| Compound ID |
Compound Name |
Compound Formula |
|
CP0339222
|
US8604061, 369
Show/Hide
|
C12H13ClN2O
|
1
|
| 1 |
EC50 = 0.6 nM
|
|
|
|
CP0095112
|
US8604061, 364
Show/Hide
|
C11H13ClN2O
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0452288
|
(4S)-4-(4-chloro-2-methylphenyl)-4,5-dihydro-1,3-oxazol-2-amine
Show/Hide
|
C10H11ClN2O
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0442393
|
2-(3-iodo-4-phenoxyphenyl)ethanamine
Show/Hide
|
C14H14INO
|
1
|
| 1 |
EC50 = 2.4 nM
|
|
|
|
CP0491924
|
2-[4-(4-fluorophenoxy)-3-iodophenyl]-N-methylethanamine
Show/Hide
|
C15H15FINO
|
1
|
| 1 |
EC50 = 2.7 nM
|
|
|
|
CP0399251
|
N-(1H-imidazol-5-ylmethyl)-N-propan-2-ylaniline
Show/Hide
|
C13H17N3
|
1
|
| 1 |
EC50 = 7.3 nM
|
|
|
|
CP0205781
|
US8604061, 91
Show/Hide
|
C9H8Cl2N2O
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0239872
|
(+)-(S)-amphetamine
Show/Hide
|
C9H13N
|
5
|
| 1 |
EC50 = 13.9 nM
|
|
|
| 2 |
EC50 = 55.6 nM
|
|
|
| 3 |
EC50 = 440 nM
|
|
|
| 4 |
EC50 = 677.4 nM
|
|
|
| 5 |
EC50 = 810 nM
|
|
|
|
CP0403658
|
(4S)-4-[(N-ethylanilino)methyl]-4,5-dihydro-1,3-oxazol-2-amine
Show/Hide
|
C12H17N3O
|
1
|
| 1 |
EC50 = 14 nM
|
|
|
|
CP0453146
|
4-[2-iodo-4-[2-(methylamino)ethyl]phenoxy]phenol
Show/Hide
|
C15H16INO2
|
1
|
| 1 |
EC50 = 18 nM
|
|
|
|
CP0459674
|
US8604061, 231
Show/Hide
|
C10H11BrN2O
|
1
|
| 1 |
EC50 = 18 nM
|
|
|
|
CP0898502
|
2-(3-phenoxyphenyl)-2-phenylethylamine hydrochloride
Show/Hide
|
C20H20ClNO
|
1
|
| 1 |
EC50 = 19 nM
|
|
|
|
CP0328861
|
4-chloro-N-(1H-imidazol-5-ylmethyl)-N-propan-2-ylaniline
Show/Hide
|
C13H16ClN3
|
1
|
| 1 |
EC50 = 25 nM
|
|
|
|
CP0351659
|
N-(1H-imidazol-5-ylmethyl)-6-methoxy-N-propan-2-ylpyridin-2-amine
Show/Hide
|
C13H18N4O
|
1
|
| 1 |
EC50 = 25 nM
|
|
|
|
CP0877959
|
2-(1-phenoxynaphthalen-4-yl)ethylamine
Show/Hide
|
C18H18ClNO
|
1
|
| 1 |
EC50 = 26 nM
|
|
|
|
CP0428087
|
3-chloro-N-(1H-imidazol-5-ylmethyl)-N-propan-2-ylaniline
Show/Hide
|
C13H16ClN3
|
1
|
| 1 |
EC50 = 27 nM
|
|
|
|
CP0847711
|
2-(4-phenoxyphenyl)-2-phenylethylamine hydrochloride
Show/Hide
|
C20H20ClNO
|
1
|
| 1 |
EC50 = 28 nM
|
|
|
|
CP0210581
|
US8604061, 105
Show/Hide
|
C9H9BrN2O
|
1
|
| 1 |
EC50 = 29 nM
|
|
|
|
CP0882579
|
2-(4-(4-hydroxyphenoxy)-3-iodophenyl)ethanaminium chloride
Show/Hide
|
C14H15ClINO2
|
1
|
| 1 |
EC50 = 33 nM
|
|
|
|
CP0391084
|
3-methyl-thyronamine
Show/Hide
|
C15H17NO2
|
1
|
| 1 |
EC50 = 33 nM
|
|
|
|
CP0372464
|
(2-butylbenzofuran-3-yl)(4-(2-(ethylamino)ethoxy)-3-iodophenyl)methanone
Show/Hide
|
C23H26INO3
|
1
|
| 1 |
EC50 = 33 nM
|
|
|
|
CP0372465
|
(2-{4-[(2-butyl-1-benzofuran-3-yl)carbonyl]-2,6-diiodophenoxy}ethyl)(ethyl)amine
Show/Hide
|
C23H25I2NO3
|
1
|
| 1 |
EC50 = 33 nM
|
|
|
|
CP0452418
|
(2-{4-[(2-butyl-1-benzofuran-3-yl)carbonyl]phenoxy}ethyl)diethylamine
Show/Hide
|
C25H31NO3
|
1
|
| 1 |
EC50 = 33 nM
|
|
|
|
CP0452419
|
(2-{4-[(2-butyl-1-benzofuran-3-yl)carbonyl]-2-iodophenoxy}ethyl)diethylamine
Show/Hide
|
C25H30INO3
|
1
|
| 1 |
EC50 = 33 nM
|
|
|
|
CP0521184
|
(2-butylbenzofuran-3-yl)(3-ethyl-4-(2-(ethylamino)ethoxy)-5-iodophenyl)methanone
Show/Hide
|
C25H30INO3
|
1
|
| 1 |
EC50 = 33 nM
|
|
|
|
CP0110511
|
(R)-amphetamine
Show/Hide
|
C9H13N
|
5
|
| 1 |
EC50 = 33.9 nM
|
|
|
| 2 |
EC50 = 169.9 nM
|
|
|
| 3 |
EC50 = 210 nM
|
|
|
| 4 |
EC50 = 214.4 nM
|
|
|
| 5 |
EC50 = 280 nM
|
|
|
|
CP0099315
|
(4S)-4-(3-fluoro-2-methylphenyl)-4,5-dihydro-1,3-oxazol-2-amine
Show/Hide
|
C10H11FN2O
|
1
|
| 1 |
EC50 = 35 nM
|
|
|
|
CP0284355
|
2-(4-Phenoxy-phenyl)-ethylamine
Show/Hide
|
C14H15NO
|
1
|
| 1 |
EC50 = 38 nM
|
|
|
|
CP0061725
|
14C-phenylethylamine
Show/Hide
|
C8H11N
|
3
|
| 1 |
EC50 = 40.33 nM
|
|
|
| 2 |
EC50 = 170.6 nM
|
|
|
| 3 |
EC50 = 261.2 nM
|
|
|
|
CP0847715
|
2-(4-phenoxyphenyl)-4-phenylbut-3-yn-1-amine hydrochloride
Show/Hide
|
C22H20ClNO
|
1
|
| 1 |
EC50 = 41 nM
|
|
|
|
CP0436590
|
3,3'-Diiodothyronamine
Show/Hide
|
C14H13I2NO2
|
1
|
| 1 |
EC50 = 41 nM
|
|
|
|
CP0436685
|
2-[4-(4-phenylbutoxy)phenyl]ethanamine
Show/Hide
|
C18H23NO
|
1
|
| 1 |
EC50 = 43 nM
|
|
|
|
CP0035003
|
4-(2-aminopropyl)phenol;hydrobromide
Show/Hide
|
C9H13NO
|
1
|
| 1 |
EC50 = 50 nM
|
|
|
|
CP0847714
|
2-(1-phenoxynaphthalen-4-yl)-2-phenylethylamine hydrochloride
Show/Hide
|
C24H22ClNO
|
1
|
| 1 |
EC50 = 52 nM
|
|
|
|
CP0381880
|
US8604061, 169
Show/Hide
|
C9H9ClN2O
|
1
|
| 1 |
EC50 = 52 nM
|
|
|
|
CP0422195
|
2-[4-[[4-(trifluoromethyl)phenyl]methoxy]phenyl]ethanamine
Show/Hide
|
C16H16F3NO
|
1
|
| 1 |
EC50 = 55 nM
|
|
|
|
CP0483553
|
3,5-Diiodothyronamine
Show/Hide
|
C14H13I2NO2
|
1
|
| 1 |
EC50 = 56 nM
|
|
|
|
CP0441305
|
4-[(2R)-2-aminopropyl]phenol
Show/Hide
|
C9H13NO
|
1
|
| 1 |
EC50 = 60 nM
|
|
|
|
CP0453149
|
N-methyl-2-[4-[[4-(trifluoromethyl)phenyl]methoxy]phenyl]ethanamine
Show/Hide
|
C17H18F3NO
|
1
|
| 1 |
EC50 = 61 nM
|
|
|
|
CP0366108
|
N-(1H-imidazol-5-ylmethyl)-3-methoxy-N-propan-2-ylaniline
Show/Hide
|
C14H19N3O
|
1
|
| 1 |
EC50 = 61 nM
|
|
|
|
CP0877538
|
2-(4-phenoxyphenyl)but-3-yn-1-amine hydrochloride
Show/Hide
|
C16H16ClNO
|
1
|
| 1 |
EC50 = 62 nM
|
|
|
|
CP0847935
|
2-(4-phenoxyphenyl)ethanaminium chloride
Show/Hide
|
C14H16ClNO
|
1
|
| 1 |
EC50 = 63 nM
|
|
|
|
CP0403661
|
(4S)-4-(2-methylphenyl)-4,5-dihydro-1,3-oxazol-2-amine
Show/Hide
|
C10H12N2O
|
1
|
| 1 |
EC50 = 63 nM
|
|
|
|
CP0462482
|
2-[4-[(4-nitrophenyl)methoxy]phenyl]ethanamine
Show/Hide
|
C15H16N2O3
|
1
|
| 1 |
EC50 = 64 nM
|
|
|
|
CP0432593
|
2-(3-iodo-4-phenylmethoxyphenyl)-N-methylethanamine
Show/Hide
|
C16H18INO
|
1
|
| 1 |
EC50 = 68 nM
|
|
|
|
CP0419527
|
2-[4-[(4-fluorophenyl)methoxy]phenyl]ethanamine
Show/Hide
|
C15H16FNO
|
1
|
| 1 |
EC50 = 72 nM
|
|
|
|
CP0459809
|
2-(3-iodo-4-phenylmethoxyphenyl)ethanamine
Show/Hide
|
C15H16INO
|
1
|
| 1 |
EC50 = 77 nM
|
|
|
|
CP0464718
|
3,3',5-triiodothyronamine
Show/Hide
|
C14H12I3NO2
|
1
|
| 1 |
EC50 = 87 nM
|
|
|
|
CP0452287
|
US8604061, 4
Show/Hide
|
C9H9ClN2O
|
1
|
| 1 |
EC50 = 87 nM
|
|
|
|
CP0432595
|
2-[4-(3-phenylpropoxy)phenyl]ethanamine
Show/Hide
|
C17H21NO
|
1
|
| 1 |
EC50 = 89 nM
|
|
|
|
CP0459808
|
2-[3-iodo-4-(4-methoxyphenoxy)phenyl]-N-methylethanamine
Show/Hide
|
C16H18INO2
|
1
|
| 1 |
EC50 = 107 nM
|
|
|
|
CP0464706
|
N-methyl-2-(4-phenylmethoxyphenyl)ethanamine
Show/Hide
|
C16H19NO
|
1
|
| 1 |
EC50 = 119 nM
|
|
|
|
CP0442569
|
4-[4-(2-aminoethyl)phenoxy]phenol
Show/Hide
|
C14H15NO2
|
1
|
| 1 |
EC50 = 131 nM
|
|
|
|
CP0125122
|
(S)Methamphetamine
Show/Hide
|
C10H15N
|
4
|
| 1 |
EC50 = 133.3 nM
|
|
|
| 2 |
EC50 = 201.8 nM
|
|
|
| 3 |
EC50 = 890 nM
|
|
|
| 4 |
EC50 = 2044 nM
|
|
|
|
CP0442211
|
2-[4-[(3,5-dimethylphenyl)methoxy]phenyl]ethanamine
Show/Hide
|
C17H21NO
|
1
|
| 1 |
EC50 = 137 nM
|
|
|
|
CP0844891
|
2-(4-phenoxyphenyl)-3-phenylpropan-1-amine hydrochloride
Show/Hide
|
C21H22ClNO
|
1
|
| 1 |
EC50 = 140 nM
|
|
|
|
CP0419528
|
2-[4-[(3-methoxyphenyl)methoxy]phenyl]ethanamine
Show/Hide
|
C16H19NO2
|
1
|
| 1 |
EC50 = 141 nM
|
|
|
|
CP0392573
|
4-[(2S)-2-aminopropyl]phenol
Show/Hide
|
C9H13NO
|
1
|
| 1 |
EC50 = 190 nM
|
|
|
|
CP0553804
|
2-[4-(2-phenylethoxy)phenyl]ethanamine
Show/Hide
|
C16H19NO
|
1
|
| 1 |
EC50 = 203 nM
|
|
|
|
CP0419530
|
2-(4-phenylmethoxyphenyl)ethanamine
Show/Hide
|
C15H17NO
|
1
|
| 1 |
EC50 = 209 nM
|
|
|
|
CP0379778
|
(R)Methamphetamine
Show/Hide
|
C10H15N
|
4
|
| 1 |
EC50 = 233.3 nM
|
|
|
| 2 |
EC50 = 330.4 nM
|
|
|
| 3 |
EC50 = 1109 nM
|
|
|
| 4 |
EC50 = 1190 nM
|
|
|
|
CP0176355
|
US8604061, 192
Show/Hide
|
C9H9ClN2O
|
1
|
| 1 |
EC50 = 246 nM
|
|
|
|
CP0877539
|
2-(4-phenoxyphenyl)propan-1-amine hydrochloride
Show/Hide
|
C15H18ClNO
|
1
|
| 1 |
EC50 = 250 nM
|
|
|
|
CP0847839
|
2-(1-methoxynaphthalen-4-yl)-2-phenylethylamine hydrochloride
Show/Hide
|
C19H20ClNO
|
1
|
| 1 |
EC50 = 270 nM
|
|
|
|
CP0462483
|
2-[4-(2-aminoethyl)phenoxy]-1-phenylethanone
Show/Hide
|
C16H17NO2
|
1
|
| 1 |
EC50 = 309 nM
|
|
|
|
CP0442394
|
2-[4-[(3,5-dimethoxyphenyl)methoxy]phenyl]ethanamine
Show/Hide
|
C17H21NO3
|
1
|
| 1 |
EC50 = 333 nM
|
|
|
|
CP0898501
|
N-methyl-3-[(4-phenoxyphenyl)oxy]propylamine hydrochloride
Show/Hide
|
C16H20ClNO2
|
1
|
| 1 |
EC50 = 370 nM
|
|
|
|
CP0844896
|
