Brief Information of the Cell Line and Protein
Cell Line ID: CL000006 , HEK293
Synonyms
Hek293
HEK-293
HEK/293
HEK 293
HEK;293
293
293 HEK
293 Ad5
Graham 293
Graham-293
Human Embryonic Kidney 293
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0045
Protein ID: PT03116 , Glutamate receptor 3
Gene Name GRIA3
Organism Rattus norvegicus, Rat
Protein Classification Ion channel
Uniprot ID P19492
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000006  Protein ID: PT03116
 
Compound ID Compound Name Compound Formula
CP0008940
(R,S)-alpha-amino-3-hydroxy-5-methyl-4-isooxazole-propionic acid
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C7H10N2O4
 1
1
EC50 = 37000 nM
   TI
   LI
   LO
   TS
CP0000105
(2S-(2alpha,3beta,4beta))-2-carboxy-4-(1-methylethenyl)-3-pyrrolidineacetic acid
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C10H15NO4
 1
1
EC50 = 40000 nM
   TI
   LI
   LO
   TS
CP0002355
(2S)-2-aminopentanedioic acid
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C5H9NO4
 1
1
EC50 = 52000 nM
   TI
   LI
   LO
   TS
CP0051516
1-[5-chloro-2-(5-oxo-4,5-dihydro-[1,2,4]oxadiazol-3-yl)-phenyl]-3-(3-bromophenyl)urea
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C15H10BrClN4O3
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0162369
2-(3-(3-bromophenyl)ureido)-4-chlorobenzoic acid
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C14H10BrClN2O3
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0312285
2-[3-(3-bromophenyl)ureido]-4-chlorobenzenesulfonic acid
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C13H10BrClN2O4S
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0346386
2-[2-[(3-bromophenyl)carbamoylamino]-4-chlorophenyl]acetic acid
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C15H12BrClN2O3
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0374730
4-Chloro-2-(3-naphthalen-2-yl-ureido)-benzoic acid
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C18H13ClN2O3
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0378727
1-(3-bromophenyl)-3-[5-chloro-2-(1H-tetrazol-5-yl-phenyl]urea
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C14H10BrClN6O
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS