151
Show/Hide
|
C16H18F3N3O2
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0539360
|
US9012651, 168
Show/Hide
|
C19H22F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0539361
|
US9012651, 193
Show/Hide
|
C18H21F3N4O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0539362
|
US9012651, 204
Show/Hide
|
C16H25FN2O2
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0539364
|
US9012651, 211
Show/Hide
|
C17H20F3N3O4S
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0546939
|
US9012651, 182
Show/Hide
|
C20H18F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0547615
|
US9012651, 152
Show/Hide
|
C16H18F3N3O2
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0547616
|
US9012651, 167
Show/Hide
|
C19H22F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0548930
|
US9012651, 176
Show/Hide
|
C16H16F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0554242
|
US9012651, 169
Show/Hide
|
C20H22F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0557347
|
US9012651, 160
Show/Hide
|
C17H18F3N3O2
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0563965
|
US9012651, 132
Show/Hide
|
C17H18F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0563969
|
US9012651, 156
Show/Hide
|
C17H20F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0563970
|
US9012651, 175
Show/Hide
|
C16H18F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0563971
|
US9012651, 179
Show/Hide
|
C15H13F6N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0564357
|
US9012651, 119
Show/Hide
|
C17H18F4N4O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0564361
|
US9012651, 149
Show/Hide
|
C16H18F3N3O2
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0564362
|
US9012651, 155
Show/Hide
|
C17H20F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0565037
|
US9012651, 197
Show/Hide
|
C17H21F3N4O3
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0569757
|
US9012651, 161
Show/Hide
|
C19H22F3N3O2
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0570667
|
US9012651, 135
Show/Hide
|
C16H16F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0573300
|
US9012651, 118
Show/Hide
|
C18H19F6N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0573304
|
US9012651, 157
Show/Hide
|
C18H20F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0573305
|
US9012651, 166
Show/Hide
|
C19H22F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0573306
|
US9012651, 174
Show/Hide
|
C17H18F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0573307
|
US9012651, 180
Show/Hide
|
C15H16F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0573308
|
US9012651, 183
Show/Hide
|
C15H16F3N3O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0573309
|
US9012651, 186
Show/Hide
|
C15H17F3N4O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0573310
|
US9012651, 192
Show/Hide
|
C16H19F3N4O
|
1
|
1 |
IC50 > 20000 nM
|
|
|
CP0101210
|
2-nitro-N-[4-(4-propan-2-ylpiperazin-1-yl)sulfonylphenyl]-4-(trifluoromethyl)benzamide
Show/Hide
|
C21H23F3N4O5S
|
1
|
1 |
IC50 > 30000 nM
|
|
|
CP0543320
|
(2S)-2-(5-phenyl-1,3-thiazol-2-yl)-N-(3-propan-2-ylphenyl)pyrrolidine-1-carboxamide
Show/Hide
|
C23H25N3OS
|
1
|
1 |
IC50 > 100000 nM
|
|
|