3-[(3-phenoxyphenyl)oxy]propylamine hydrochloride
Show/Hide
|
C15H18ClNO2
|
1
|
| 1 |
EC50 = 373 nM
|
|
|
|
CP0462140
|
3-chloro-N-(1H-imidazol-2-ylmethyl)-N-propan-2-ylaniline
Show/Hide
|
C13H16ClN3
|
1
|
| 1 |
EC50 = 400 nM
|
|
|
|
CP0389567
|
(4S)-4-(4-phenylphenyl)-4,5-dihydro-1,3-oxazol-2-amine
Show/Hide
|
C15H14N2O
|
1
|
| 1 |
EC50 = 428 nM
|
|
|
|
CP0397938
|
US8604061, 180
Show/Hide
|
C10H11ClN2O
|
1
|
| 1 |
EC50 = 560 nM
|
|
|
|
CP0898503
|
2-(1-hydroxynaphthalen-4-yl)-2-phenylethylamine hydrochloride
Show/Hide
|
C18H18ClNO
|
1
|
| 1 |
EC50 = 716 nM
|
|
|
|
CP0880571
|
3-[(4-phenoxyphenyl)oxy]propylamine hydrochloride
Show/Hide
|
C15H18ClNO2
|
1
|
| 1 |
EC50 = 758 nM
|
|
|
|
CP0449800
|
3'-iodothyronamine
Show/Hide
|
C14H14INO2
|
1
|
| 1 |
EC50 = 800 nM
|
|
|
|
CP0121744
|
3-{[4-(2-aminoethoxy)-3,5-diiodophenyl]carbonyl}-2-butyl-1-benzofuran
Show/Hide
|
C21H21I2NO3
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0010255
|
(RS)-3,4-(methylenedioxy)methamphetamine
Show/Hide
|
C11H15NO2
|
1
|
| 1 |
EC50 = 1700 nM
|
|
|
|
CP0381901
|
US8604061, 199
Show/Hide
|
C9H9FN2O
|
1
|
| 1 |
EC50 = 1920 nM
|
|
|
|
CP0847934
|
5-(4-phenoxybenzamido)pentylamine hydrochloride
Show/Hide
|
C18H23ClN2O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0844892
|
2-methyl-2-(4-phenoxyphenyl)propan-1-amine hydrochloride
Show/Hide
|
C16H20ClNO
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0844895
|
3-(4-phenoxybenzamido)propylamine hydrochloride
Show/Hide
|
C16H19ClN2O2
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0844897
|
N,N-dimethyl-3-[(4-phenoxyphenyl)oxy]propylamine hydrochloride
Show/Hide
|
C17H22ClNO2
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0847713
|
N,N-dimethyl-5-(4-phenoxybenzamido)pentylamine hydrochloride
Show/Hide
|
C20H27ClN2O2
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0847840
|
2-(4-phenoxybenzamido)ethylamine hydrochloride
Show/Hide
|
C15H17ClN2O2
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0868921
|
N,N-dimethyl-3-(4-phenoxybenzamido)propylamine hydrochloride
Show/Hide
|
C18H23ClN2O2
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0877540
|
N,N-dimethyl-4-(4-phenoxybenzamido)butylamine hydrochloride
Show/Hide
|
C19H25ClN2O2
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0877741
|
N,N-dimethyl-2-(4-phenoxybenzamido)ethylamine hydrochloride
Show/Hide
|
C17H21ClN2O2
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0918263
|
4-(4-phenoxybenzamido)butylamine hydrochloride
Show/Hide
|
C17H21ClN2O2
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0919876
|
7-phenoxy-1-phenyl-2,3,4,5-tetrahydro-3-benzazepine hydrochloride
Show/Hide
|
C22H22ClNO
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0921536
|
8-phenoxy-1-phenyl-2,3,4,5-tetrahydro-3-benzazepine hydrochloride
Show/Hide
|
C22H22ClNO
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0419533
|
2-[4-[(2,3,4,5,6-pentafluorophenyl)methoxy]phenyl]ethanamine
Show/Hide
|
C15H12F5NO
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0432594
|
2-[3-iodo-4-(p-hydroxy)phenoxyphenyl]ethanol
Show/Hide
|
C14H13IO3
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0436589
|
N-[2-(4-phenylmethoxyphenyl)ethyl]butan-1-amine
Show/Hide
|
C19H25NO
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0436591
|
3,3',5,5'-tetraiodothyronamine
Show/Hide
|
C14H11I4NO2
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0439414
|
3,3',5'-triiodothyronamine
Show/Hide
|
C14H12I3NO2
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0441793
|
2-[3-iodo-4-[[4-(trifluoromethyl)phenyl]methoxy]phenyl]ethanamine
Show/Hide
|
C16H15F3INO
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0442208
|
N-ethyl-2-(4-phenylmethoxyphenyl)ethanamine
Show/Hide
|
C17H21NO
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0442395
|
N-benzyl-2-(4-phenylmethoxyphenyl)ethanamine
Show/Hide
|
C22H23NO
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0462481
|
N-[2-(4-phenylmethoxyphenyl)ethyl]propan-1-amine
Show/Hide
|
C18H23NO
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0485667
|
N,N-dimethyl-2-(4-phenylmethoxyphenyl)ethanamine
Show/Hide
|
C17H21NO
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0491925
|
3',5'-diiodothyronamine
Show/Hide
|
C14H13I2NO2
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0515820
|
2-[3-iodo-4-[4-(trifluoromethyl)phenoxy]phenyl]-N-methylethanamine
Show/Hide
|
C16H15F3INO
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0406846
|
US9416127, 10
Show/Hide
|
C20H18F3N5O2
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0476857
|
US9416127, 12
Show/Hide
|
C19H18ClN5O2
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0518693
|
US9416127, 7
Show/Hide
|
C20H21N5O2
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0537360
|
US9416127, 6
Show/Hide
|
C19H18ClN5O2
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0548106
|
US11697636, Example 154
Show/Hide
|
C19H20Cl2N2O
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0472162
|
US11697636, Example 152
Show/Hide
|
C18H18Cl2N2O
|
1
|
| 1 |
Ki = 0.3 nM
|
|
|
|
CP0484426
|
US10501411, Example 128
Show/Hide
|
C20H23ClN2O2
|
1
|
| 1 |
Ki = 0.3 nM
|
|
|
|
CP0386662
|
US10501411, Example 121
Show/Hide
|
C19H21ClN2O2
|
1
|
| 1 |
Ki = 0.4 nM
|
|
|
|
CP0515644
|
US10501411, Example 142
Show/Hide
|
C19H21ClN2O
|
1
|
| 1 |
Ki = 0.4 nM
|
|
|
|
CP0536957
|
US11697636, Example 150
Show/Hide
|
C18H18Cl2N2O
|
1
|
| 1 |
Ki = 0.4 nM
|
|
|
|
CP0561207
|
US9416127, 23
Show/Hide
|
C20H21N5O2
|
1
|
| 1 |
Ki = 0.5 nM
|
|
|
|
CP0512910
|
US11697636, Example 153
Show/Hide
|
C18H19ClN2O
|
1
|
| 1 |
Ki = 0.5 nM
|
|
|
|
CP0548089
|
US10501411, Example 303
Show/Hide
|
C17H18ClN3O2
|
1
|
| 1 |
Ki = 0.5 nM
|
|
|
|
CP0557247
|
US10501411, Example 57
Show/Hide
|
C18H19ClN2O
|
1
|
| 1 |
Ki = 0.5 nM
|
|
|
|
CP0468231
|
US9029370, 96
Show/Hide
|
C21H19ClF2N4O3
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0542940
|
US9029370, 12
Show/Hide
|
C20H18F2N4O2
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0493420
|
US9416127, 29
Show/Hide
|
C20H19F2N5O3
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0561195
|
US9416127, 13
Show/Hide
|
C20H18F3N5O2
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0405834
|
US10501411, Example 143
Show/Hide
|
C17H17ClN2O2
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0540643
|
US10501411, Example 235
Show/Hide
|
C19H21ClN2O2
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0554037
|
US10501411, Example 225
Show/Hide
|
C19H21ClN2O
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0474480
|
US9029370, 63
Show/Hide
|
C18H16F2N4O2
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0541862
|
US9029370, 90
Show/Hide
|
C21H19F3N4O3
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0556583
|
US9029370, 86
Show/Hide
|
C21H19F3N4O3
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0387660
|
US11697636, Example 157
Show/Hide
|
C19H21ClN2O
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0539902
|
US10501411, Example 125
Show/Hide
|
C20H21F3N2O3
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0544344
|
US9416127, 8
Show/Hide
|
C19H19N5O2
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0545134
|
US9416127, 2
Show/Hide
|
C20H21N5O2
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0405832
|
US10501411, Example 136
Show/Hide
|
C18H17ClN2O2
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0490926
|
US10501411, Example 237
Show/Hide
|
C20H24N2OS
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0512923
|
US11697636, Example 151
Show/Hide
|
C18H19ClN2O
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0555546
|
US10501411, Example 276
Show/Hide
|
C19H22N2O3
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0899550
|
US9029370, 2
Show/Hide
|
C18H16F2N4O2
|
1
|
| 1 |
Ki = 0.9 nM
|
|
|
|
CP0413259
|
US10501411, Example 211
Show/Hide
|
C26H26N2O5
|
1
|
| 1 |
Ki = 0.9 nM
|
|
|
|
CP0484079
|
US10501411, Example 259
Show/Hide
|
C19H22N2OS
|
1
|
| 1 |
Ki = 0.9 nM
|
|
|
|
CP0556172
|
US11697636, Example 155
Show/Hide
|
C20H21F3N2O
|
1
|
| 1 |
Ki = 0.9 nM
|
|
