| Compound ID |
Compound Name |
Compound Formula |
|
CP0052187
|
4-methoxy-3-(1-methylpiperidin-4-yl)oxy-N-[(3-propan-2-yl-1,2-oxazol-5-yl)methyl]benzamide
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|
C21H29N3O4
|
3
|
| 1 |
IC50 = 72 nM
|
|
|
| 2 |
IC50 = 90 nM
|
|
|
| 3 |
IC50 = 270 nM
|
|
|
|
CP0071979
|
4-methoxy-N-[(3-propan-2-yl-1,2-oxazol-5-yl)methyl]-3-(1-propan-2-ylpiperidin-4-yl)oxybenzamide
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|
C23H33N3O4
|
2
|
| 1 |
IC50 = 100 nM
|
|
|
| 2 |
IC50 = 240 nM
|
|
|
|
CP0091214
|
4-chloro-3-(1-methylpiperidin-4-yl)oxy-N-[(3-propan-2-yl-1,2-oxazol-5-yl)methyl]benzamide
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|
C20H26ClN3O3
|
1
|
| 1 |
IC50 = 270 nM
|
|
|
|
CP0399368
|
4-fluoro-3-(1-methylpiperidin-4-yl)oxy-N-[(3-propan-2-yl-1,2-oxazol-5-yl)methyl]benzamide
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|
C20H26FN3O3
|
1
|
| 1 |
IC50 = 467 nM
|
|
|
|
CP0052185
|
4-methoxy-3-(2-piperidin-1-ylethoxy)-N-[(3-propan-2-yl-1,2-oxazol-5-yl)methyl]benzamide
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|
C22H31N3O4
|
2
|
| 1 |
IC50 = 530 nM
|
|
|
| 2 |
IC50 = 760 nM
|
|
|
|
CP0523221
|
MLS001100779
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|
C22H31N3O4
|
1
|
| 1 |
IC50 = 600 nM
|
|
|
|
CP0408990
|
3-(1-methylpiperidin-4-yl)oxy-N-[(3-propan-2-yl-1,2-oxazol-5-yl)methyl]benzamide
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|
C20H27N3O3
|
1
|
| 1 |
IC50 = 640 nM
|
|
|
|
CP0432592
|
MLS001126544
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|
C22H31N3O3S
|
1
|
| 1 |
IC50 = 760 nM
|
|
|
|
CP0093046
|
N-[(1-ethyl-3,5-dimethylpyrazol-4-yl)methyl]-4-methoxy-3-(1-propan-2-ylpiperidin-4-yl)oxybenzamide
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|
C24H36N4O3
|
2
|
| 1 |
IC50 = 910 nM
|
|
|
| 2 |
IC50 = 1580 nM
|
|
|
|
CP0523220
|
4-methoxy-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-3-(1-propan-2-ylpiperidin-4-yl)oxybenzamide
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|
C21H29N3O3S
|
2
|
| 1 |
IC50 = 1020 nM
|
|
|
| 2 |
IC50 = 3480 nM
|
|
|
|
CP0432646
|
4-methoxy-3-(1-methylpiperidin-3-yl)oxy-N-[(3-propan-2-yl-1,2-oxazol-5-yl)methyl]benzamide
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|
C21H29N3O4
|
2
|
| 1 |
IC50 = 1250 nM
|
|
|
| 2 |
IC50 = 4540 nM
|
|
|
|
CP0523186
|
MLS000733239
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|
C26H29N3O2
|
1
|
| 1 |
IC50 = 1260 nM
|
|
|
|
CP0379119
|
4-methoxy-3-(1-propan-2-ylpiperidin-4-yl)oxy-N-(2-pyrrolidin-1-ylethyl)benzamide
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|
C22H35N3O3
|
2
|
| 1 |
IC50 = 1560 nM
|
|
|
| 2 |
IC50 = 2130 nM
|
|
|
|
CP0239947
|
4-methoxy-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(1-propan-2-ylpiperidin-4-yl)oxybenzamide
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|
C21H29N3O3S
|
2
|
| 1 |
IC50 = 1640 nM
|
|
|
| 2 |
IC50 = 4930 nM
|
|
|
|
CP0068994
|
4-methoxy-3-(1-propan-2-ylpiperidin-4-yl)oxy-N-(1-pyridin-2-ylpropan-2-yl)benzamide
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|
C24H33N3O3
|
2
|
| 1 |
IC50 = 1730 nM
|
|
|
| 2 |
IC50 = 4120 nM
|
|
|
|
CP0379013
|
4-methoxy-3-(2-morpholin-4-ylethoxy)-N-[(3-propan-2-yl-1,2-oxazol-5-yl)methyl]benzamide
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|
C21H29N3O5
|
2
|
| 1 |
IC50 = 1770 nM
|
|
|
| 2 |
IC50 = 6120 nM
|
|
|
|
CP0534056
|
N-[(3-propan-2-yl-1,2-oxazol-5-yl)methyl]-3-(1-propan-2-ylpiperidin-4-yl)oxybenzamide
Show/Hide
|
C22H31N3O3
|
1
|
| 1 |
IC50 = 1840 nM
|
|
|
|
CP0468988
|
N-[(1-ethylpyrazol-4-yl)methyl]-4-methoxy-3-(1-propan-2-ylpiperidin-4-yl)oxybenzamide
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|
C22H32N4O3
|
2
|
| 1 |
IC50 = 1850 nM
|
|
|
| 2 |
IC50 = 9270 nM
|
|
|
|
CP0379120
|
N-[(1,5-dimethylpyrazol-3-yl)methyl]-4-methoxy-3-(1-propan-2-ylpiperidin-4-yl)oxybenzamide
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|
C22H32N4O3
|
2
|
| 1 |
IC50 = 2510 nM
|
|
|
| 2 |
IC50 = 8090 nM
|
|
|
|
CP0413202
|
MLS001082585
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|
C24H36N2O3
|
1
|
| 1 |
IC50 = 3160 nM
|
|
|
|
CP0534057
|
4-cyano-3-(1-methylpiperidin-4-yl)oxy-N-[(3-propan-2-yl-1,2-oxazol-5-yl)methyl]benzamide
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|
C21H26N4O3
|
1
|
| 1 |
IC50 = 3350 nM
|
|
|
|
CP0418546
|
MLS001122453
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|
C25H32N2O3
|
1
|
| 1 |
IC50 = 3360 nM
|
|
|
|
CP0504584
|
MLS001101393
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|
C23H30N2O2
|
1
|
| 1 |
IC50 = 4220 nM
|
|
|
|
CP0523222
|
3-[(1-isopropyl-4-piperidyl)oxy]-4-methoxy-N-(1-methyl-2-pyrazin-2-yl-ethyl)benzamide
Show/Hide
|
C23H32N4O3
|
1
|
| 1 |
IC50 = 4470 nM
|
|
|
|
CP0408992
|
3-(1-methylpiperidin-4-yl)oxy-N-[(3-propan-2-yl-1,2-oxazol-5-yl)methyl]-4-(trifluoromethyl)benzamide
Show/Hide
|
C21H26F3N3O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
