Compound ID |
Compound Name |
Compound Formula |
CP0126502
|
US10865208, Compound I-115
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|
C11H15FN6O5S2
|
1
|
1 |
IC50 = 47 nM
|
|
|
CP0571688
|
US10865208, Compound I-141
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|
C17H19FN6O5S2
|
2
|
1 |
IC50 = 51 nM
|
|
|
2 |
IC50 = 140 nM
|
|
|
CP0126501
|
US10865208, Compound I-106
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|
C16H16ClFN6O5S2
|
2
|
1 |
IC50 = 56 nM
|
|
|
2 |
IC50 = 198 nM
|
|
|
CP0126513
|
US10865208, Compound I-139
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|
C13H19FN6O5S2
|
2
|
1 |
IC50 = 56 nM
|
|
|
2 |
IC50 = 199 nM
|
|
|
CP0142433
|
US10865208, Compound I-42
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|
C11H16N6O6S2
|
2
|
1 |
IC50 = 83 nM
|
|
|
2 |
IC50 = 431 nM
|
|
|
CP0343953
|
US10865208, Compound I-200
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|
C11H16N6O5S2
|
2
|
1 |
IC50 = 86 nM
|
|
|
2 |
IC50 = 280 nM
|
|
|
CP0422146
|
US10865208, Compound I-181
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|
C13H20N6O5S2
|
2
|
1 |
IC50 = 150 nM
|
|
|
2 |
IC50 = 438 nM
|
|
|
CP0136720
|
US10865208, Compound I-51
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|
C12H18N6O6S2
|
1
|
1 |
IC50 = 160 nM
|
|
|
CP0343947
|
US10865208, Compound I-27
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|
C11H14F2N6O7S
|
2
|
1 |
IC50 = 162 nM
|
|
|
2 |
IC50 = 479 nM
|
|
|
CP0571799
|
US10865208, Compound I-69
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|
C17H20N6O6S2
|
1
|
1 |
IC50 = 178 nM
|
|
|
CP0232840
|
US10865208, Compound I-82
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|
C16H18N6O6S2
|
1
|
1 |
IC50 = 201 nM
|
|
|
CP0098630
|
US10865208, Compound I-58
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|
C13H20N6O6S2
|
2
|
1 |
IC50 = 284 nM
|
|
|
2 |
IC50 = 1250 nM
|
|
|
CP0098617
|
US10865208, Compound I-219
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|
C11H16N6O5S2
|
1
|
1 |
IC50 = 295 nM
|
|
|
CP0219491
|
US10865208, Compound I-105
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|
C11H15FN6O6S
|
1
|
1 |
IC50 = 317 nM
|
|
|
CP0098628
|
US10865208, Compound I-52
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|
C17H20N6O6S2
|
2
|
1 |
IC50 = 322 nM
|
|
|
2 |
IC50 = 604 nM
|
|
|
CP0301792
|
US10865208, Compound I-1
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|
C11H16N6O7S
|
1
|
1 |
IC50 = 335 nM
|
|
|
CP0126531
|
US10865208, Compound I-172
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|
C12H18N6O5S2
|
1
|
1 |
IC50 = 367 nM
|
|
|
CP0422145
|
US10865208, Compound I-205
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|
C17H20N6O5S2
|
1
|
1 |
IC50 = 422 nM
|
|
|
CP0126518
|
US10865208, Compound I-99
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|
C11H13F3N6O6S
|
1
|
1 |
IC50 = 453 nM
|
|
|
CP0115955
|
US10865208, Compound I-220
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|
C13H20N6O5S2
|
1
|
1 |
IC50 = 468 nM
|
|
|
CP0239911
|
US10865208, Compound I-179
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|
C16H17ClN6O5S2
|
1
|
1 |
IC50 = 499 nM
|
|
|
CP0343931
|
US10865208, Compound I-195
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|
C11H14F2N6O6S
|
1
|
1 |
IC50 = 545 nM
|
|
|
CP0232854
|
US10865208, Compound I-95
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|
C13H20N6O6S2
|
1
|
1 |
IC50 = 882 nM
|
|
|
CP0098595
|
US10865208, Compound I-76
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|
C17H20N6O7S
|
1
|
1 |
IC50 = 1280 nM
|
|
|
CP0126503
|
US10865208, Compound I-94
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|
C11H16N6O6S2
|
1
|
1 |
IC50 = 1280 nM
|
|
|
CP0678838
|
{(2R,3S,4R,5R)-5-[4-amino-3-(1H-pyrazol-4-ylsulfanyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl]-3,4-dihydroxytetrahydrofuran-2-yl}methyl sulfamate
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|
C13H16N8O6S2
|
1
|
1 |
IC50 = 1280 nM
|
|
|