|
|
CP0561161
|
US10501411, Example 240
Show/Hide
|
C19H21ClN2O2
|
1
|
| 1 |
Ki = 0.9 nM
|
|
|
|
CP0474479
|
US9029370, 60
Show/Hide
|
C19H17BrF2N4O3
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0516792
|
US9029370, 59
Show/Hide
|
C18H16F2N4O2
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0533139
|
US9029370, 72
Show/Hide
|
C19H17F3N4O3
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0406824
|
US9416127, 34
Show/Hide
|
C19H19N5O
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0406847
|
US9416127, 22
Show/Hide
|
C21H23N5O3
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0387668
|
US10501411, Example 226
Show/Hide
|
C19H21ClN2O
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0393350
|
US11697636, Example 149
Show/Hide
|
C18H19ClN2O
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0425528
|
US10501411, Example 146
Show/Hide
|
C17H16ClFN2O2
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0425534
|
US10501411, Example 213
Show/Hide
|
C25H23ClN2O5
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0429136
|
US10501411, Example 2
Show/Hide
|
C18H20Cl2N4O
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0469603
|
US10501411, Example 196
Show/Hide
|
C18H20N2O2
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0470652
|
US10501411, Example 234
Show/Hide
|
C19H19F3N2O
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0484081
|
US10501411, Example 292
Show/Hide
|
C17H18ClN3O2
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0491899
|
US11697636, Example 176
Show/Hide
|
C20H22Cl2N2O
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0488840
|
US9029370, 75
Show/Hide
|
C21H19F3N4O3
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0393349
|
US10501411, Example 46
Show/Hide
|
C19H21FN2O2
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0413466
|
US10501411, Example 312
Show/Hide
|
C18H18F3N3O2
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0419408
|
US10501411, Example 206
Show/Hide
|
C23H21ClN2O3
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0481202
|
US10501411, Example 263
Show/Hide
|
C17H17ClN2O2
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0491876
|
US10501411, Example 122
Show/Hide
|
C20H21F3N2O2
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0544298
|
US9452980, 267
Show/Hide
|
C18H20N2O2S
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0544404
|
US10501411, Example 144
Show/Hide
|
C17H17ClN2O2
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0474482
|
US9029370, 71
Show/Hide
|
C19H17F3N4O3
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0503634
|
US9029370, 31
Show/Hide
|
C20H18ClFN4O2
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0506777
|
US9029370, 30
Show/Hide
|
C20H18ClFN4O2
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0520270
|
US9029370, 47
Show/Hide
|
C19H17ClF2N4O3
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0538899
|
US9029370, 32
Show/Hide
|
C20H18ClFN4O2
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0542953
|
US9029370, 93
Show/Hide
|
C21H19ClF2N4O3
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0413465
|
US10501411, Example 304
Show/Hide
|
C18H21N3O2
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0419409
|
US10501411, Example 216
Show/Hide
|
C18H20N2O2S
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0478326
|
US10501411, Example 227
Show/Hide
|
C20H24N2O
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0515635
|
US10501411, Example 260
Show/Hide
|
C20H24N2O
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0516922
|
US10501411, Example 246
Show/Hide
|
C20H24N2OS
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0531534
|
US10501411, Example 267
Show/Hide
|
C18H20N2O2S
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0515465
|
US9029370, 5
Show/Hide
|
C18H17ClN4O2
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0419343
|
US9416127, 1
Show/Hide
|
C19H19N5O2
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0387673
|
US10501411, Example 262
Show/Hide
|
C17H17ClN2O2
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0393352
|
US10501411, Example 120
Show/Hide
|
C19H21ClN2O2
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0516917
|
US10501411, Example 145
Show/Hide
|
C18H19ClN2O2
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0531537
|
US10501411, Example 323
Show/Hide
|
C18H19ClN2O2
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0488839
|
US9029370, 55
Show/Hide
|
C16H16Cl2N4O2
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0499889
|
US9029370, 50
Show/Hide
|
C17H16ClF3N4O2
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0393341
|
US10501411, Example 59
Show/Hide
|
C17H18ClN3O
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0405866
|
US10501411, Example 281
Show/Hide
|
C17H17Cl2N3O
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0413258
|
US10501411, Example 203
Show/Hide
|
C19H21ClN2O2
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0481210
|
US10501411, Example 299
Show/Hide
|
C20H20N4O2
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0491874
|
US10501411, Example 116
Show/Hide
|
C19H22ClN3O
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0491895
|
US11697636, Example 158
Show/Hide
|
C21H26N2O2
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0493428
|
US10501411, Example 311
Show/Hide
|
C18H18F3N3O2
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0518650
|
US10501411, Example 293
Show/Hide
|
C18H21N3O2
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0531533
|
US10501411, Example 236
Show/Hide
|
C19H22N2OS
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0555964
|
US10501411, Example 231
Show/Hide
|
C20H19N3O2S
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0555965
|
US10501411, Example 233
Show/Hide
|
C20H19N3O2S
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0503631
|
US9029370, 3
Show/Hide
|
C18H17FN4O2
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
|
CP0506780
|
US9029370, 49
Show/Hide
|
C17H16ClF3N4O2
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
|
CP0405836
|
US10501411, Example 202
Show/Hide
|
C19H21ClN2O2
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
|
CP0423318
|
US10501411, Example 27
Show/Hide
|
C18H18F3N3O
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
|
CP0515676
|
US10501411, Example 261
Show/Hide
|
C19H19F3N2O
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
|
CP0516915
|
US10501411, Example 137
Show/Hide
|
C21H26N2O
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
|
CP0441928
|
US9029370, 7
Show/Hide
|
C18H17ClN4O2
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0488841
|
US9029370, 82
Show/Hide
|
C21H17F3N4O4
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0541869
|
US9029370, 127
Show/Hide
|
C19H16F4N6O2
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0553586
|
US9416127, 18
Show/Hide
|
C20H21N5O2
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0405864
|
US10501411, Example 214
Show/Hide
|
C21H24N2O3
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0425531
|
US10501411, Example 197
Show/Hide
|
C19H22N2O3
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0484094
|
US10501411, Example 189
Show/Hide
|
C18H20N2O2
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0484095
|
US10501411, Example 209
Show/Hide
|
C17H17ClN2O2
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0518652
|
US10501411, Example 3
Show/Hide
|
C17H17Cl2N3O
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0539906
|
US10501411, Example 230
Show/Hide
|
C17H16ClFN2O2
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0524300
|
US9029370, 53
Show/Hide
|
C17H16ClF3N4O2
|
1
|
| 1 |
Ki = 1.7 nM
|
|
|
|
CP0529262
|
US9029370, 6
Show/Hide
|
C18H17ClN4O2
|
1
|
| 1 |
Ki = 1.7 nM
|
|
|
|
CP0537359
|
US9416127, 35
Show/Hide
|
C20H21N5O
|
1
|
| 1 |
Ki = 1.7 nM
|
|
|
|
CP0486274
|
US10501411, Example 291
Show/Hide
|
C18H18F3N3O2
|
1
|
| 1 |
Ki = 1.7 nM
|
|
|
|
CP0516923
|
US10501411, Example 322
Show/Hide
|
C18H19ClN2O2
|
1
|
| 1 |
Ki = 1.7 nM
|
|
|
|
CP0468230
|
US9029370, 76
Show/Hide
|
C21H19F3N4O3
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0506940
|
US9029370, 48
Show/Hide
|
C19H17ClF2N4O3
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0551020
|
US9029370, 54
Show/Hide
|
C17H16ClF3N4O2
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0470708
|
US10501411, Example 223
Show/Hide
|
C19H20F3N3O2
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0515745
|
US10501411, Example 119
Show/Hide
|
C20H24ClN3O
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0516911
|
US10501411, Example 308
Show/Hide
|
C18H19ClN2O2
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0536956
|
US10501411, Example 112
Show/Hide
|
C18H19ClN2O
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0551901
|
US10501411, Example 56
Show/Hide
|
C17H16Cl2N2O
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0516793
|
US9029370, 73
Show/Hide
|
C20H21FN4O3
|
1
|
| 1 |
Ki = 1.9 nM
|
|
|
|
CP0481228
|
US9416127, 20
Show/Hide
|
C20H21N5O3
|
1
|
| 1 |
Ki = 1.9 nM
|
|
|
|
CP0536960
|
US10501411, Example 229
Show/Hide
|
C17H16ClFN2O2
|
1
|
| 1 |
Ki = 1.9 nM
|
|
|
|
CP0529263
|
US9029370, 26
Show/Hide
|
C18H16F2N4O2
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0919389
|
US9181230, 8
Show/Hide
|
C19H18ClN3O
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0405868
|
US10501411, Example 300
Show/Hide
|
C18H21N3O3
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0423325
|
US11697636, Example 156
Show/Hide
|
C19H21FN2O
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0469621
|
US10501411, Example 127
Show/Hide
|
C19H21ClN2O2
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0512889
|
US11697636, Example 178
Show/Hide
|
C19H20F3N3O2
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0922778
|
US9181230, 9
Show/Hide
|
C19H18ClN3O
|
1
|
| 1 |
Ki = 2.1 nM
|
|
|
|
CP0548109
|
US10501411, Example 190
Show/Hide
|
C18H20N2O3
|
1
|
| 1 |
Ki = 2.1 nM
|
|
|
|
CP0506774
|
US9029370, 21
Show/Hide
|
C20H18F2N4O2
|
1
|
| 1 |
Ki = 2.2 nM
|
|
|
|
CP0393340
|
US10501411, Example 58
Show/Hide
|
C18H19ClN2O
|
1
|
| 1 |
Ki = 2.2 nM
|
|
|
|
CP0404997
|
US10501411, Example 44
Show/Hide
|
C16H17ClN4O
|
1
|
| 1 |
Ki = 2.2 nM
|
|
|
|
CP0413447
|
US10501411, Example 195
Show/Hide
|
C18H20N2O2
|
1
|
| 1 |
Ki = 2.2 nM
|
|
|
|
CP0419337
|
US10501411, Example 200
Show/Hide
|
C19H21ClN2O2
|
1
|
| 1 |
Ki = 2.2 nM
|
|
|
|
CP0484093
|
US11697636, Example 179
Show/Hide
|
C19H23N3O2
|
1
|
| 1 |
Ki = 2.2 nM
|
|
|
|
CP0491877
|
US10501411, Example 126
Show/Hide
|
C19H20Cl2N2O2
|
1
|
| 1 |
Ki = 2.2 nM
|
|
|
|
CP0495812
|
US10501411, Example 123
Show/Hide
|
C20H21F3N2O2
|
1
|
| 1 |
Ki = 2.2 nM
|
|
|
|
CP0512929
|
US10501411, Example 201
Show/Hide
|
C19H21ClN2O2
|
1
|
| 1 |
Ki = 2.2 nM
|
|
|
|
CP0544304
|
US10501411, Example 309
Show/Hide
|
C18H19ClN2O2
|
1
|
| 1 |
Ki = 2.3 nM
|
|
|
|
CP0499843
|
US9029370, 13
Show/Hide
|
C20H18F2N4O2
|
1
|
| 1 |
Ki = 2.4 nM
|
|
|
|
CP0451533
|
US10501411, Example 249
Show/Hide
|
C20H19N3O3
|
1
|
| 1 |
Ki = 2.4 nM
|
|
|
|
CP0516916
|
US10501411, Example 141
Show/Hide
|
C17H16F3N3O2
|
1
|
| 1 |
Ki = 2.4 nM
|
|
|
|
CP0539905
|
US10501411, Example 220
Show/Hide
|
C22H27ClN2O4
|
1
|
| 1 |
Ki = 2.4 nM
|
|
|
|
CP0540193
|
US10501411, Example 268
Show/Hide
|
C18H18F3N3O3
|
1
|
| 1 |
Ki = 2.4 nM
|
|
|
|
CP0488325
|
US9029370, 129
Show/Hide
|
C19H16F4N6O2
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0514647
|
US9029370, 128
Show/Hide
|
C19H16ClF3N6O2
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0516231
|
US9029370, 61
Show/Hide
|
C19H17BrF2N4O3
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0425530
|
US10501411, Example 182
Show/Hide
|
C18H20N2O
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0486679
|
US10501411, Example 23
Show/Hide
|
C17H17ClN2O2
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0429150
|
US11697636, Example 168
Show/Hide
|
C17H18ClN3O
|
1
|
| 1 |
Ki = 2.6 nM
|
|
|
|
CP0539904
|
US10501411, Example 185
Show/Hide
|
C19H22N2O
|
1
|
| 1 |
Ki = 2.6 nM
|
|
|
|
CP0551022
|
US9029370, 105
Show/Hide
|
C21H18ClN5O2
|
1
|
| 1 |
Ki = 2.7 nM
|
|
|
|
CP0405867
|
US10501411, Example 289
Show/Hide
|
C20H25N3O
|
1
|
| 1 |
Ki = 2.7 nM
|
|
|
|
CP0491898
|
US11697636, Example 169
Show/Hide
|
C20H23ClN2O
|
1
|
| 1 |
Ki = 2.7 nM
|
|
|
|
CP0516931
|
US10501411, Example 5
Show/Hide
|
C17H18ClN3O
|
1
|
| 1 |
Ki = 2.7 nM
|
|
|
|
CP0519675
|
US11697636, Example 175
Show/Hide
|
C21H23F3N2O
|
1
|
| 1 |
Ki = 2.7 nM
|
|
|
|
CP0548108
|
US10501411, Example 186
Show/Hide
|
C19H22N2O2
|
1
|
| 1 |
Ki = 2.7 nM
|
|
|
|
CP0488316
|
US9029370, 4
Show/Hide
|
C18H17FN4O2
|
1
|
| 1 |
Ki = 2.8 nM
|
|
|
|
CP0515466
|
US9029370, 62
Show/Hide
|
C18H16F2N4O2
|
1
|
| 1 |
Ki = 2.8 nM
|
|
|
|
CP0552500
|
US10501411, Example 198
Show/Hide
|
C19H22N2O2
|
1
|
| 1 |
Ki = 2.8 nM
|
|
|
|
CP0512930
|
US10501411, Example 117
Show/Hide
|
C18H20ClN3O
|
1
|
| 1 |
Ki = 2.9 nM
|
|
|
|
CP0519676
|
US10501411, Example 224
Show/Hide
|
C19H20F3N3O2
|
1
|
| 1 |
Ki = 2.9 nM
|
|
|
|
CP0553386
|
US9029370, 64
Show/Hide
|
C16H16Cl2N4O2
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0557330
|
US9029370, 91
Show/Hide
|
C18H20ClN3O3
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0484080
|
US10501411, Example 269
Show/Hide
|
C18H18F3N3O3
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0561904
|
US9029370, 103
Show/Hide
|
C21H18ClN5O2
|
1
|
| 1 |
Ki = 3.1 nM
|
|
|
|
CP0548074
|
US10501411, Example 219
Show/Hide
|
C16H15Cl2N3O2
|
1
|
| 1 |
Ki = 3.1 nM
|
|
|
|
CP0518695
|
US9416127, 26
Show/Hide
|
C21H23N5O3
|
1
|
| 1 |
Ki = 3.2 nM
|
|
|
|
CP0441571
|
US9029370, 18
Show/Hide
|
C20H18ClFN4O2
|
1
|
| 1 |
Ki = 3.3 nM
|
|
|
|
CP0451904
|
US9029370, 10
Show/Hide
|
C17H16F4N4O2
|
1
|
| 1 |
Ki = 3.3 nM
|
|
|
|
CP0466965
|
US9029370, 23
Show/Hide
|
C21H21FN4O2
|
1
|
| 1 |
Ki = 3.3 nM
|
|
|
|
CP0484441
|
US10501411, Example 222
Show/Hide
|
C18H18F3N3O3
|
1
|
| 1 |
Ki = 3.3 nM
|
|
|
|
CP0495845
|
US10501411, Example 61
Show/Hide
|
C20H21F3N2O
|
1
|
| 1 |
Ki = 3.3 nM
|
|
|
|
CP0488318
|
US9029370, 19
Show/Hide
|
C16H16Cl2N4O2
|
1
|
| 1 |
Ki = 3.4 nM
|
|
|
|
CP0939770
|
US9181230, 3
Show/Hide
|
C19H18ClN3O
|
1
|
| 1 |
Ki = 3.4 nM
|
|
|
|
CP0405835
|
US10501411, Example 193
Show/Hide
|
C16H16ClN3O2
|
1
|
| 1 |
Ki = 3.4 nM
|
|
|
|
CP0506781
|
US9029370, 56
Show/Hide
|
C18H16F2N4O2
|
1
|
| 1 |
Ki = 3.5 nM
|
|
|
|
CP0481201
|
US10501411, Example 253
Show/Hide
|
C19H22N2O
|
1
|
| 1 |
Ki = 3.5 nM
|
|
|
|
CP0491900
|
US10501411, Example 205
Show/Hide
|
C18H18F3N3O2
|
1
|
| 1 |
Ki = 3.5 nM
|
|
|
|
CP0506775
|
US9029370, 22
Show/Hide
|
C20H18F2N4O2
|
1
|
| 1 |
Ki = 3.6 nM
|
|
|
|
CP0518578
|
US9029370, 29
Show/Hide
|
C20H18ClFN4O2
|
1
|
| 1 |
Ki = 3.6 nM
|
|
|
|
CP0561011
|
US9029370, 132
Show/Hide
|
C19H16F4N6O2
|
1
|
| 1 |
Ki = 3.6 nM
|
|
|
|
CP0902148
|
US9181230, 31
Show/Hide
|
C19H18FN3O
|
1
|
| 1 |
Ki = 3.6 nM
|
|
|
|
CP0404995
|
US10501411, Example 18
Show/Hide
|
C18H17F3N2O
|
1
|
| 1 |
Ki = 3.6 nM
|
|
|
|
CP0423948
|
US10501411, Example 275
Show/Hide
|
C19H22N2O3
|
1
|
| 1 |
Ki = 3.6 nM
|
|
|
|
CP0475692
|
US10501411, Example 277
Show/Hide
|
C18H20N2O2
|
1
|
| 1 |
Ki = 3.6 nM
|
|
|
|
CP0512888
|
US10501411, Example 124
Show/Hide
|
C19H20F2N2O2
|
1
|
| 1 |
Ki = 3.6 nM
|
|
|
|
CP0531313
|
US10501411, Example 7
Show/Hide
|
C17H17Cl2N3O
|
1
|
| 1 |
Ki = 3.6 nM
|
|
|
|
CP0478763
|
US10501411, Example 221
Show/Hide
|
C16H15Cl2N3O2
|
1
|
| 1 |
Ki = 3.7 nM
|
|
|
|
CP0488843
|
US9029370, 109
Show/Hide
|
C21H17ClFN5O2
|
1
|
| 1 |
Ki = 3.8 nM
|
|
|
|
CP0499848
|
US9029370, 67
Show/Hide
|
C16H16BrClN4O2
|
1
|
| 1 |
Ki = 3.8 nM
|
|
|
|
CP0535911
|
US9029370, 130
Show/Hide
|
C20H17F4N5O2
|
1
|
| 1 |
Ki = 3.8 nM
|
|
|
|
CP0538898
|
US9029370, 27
Show/Hide
|
C18H16F2N4O2
|
1
|
| 1 |
Ki = 3.8 nM
|
|
|
|
CP0386656
|
US10501411, Example 306
Show/Hide
|
C19H23N3O2
|
1
|
| 1 |
Ki = 3.8 nM
|
|
|
|
CP0481211
|
US10501411, Example 305
Show/Hide
|
C17H18ClN3O2
|
1
|
| 1 |
Ki = 3.8 nM
|
|
|
|
CP0441604
|
US9029370, 78
Show/Hide
|
C19H20F3N3O3
|
1
|
| 1 |
Ki = 3.9 nM
|
|
|
|
CP0542939
|
US9029370, 8
Show/Hide
|
C16H16ClFN4O2
|
1
|
| 1 |
Ki = 3.9 nM
|
|
|
|
CP0542941
|
US9029370, 14
Show/Hide
|
C16H16Cl2N4O2
|
1
|
| 1 |
Ki = 3.9 nM
|
|
|
|
CP0554637
|
US9029370, 74
Show/Hide
|
C20H21FN4O3
|
1
|
| 1 |
Ki = 3.9 nM
|
|
|
|
CP0512018
|
US9029370, 134
Show/Hide
|
C19H16F4N6O2
|
1
|
| 1 |
Ki = 4 nM
|
|
|
|
CP0490993
|
US10501411, Example 257
Show/Hide
|
C17H20N4OS
|
1
|
| 1 |
Ki = 4 nM
|
|
|
|
CP0512890
|
US10501411, Example 113
Show/Hide
|
C18H19ClN2O
|
1
|
| 1 |
Ki = 4 nM
|
|
|
|
CP0515636
|
US10501411, Example 271
Show/Hide
|
C16H15Cl2N3O2
|
1
|
| 1 |
Ki = 4 nM
|
|
|
|
CP0548073
|
US10501411, Example 207
Show/Hide
|
C16H16ClN3O2
|
1
|
| 1 |
Ki = 4.2 nM
|
|
|
|
CP0868677
|
US9181230, 41
Show/Hide
|
C19H17F2N3O
|
1
|
| 1 |
Ki = 4.3 nM
|
|
|
|
CP0405863
|
US10501411, Example 204
Show/Hide
|
C18H18F3N3O2
|
1
|
| 1 |
Ki = 4.3 nM
|
|
|
|
CP0553955
|
US10501411, Example 16
Show/Hide
|
C17H17ClN2O
|
1
|
| 1 |
Ki = 4.3 nM
|
|
|
|
CP0556581
|
US9029370, 45
Show/Hide
|
C19H19ClN4O3
|
1
|
| 1 |
Ki = 4.4 nM
|
|
|
|
CP0939771
|
US9181230, 29
Show/Hide
|
C19H18FN3O
|
1
|
| 1 |
Ki = 4.4 nM
|
|
|
|
CP0387675
|
US10501411, Example 8
Show/Hide
|
C17H18ClN3O
|
1
|
| 1 |
Ki = 4.4 nM
|
|
|
|
CP0425535
|
US10501411, Example 279
Show/Hide
|
C20H24N4O2
|
1
|
| 1 |
Ki = 4.4 nM
|
|
|
|
CP0490765
|
US10501411, Example 252
Show/Hide
|
C17H18BrN3O
|
1
|
| 1 |
Ki = 4.4 nM
|
|
|
|
CP0518664
|
US10501411, Example 208
Show/Hide
|
C16H16ClN3O2
|
1
|
| 1 |
Ki = 4.4 nM
|
|
|
|
CP0548081
|
US10501411, Example 297
Show/Hide
|
C19H23N3O
|
1
|
| 1 |
Ki = 4.4 nM
|
|
|
|
CP0574106
|
US10501411, Example 286
Show/Hide
|
C17H18ClN3O2
|
1
|
| 1 |
Ki = 4.4 nM
|
|
|
|
CP0450282
|
US9029370, 92
Show/Hide
|
C18H20ClN3O3
|
1
|
| 1 |
Ki = 4.5 nM
|
|
|
|
CP0515677
|
US10501411, Example 270
Show/Hide
|
C16H15Cl2N3O2
|
1
|
| 1 |
Ki = 4.5 nM
|
|
|
|
CP0413221
|
US10501411, Example 62
Show/Hide
|
C20H21F3N2O2
|
1
|
| 1 |
Ki = 4.6 nM
|
|
|
|
CP0480771
|
US11697636, Example 160
Show/Hide
|
C16H17ClN4O
|
1
|
| 1 |
Ki = 4.6 nM
|
|
|
|
CP0512620
|
US9029370, 126
Show/Hide
|
C19H16ClF3N6O2
|
1
|
| 1 |
Ki = 4.7 nM
|
|
|
|
CP0538891
|
US9029370, 84
Show/Hide
|
C18H20FN3O3
|
1
|
| 1 |
Ki = 4.7 nM
|
|
|
|
CP0491897
|
US11697636, Example 167
Show/Hide
|
C17H18ClN3O
|
1
|
| 1 |
Ki = 4.8 nM
|
|
|
|
CP0512885
|
US10501411, Example 282
Show/Hide
|
C18H20ClN3O
|
1
|
| 1 |
Ki = 4.8 nM
|
|
|
|
CP0516910
|
US10501411, Example 47
Show/Hide
|
C18H19FN2O2
|
1
|
| 1 |
Ki = 4.8 nM
|
|
|
|
CP0488370
|
US10501411, Example 244
Show/Hide
|
C18H21N3OS
|
1
|
| 1 |
Ki = 4.9 nM
|
|
|
|
CP0539903
|
US9452980, 148
Show/Hide
|
C16H16ClN3O2
|
1
|
| 1 |
Ki = 4.9 nM
|
|
|
|
CP0468227
|
US9029370, 20
Show/Hide
|
C16H16Cl2N4O2
|
1
|
| 1 |
Ki = 5 nM
|
|
|
|
CP0469602
|
US10501411, Example 194
Show/Hide
|
C17H16N4O2
|
1
|
| 1 |
Ki = 5 nM
|
|
|
|
CP0490769
|
US10501411, Example 284
Show/Hide
|
C17H16F3N3O2
|
1
|
| 1 |
Ki = 5 nM
|
|
|
|
CP0544299
|
US10501411, Example 285
Show/Hide
|
C17H18ClN3O2
|
1
|
| 1 |
Ki = 5 nM
|
|
|
|
CP0919298
|
US9029370, 1
Show/Hide
|
C18H16F2N4O2
|
1
|
| 1 |
Ki = 5.1 nM
|
|
|
|
CP0557248
|
US10501411, Example 139
Show/Hide
|
C17H16F3N3O
|
1
|
| 1 |
Ki = 5.1 nM
|
|
|
|
CP0524299
|
US9029370, 37
Show/Hide
|
C16H16BrClN4O2
|
1
|
| 1 |
Ki = 5.3 nM
|
|
|
|
CP0478329
|
US10501411, Example 53
Show/Hide
|
C20H24N2O
|
1
|
| 1 |
Ki = 5.3 nM
|
|
|
|
CP0486271
|
US10501411, Example 251
Show/Hide
|
C16H17BrN4O
|
1
|
| 1 |
Ki = 5.4 nM
|
|
|
|
CP0536959
|
US10501411, Example 188
Show/Hide
|
C17H18N2O2
|
1
|
| 1 |
Ki = 5.5 nM
|
|
|
|
CP0488372
|
US10501411, Example 302
Show/Hide
|
C16H17ClN4O2
|
1
|
| 1 |
Ki = 5.6 nM
|
|
|
|
CP0499605
|
US10501411, Example 238
Show/Hide
|
C16H17ClN4O
|
1
|
| 1 |
Ki = 5.6 nM
|
|
|
|
CP0549631
|
US10501411, Example 250
Show/Hide
|
C18H19F3N4O2
|
1
|
| 1 |
Ki = 5.6 nM
|
|
|
|
CP0513417
|
US9029370, 52
Show/Hide
|
C16H15ClF3N5O2
|
1
|
| 1 |
Ki = 5.8 nM
|
|
|
|
CP0488319
|
US9029370, 28
Show/Hide
|
C21H18FN5O2
|
1
|
| 1 |
Ki = 5.9 nM
|
|
|
|
CP0488838
|
US9029370, 44
Show/Hide
|
C19H19FN4O3
|
1
|
| 1 |
Ki = 5.9 nM
|
|
|
|
CP0541863
|
US9029370, 108
Show/Hide
|
C21H17F2N5O2
|
1
|
| 1 |
Ki = 5.9 nM
|
|
|
|
CP0913787
|
US9181230, 4
Show/Hide
|
C19H18FN3O
|
1
|
| 1 |
Ki = 5.9 nM
|
|
|
|
CP0405833
|
US10501411, Example 138
Show/Hide
|
C18H18F3N3O
|
1
|
| 1 |
Ki = 5.9 nM
|
|
|
|
CP0481204
|
US10501411, Example 265
Show/Hide
|
C18H18F3N3O
|
1
|
| 1 |
Ki = 5.9 nM
|
|
|
|
CP0516909
|
US10501411, Example 283
Show/Hide
|
C17H16F3N3O2
|
1
|
| 1 |
Ki = 5.9 nM
|
|
|
|
CP0491893
|
US10501411, Example 89
Show/Hide
|
C18H18F3N3O2
|
1
|
| 1 |
Ki = 6 nM
|
|
|
|
CP0387670
|
US10501411, Example 243
Show/Hide
|
C18H21N3O
|
1
|
| 1 |
Ki = 6.2 nM
|
|
|
|
CP0478325
|
US10501411, Example 210
Show/Hide
|
C16H16ClN3O2
|
1
|
| 1 |
Ki = 6.2 nM
|
|
|
|
CP0478331
|
US10501411, Example 314
Show/Hide
|
C18H19ClN2O2
|
1
|
| 1 |
Ki = 6.2 nM
|
|
|
|
CP0515643
|
US10501411, Example 129
Show/Hide
|
C20H22N2O2
|
1
|
| 1 |
Ki = 6.2 nM
|
|
|
|
CP0548076
|
US10501411, Example 258
Show/Hide
|
C21H24N2O2
|
1
|
| 1 |
Ki = 6.2 nM
|
|
|
|
CP0387671
|
US10501411, Example 245
Show/Hide
|
C18H21N3O3
|
1
|
| 1 |
Ki = 6.3 nM
|
|
|
|
CP0506938
|
US9029370, 46
Show/Hide
|
C19H19ClN4O3
|
1
|
| 1 |
Ki = 6.4 nM
|
|
|
|
CP0538901
|
US9029370, 77
Show/Hide
|
C19H20F3N3O3
|
1
|
| 1 |
Ki = 6.4 nM
|
|
|
|
CP0566771
|
US9029370, 107
Show/Hide
|
C18H17FN4O3
|
1
|
| 1 |
Ki = 6.5 nM
|
|
|
|
CP0514621
|
US9029370, 85
Show/Hide
|
C18H20FN3O3
|
1
|
| 1 |
Ki = 6.7 nM
|
|
|
|
CP0544394
|
US10501411, Example 96
Show/Hide
|
C18H18Cl2N2O
|
1
|
| 1 |
Ki = 6.7 nM
|
|
|
|
CP0560152
|
US11697636, Example 177
Show/Hide
|
C22H24N2O
|
1
|
| 1 |
Ki = 6.7 nM
|
|
|
|
CP0553587
|
US9416127, 24
Show/Hide
|
C20H21N5O2
|
1
|
| 1 |
Ki = 6.9 nM
|
|
|
|
CP0486273
|
US10501411, Example 280
Show/Hide
|
C17H16F3N3O2
|
1
|
| 1 |
Ki = 6.9 nM
|
|
|
|
CP0441930
|
US9029370, 24
Show/Hide
|
C17H17ClFN3O3
|
1
|
| 1 |
Ki = 7 nM
|
|
|
|
CP0512886
|
US10501411, Example 301
Show/Hide
|
C17H16ClIN2O2
|
1
|
| 1 |
Ki = 7 nM
|
|
|
|
CP0413211
|
US10501411, Example 1
Show/Hide
|
C22H29N3O
|
1
|
| 1 |
Ki = 7.2 nM
|
|
|
|
CP0405000
|
US10501411, Example 191
Show/Hide
|
C19H20F3N3O2
|
1
|
| 1 |
Ki = 7.4 nM
|
|
|
|
CP0425494
|
US10501411, Example 114
Show/Hide
|
C18H21ClN4O
|
1
|
| 1 |
Ki = 7.4 nM
|
|
|
|
CP0563898
|
US9029370, 83
Show/Hide
|
C17H15F4N3O2
|
1
|
| 1 |
Ki = 7.5 nM
|
|
|
|
CP0555547
|
US10501411, Example 288
Show/Hide
|
C18H17N5O2S
|
1
|
| 1 |
Ki = 7.5 nM
|
|
|
|
CP0514637
|
US9029370, 125
Show/Hide
|
C19H16F4N6O2
|
1
|
| 1 |
Ki = 7.6 nM
|
|
|
|
CP0478803
|
US10501411, Example 20
Show/Hide
|
C17H17ClN2O
|
1
|
| 1 |
Ki = 7.7 nM
|
|
|
|
CP0484103
|
US10501411, Example 45
Show/Hide
|
C17H22F2N2O2
|
1
|
| 1 |
Ki = 7.7 nM
|
|
|
|
CP0484440
|
US11697636, Example 172
Show/Hide
|
C20H25N3O2
|
1
|
| 1 |
Ki = 7.7 nM
|
|
|
|
CP0481206
|
US10501411, Example 273
Show/Hide
|
C17H18ClN3O2
|
1
|
| 1 |
Ki = 8 nM
|
|
|
|
CP0474481
|
US9029370, 68
Show/Hide
|
C16H16BrClN4O2
|
1
|
| 1 |
Ki = 8.1 nM
|
|
|
|
CP0429137
|
US10501411, Example 15
Show/Hide
|
C17H17FN2O2
|
1
|
| 1 |
Ki = 8.1 nM
|
|
|
|
CP0480822
|
US10501411, Example 118
Show/Hide
|
C19H22ClN3O
|
1
|
| 1 |
Ki = 8.1 nM
|
|
|
|
CP0539900
|
US10501411, Example 108
Show/Hide
|
C20H18ClN3O
|
1
|
| 1 |
Ki = 8.1 nM
|
|
|
|
CP0493481
|
US9416127, 30
Show/Hide
|
C20H21N5O3
|
1
|
| 1 |
Ki = 8.2 nM
|
|
|
|
CP0466478
|
US9029370, 39
Show/Hide
|
C19H19FN4O3
|
1
|
| 1 |
Ki = 8.5 nM
|
|
|
|
CP0387669
|
US10501411, Example 239
Show/Hide
|
C16H17ClN4O
|
1
|
| 1 |
Ki = 8.5 nM
|
|
|
|
CP0468232
|
US9029370, 111
Show/Hide
|
C21H18FN5O2
|
1
|
| 1 |
Ki = 8.6 nM
|
|
|
|
CP0413450
|
US10501411, Example 218
Show/Hide
|
C16H16ClN3O2
|
1
|
| 1 |
Ki = 8.7 nM
|
|
|
|
CP0478327
|
US10501411, Example 242
Show/Hide
|
C18H18F3N3O
|
1
|
| 1 |
Ki = 8.9 nM
|
|
|
|
CP0533136
|
US9029370, 41
Show/Hide
|
C17H18Cl2N4O
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0516912
|
US10501411, Example 315
Show/Hide
|
C17H18ClN3O2
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0493418
|
US9416127, 25
Show/Hide
|
C20H21N5O3
|
1
|
| 1 |
Ki = 9.2 nM
|
|
|
|
CP0491896
|
US11697636, Example 162
Show/Hide
|
C17H18ClN3O
|
1
|
| 1 |
Ki = 9.2 nM
|
|
|
|
CP0466964
|
US9029370, 11
Show/Hide
|
C17H16F4N4O2
|
1
|
| 1 |
Ki = 9.5 nM
|
|
|
|
CP0512911
|
US11697636, Example 161
Show/Hide
|
C17H18ClN3O
|
1
|
| 1 |
Ki = 10.1 nM
|
|
|
|
CP0513469
|
US10501411, Example 90
Show/Hide
|
C21H21N3O2
|
1
|
| 1 |
Ki = 10.1 nM
|
|
|
|
CP0536958
|
US11697636, Example 171
Show/Hide
|
C19H22ClN3O
|
1
|
| 1 |
Ki = 10.1 nM
|
|
|
|
CP0506783
|
US9029370, 70
Show/Hide
|
C16H15BrF3N5O2
|
1
|
| 1 |
Ki = 10.3 nM
|
|
|
|
CP0553385
|
US9029370, 9
Show/Hide
|
C16H16ClFN4O2
|
1
|
| 1 |
Ki = 10.5 nM
|
|
|
|
CP0493123
|
US10501411, Example 310
Show/Hide
|
C17H18ClN3O2
|
1
|
| 1 |
Ki = 10.8 nM
|
|
|
|
CP0405853
|
US10501411, Example 52
Show/Hide
|
C19H22N2O2
|
1
|
| 1 |
Ki = 10.9 nM
|
|
|
|
CP0413446
|
US10501411, Example 192
Show/Hide
|
C24H24N2O3
|
1
|
| 1 |
Ki = 11.3 nM
|
|
|
|
CP0425522
|
US10501411, Example 37
Show/Hide
|
C19H21ClN2O
|
1
|
| 1 |
Ki = 11.4 nM
|
|
|
|
CP0513442
|
US10501411, Example 98
Show/Hide
|
C19H19F3N2O
|
1
|
| 1 |
Ki = 11.4 nM
|
|
|
|
CP0405856
|
US10501411, Example 115
Show/Hide
|
C19H23ClN4O
|
1
|
| 1 |
Ki = 11.8 nM
|
|
|
|
CP0481208
|
US10501411, Example 278
Show/Hide
|
C19H24N4O
|
1
|
| 1 |
Ki = 11.8 nM
|
|
|
|
CP0387656
|
US10501411, Example 83
Show/Hide
|
C17H19ClN4O
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0512905
|
US10501411, Example 256
Show/Hide
|
C19H23N3O2
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0491891
|
US10501411, Example 71
Show/Hide
|
C17H17ClN2O2
|
1
|
| 1 |
Ki = 12.1 nM
|
|
|
|
CP0516914
|
US11697636, Example 164
Show/Hide
|
C17H19ClN4O
|
1
|
| 1 |
Ki = 12.1 nM
|
|
|
|
CP0554132
|
US11697636, Example 163
Show/Hide
|
C15H15ClN4O
|
1
|
| 1 |
Ki = 12.1 nM
|
|
|
|
CP0561164
|
US10501411, Example 316
Show/Hide
|
C19H20F3N3O3
|
1
|
| 1 |
Ki = 12.1 nM
|
|
|
|
CP0512216
|
US9181230, 26
Show/Hide
|
C19H18FN3O
|
1
|
| 1 |
Ki = 12.2 nM
|
|
|
|
CP0555960
|
US10501411, Example 187
Show/Hide
|
C17H18ClN3O
|
1
|
| 1 |
Ki = 12.3 nM
|
|
|
|
CP0419307
|
US10501411, Example 81
Show/Hide
|
C20H20N4O
|
1
|
| 1 |
Ki = 12.4 nM
|
|
|
|
CP0533137
|
US9029370, 51
Show/Hide
|
C16H15ClF3N5O2
|
1
|
| 1 |
Ki = 12.6 nM
|
|
|
|
CP0450169
|
US9029370, 57
Show/Hide
|
C19H19BrN4O3
|
1
|
| 1 |
Ki = 12.7 nM
|
|
|
|
CP0451905
|
US9029370, 25
Show/Hide
|
C17H17ClFN3O3
|
1
|
| 1 |
Ki = 12.7 nM
|
|
|
|
CP0441929
|
US9029370, 17
Show/Hide
|
C21H21FN4O2
|
1
|
| 1 |
Ki = 12.8 nM
|
|
|
|
CP0930210
|
US9181230, 7
Show/Hide
|
C16H15BrN4O
|
1
|
| 1 |
Ki = 12.8 nM
|
|
|
|
CP0554134
|
US11697636, Example 180
Show/Hide
|
C17H18FN3O
|
1
|
| 1 |
Ki = 13.1 nM
|
|
|
|
CP0405858
|
US10501411, Example 135
Show/Hide
|
C19H21F2N3O
|
1
|
| 1 |
Ki = 13.4 nM
|
|
|
|
CP0491894
|
US10501411, Example 105
Show/Hide
|
C21H23F3N2O2
|
1
|
| 1 |
Ki = 13.5 nM
|
|
|
|
CP0387672
|
US10501411, Example 248
Show/Hide
|
C17H17F3N4O
|
1
|
| 1 |
Ki = 14.3 nM
|
|
|
|
CP0488371
|
US10501411, Example 298
Show/Hide
|
C19H19N5O2S
|
1
|
| 1 |
Ki = 14.3 nM
|
|
|
|
CP0572282
|
US10501411, Example 264
Show/Hide
|
C18H21N3O
|
1
|
| 1 |
Ki = 14.3 nM
|
|
|
|
CP0553384
|
US9029370, 131
Show/Hide
|
C19H16FN7O2
|
1
|
| 1 |
Ki = 14.4 nM
|
|
|
|
CP0514623
|
US9029370, 110
Show/Hide
|
C21H17F2N5O2
|
1
|
| 1 |
Ki = 15.2 nM
|
|
|
|
CP0387654
|
US10501411, Example 54
Show/Hide
|
C19H18N2O
|
1
|
| 1 |
Ki = 15.2 nM
|
|
|
|
CP0928189
|
US9181230, 32
Show/Hide
|
C20H18N4O
|
1
|
| 1 |
Ki = 15.4 nM
|
|
|
|
CP0553588
|
US9416127, 27
Show/Hide
|
C20H18F3N5O3
|
1
|
| 1 |
Ki = 15.4 nM
|
|
|
|
CP0478817
|
US10501411, Example 313
Show/Hide
|
C18H19ClN2O2
|
1
|
| 1 |
Ki = 15.4 nM
|
|
|
|
CP0865216
|
US9181230, 40
Show/Hide
|
C19H17F2N3O
|
1
|
| 1 |
Ki = 15.5 nM
|
|
|
|
CP0553281
|
US9416127, 28
Show/Hide
|
C20H18F3N5O3
|
1
|
| 1 |
Ki = 15.6 nM
|
|
|
|
CP0514646
|
US9029370, 121
Show/Hide
|
C18H17FN4O3
|
1
|
| 1 |
Ki = 15.8 nM
|
|
|
|
CP0425529
|
US11697636, Example 170
Show/Hide
|
C20H23FN2O
|
1
|
| 1 |
Ki = 15.8 nM
|
|
|
|
CP0554133
|
US11697636, Example 174
Show/Hide
|
C18H21ClN4O
|
1
|
| 1 |
Ki = 15.9 nM
|
|
|
|
CP0503635
|
US9029370, 66
Show/Hide
|
C17H16BrN5O2
|
1
|
| 1 |
Ki = 16.1 nM
|
|
|
|
CP0549961
|
US9029370, 58
Show/Hide
|
C19H19BrN4O3
|
1
|
| 1 |
Ki = 16.1 nM
|
|
|
|
CP0902147
|
US9181230, 28
Show/Hide
|
C20H18N4O
|
1
|
| 1 |
Ki = 16.8 nM
|
|
|
|
CP0497611
|
US10501411, Example 272
Show/Hide
|
C17H16F3N3O2
|
1
|
| 1 |
Ki = 16.9 nM
|
|
|
|
CP0548066
|
US10501411, Example 130
Show/Hide
|
C19H18ClF3N2O2
|
1
|
| 1 |
Ki = 16.9 nM
|
|
|
|
CP0425526
|
US10501411, Example 87
Show/Hide
|
C16H16BrN3O
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0910427
|
US9181230, 42
Show/Hide
|
C18H17ClN4O
|
1
|
| 1 |
Ki = 17.1 nM
|
|
|
|
CP0561196
|
US9416127, 17
Show/Hide
|
C20H21N5O2
|
1
|
| 1 |
Ki = 17.4 nM
|
|
|
|
CP0405865
|
US10501411, Example 274
Show/Hide
|
C18H22N4O
|
1
|
| 1 |
Ki = 17.4 nM
|
|
|
|
CP0516913
|
US10501411, Example 133
Show/Hide
|
C18H19F2N3O
|
1
|
| 1 |
Ki = 17.4 nM
|
|
|
|
CP0423322
|
US10501411, Example 109
Show/Hide
|
C19H21ClN2O
|
1
|
| 1 |
Ki = 17.6 nM
|
|
|
|
CP0462835
|
US9029370, 133
Show/Hide
|
C17H14ClFN4O2
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0506782
|
US9029370, 69
Show/Hide
|
C16H15BrF3N5O2
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0868682
|
US9181230, 49
Show/Hide
|
C16H14F3N3O
|
1
|
| 1 |
Ki = 18.2 nM
|
|
|
|
CP0413264
|
US9416127, 33
Show/Hide
|
C20H19F2N5O2
|
1
|
| 1 |
Ki = 18.9 nM
|
|
|
|
CP0491889
|
US10501411, Example 19
Show/Hide
|
C17H16Cl2N2O
|
1
|
| 1 |
Ki = 18.9 nM
|
|
|
|
CP0554845
|
US9029370, 38
Show/Hide
|
C16H16Cl2N4O
|
1
|
| 1 |
Ki = 19.1 nM
|
|
|
|
CP0488377
|
US10501411, Example 97
Show/Hide
|
C20H24N2O2
|
1
|
| 1 |
Ki = 19.3 nM
|
|
|
|
CP0865215
|
US9181230, 23
Show/Hide
|
C18H17FN4O
|
1
|
| 1 |
Ki = 19.6 nM
|
|
|
|
CP0930207
|
US9181230, 33
Show/Hide
|
C20H17FN4O
|
1
|
| 1 |
Ki = 20.1 nM
|
|
|
|
CP0450281
|
US9029370, 87
Show/Hide
|
C17H15F4N3O2
|
1
|
| 1 |
Ki = 20.2 nM
|
|
|
|
CP0556585
|
US9029370, 100
Show/Hide
|
C17H15ClN4O2
|
1
|
| 1 |
Ki = 20.2 nM
|
|
|
|
CP0386666
|
US10501411, Example 85
Show/Hide
|
C20H19N3O
|
1
|
| 1 |
Ki = 20.5 nM
|
|
|
|
CP0561165
|
US10501411, Example 319
Show/Hide
|
C17H18ClN3O2
|
1
|
| 1 |
Ki = 20.6 nM
|
|
|
|
CP0387661
|
US11697636, Example 166
Show/Hide
|
C18H20FN3O
|
1
|
| 1 |
Ki = 21.2 nM
|
|
|
|
CP0519668
|
US10501411, Example 64
Show/Hide
|
C26H26N2O2
|
1
|
| 1 |
Ki = 21.5 nM
|
|
|
|
CP0468229
|
US9029370, 65
Show/Hide
|
C17H16BrN5O2
|
1
|
| 1 |
Ki = 21.8 nM
|
|
|
|
CP0470707
|
US11697636, Example 173
Show/Hide
|
C19H22ClN3O
|
1
|
| 1 |
Ki = 21.8 nM
|
|
|
|
CP0386663
|
US10501411, Example 131
Show/Hide
|
C15H19F3N2O2
|
1
|
| 1 |
Ki = 21.9 nM
|
|
|
|
CP0515740
|
US10501411, Example 91
Show/Hide
|
C21H21N3O2
|
1
|
| 1 |
Ki = 22.3 nM
|
|
|
|
CP0537351
|
US10501411, Example 317
Show/Hide
|
C18H19ClN2O2
|
1
|
| 1 |
Ki = 22.6 nM
|
|
|
|
CP0539161
|
US9029370, 34
Show/Hide
|
C17H16Cl2N2O2
|
1
|
| 1 |
Ki = 22.9 nM
|
|
|
|
CP0556174
|
US10501411, Example 69
Show/Hide
|
C17H16ClFN2O
|
1
|
| 1 |
Ki = 23 nM
|
|
|
|
CP0553383
|
US9029370, 124
Show/Hide
|
C18H17ClN4O3
|
1
|
| 1 |
Ki = 23.1 nM
|
|
|
|
CP0480811
|
US10501411, Example 77
Show/Hide
|
C17H16ClFN2O
|
1
|
| 1 |
Ki = 23.8 nM
|
|
|
|
CP0554659
|
US10501411, Example 92
Show/Hide
|
C18H19ClN2O
|
1
|
| 1 |
Ki = 23.8 nM
|
|
|
|
CP0553956
|
US10501411, Example 43
Show/Hide
|
C16H16ClN3O
|
1
|
| 1 |
Ki = 24.2 nM
|
|
|
|
CP0561411
|
US9029370, 112
Show/Hide
|
C18H17ClN4O2
|
1
|
| 1 |
Ki = 24.8 nM
|
|
|
|
CP0577304
|
US10501411, Example 320
Show/Hide
|
C18H18F3N3O2
|
1
|
| 1 |
Ki = 24.9 nM
|
|
|
|
CP0441068
|
US9181230, 35
Show/Hide
|
C18H17FN4O
|
1
|
| 1 |
Ki = 25.2 nM
|
|
|
|
CP0553387
|
US9029370, 89
Show/Hide
|
C18H20FN3O3
|
1
|
| 1 |
Ki = 25.4 nM
|
|
|
|
CP0953394
|
US9181230, 38
Show/Hide
|
C18H17ClN4O
|
1
|
| 1 |
Ki = 25.7 nM
|
|
|
|
CP0512928
|
US10501411, Example 73
Show/Hide
|
C19H19N5O
|
1
|
| 1 |
Ki = 25.7 nM
|
|
|
|
CP0537352
|
US10501411, Example 321
Show/Hide
|
C18H18F3N3O2
|
1
|
| 1 |
Ki = 26 nM
|
|
|
|
CP0539899
|
US10501411, Example 101
Show/Hide
|
C20H23ClN2O
|
1
|
| 1 |
Ki = 26.3 nM
|
|
|
|
CP0491061
|
US10501411, Example 104
Show/Hide
|
C21H23F3N2O
|
1
|
| 1 |
Ki = 27.6 nM
|
|
|
|
CP0413218
|
US10501411, Example 26
Show/Hide
|
C16H17ClN4O
|
1
|
| 1 |
Ki = 27.9 nM
|
|
|
|
CP0928984
|
US9181230, 43
Show/Hide
|
C17H16FN3O
|
1
|
| 1 |
Ki = 29.1 nM
|
|
|
|
CP0481229
|
US9416127, 21
Show/Hide
|
C21H23N5O3
|
1
|
| 1 |
Ki = 29.3 nM
|
|
|
|
CP0393346
|
US10501411, Example 6
Show/Hide
|
C17H19N3O
|
1
|
| 1 |
Ki = 29.5 nM
|
|
|
|
CP0493419
|
US9416127, 36
Show/Hide
|
C18H17BrN6O2
|
1
|
| 1 |
Ki = 30 nM
|
|
|
|
CP0468233
|
US9029370, 137
Show/Hide
|
C16H14F4N4O2
|
1
|
| 1 |
Ki = 30.1 nM
|
|
|
|
CP0928985
|
US9181230, 13
Show/Hide
|
C19H17F2N3O
|
1
|
| 1 |
Ki = 30.5 nM
|
|
|
|
CP0491888
|
US10501411, Example 307
Show/Hide
|
C17H25N3O2
|
1
|
| 1 |
Ki = 30.5 nM
|
|
|
|
CP0386669
|
US10501411, Example 100
Show/Hide
|
C18H18ClFN2O
|
1
|
| 1 |
Ki = 30.8 nM
|
|
|
|
CP0425536
|
US10501411, Example 318
Show/Hide
|
C18H19ClN2O2
|
1
|
| 1 |
Ki = 31.2 nM
|
|
|
|
CP0386658
|
US10501411, Example 11
Show/Hide
|
C17H18N2O2
|
1
|
| 1 |
Ki = 31.5 nM
|
|
|
|
CP0470651
|
US10501411, Example 232
Show/Hide
|
C21H25N3O4
|
1
|
| 1 |
Ki = 31.7 nM
|
|
|
|
CP0530371
|
US9181230, 39
Show/Hide
|
C18H17FN4O
|
1
|
| 1 |
Ki = 32.2 nM
|
|
|
|
CP0538890
|
US9029370, 80
Show/Hide
|
C17H15FN4O2
|
1
|
| 1 |
Ki = 32.5 nM
|
|
|
|
CP0929265
|
US9181230, 6
Show/Hide
|
C20H18N4O
|
1
|
| 1 |
Ki = 33.5 nM
|
|
|
|
CP0565578
|
US9029370, 104
Show/Hide
|
C20H18F3N5O3
|
1
|
| 1 |
Ki = 34 nM
|
|
|
|
CP0450284
|
US9029370, 115
Show/Hide
|
C18H17FN4O2
|
1
|
| 1 |
Ki = 34.3 nM
|
|
|
|
CP0555915
|
US9029370, 95
Show/Hide
|
C18H20ClN3O3
|
1
|
| 1 |
Ki = 35 nM
|
|
|
|
CP0576484
|
US10501411, Example 42
Show/Hide
|
C16H16ClN3O
|
1
|
| 1 |
Ki = 35.4 nM
|
|
|
|
CP0480769
|
US10501411, Example 140
Show/Hide
|
C16H16ClN3O
|
1
|
| 1 |
Ki = 35.8 nM
|
|
|
|
CP0387684
|
US10501411, Example 17
Show/Hide
|
C18H19ClN2O
|
1
|
| 1 |
Ki = 36.3 nM
|
|
|
|
CP0423323
|
US10501411, Example 110
Show/Hide
|
C20H23ClN2O
|
1
|
| 1 |
Ki = 37.5 nM
|
|
|
|
CP0474483
|
US9029370, 94
Show/Hide
|
C18H20ClN3O3
|
1
|
| 1 |
Ki = 38.1 nM
|
|
|
|
CP0405854
|
US10501411, Example 84
Show/Hide
|
C20H19N3O
|
1
|
| 1 |
Ki = 38.1 nM
|
|
|
|
CP0405855
|
US10501411, Example 111
Show/Hide
|
C20H23ClN2O
|
1
|
| 1 |
Ki = 38.2 nM
|
|
|
|
CP0545113
|
US9416127, 19
Show/Hide
|
C20H21N5O3
|
1
|
| 1 |
Ki = 38.8 nM
|
|
|
|
CP0472163
|
US11697636, Example 165
Show/Hide
|
C17H16N4O
|
1
|
| 1 |
Ki = 41.1 nM
|
|
|
|
CP0537492
|
US10501411, Example 107
Show/Hide
|
C18H19ClN2O
|
1
|
| 1 |
Ki = 44.5 nM
|
|
|
|
CP0488314
|
US9029370, 117
Show/Hide
|
C19H21FN4O3
|
1
|
| 1 |
Ki = 45 nM
|
|
|
|
CP0413263
|
US9416127, 32
Show/Hide
|
C20H19F2N5O3
|
1
|
| 1 |
Ki = 45 nM
|
|
|
|
CP0554033
|
US10501411, Example 60
Show/Hide
|
C19H21ClN2O2
|
1
|
| 1 |
Ki = 45.7 nM
|
|
|
|
CP0514622
|
US9029370, 88
Show/Hide
|
C18H20FN3O3
|
1
|
| 1 |
Ki = 45.8 nM
|
|
|
|
CP0548062
|
US10501411, Example 78
Show/Hide
|
C17H18ClN3O
|
1
|
| 1 |
Ki = 46.6 nM
|
|
|
|
CP0542938
|
US9029370, 123
Show/Hide
|
C18H17ClN4O2
|
1
|
| 1 |
Ki = 47.4 nM
|
|
|
|
CP0484425
|
US10501411, Example 24
Show/Hide
|
C19H19F3N2O
|
1
|
| 1 |
Ki = 49.7 nM
|
|
|
|
CP0406784
|
US10501411, Example 29
Show/Hide
|
C19H22N2O
|
1
|
| 1 |
Ki = 50.1 nM
|
|
|
|
CP0513443
|
US10501411, Example 99
Show/Hide
|
C18H18Cl2N2O
|
1
|
| 1 |
Ki = 50.1 nM
|
|
|
|
CP0563897
|
US9029370, 15
Show/Hide
|
C19H19FN4O2
|
1
|
| 1 |
Ki = 54.4 nM
|
|
|
|
CP0404996
|
US10501411, Example 33
Show/Hide
|
C19H21ClN2O
|
1
|
| 1 |
Ki = 54.5 nM
|
|
|
|
CP0386665
|
US10501411, Example 67
Show/Hide
|
C20H24N2O2
|
1
|
| 1 |
Ki = 55.5 nM
|
|
|
|
CP0531619
|
US9181230, 27
Show/Hide
|
C18H17FN4O
|
1
|
| 1 |
Ki = 56.5 nM
|
|
|
|
CP0868679
|
US9181230, 44
Show/Hide
|
C17H16FN3O
|
1
|
| 1 |
Ki = 57.1 nM
|
|
|
|
CP0535912
|
US9029370, 136
Show/Hide
|
C18H17FN4O2
|
1
|
| 1 |
Ki = 58.5 nM
|
|
|
|
CP0910994
|
US9181230, 11
Show/Hide
|
C17H15F2N3O
|
1
|
| 1 |
Ki = 59.7 nM
|
|
|
|
CP0387685
|
US10501411, Example 38
Show/Hide
|
C20H24N2O
|
1
|
| 1 |
Ki = 60.6 nM
|
|
|
|
CP0484442
|
US10501411, Example 228
Show/Hide
|
C22H26N2O4
|
1
|
| 1 |
Ki = 60.8 nM
|
|
|
|
CP0484102
|
US10501411, Example 31
Show/Hide
|
C19H21ClN2O
|
1
|
| 1 |
Ki = 61.3 nM
|
|
|
|
CP0512214
|
US9181230, 12
Show/Hide
|
C20H18N4O
|
1
|
| 1 |
Ki = 61.5 nM
|
|
|
|
CP0959316
|
US9181230, 5
Show/Hide
|
C18H17ClN4O
|
1
|
| 1 |
Ki = 63.1 nM
|
|
|
|
CP0469619
|
US10501411, Example 103
Show/Hide
|
C20H23ClN2O
|
1
|
| 1 |
Ki = 64.6 nM
|
|
|
|
CP0524304
|
US9029370, 113
Show/Hide
|
C18H17FN4O2
|
1
|
| 1 |
Ki = 65.4 nM
|
|
|
|
CP0438865
|
US9181230, 19
Show/Hide
|
C19H18FN3O
|
1
|
| 1 |
Ki = 66.9 nM
|
|
|
|
CP0512887
|
US10501411, Example 74
Show/Hide
|
C17H18ClN3O
|
1
|
| 1 |
Ki = 67.2 nM
|
|
|
|
CP0445130
|
US10501411, Example 247
Show/Hide
|
C17H20N4O
|
1
|
| 1 |
Ki = 67.7 nM
|
|
|
|
CP0488317
|
US9029370, 16
Show/Hide
|
C19H19FN4O2
|
1
|
| 1 |
Ki = 67.9 nM
|
|
|
|
CP0865217
|
US9181230, 46
Show/Hide
|
C16H14F3N3O
|
1
|
| 1 |
Ki = 69.8 nM
|
|
|
|
CP0943110
|
US9181230, 2
Show/Hide
|
C17H16ClN3O
|
1
|
| 1 |
Ki = 71.1 nM
|
|
|
|
CP0914173
|
US9181230, 24
Show/Hide
|
C18H23N3O2
|
1
|
| 1 |
Ki = 72.2 nM
|
|
|
|
CP0429139
|
US10501411, Example 30
Show/Hide
|
C19H22N2O
|
1
|
| 1 |
Ki = 72.2 nM
|
|
|
|
CP0512927
|
US10501411, Example 55
Show/Hide
|
C18H17N3O
|
1
|
| 1 |
Ki = 74.5 nM
|
|
|
|
CP0868681
|
US9181230, 47
Show/Hide
|
C15H14ClN3O
|
1
|
| 1 |
Ki = 75 nM
|
|
|
|
CP0406783
|
US10501411, Example 25
Show/Hide
|
C19H22N2O
|
1
|
| 1 |
Ki = 75.8 nM
|
|
|
|
CP0879626
|
US9181230, 20
Show/Hide
|
C18H17FN4O
|
1
|
| 1 |
Ki = 77.9 nM
|
|
|
|
CP0488375
|
US10501411, Example 35
Show/Hide
|
C25H25ClN2O
|
1
|
| 1 |
Ki = 78 nM
|
|
|
|
CP0488373
|
US10501411, Example 4
Show/Hide
|
C21H23N5O2
|
1
|
| 1 |
Ki = 83.7 nM
|
|
|
|
CP0561163
|
US10501411, Example 296
Show/Hide
|
C18H19N5O2S
|
1
|
| 1 |
Ki = 84.7 nM
|
|
|
|
CP0550187
|
US9181230, 36
Show/Hide
|
C18H17FN4O
|
1
|
| 1 |
Ki = 85.7 nM
|
|
|
|
CP0555958
|
US10501411, Example 32
Show/Hide
|
C18H19ClN2O
|
1
|
| 1 |
Ki = 85.8 nM
|
|
|
|
CP0438896
|
US9181230, 52
Show/Hide
|
C18H19N3O3
|
1
|
| 1 |
Ki = 87.3 nM
|
|
|
|
CP0393351
|
US10501411, Example 102
Show/Hide
|
C19H21ClN2O
|
1
|
| 1 |
Ki = 89.4 nM
|
|
|
|
CP0902151
|
US9181230, 51
Show/Hide
|
C17H20N4O2
|
1
|
| 1 |
Ki = 90.4 nM
|
|
|
|
CP0425524
|
US10501411, Example 79
Show/Hide
|
C17H19ClN4O
|
1
|
| 1 |
Ki = 92.4 nM
|
|
|
|
CP0450283
|
US9029370, 106
Show/Hide
|
C17H14ClFN4O2
|
1
|
| 1 |
Ki = 93.8 nM
|
|
|
|
CP0405837
|
US10501411, Example 217
Show/Hide
|
C15H17N3O2S
|
1
|
| 1 |
Ki = 94.1 nM
|
|
|
|
CP0491057
|
US10501411, Example 51
Show/Hide
|
C19H22N2O2
|
1
|
| 1 |
Ki = 98.5 nM
|
|
|
|
CP0386659
|
US10501411, Example 13
Show/Hide
|
C17H18N2O
|
1
|
| 1 |
Ki = 99.5 nM
|
|
|
|
CP0491892
|
US10501411, Example 88
Show/Hide
|
C18H19FN2O2
|
1
|
| 1 |
Ki = 101.6 nM
|
|
|
|
CP0469618
|
US10501411, Example 68
Show/Hide
|
C20H21N3O
|
1
|
| 1 |
Ki = 102 nM
|
|
|
|
CP0512994
|
US9416127, 31
Show/Hide
|
C21H23N5O3
|
1
|
| 1 |
Ki = 106.6 nM
|
|
|
|
CP0484092
|
US10501411, Example 72
Show/Hide
|
C17H17ClN2O2
|
1
|
| 1 |
Ki = 107.2 nM
|
|
|
|
CP0488321
|
US9029370, 35
Show/Hide
|
C16H15Cl2N3O2
|
1
|
| 1 |
Ki = 110.9 nM
|
|
|
|
CP0425525
|
US10501411, Example 86
Show/Hide
|
C16H16ClN3O
|
1
|
| 1 |
Ki = 115.6 nM
|
|
|
|
CP0515673
|
US10501411, Example 241
Show/Hide
|
C20H24N4O3
|
1
|
| 1 |
Ki = 116 nM
|
|
|
|
CP0468228
|
US9029370, 40
Show/Hide
|
C17H19ClN4O2
|
1
|
| 1 |
Ki = 120.4 nM
|
|
|
|
CP0413220
|
US10501411, Example 50
Show/Hide
|
C19H21BrN2O2
|
1
|
| 1 |
Ki = 121.7 nM
|
|
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CP0419405
|
US9181230, 25
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C18H17FN4O
|
1
|
| 1 |
Ki = 140.2 nM
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|
CP0423324
|
US10501411, Example 132
Show/Hide
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C18H20FN3O
|
1
|
| 1 |
Ki = 140.6 nM
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CP0488324
|
US9029370, 99
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C17H15ClN4O2
|
1
|
| 1 |
Ki = 154.4 nM
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|
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CP0531620
|
US9181230, 34
Show/Hide
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C18H16FN3O2
|
1
|
| 1 |
Ki = 156 nM
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|
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|
CP0450285
|
US9029370, 116
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C17H16ClFN4O3
|
1
|
| 1 |
Ki = 162.3 nM
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|
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CP0386667
|
US10501411, Example 93
Show/Hide
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C18H17N3OS
|
1
|
| 1 |
Ki = 172.9 nM
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CP0484075
|
US10501411, Example 63
Show/Hide
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C17H17ClN2O2
|
1
|
| 1 |
Ki = 174.3 nM
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CP0868674
|
US9181230, 14
Show/Hide
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C19H17F2N3O
|
1
|
| 1 |
Ki = 183 nM
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CP0488323
|
US9029370, 97
Show/Hide
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C17H15ClN4O2
|
1
|
| 1 |
Ki = 184 nM
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CP0488322
|
US9029370, 79
Show/Hide
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C17H15FN4O2
|
1
|
| 1 |
Ki = 196.3 nM
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|
|
|
CP0488374
|
US10501411, Example 34
Show/Hide
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C24H23ClN2O
|
1
|
| 1 |
Ki = 213.6 nM
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|
|
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CP0419406
|
US9181230, 53
Show/Hide
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C17H14F3N3O2
|
1
|
| 1 |
Ki = 226.1 nM
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|
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|
CP0539232
|
US9181230, 17
Show/Hide
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C18H16FN3O2
|
1
|
| 1 |
Ki = 228.5 nM
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|
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CP0419335
|
US10501411, Example 199
Show/Hide
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C17H18N2O3
|
1
|
| 1 |
Ki = 238.1 nM
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|
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CP0512215
|
US9181230, 18
Show/Hide
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C18H17FN4O
|
1
|
| 1 |
Ki = 254.3 nM
|
|
|
|
CP0474477
|
US9029370, 118
Show/Hide
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C18H19ClN4O3
|
1
|
| 1 |
Ki = 263.6 nM
|
|
|
|
CP0561419
|
US9029370, 114
Show/Hide
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C18H19FN4O3
|
1
|
| 1 |
Ki = 265.4 nM
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|
|
|
CP0868675
|
US9181230, 15
Show/Hide
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C17H16FN3O
|
1
|
| 1 |
Ki = 284.6 nM
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|
CP0387676
|
US10501411, Example 12
Show/Hide
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C18H20N2O
|
1
|
| 1 |
Ki = 289.9 nM
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|
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CP0425533
|
US10501411, Example 212
Show/Hide
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C25H24N2O5
|
1
|
| 1 |
Ki = 295.8 nM
|
|
|
|
CP0914326
|
US9452980, 76
Show/Hide
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C18H18N4O
|
1
|
| 1 |
Ki = 295.8 nM
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|
|
|
CP0419407
|
US9181230, 55
Show/Hide
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C17H14F3N3O2
|
1
|
| 1 |
Ki = 303.6 nM
|
|
|
|
CP0910425
|
US9181230, 37
Show/Hide
|
C18H17ClN4O
|
1
|
| 1 |
Ki = 303.6 nM
|
|
|
|
CP0512019
|
US9029370, 138
Show/Hide
|
C18H20FN3O3
|
1
|
| 1 |
Ki = 308.2 nM
|
|
|
|
CP0531314
|
US10501411, Example 10
Show/Hide
|
C17H25N3O
|
1
|
| 1 |
Ki = 309.2 nM
|
|
|
|
CP0513470
|
US10501411, Example 95
Show/Hide
|
C18H21N3O3
|
1
|
| 1 |
Ki = 321.6 nM
|
|
|
|
CP0481209
|
US10501411, Example 290
Show/Hide
|
C18H17N5O2S
|
1
|
| 1 |
Ki = 323.6 nM
|
|
|
|
CP0548091
|
US10501411, Example 36
Show/Hide
|
C23H21ClN2O
|
1
|
| 1 |
Ki = 323.9 nM
|
|
|
|
CP0387655
|
US10501411, Example 65
Show/Hide
|
C19H22N2O2
|
1
|
| 1 |
Ki = 352.3 nM
|
|
|
|
CP0574114
|
US10501411, Example 21
Show/Hide
|
C15H21N3O2
|
1
|
| 1 |
Ki = 359.1 nM
|
|
|
|
CP0499888
|
US9029370, 43
Show/Hide
|
C17H17Cl2N3O
|
1
|
| 1 |
Ki = 367.2 nM
|
|
|
|
CP0910426
|
US9181230, 30
Show/Hide
|
C20H19FN4O2
|
1
|
| 1 |
Ki = 373.6 nM
|
|
|
|
CP0386668
|
US10501411, Example 94
Show/Hide
|
C17H19N3O2
|
1
|
| 1 |
Ki = 378.7 nM
|
|
|
|
CP0561162
|
US10501411, Example 287
Show/Hide
|
C20H25N5O2
|
1
|
| 1 |
Ki = 378.9 nM
|
|
|
|
CP0532976
|
US9029370, 102
Show/Hide
|
C17H15ClN4O2
|
1
|
| 1 |
Ki = 409.9 nM
|
|
|
|
CP0468226
|
US9029370, 120
Show/Hide
|
C18H19FN4O4
|
1
|
| 1 |
Ki = 425.6 nM
|
|
|
|
CP0540192
|
US10501411, Example 255
Show/Hide
|
C18H26N2O3
|
1
|
| 1 |
Ki = 427.8 nM
|
|
|
|
CP0516887
|
US9181230, 54
Show/Hide
|
C17H14F3N3O2
|
1
|
| 1 |
Ki = 447.9 nM
|
|
|
|
CP0419305
|
US10501411, Example 28
Show/Hide
|
C16H23N3O
|
1
|
| 1 |
Ki = 473.3 nM
|
|
|
|
CP0557327
|
US9029370, 36
Show/Hide
|
C16H15Cl2N3O2
|
1
|
| 1 |
Ki = 488.3 nM
|
|
|
|
CP0425523
|
US9452980, 40
Show/Hide
|
C25H26ClN3O
|
1
|
| 1 |
Ki = 521.8 nM
|
|
|
|
CP0488842
|
US9029370, 101
Show/Hide
|
C17H15ClN4O2
|
1
|
| 1 |
Ki = 524 nM
|
|
|
|
CP0474484
|
US9029370, 98
Show/Hide
|
C17H15ClN4O2
|
1
|
| 1 |
Ki = 565 nM
|
|
|
|
CP0466882
|
US9029370, 135
Show/Hide
|
C18H17FN4O2
|
1
|
| 1 |
Ki = 578.3 nM
|
|
|
|
CP0563304
|
US10501411, Example 48
Show/Hide
|
C19H22N2O2
|
1
|
| 1 |
Ki = 613.2 nM
|
|
|
|
CP0565150
|
US11697636, Example 159
Show/Hide
|
C18H19ClN2O
|
1
|
| 1 |
Ki = 629.8 nM
|
|
|
|
CP0552284
|
US10501411, Example 66
Show/Hide
|
C19H19N3O
|
1
|
| 1 |
Ki = 644.7 nM
|
|
|
|
CP0393347
|
US10501411, Example 14
Show/Hide
|
C18H21N3O
|
1
|
| 1 |
Ki = 644.9 nM
|
|
|
|
CP0462834
|
US9029370, 119
Show/Hide
|
C18H19FN4O3
|
1
|
| 1 |
Ki = 686.8 nM
|
|
|
|
CP0548075
|
US10501411, Example 254
Show/Hide
|
C18H26N2O3
|
1
|
| 1 |
Ki = 725.5 nM
|
|
|
|
CP0423321
|
US10501411, Example 80
Show/Hide
|
C18H19ClN2O2
|
1
|
| 1 |
Ki = 741.8 nM
|
|
|
|
CP0488315
|
US9029370, 122
Show/Hide
|
C18H19ClN4O3
|
1
|
| 1 |
Ki = 758 nM
|
|
|
|
CP0965647
|
US9181230, 1
Show/Hide
|
C17H17N3O
|
1
|
| 1 |
Ki = 760 nM
|
|
|
|
CP0870565
|
US9181230, 21
Show/Hide
|
C18H17FN4O2
|
1
|
| 1 |
Ki = 895 nM
|
|
|
|
CP0554846
|
US9029370, 81
Show/Hide
|
C17H15FN4O2
|
1
|
| 1 |
Ki = 959.3 nM
|
|
|
|
CP0868680
|
US9181230, 45
Show/Hide
|
C15H15N3O
|
1
|
| 1 |
Ki = 1002.1 nM
|
|
|
|
CP0519674
|
US10501411, Example 9
Show/Hide
|
C18H21N3O
|
1
|
| 1 |
Ki = 1112.8 nM
|
|
|
|
CP0910995
|
US9181230, 16
Show/Hide
|
C19H21N3O
|
1
|
| 1 |
Ki = 1144.5 nM
|
|
|
|
CP0491062
|
US10501411, Example 106
Show/Hide
|
C17H17F2N3O
|
1
|
| 1 |
Ki = 1427.3 nM
|
|
|
|
CP0484076
|
US10501411, Example 75
Show/Hide
|
C16H15F2N3O
|
1
|
| 1 |
Ki = 1476.8 nM
|
|
|
|
CP0419404
|
US9181230, 22
Show/Hide
|
C19H19FN2O2
|
1
|
| 1 |
Ki = 1509.8 nM
|
|
|
|
CP0488320
|
US9029370, 33
Show/Hide
|
C19H17N5O2
|
1
|
| 1 |
Ki = 1511.2 nM
|
|
|
|
CP0942245
|
US9181230, 10
Show/Hide
|
C17H16FN3O
|
1
|
| 1 |
Ki = 1662.6 nM
|
|
|
|
CP0554032
|
US10501411, Example 49
Show/Hide
|
C19H22N2O2
|
1
|
| 1 |
Ki = 1684.8 nM
|
|
|
|
CP0566259
|
US10501411, Example 82
Show/Hide
|
C16H16FN3O
|
1
|
| 1 |
Ki = 1768.8 nM
|
|
|
|
CP0484057
|
US10501411, Example 215
Show/Hide
|
C24H21ClN2O5
|
1
|
| 1 |
Ki = 2310.1 nM
|
|
|
|
CP0549632
|
US10501411, Example 22
Show/Hide
|
C18H20N2O2
|
1
|
| 1 |
Ki = 2369.7 nM
|
|
|
|
CP0548092
|
US10501411, Example 41
Show/Hide
|
C18H20N2O
|
1
|
| 1 |
Ki = 2980.9 nM
|
|
|
|
CP0557328
|
US9029370, 42
Show/Hide
|
C17H18ClN3O2
|
1
|
| 1 |
Ki = 3989 nM
|
|
|
